دانلود مقالات ISI درباره Sar + ترجمه فارسی

Landslide deformation monitoring using point-like target offset tracking with multi-mode high-resolution TerraSAR-X data

Keywords: Landslide; SAR; Point-like target offset tracking; Displacement; Water level; Three Gorges

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

Motor and Nonmotor Circuitry Activation Induced by Subthalamic Nucleus Deep Brain Stimulation in Patients With Parkinson Disease

Keywords: BOLD; blood oxygen level-dependent; DBS; deep brain stimulation; FDR; false discovery rate; fMRI; functional magnetic resonance imaging; GE-EPI; gradient echo-echo planar imaging; MP-RAGE; magnetization-prepared rapid gradient-echo; PD; Parkinson dise

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

Design, synthesis and biological evaluation of novel tetrahydroisoquinoline derivatives as potential PDE4 inhibitors

Keywords: 7-(Cyclopentyloxy)-6-methoxy-1,2,3,4-tetrahydroisoquinoline derivatives; Synthesis; PDE4 inhibitor; SAR; Molecular simulation;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

Use of read-across and computer-based predictive analysis for the safety assessment of PEG cocamines

Keywords: CIR; Cosmetic Ingredient Review; GD; gestation day; LOAEL; lowest observed adverse effect level; NOAEL; no observed adverse effect level; NOEL; no observed effect level; PEG; polyethylene glycol; SAR; structure-activity relationship; SOI; structure of i

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Targeting G-quadruplex nucleic acids with heterocyclic alkaloids and their derivatives

Keywords: G-Quadruplex; Heterocyclic alkaloid; Alkaloid derivative; Bioactivity; Anti-cancer; G4s; G-quadruplexes; rDNA; ribosomal DNA; PQS; putative G-quadruplex forming sequences; POT1; the protection of telomeres 1; TRF1 and TRF2; the telomeric repeat binding fa

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Design, synthesis and biological activities of novel oxazolo[4,5-g]quinazolin-2(1H)-one derivatives as EGFR inhibitors

Keywords: EGFR inhibitor; Oxazolo[4,5-g]quinazolin-2(1H)-one scaffold; Protein tyrosine kinases (PTK); Docking; SAR;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Benzoic acid derivatives with improved antifungal activity: Design, synthesis, structure-activity relationship (SAR) and CYP53 docking studies

Keywords: Benzoic acid; CYP53; Cytochrome P450; SAR; Molecular modeling; Molecular docking; Antifungal activity;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Soil moisture retrieval model by using RISAT-1, C-band data in tropical dry and sub-humid zone of Bankura district of India

Keywords: SAR; RISAT-1; Soil moisture; Semi-empirical model

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Evaluation of the operational SAR based Baltic Sea ice concentration products

Keywords: SAR; Sea ice; Ice concentration; Operational; Evaluation;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-activity relationship studies of pyrimidine-2,4-dione derivatives as potent P2X7 receptor antagonists

Keywords: P2X7 receptor; Antagonists; KN-62; Structure-activity relationships; IL-1β; Inflammation; AcCl; acetyl chloride; ACN; acetonitrile; ATP; adenosine-5′-triphosphate; BzATP; 2′(3′)-O-(4-benzoylbenzoyl)-ATP; DCM; dichloromethane; DMEM; Dulbecco's Mod

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

4G antennas for wireless eyewear devices and related SAR

Keywords: Eyewear device; Coupling element; LTE; SAR; Lunettes connectées; Élément de couplage; LTE; DAS;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2015 سفارش ترجمه

Conformationally restricted κ-opioid receptor agonists: Synthesis and pharmacological evaluation of diastereoisomeric and enantiomeric decahydroquinoxalines

Keywords: κ agonists; κ-Opioid receptor; Decahydroquinoxalines; Diastereoisomers; Resolution of enantiomers; Hydrogenation; SAR; Relationship between configuration and κ affinity;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2015 سفارش ترجمه

