Keywords: کیناز پولو مانند; Polo-like kinase; Acute myeloid leukemia; Myelodysplastic syndromes; Drug development;
مقالات ISI کیناز پولو مانند (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: کیناز پولو مانند; Anti-cancer drugs; Polo-like kinase; Structure-based drug design; Homology modelling; Molecular docking; Molecular dynamics simulation
Keywords: کیناز پولو مانند; Plk1; Polo-like kinase; Polo-box domain; Phosphoamino acid mimetic;
Novel compounds with potent CDK9 inhibitory activity for the treatment of myeloma
Keywords: کیناز پولو مانند; Cyclin dependent kinase inhibitor; 2,4-Disubstituted pyrimidine; Multiple myeloma; Polo-like kinase; DGGRGPAHRNGGGK-UHFFFAOYSA-N; IZZPOWGOQQEMLG-UHFFFAOYSA-N; XXDWIVIRVZIFRJ-UHFFFAOYSA-N; LJDYPDFYDYUVQU-UHFFFAOYSA-N; UCWVJKDAOWZSON-UHFFFAOYSA-N; POGNPTQDN
AGC kinases, mechanisms of regulation âand innovative drug development
Keywords: کیناز پولو مانند; AGC kinase; group of kinases related to PKA PKG and PKC; PKA; protein kinase A; PKC; protein kinase C; PKG; protein kinase G; PRK; protein kinase C related kinase (also termed PKN protein kinase N); PDK1; 3-phosphoinositide-dependent protein kinase 1; PKB
An open-label, phase II study of the polo-like kinase-1 (Plk-1) inhibitor, BI 2536, in patients with relapsed small cell lung cancer (SCLC)
Keywords: کیناز پولو مانند; Small cell lung cancer; Plk-1 inhibition; Polo-like kinase; BI 2536;
RNAi prodrugs targeting Plk1 induce specific gene silencing in primary cells from pediatric T-acute lymphoblastic leukemia patients
Keywords: کیناز پولو مانند; RNAi prodrug; RNA interference; Polo-like kinase; Pediatric leukemia; Drug delivery; BI6727;
Depletion of the mitotic kinase Cdc5p in Candida albicans results in the formation of elongated buds that switch to the hyphal fate over time in a Ume6p and Hgc1p-dependent manner
Keywords: کیناز پولو مانند; Candida albicans; Cdc5p; Polo-like kinase; Hyphae; Mitosis; Hyphal-specific genes expression; UME6;
Modulating angiogenesis with integrin-targeted nanomedicines
Keywords: کیناز پولو مانند; (RGD)m; RGD mimetics; 4-NQO; 4-nitroquinoline 1-oxide; AAA; Abdominal Aortic Aneurysms; ADA; 8-Amino-3,6-Dioxaoctonoic Acid; AH-GDM; Aminohexyl-Geldanamycin; ami; Amide; AP-2α; Activating Protein 2α; ARMS; Alveolar Rhabdomyosarcoma; ATO; Arsenic Trioxid
Studying mechanisms of cAMP and cyclic nucleotide phosphodiesterase signaling in Leydig cell function with phosphoproteomics
Keywords: کیناز پولو مانند; AC; adenylyl cyclase; ACTH; adrenocorticotropic hormone; AKAP; A-kinase anchor protein; AMP; 5â² adenosine monophosphate; AMPK; AMP-activated protein kinase; Arfgap1; ADP-ribosylation factor GTPase-activating protein 1; Arhgef2; Rho guanine nucleotide ex
Emerging role of protein phosphatases changes the landscape of phospho-signaling in DNA damage response
Keywords: کیناز پولو مانند; 53BP1; p53 binding protein 1; ATM; ataxia-telangiectasia mutated; ATR; ataxia telangiectasia and Rad3 related; BLM; blooms syndrome RecQ helicase-like, human homolog of SGS1; BRCA1; breast cancer 1, early onset; CDC; cell division cycle; CDK; cyclin depen
Ser129 phosphorylation of endogenous α-synuclein induced by overexpression of polo-like kinases 2 and 3 in nigral dopamine neurons is not detrimental to their survival and function
Keywords: کیناز پولو مانند; α-Synuclein; Phosphorylation; Polo-like kinase; Adeno-associated vector; Parkinson's disease
In vivo modulation of polo-like kinases supports a key role for PLK2 in Ser129 α-synuclein phosphorylation in mouse brain
Keywords: کیناز پولو مانند; ANOVA; analysis of variance; Ce; cerebellum; CEB; cell extraction buffer; CHAPS; 3-[(3-cholamidopropyl)dimethylammonio]-1-propanesulfonate; Co; cerebral cortex; CSNK2a2; alpha prime subunit of casein kinase II; EDTA; ethylenediaminetetraacetic acid; EGTA;
Sequential Cdk1 and Plk1 phosphorylation of caspase-8 triggers apoptotic cell death during mitosis
Keywords: کیناز پولو مانند; Cell cycle; Apoptosis; Polo-like kinase;
Small-molecular, non-peptide, non-ATP-competitive polo-like kinase 1 (Plk1) inhibitors with a terphenyl skeleton
Keywords: کیناز پولو مانند; Polo-like kinase; Inhibitor; Small molecule; Terphenyl skeleton; Non-peptide; Non-ATP-competitive
Enhanced gemcitabine-mediated cell killing of human lung adenocarcinoma by vector-based RNA interference against PLK1
Keywords: کیناز پولو مانند; RNA interference; Polo-like kinase; Gemcitabine
5-(2-Amino-pyrimidin-4-yl)-1H-pyrrole and 2-(2-amino-pyrimidin-4-yl)-1,5,6,7-tetrahydro-pyrrolo[3,2-c]pyridin-4-one derivatives as new classes of selective and orally available Polo-like kinase 1 inhibitors
