Keywords: Multiple Sclerosis (MS); Normal-appearing white matter (NAWM); Microglia; Axon; Inflammation; VCAM-1; Sphingosine; S1P1; Wallerian degeneration;
مقالات ISI (ترجمه نشده)
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Keywords: ASC; apoptosis-associated speck-like protein containing a caspase recruitment domain; DAMPs; danger associated molecular patterns; EAE; experimental autoimmune encephalomyelitis; HER2; human epidermal growth factor related receptor 2; ERK; extracellular s
Keywords: Sphingosine 1-phosphate; Sphingosine 1-phosphate receptor; S1P1; S1pr1; GPCR; Cardiomyocyte; Noncompaction; Heart development;
Keywords: SSc; systemic sclerosis; SRC; scleroderma renal crisis; PAH; pulmonary arterial hypertension; SMR; standardized mortality ratio; DNMTs; DNA methyltransferases; SAM; S-adenosyl-methionine; 5mC; 5-methylcytosine; MBD; methyl-CpG-binding domain; Tet; ten-e
Keywords: SphK1; sphingosine kinase 1; S1P1; sphingosine-1-phosphate (S1P) receptor 1; ECs; endothelial cells; E2; 17β-estradiol; ER; estrogen receptor; Akt; protein kinase B; eNOS; endothelial nitric oxide (NO) synthase; HUVEC; human umbilical vein endothelial ce
Keywords: αSMA; α-smooth muscle actin; ATX; autotaxin or ectonucleotide pyrophosphatase/phosphodiesterase 2; Cd; cadmium; CdCl2; cadmium chloride; LC-MS/MS; chromatography-tandem mass spectrometry; DMEM; dulbecco's modified Eagle's medium; FCS; fetal calf
Long noncoding RNA LISPR1 is required for S1P signaling and endothelial cell function
Keywords: COPD; Chronic obstructive pulmonary disease; CTEPH; Chronic thromboembolic pulmonary hypertension; CRISPR/Cas9; Clustered Regularly Interspaced Short Palindromic Repeats/CRISPR associated protein 9; HUVEC; Human umbilical vein endothelial cells; IPAH; Idi
FOXOs in cancer immunity: Knowns and unknowns
Keywords: 2B4; CD244 molecule; AKT or PKB; protein kinase B; APCs; antigen-presenting cells; ARG1; arginase 1; BEC; blood endothelial cell; BLNK; B cell Linker protein; BMP; bone morphogenetic protein; BTK; Bruton tyrosine kinase; C/EBP; CCAAT/enhancer-binding prot
Identification and synthesis of potent and selective pyridyl-isoxazole based agonists of sphingosine-1-phosphate 1 (S1P1)
Keywords: Sphingosine-1-phosphate; Sphingosine-1-phosphate 1; S1P1; Isoxazole; FTY720; Fingolimod;
Synthesis, identification, and biological activity of metabolites of two novel selective S1P1 agonists
Keywords: S1P1; Metabolites; Monohydroxylated products;
Late-stage optimization of a tercyclic class of S1P3-sparing, S1P1 receptor agonists
Keywords: SFBFJQXHRYGKHV-INIZCTEOSA-N; SDCQNJRPSLMFIT-SFHVURJKSA-N; GMEODUAZQQLOFF-MRXNPFEDSA-N; MUINZQQLLPFAQS-OAHLLOKOSA-N; S1P1; S1P3; Solubility; Autoimmune;
Functional role of inorganic trace elements in angiogenesis part III: (Ti, Li, Ce, As, Hg, Va, Nb and Pb)
Keywords: As; arsenic; FGF-2; basic fibroblast growth factor; BMP-2; bone morphogenetic protein-2; Ce; cerium; COX; cyclooxygenase; EC; endothelial cells; EPCR; endothelial cell protein C receptor; EPCs; endothelial progenitor cells; EMT; epithelial to mesenchymal
Imaging S1P1 activation in vivo
Keywords: S1P1; sphingosine-1-phosphate receptor 1; S1P; sphingosine-1-phosphate; GPCR; G protein-coupled receptor; ApoM; apolipoprotein M; HDL; high-density lipoprotein; HEV; high endothelial venules; MS; multiple sclerosis; tTA; tetracycline transcriptional activ