An overview of integrated remote sensing and GIS for groundwater mapping in Egypt

Keywords: ALOS; Advanced Land Observing Satellite; ASTER; Advanced Spaceborne Thermal Emission and Reflection Radiometer; IWACO; Consultants for Water and Environment; DEM; Digital Elevation Model; FAO; Food and Agricultural Organization; GIS; Geographic Informatio

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2015 سفارش ترجمه

Molecular descriptors calculation as a tool in the analysis of the antileishmanial activity achieved by two series of diselenide derivatives. An insight into its potential action mechanism

Keywords: Leishmania; Diselenide; Diselenosulfonamides; Molecular descriptors; SAR

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

Novel benzidine and diaminofluorene prolinamide derivatives as potent hepatitis C virus NS5A inhibitors

Keywords: HCV; NS5A inhibitor; Benzidine; Diaminofluorene; Structure-activity relationship; HCV; hepatitis C virus; Peg-IFNα; pegylated interferon α; SVR; sustained virological response; GT1a; hepatitis C virus genotype 1a, a subtype of hepatitis C virus genoty

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

The importance of the 6- and 7-positions of tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor

Keywords: BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium 3-oxid hexafluorophosphate; HPLC; high performance liquid chromatography; OX1; orexin 1 receptor; OX2;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

Design, synthesis and evaluation of novel 5-phenylpyridin-2(1H)-one derivatives as potent reversible Bruton’s tyrosine kinase inhibitors

Keywords: Reversible Btk inhibitors; Structure; SAR; Efficacy; In vivo

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

Savannah woody structure modelling and mapping using multi-frequency (X-, C- and L-band) Synthetic Aperture Radar data

Keywords: Woody structure; Savannahs; SAR; Multi-frequency; LiDAR; Random Forest

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase

Keywords: TB; tuberculosis; Mtb; Mycobacterium tuberculosis; MIC; minimal inhibitory concentration; CYP; cytochrome P450; SAR; structure-activity relationships; MMIC; mammalian cytotoxicity; DprE1; decaprenylphosphoryl-β-d-ribose 2′-oxidase; TEA; triethylamine

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

Offshore wind climatology based on synergetic use of Envisat ASAR, ASCAT and QuikSCAT

Keywords: Offshore wind; SAR; QuikSCAT; ASCAT; Wind energy; Resource; Northern Europe;

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

Strengths and weaknesses of multi-year Envisat ASAR backscatter measurements to map permanent open water bodies at global scale

Keywords: Water body; SAR; Backscatter; Envisat ASAR; C-band; Land cover;

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

The Kennaugh element framework for multi-scale, multi-polarized, multi-temporal and multi-frequency SAR image preparation

Keywords: Radar; SAR; Imagery; Multifrequency; Multisensor; Multitemporal; Multiresolution; Change detection; Application; Combination; Polarization;

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2015 سفارش ترجمه

(Q)SAR modelling of nanomaterial toxicity: A critical review

Keywords: AES; Auger electron spectroscopy; AFM; atomic force microscopy; ANNs; artificial neural networks; APO or Apop.; apoptosis; ATP; adenosine triphosphate (ATP); BET; Brunauer-Emmett-Teller; BSAI; biological surface adsorption index; CNTs; carbon nanotube

دانلود رایگان متن کامل مقاله ISI 19 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-activity relationship of flavonoids as potent inhibitors of carbonyl reductase 1 (CBR1)

Keywords: CBR; carbonyl reductase; DOX; doxorubicin; Hydroxy-PP; 3-(1-tert-butyl-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenol; SAR; structure-activity relationship; S-Tetralol; (S)-(+)-1,2,3,4-tetrahydro-1-naphthol; Acacetin (PubChem CID: 5280442); Apigenin (P

دانلود رایگان متن کامل مقاله ISI 22 صفحه سال انتشار : 2015 سفارش ترجمه

Design, synthesis and SAR studies of GABA uptake inhibitors derived from 2-substituted pyrrolidine-2-yl-acetic acids