Keywords: کیناز پولو مانند; PLK1; Polo-like kinase; PLK2 and PLK3; Cell cycle; Cellular activity; Crystal structure;
Synthesis and biological evaluation of benzyl styrylsulfonyl derivatives as potent anticancer mitotic inhibitors
Keywords: کیناز پولو مانند; Mitotic inhibitor; Polo-like kinase; Serine/threonine kinase; Anticancer therapy
NMS-P937, a 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivative as potent and selective Polo-like kinase 1 inhibitor
Keywords: کیناز پولو مانند; PLK1; Polo-like kinase; Kinase inhibitor; In vivo activity; Phase I clinical trials
Serine phosphorylation regulates disabled-1 early isoform turnover independently of Reelin
Keywords: کیناز پولو مانند; ApoER2; apolipoprotein E receptor 2; CsA; cyclosporine A; Cdk; cyclin dependent kinase; Dab1; Disabled-1; CHX; cycloheximide; CPTS; 3,4',4â³,4-copper phthalocyanine tetrasulfonic acid, tetrasodium salt; CsA; cyclosporine A; ED; embryonic day; GSK3; glyco
4,5-Dihydro-1H-pyrazolo[4,3-h]quinazolines as potent and selective Polo-like kinase 1 (PLK1) inhibitors
Keywords: کیناز پولو مانند; PLK1; Polo-like kinase; Kinase inhibitor; In vivo activity
Heteroaryl-linked 5-(1H-benzimidazol-1-yl)-2-thiophenecarboxamides: Potent inhibitors of polo-like kinase 1 (PLK1) with improved drug-like properties
Keywords: کیناز پولو مانند; PLK1; Polo-like kinase; Kinase inhibitor; CYP450 inhibition; Mouse iv clearance; Solubility;
Schistosoma mansoni Polo-like kinase 1: A mitotic kinase with key functions in parasite reproduction
Keywords: کیناز پولو مانند; Schistosoma mansoni; Polo-like kinase; Reproduction; Kinase inhibitor
Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein binding
Keywords: کیناز پولو مانند; Polo-like kinase; Anti-mitotic; Cell cycle inhibitor; Thiophene; Solubility; Protein binding
Imidazopyridine derivatives as potent and selective Polo-like kinase (PLK) inhibitors
Keywords: کیناز پولو مانند; PLK1; Polo-like kinase; Imidazopyridine
Development of high-throughput assays based on fluorescence polarization for inhibitors of the polo-box domains of polo-like kinases 2 and 3
Keywords: کیناز پولو مانند; Assay; Fluorescence polarization; High-throughput screening; Polo-like kinase; PBD; Plk2; Plk3;
Theoretical model of treatment strategies for clear cell carcinoma of the ovary: Focus on perspectives
Keywords: کیناز پولو مانند; Ovarian clear cell carcinoma; Renal cell carcinoma; Hepatocyte nuclear factor-1beta; Polo-like kinase; Molecular target
Transcriptional regulation of human polo-like kinases and early mitotic inhibitor
Keywords: کیناز پولو مانند; polo-like kinase; early mitotic inhibitor; cell cycle; E2F; promoter; gene regulation
Anti-breast cancer activity of LFM-A13, a potent inhibitor of Polo-like kinase (PLK)
Keywords: کیناز پولو مانند; Polo-like kinase; Mitosis; Transgenic mouse; Cancer
Mitotic drug targets and the development of novel anti-mitotic anticancer drugs
Keywords: کیناز پولو مانند; Mitosis; Chemotherapy; Spindle checkpoint; Aurora kinase; Polo-like kinase; KSP; Eg5; Microtubules; Taxanes; Vinca alkaloids; UCN-01; G2 checkpoint; Anticancer drug resistance
What's new in pancreatic cancer treatment pipeline?
Keywords: کیناز پولو مانند; vascular endothelial growth factor (VEGF); epidermal growth factor receptor (EGFR); gastrin; hypoxia inducible factor alpha (HIF-1α); vaccine; thioredoxin reductase; polo-like kinase; thioredoxin; gemcitabine; bevacizumab; cetuximab; TNFerade; sorafenib;
Overexpression of polo-like kinase 1 is a common and early event in pancreatic cancer
Keywords: کیناز پولو مانند; Polo-like kinase; Pancreatic carcinoma; Immunohistochemistry; Pancreatic intraepithelial neoplasia; Prognosis;
Influence of neuroendocrine tumor cells on proliferation in prostatic carcinoma
Keywords: کیناز پولو مانند; PLK; Polo-like kinase; PCa; Prostatic carcinoma; CgA; Chromogranin A; NE; Neuroendocrine; HNE; High neuroendocrine differentiation; LNE; Low neuroendocrine differentiation; PI; Proliferation index; Ki-67; Neuroendocrine tumor differentiation; PLK1; Prolif
Protective effect of FK506 against apoptosis of SH-SY5Y cells correlates with regulation of the serum inducible kinase gene
Keywords: کیناز پولو مانند; FK506; the immunosuppressive macrolactamlactone tacrolimus; SNK; serum inducible kinase; FNK; fibroblast growth factor inducible kinase; Plk; polo-like kinase; NF-IL3; nuclear factor interleukin-3; CRE; cAMP response element; CREB; cAMP response element b