Design and synthesis of new tricyclic indoles as potent modulators of the S1P1 receptor
Keywords: S1P1; Sphingosine-1-phosphate; Gilenya®
Different Correlation of Sphingosine-1-Phosphate Receptor 1 with Receptor Activator of Nuclear Factor Kappa B Ligand and Regulatory T Cells in Rat Periapical Lesions
Keywords: Bone resorption; osteoclast; periapical lesions; RANKL; regulatory T cells; S1P1;
Cbl-b-deficient mice express alterations in trafficking-related molecules but retain sensitivity to the multiple sclerosis therapeutic agent, FTY720
Keywords: CBLB/Cbl-b; Casitas-B lineage lymphoma-b; Cbl-bâ/â; Cbl-b-deficient; RRMS; relapsing remitting MS; S1P; sphingosine-1-phosphate; S1P1; sphingosine-1-phosphate receptor 1; THI; 2-acetyl-4-tetrahydroxybutyl imidazole; SEW2871; 5-[4-phenyl-5-(trifluorome
Sphingosine 1-phosphate induced anti-atherogenic and atheroprotective M2 macrophage polarization through IL-4
Keywords: S1P; sphingosine 1-phosphate; GPCR; G-protein-coupled receptor; S1P1; sphingosine 1-phosphate receptor type 1 (EDG1); LPS; lipopolysaccharide; iNOS; inducible nitric oxide synthase; COX-2; cyclooxygenase 2; NF-κB; nuclear factor kappa B; STAT6; signal tr
Second generation S1P pathway modulators: Research strategies and clinical developments
Keywords: Immunomodulator; S1P modulator; S1P1; Fingolimod
Isoform-selective thiazolo[5,4-b]pyridine S1P1 agonists possessing acyclic amino carboxylate head-groups
Keywords: Sphingosine-1-phosphate receptor; S1P1; Thiazolo[5,4-b]pyridine; Agonist; Immunosuppression
Discovery of CS-2100, a potent, orally active and S1P3-sparing S1P1 agonist
Keywords: S1P1; Agonist; CS-2100; Lymphocyte; HvGR
Synthesis and SAR of 1,3-thiazolyl thiophene and pyridine derivatives as potent, orally active and S1P3-sparing S1P1 agonists
Keywords: S1P1; Agonist; Lymphocyte; HvGR;
Blocking S1P interaction with S1P1 receptor by a novel competitive S1P1-selective antagonist inhibits angiogenesis
Keywords: S1P; sphingosine 1-phosphate; S1P1; the type 1 sphingosine 1-phosphate (S1P) G protein-coupled receptor; Ab; antibody; HUVEC; human umbilical vein endothelial cells; FBS; fetal bovine serum; BSA; bovine serum albumin; ECs; endothelial cells; PDGF; platele
Lymphopenia induced by a novel selective S1P1 antagonist structurally unrelated to S1P
Keywords: S1P; sphingosine 1-phosphate; S1P1; type 1 sphingosine 1-phosphate receptor; CHS; contact hypersensitivity response; HEK293; human embryonic kidney cell line; CHO-K1; Chinese hamster ovary cell line; HTS; high-throughput screening; GTP; guanosine-5â²-tri
Synthesis and evaluation of CS-2100, a potent, orally active and S1P3- sparing S1P1 agonist
Keywords: S1P1; Agonist; CS-2100; Lymphocyte; Adjuvant-induced arthritis; EAE; Multiple sclerosis
A polysaccharides MDG-1 augments survival in the ischemic heart by inducing S1P release and S1P1 expression
Keywords: HMEC-1; human microvascular endothelial cells-1; OGD; oxygen glucose deprivation; S1P; sphingosine 1-phosphate; SPHK; sphingosine kinase; S1P1; sphingosine 1-phosphate receptor 1; ERK; extracellular signal regulated kinase; SH; sham operation; AMI; acute
Propentofylline, a CNS glial modulator does not decrease pain in post-herpetic neuralgia patients: In vitro evidence for differential responses in human and rodent microglia and macrophages
Keywords: ATP; adenosine tri-phosphate; BPI-sf; brief pain inventory short form; CNS; central nervous system; GFAP; glial fibrillary acidic protein; GM-CSF; granulocyte macrophage colony stimulating factor; Iba-1; ionized calcium binding adaptor molecule 1; IC50; i