Keywords: CNS; GABA uptake; SAR; 2-Substituted pyrrolidine-2-yl-acetic acid; N-Acylpyrrolidinium ion

دانلود رایگان متن کامل مقاله ISI 23 صفحه سال انتشار : 2015 سفارش ترجمه

Flupyradifurone (Sivanto™) and its novel butenolide pharmacophore: Structural considerations

Keywords: ACh; acetylcholine; BgTx; bungarotoxin; CNS; central nervous system; DFT; density functional theory; FPF; flupyradifurone; IMD; imidacloprid; IRM; insect resistance management; IRAC; Insecticide Resistance Action Committee; nAChR; nicotinic acetylcholine

دانلود رایگان متن کامل مقاله ISI 23 صفحه سال انتشار : 2015 سفارش ترجمه

Structure activity relationship (SAR) study of benzimidazole scaffold for different biological activities: A mini-review

Keywords: Anthelmintics; Benzimidazole; Heterocyclic ring systems; Pharmacological activities; SAR study; NPY; neuropeptide; CYP450; cytochrome P450; HBV; hepatitis B virus; HCV; hepatitis C virus; RSV; respiratory syncytial virus; VV; varicella virus; BVDV; bovine

دانلود رایگان متن کامل مقاله ISI 25 صفحه سال انتشار : 2015 سفارش ترجمه

Segmented TOF at 7 T MRI: Technique and clinical applications

Keywords: Segmented TOF; 7 T; Venous suppression; SAR; MR angiography;

دانلود رایگان متن کامل مقاله ISI 28 صفحه سال انتشار : 2015 سفارش ترجمه

Pyrrolo[2,3-b]pyridine derivatives as potent Bruton's tyrosine kinase inhibitors

Keywords: BTK kinase; Inhibitor; Pyrrolo[2,3-b]pyridine; SAR;

دانلود رایگان متن کامل مقاله ISI 33 صفحه سال انتشار : 2015 سفارش ترجمه

Discovery of novel Bruton's tyrosine kinase (BTK) inhibitors bearing a pyrrolo[2,3-d]pyrimidine scaffold

Keywords: BTK inhibitors; Pyrrolo[23-d]pyrimidine; SAR;

دانلود رایگان متن کامل مقاله ISI 35 صفحه سال انتشار : 2015 سفارش ترجمه

A subset of N-substituted phenothiazines inhibits NADPH oxidases

Keywords: CHO; Chinese hamster ovary; DMSO; dimethyl sulfoxide; DUOX; dual oxidase; DMEM; Dulbecco׳s modified Eagle medium; DPI; diphenyleneiodonium; ESP; electrostatic potential; FBS; fetal bovine serum; GFP; green fluorescent protein; HBSS; Hanks׳ buffered salt

دانلود رایگان متن کامل مقاله ISI 37 صفحه سال انتشار : 2015 سفارش ترجمه

Interrogating alkyl and arylalkylpolyamino (bis)urea and (bis)thiourea isosteres as potent antimalarial chemotypes against multiple lifecycle forms of Plasmodium falciparum parasites

Keywords: GVBYQYRUQTVCSX-UHFFFAOYSA-N; CWGWQODLMSBNJO-UHFFFAOYSA-N; RIJOLQPUEHMLBL-UHFFFAOYSA-N; INWXGCBOYRSOBH-UHFFFAOYSA-N; PHXRNBAPWQWFIU-UHFFFAOYSA-N; ITLCJTLROKBPIR-UHFFFAOYSA-N; WRZLHNOERLQPKX-UHFFFAOYSA-N; OQVYIEDMQNROCP-UHFFFAOYSA-N; BRVMEZRDZYMOLC-UHFFFAOY

دانلود رایگان متن کامل مقاله ISI 39 صفحه سال انتشار : 2015 سفارش ترجمه

Post-HTS case report and structural alert: Promiscuous 4-aroyl-1,5-disubstituted-3-hydroxy-2H-pyrrol-2-one actives verified by ALARM NMR

Keywords: acetyl-CoA; acetyl coenzyme A; ALARM NMR; a La assay to detect reactive molecules by nuclear magnetic resonance; Asf1; anti-silencing function 1; AZ; AstraZeneca; BME; β-mercaptoethanol; BSA; bovine serum albumin; CoA; coenzyme A; CPM; N-[4-(7-diethylami

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2015 سفارش ترجمه

Pyrazoloquinazolines: Synthetic strategies and bioactivities

Keywords: Pyrazoloquinazolines; Synthetic strategies; Biological activities; SAR; QSAR; Docking;

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2015 سفارش ترجمه

Design, chemical synthesis and biological evaluation of 3-spiromorpholinone/3-spirocarbamate androsterone derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 3

Keywords: ADT; androsterone; AR; androgen receptor; Ar; aryl group; DBD; DNA binding domain; DCM; dichloromethane; DHT; dihydrotestosterone; DIPEA; N,N-diisopropylethylamine; DMF; dimethylformamide; DMSO; dimethylsulfoxide; Δ4-dione; 4-androstene-3,17-dione; EtOAc

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2015 سفارش ترجمه

Discovery of InhA inhibitors with anti-mycobacterial activity through a matched molecular pair approach

Keywords: Antibiotics; Enoyl-acyl carrier protein reductase (InhA); In silico drug screening; Mycobacterium tuberculosis; Matched molecular pair (MMP); TB; tuberculosis; MDR; multi-drug-resistant; XDR; extensively drug-resistant; HIV; human immunodeficiency virus;

دانلود رایگان متن کامل مقاله ISI 45 صفحه سال انتشار : 2015 سفارش ترجمه

Naturally occurring plant isoquinoline N-oxide alkaloids: Their pharmacological and SAR activities

Keywords: Alkaloids; Isoquinoline; Anticancer; Antibacterial; SAR; Activities;

دانلود رایگان متن کامل مقاله ISI 48 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-based design and synthesis of covalent-reversible inhibitors to overcome drug resistance in EGFR

Keywords: CRI; covalent reversible inhibitor; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt; hydroxybenzotriazole; DIPEA; N,N-diisopropylethylamine; EGFR; epidermal growth factor receptor; NOE; nuclear Overhauser effect; NSCLC; non-sma

دانلود رایگان متن کامل مقاله ISI 48 صفحه سال انتشار : 2015 سفارش ترجمه

3-Nitrotriazole-based piperazides as potent antitrypanosomal agents

Keywords: Nitrotriazoles; Piperazides; Trypanocidal; Leishmanicidal; Chagas disease; NTD; neglected tropical diseases; T. brucei; Trypanosoma brucei; HAT; human African trypanosomiasis; T. cruzi; Trypanosoma cruzi; Bnz; benznidazole (N-benzyl-2-(2-nitro-1H-imidaz

دانلود رایگان متن کامل مقاله ISI 60 صفحه سال انتشار : 2015 سفارش ترجمه

Stereoselective synthesis, biological evaluation, and modeling of novel bile acid-derived G-protein coupled Bile acid receptor 1 (GP-BAR1, TGR5) agonists

Keywords: GPCR; G protein-coupled receptor; BAs; bile acids; CDCA; chenodeoxycholic acid; CA; cholic acid; LCA; lithocholic acid; UDCA; ursodeoxycholic acid; FXR; farnesoid X receptor; NRs; nuclear receptors; LBD; ligand-binding domain; cAMP; cyclic adenosine monop

دانلود رایگان متن کامل مقاله ISI 62 صفحه سال انتشار : 2015 سفارش ترجمه

Metabolically programmed iron chelators

Keywords: NTBI; nontransferrin-bound iron; DFO; desferrioxamine; sc; subcutaneously; DFT; desferrithiocin; DADFT; desazadesferrithiocin; s.i.d.; once daily; b.i.d.; twice daily; BUN; blood urea nitrogen; SCr; serum creatinine; GI; gastrointestinal; ICE; iron cleari