The sphingosine-1-phosphate receptor-1 antagonist, W146, causes early and short-lasting peripheral blood lymphopenia in mice
Keywords: S1P; sphigosine-1-phosphate; S1P1; sphingosine-1-phosphate receptor 1; Sphingosine-1-phosphate receptors; Lymphocytes; Lymph nodes; Lymphopenia; W146; S1P1 agonists;
Discovery of a novel series of potent S1P1 agonists
Keywords: S1P1; Sphingosine-1-phosphate; Structure–activity relationships; Hit-to-lead; Lymphopenia
Sphingosine-1-phosphate receptor S1P1 is regulated by direct interactions with P-Rex1, a Rac guanine nucleotide exchange factor
Keywords: Sphingosine-1-phosphate; S1P1; P-Rex1; Cell migration; PDZ domain
Sphingosine kinase-1/S1P1 signalling axis negatively regulates mitogenic response elicited by PDGF in mouse myoblasts
Keywords: S1P; sphingosine 1-phoshate; SK; sphingosine kinase; S1PR; S1P receptor; DMEM; Dulbecco's modified Eagle's medium; BSA; bovine serum albumin; FCS; fetal calf serum; siRNA; short interfering RNA; SDS; sodium dodecyl sulphate; PAGE; polyacrylamide gel elect
Role of sphingosine kinase 1 in allergen-induced pulmonary vascular remodeling and hyperresponsiveness
Keywords: Pulmonary arterial hypertension; allergen-induced lung inflammation; vascular remodeling; perfused mouse lung; sphingosine kinase; sphingosine 1-phosphate; BAL; Bronchoalveolar lavage; CT; Threshold cycle; G-CSF; Granulocyte colony-stimulating factor; HPR
S1P1 overexpression stimulates S1P-dependent chemotaxis of human CD34+ hematopoietic progenitor cells but strongly inhibits SDF-1/CXCR4-dependent migration and in vivo homing
Keywords: PBPCs, mobilized peripheral blood progenitor cells; HSC, hematopoietic stem cells; S1P, sphingosine-1-phophate; LPA, lysophosphatidic acid; SDF-1stromal cell-derived, factor 1HSC; S1P1; CXCR4; SDF-1; Migration; Homing
Sphingosine 1-phosphate regulates inflammation-related genes in human endothelial cells through S1P1 and S1P3
Keywords: S1P; S1P1; S1P3; Endothelial cells
Trichostatin A and 5-aza-2′-deoxycytidine switch S1P from an inhibitor to a stimulator of motility through epigenetic regulation of S1P receptors
Keywords: Sphingosine-1-phosphate; S1P1; S1P2; S1P3; Trichostatin A; Motility; EpigeneticAza-dC, 5′-aza-2′-deoxycytidine; ATX, autotaxin; DMEM, Dulbecco’s minimum essential medium; DNMT, DNA methyltransferase; EDG, endothelial differentiation gene; GPCR, G-protein-
Changes in S1P1 and S1P2 expression during embryonal development and primitive endoderm differentiation of F9 cells
Keywords: Sphingolipid; Sphingosine 1-phosphate; S1P receptor; S1P1; Embryonal development; Differentiation; Endoderm; F9 cells
Synthesis of 4(5)-phenylimidazole-based analogues of sphingosine-1-phosphate and FTY720: Discovery of potent S1P1 receptor agonists
Keywords: S1P receptor agonists; FTY720; S1P1; Bradycardia; Phosphothioate; Sphingosine-1-phosphate
FTY720, a new class of immunomodulator, inhibits lymphocyte egress from secondary lymphoid tissues and thymus by agonistic activity at sphingosine 1-phosphate receptors
Keywords: AZ; azathioprine; CI; combination index; CsA; cyclosporin A; EAE; experimental autoimmune encephalomyelitis; FK506; tacrolimus; FTY720; 2-amino-2-[2-(4-octylphenyl)ethyl]propane-1,3-diol hydrochloride; FTY720-P; FTY720-phosphate; GvHR; graft versus host r