دانلود رایگان متن کامل مقاله ISI 65 صفحه سال انتشار : 2015 سفارش ترجمه

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 5

Keywords: Pyrido[1,2-c]pyrimidines; Antidepressants; Dual SSRI/5-HT1A activity; Quinoline derivatives; SERT; serotonin transporter; SAR; structure-activity relationship; 5-HT1AR; serotonin 5-HT1A receptors; 8-OH-DPAT; 8-hydroxy-2-(di-n-propylamino)tetralin; Ki; inh

دانلود رایگان متن کامل مقاله ISI 65 صفحه سال انتشار : 2015 سفارش ترجمه

Coumarins as anticancer agents: A review on synthetic strategies, mechanism of action and SAR studies

Keywords: Coumarins; Anticancer; Synthesis; Targets; SAR; IC50; ARI; aromatase inhibitor; CAM; choriallanotoic membrane; CDC; cell cycle division protein; CDK2; cyclin dependent kinase 2; CDKN1A; cyclin-dependent kinase inhibitor 1A; CYP; cytochromes P450; DDIT4; D

دانلود رایگان متن کامل مقاله ISI 72 صفحه سال انتشار : 2015 سفارش ترجمه

Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1

Keywords: Imidazo[1,2-b]pyridazine; Anti-apicomplexan; Toxoplasma gondii; Toxoplasma gondii calcium-dependent protein kinase 1; IC50; 50% inhibitory concentration; EC50; 50% effective concentration; CC50; 50% cytotoxic concentration; SAR; structure-activity relatio

دانلود رایگان متن کامل مقاله ISI 129 صفحه سال انتشار : 2015 سفارش ترجمه

A facile synthesis and microtubule-destabilizing properties of 4-(1H-benzo[d]imidazol-2-yl)-furazan-3-amines

Keywords: Benzoimidazolfurazanamines; Inhibitors of tubulin polymerization; Sea urchin embryo; Cytotoxicity; BIFA; 4-(1H-benzo[d]imidazol-2-yl)-furazan-3-amine; SAR; structure-activity relationship; CZSWDLNVZBRZKA-UHFFFAOYSA-N; OVKMKVJRZIKUQA-UHFFFAOYSA-N; RZHUNSKD

دانلود رایگان متن کامل مقاله ISI 133 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-activity relationship and properties optimization of a series of Quinazoline-2,4-diones as inhibitors of the canonical Wnt pathway

Keywords: Wnt pathway; β-catenin; Small molecule; Structure-activity relationship; Glioblastoma; Fz; Frizzled; LRP; lipoprotein receptor-related protein; ACN; acetonitrile; APC; adenomatous polyposis coli; B/P; brain to plasma ratio; CDI; N,N′-carbonyl-diimida

دانلود رایگان متن کامل مقاله ISI 136 صفحه سال انتشار : 2015 سفارش ترجمه

Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives

Keywords: AcOH; acetic acid; Boc; tert-butyloxycarbonyl; CCL2; chemokine ligand 2; CCR2; chemokine receptor 2; DCE; dichloroethane; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMAP; N,N-dimethylaminopyridine; DMSO; dimethylsulfoxide; INCB3344; N-(2-(((3

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Synthesis and evaluation of N-alkyl-9-aminoacridines with antibacterial activity

Keywords: Acridines; Antimicrobials; SAR; MRSA; Intercalation; Amphiphiles; Drug design; Synthesis; Topoisomerase;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Design, synthesis, in vitro evaluation and preliminary SAR studies of N-(2-(heteroaryloxy)propyl)phenothiazines against Rhipicephalus microplus cattle tick

Keywords: Ticks; Phenothiazines; Pyridines; Acaricides; SAR; Rhipicephalus microplus;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Novel Roflumilast analogs as soft PDE4 inhibitors

Keywords: PDE4 inhibitors; Soft drug; SAR; Esterase; COPD

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه