دانلود مقالات ISI درباره Sar + ترجمه فارسی

Modification of the length and structure of the linker of N6-benzyladenosine modulates its selective antiviral activity against enterovirus 71

Keywords: N6-benzyladenosine derivatives; Synthesis and antiviral activity; SAR; Enterovirus 71;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Spatiotemporal variations in surface velocity of the Gangotri glacier, Garhwal Himalaya, India: Study using synthetic aperture radar data

Keywords: Glacier velocity; Gangotri glacier dynamics; Garhwal Himalaya; Seasonal fluctuations; Interannual fluctuations; SAR; PALSAR; ASAR;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Safety assessment of widely used fermented virgin coconut oil (Cocos nucifera) in Malaysia: Chronic toxicity studies and SAR analysis of the active components

Keywords: Safety; Toxicity; Fermented virgin coconut oil; Southeast Asia; SAR;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

L-band Synthetic Aperture Radar imagery performs better than optical datasets at retrieving woody fractional cover in deciduous, dry savannahs

Keywords: Woody canopy cover; SAR; LandSAT-5; Textures; Spectral vegetation indices; Random Forest;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Pyrazolo[3,4-d]pyrimidine based scaffold derivatives targeting kinases as anticancer agents

Keywords: Protein kinase; Bioisostere; Pyrazolo[3,4-d]pyrimidine; Synthetic strategy; SAR

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

High resolution multisensor fusion of SAR, optical and LiDAR data based on crisp vs. fuzzy and feature vs. decision ensemble systems

Keywords: SAR; Optical data; LiDAR; Multisensor fusion;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Response of phytohormones and correlation of SAR signal pathway genes to the different resistance levels of grapevine against Plasmopara viticola infection

Keywords: Phytohormones; Grapevine; Resistance; SAR; SA; salicylic acid; ABA; abscisic acid; ETI; effector-triggered immunity; EDS1; enhanced disease susceptibility 1; HR; hypersensitive response; ICS2; isochorismate synthase 2; JA; jasmonic acid; NPR1; non-express

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Extracting hurricane eye morphology from spaceborne SAR images using morphological analysis

Keywords: Meteorology; Oceanography; SAR; RADARSAT; Feature extraction; Pattern recognition; Segmentation mathematical morphology

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and in vitro acetylcholinesterase and butyrylcholinesterase inhibitory potential of hydrazide based Schiff bases

Keywords: Synthesis; Acetylcholinesterase; Butyrylcholinesterase; Molecular docking; Schiff bases; SAR;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

A 210Pb-based chronological model for recent sediments with random entries of mass and activities: Model development

Keywords: 210Pb dating; Sediment dating; Random SAR; Random initial activity; TERESA model; TERESA; Time estimates from random entries of sediments and activities; SWI; sediment-water interface; SAR; mass sediment accumulation rate;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Infrared thermography based magnetic hyperthermia study in Fe3O4 based magnetic fluids

Keywords: Infrared thermography; Magnetic fluid hyperthermia; SAR; Magnetic fluids

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2016 سفارش ترجمه

Design of α7 nicotinic acetylcholine receptor ligands using the (het)Aryl-1,2,3-triazole core: Synthesis, in vitro evaluation and SAR studies

Keywords: Alpha 7 nicotinic acetylcholine receptors; Quinuclidine; Tropane; Triazole synthesis; SAR; In vitro evaluation;

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2016 سفارش ترجمه

Structure-guided design of novel Trypanosoma brucei Methionyl-tRNA synthetase inhibitors

Keywords: Human African trypanosomiasis; Methionyl-tRNA synthetase; Structure-guided design; AP; auxiliary pocket; CNS; central nervous system; EMP; enlarged methionine pocket; HAT; human African trypanosomiasis; MetRS; methionyl-tRNA synthetase; SAR; structure-act

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2016 سفارش ترجمه

Structural requirements of acylated Gly-l-Ala-d-Glu analogs for activation of the innate immune receptor NOD2

Keywords: Muramyl dipeptide; Immunomodulator; Desmuramylpeptide; NOD2 agonist; Immunostimulant; Immunoadjuvant; CARD; caspase activation and recruitment domain; DCC; dicyclohexylcarbodiimide; DMAP; 4-dimethylaminopyridine; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carb

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2016 سفارش ترجمه

Mexico City land subsidence in 2014-2015 with Sentinel-1 IW TOPS: Results using the Intermittent SBAS (ISBAS) technique

Keywords: SAR; InSAR; Sentinel-1; Land subsidence; TOPS;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2016 سفارش ترجمه

The Costa Concordia last cruise: The first application of high frequency monitoring based on COSMO-SkyMed constellation for wreck removal

Keywords: Costa Concordia; SAR; COSMO-SkyMed; Oil spill; Wreck;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2016 سفارش ترجمه

An innovative procedure for monitoring the change in soil seismic response by InSAR data: application to the Mexico City subsidence

Keywords: Subsidence; Resonant period; SAR; GEP; Seismic hazard;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2016 سفارش ترجمه

Minimal Clinically Important Difference (MCID) in Allergic Rhinitis: Agency for Healthcare Research and Quality or Anchor-Based Thresholds?

Keywords: Allergic rhinitis; Oral antihistamine; Intranasal antihistamine; Intranasal corticosteroid; Leukotriene receptor antagonist; Minimal clinically important difference (MCID); Seasonal allergic rhinitis (SAR); Total nasal symptom score (TNSS); AHRQ; Agency f

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2016 سفارش ترجمه

Accounting for land use in life cycle assessment: The value of NPP as a proxy indicator to assess land use impacts on ecosystems

Keywords: AoP; area of protection; BDP; Biodiversity Damage Potential; BPP; biotic production potential; CF; characterization factor; CEENE; Cumulative Exergy Extraction from the Natural Environment; CSP; Carbon Sequestration Potential; EDP; Ecosystem Damage Potent

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2016 سفارش ترجمه

Middle–Late Holocene earthquake history of the Gyrtoni Fault, Central Greece: Insight from optically stimulated luminescence (OSL) dating and paleoseismology

Keywords: OSL (optically stimulated luminescence) dating; SAR; Paleoseismology; Gyrtoni Fault; Central Greece

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2016 سفارش ترجمه

Design and synthesis of new potent PTP1B inhibitors with the skeleton of 2-substituted imino-3-substituted-5-heteroarylidene-1,3-thiazolidine-4-one: Part I

Keywords: 1,3-Thiazolidine-4-one; PTP1B; Pyrrole; Pyridine; Dock; SAR

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2016 سفارش ترجمه

Improved inland water levels from SAR altimetry using novel empirical and physical retrackers

Keywords: CryoSat-2; Satellite altimetry; Retracking; SAR; Inland water; SAMOSA;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2016 سفارش ترجمه

Biological characterization of the hygrobafilomycin antibiotic JBIR-100 and bioinformatic insights into the hygrolide family of natural products

Keywords: DiOC2(3); 3,3′-diethyloxacarbocyanine iodide; ACP; acyl carrier protein; AT; acyltransferase; BGC; biosynthetic gene cluster; CCDC; Cambridge Crystallographic Data Centre; CID; collision-induced dissociation; DIC; differential interference contrast; DTT

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and biological activities of indolizine derivatives as alpha-7 nAChR agonists

Keywords: α7 nAChR; Indolizine; Agonists; SAR; Schizophrenia; ACh; acetylcholine; THF; tetrahydrofuran; DMSO; dimethylsulfoxide; CNS; central nervous system; HRMS; high resolution mass; DIPEA; diisopropylethylamine; AChBP; acetylcholine binding protein; SAR; struc

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2016 سفارش ترجمه

New telmisartan-derived PPARγ agonists: Impact of the 3D-binding mode on the pharmacological profile

Keywords: PPARγ; Transactivation; Cytotoxicity; Binding mode; Molecular modeling; Amax; maximum intrinsic activity; BPO; benzoyl peroxide; DMEM; Dulbecco's modified Eagle medium; LBD; ligand binding domaine; mp; melting point; NBS; N-bromosuccinimide; PPAR; peroxi

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2016 سفارش ترجمه

Discovery of a novel small molecule agonist scaffold for the APJ receptor

Keywords: AT1; angiotensin 2 receptor 1; CB1; cannabinoid receptor 1; CB2; cannabinoid receptor 2; NPS; neuropeptide S receptor; NTR-1; neurotensin receptor 1; BOP; benzotriazole-1-yl-oxy-tris-(dimethylamino)-phosphonium hexafluorophosphate; LiOH·H2O; lithium hydr

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2016 سفارش ترجمه

Discovery of a 7-arylaminobenzimidazole series as novel CRF1 receptor antagonists

Keywords: WMCIXFXVIWSRFJ-UHFFFAOYSA-N; CRF; corticotropin-releasing factor; HPA; hypothalamus-pituitary-adrenocortical; ACTH; adrenocorticotropic hormone; SAR; structure-activity-relationship; HBA; hydrogen-bonding acceptor; CDI; N,N′-carbonyldiimidazole; o

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2016 سفارش ترجمه

Novel S1P1 receptor agonists - Part 4: Alkylaminomethyl substituted aryl head groups

Keywords: S1P1 receptor agonist; Immunomodulator; Lymphocyte count; Aminomethyl pyridine; Aminomethyl benzene; Aminomethyl thiophene; Phototoxicity; BuLi; n-butyl lithium; CC; column chromatography; DCM; dichloromethane; DIPEA; diisopropylethylamine; DEAD; diethyl

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2016 سفارش ترجمه

'Looting marks' in space-borne SAR imagery: Measuring rates of archaeological looting in Apamea (Syria) with TerraSAR-X Staring Spotlight

Keywords: TerraSAR-X; Staring Spotlight; SAR; Amplitude change detection; Archaeological remote sensing; Archaeological looting; Looting marks; Cultural heritage; Apamea; Syria;

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and biological evaluation of novel 6,7-dihydro-5H-cyclopenta[d]pyrimidine and 5,6,7,8-tetrahydroquinazoline derivatives as sigma-1 (σ1) receptor antagonists for the treatment of pain

Keywords: σ1R; sigma-1 receptor; σ2R; sigma-2 receptor; NMDA; N-methyl-d-aspartate; CNS; central nervous system; PNS; peripheral nervous system; KO; knockout; WT; wild-type; [3H]-DTG; [3H]-di-o-tolylguanidine; SAR; structure-active relationship; FRET; fluorescenc

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis, radiolabeling and evaluation of novel amine guanidine derivatives as potential positron emission tomography tracers for the ion channel of the N-methyl-d-aspartate receptor

Keywords: PET; NMDA; Radiolabeling; SAR; Non-competitive antagonists;

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis of 2-acylated and sulfonated 4-hydroxycoumarins: In vitro urease inhibition and molecular docking studies

Keywords: Synthesis; 2-Acylated and sulfonated 4-hydroxycoumarin; Urease inhibition; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 19 صفحه سال انتشار : 2016 سفارش ترجمه

A review on ROCK-II inhibitors: From molecular modelling to synthesis

Keywords: XHJYFLXYQPATSO-OAQYLSRUSA-N; NGOKTEXAUPRBFP-UHFFFAOYSA-N; OMVMGDVRMSCTFN-UHFFFAOYSA-N; MUVYYVZAJFICKR-UHFFFAOYSA-N; JAWPAUHQCGKVGI-GFCCVEGCSA-N; ROFMCPHQNWGXGE-UHFFFAOYSA-N; WEEWAVMLLVLCNC-UHFFFAOYSA-N; PZWKXWPMVNKURA-UHFFFAOYSA-N; RHQHGEJBKFGHSM-RUZDIDTE

دانلود رایگان متن کامل مقاله ISI 20 صفحه سال انتشار : 2016 سفارش ترجمه

2-Methyl-4/5-nitroimidazole derivatives potentiated against sexually transmitted Trichomonas: Design, synthesis, biology and 3D-QSAR study

Keywords: Anti-Trichomonas; Dithiocarbamate; 4/5-Nitroimidazoles; Resistant Trichomonas; Hybridization; STDs; sexually transmitted diseases; TV; Trichomonas vaginalis; DTC; dithiocarbamate; SAR; structure activity relationship; MTZ; Metronidazole; NI; nitroimidazol

دانلود رایگان متن کامل مقاله ISI 20 صفحه سال انتشار : 2016 سفارش ترجمه

New insights into selective PDE4D inhibitors: 3-(Cyclopentyloxy)-4-methoxybenzaldehyde O-(2-(2,6-dimethylmorpholino)-2-oxoethyl) oxime (GEBR-7b) structural development and promising activities to restore memory impairment

Keywords: PDE4D inhibitors; cAMP enhancers; Memory behavior test; Pharmacokinetic analyses; Molecular dynamics simulation; In silico ADMET properties; AD; Alzheimer Disease; cAMP; cyclic adenosine monophosphate; CR3; conserved region 3; CREB; cAMP response element-

دانلود رایگان متن کامل مقاله ISI 21 صفحه سال انتشار : 2016 سفارش ترجمه

Influence of intramolecular hydrogen bonds on regioselectivity of glycosylation. Synthesis of lupane-type saponins bearing the OSW-1 saponin disaccharide unit and its isomers

Keywords: OSW-1 disaccharide; Glycosylation; Lupane saponins; SAR; Hydrogen bond network;

دانلود رایگان متن کامل مقاله ISI 21 صفحه سال انتشار : 2016 سفارش ترجمه

Microwave assisted synthesis of novel acridine-acetazolamide conjugates and investigation of their inhibition effects on human carbonic anhydrase isoforms hCA I, II, IV and VII

Keywords: CA; carbonic anhydrase; hCA; human carbonic anhydrase; Quinacrine; (RS)-N′-(6-Chloro-2-methoxy-acridin-9-yl)-N,N-diethylpentane-1,4-diamine; Proflavine; acridine-3,6-di-amine; Amsacrine; N-(4-(acridin-9-ylamino)-3-methoxyphenyl)methanesulfonamide; IR; i

دانلود رایگان متن کامل مقاله ISI 23 صفحه سال انتشار : 2016 سفارش ترجمه

The versatile ruthenium(II/III) tetraazamacrocycle complexes and their nitrosyl derivatives

Keywords: acn; acetonitrile; 4-acpy; pyridine-4-acetyl; acv; (acyclovir), 2-amino-1,9-dihydro-9-[(2-hydroxyethoxy)methyl]-6H-purin-6-one); am(m)ine; ammine, amine, and/or tetraazamacrocycle; ampy; 2-aminomethylpyridine; [15]aneN4; 1,4,8,12-tetraazacyclopentadecane;

دانلود رایگان متن کامل مقاله ISI 26 صفحه سال انتشار : 2016 سفارش ترجمه

PI3K/Akt/mTOR and Ras/Raf/MEK/ERK signaling pathways inhibitors as anticancer agents: Structural and pharmacological perspectives

Keywords: Cancer; Inhibitors; PI3K; Ras; SAR; Signaling pathways

دانلود رایگان متن کامل مقاله ISI 28 صفحه سال انتشار : 2016 سفارش ترجمه

Design, synthesis and evaluation of pyrazole derivatives as non-nucleoside hepatitis B virus inhibitors

Keywords: HBV; Bioisosterism; Hybrid pharmacophore-based; Non-nucleoside; SAR;

دانلود رایگان متن کامل مقاله ISI 31 صفحه سال انتشار : 2016 سفارش ترجمه

Tissue-specific expression of Arabidopsis NPR1 gene in rice for sheath blight resistance without compromising phenotypic cost

Keywords: SAR; systemic acquired resistance; PDA; potato dextrose agar; BDL; bioassay using detached leaf; DPI; days post inoculation; PDI; percent disease index; MS; Murashige and Skoog; Yield penalty; Transgenic rice; Systemic acquired resistance; Green tissue-sp

دانلود رایگان متن کامل مقاله ISI 37 صفحه سال انتشار : 2016 سفارش ترجمه

Development, synthesis and structure-activity-relationships of inhibitors of the macrophage infectivity potentiator (Mip) proteins of Legionella pneumophila and Burkholderia pseudomallei

Keywords: Mip; macrophage infectivity potentiator; PPIase; peptidyl-prolyl cis/trans isomerase; LpMip; L. pneumophila Mip; BpMip; B. pseudomallei Mip; SAR; structure-activity relationship; HSQC; Heteronuclear Single Quantum Coherence; NMM; N-methylmorpholine; DIP

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2016 سفارش ترجمه

Design, synthesis and biological evaluation of novel EGFR/HER2 dual inhibitors bearing a oxazolo[4,5-g]quinazolin-2(1H)-one scaffold

Keywords: EGFR/HER2 dual inhibitor; Oxazolo[4,5-g]quinazolin-2(1H)-one scaffold; Antitumor proliferation; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 44 صفحه سال انتشار : 2016 سفارش ترجمه

Recent developments of C-4 substituted coumarin derivatives as anticancer agents

Keywords: C-4 substituted coumarin; Anticancer; Synthesis; Mechanism of action; SAR;

دانلود رایگان متن کامل مقاله ISI 53 صفحه سال انتشار : 2016 سفارش ترجمه

5,10b-Ethanophenanthridine amaryllidaceae alkaloids inspire the discovery of novel bicyclic ring systems with activity against drug resistant cancer cells

Keywords: Glioblastoma; Apoptosis resistance; Multidrug resistance; Translation inhibition; Lycorine; Haemanthamine; ATCC; American Type Culture Collection; DAPI; 4′,6-diamidino-2-phenylindole; DMEM; Dulbecco's modified Eagle's medium; DMF; dimethylformamide; DMS

دانلود رایگان متن کامل مقاله ISI 54 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors

Keywords: Coumarins; Factor XIIa; Factor XII; FXII; Antithrombotic agents; Benzopyrans; ADME; absorption, distribution, metabolism and excretion; FXIIa; activated coagulation factor XII; FXa; activated coagulation factor X; THR; thrombin; FVIIa; activated factor VI

دانلود رایگان متن کامل مقاله ISI 55 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and biological evaluation of indole-2-carboxamides bearing photoactivatable functionalities as novel allosteric modulators for the cannabinoid CB1 receptor

Keywords: Cannabinoid receptor; Allosteric modulator; Photoaffinity labeling; Photoactivatable ligands; CB1; Cannabinoid type 1 receptor; GPCR; G-protein coupled receptor; nAChRs; nicotinic acetylcholine receptors; BP; benzophenone; PTFMD; phenyltrifluoromethyldiaz

دانلود رایگان متن کامل مقاله ISI 56 صفحه سال انتشار : 2016 سفارش ترجمه

Balancing potency, metabolic stability and permeability in pyrrolopyrimidine-based EGFR inhibitors

Keywords: EGFR; Pyrrolopyrimidine; SAR; ADME; Metabolism; Erlotinib;

دانلود رایگان متن کامل مقاله ISI 61 صفحه سال انتشار : 2016 سفارش ترجمه

DNA repair targeted therapy: The past or future of cancer treatment?

Keywords: DNA damage; DNA repair; Cancer; Radiation; Replication protein A; NER; nucleotide excision repair; MMR; DNA mismatch repair; BER; base excision repair; HDR; homology directed repair; FA; Fanconi anemia; HR; homologous recombination; DDR; DNA damage respon

دانلود رایگان متن کامل مقاله ISI 64 صفحه سال انتشار : 2016 سفارش ترجمه

Amphiphilic xanthones as a potent chemical entity of anti-mycobacterial agents with membrane-targeting properties

Keywords: Mycobacteria; Tuberculosis; Xanthone; Membrane targeting; ACN; acetonitrile; ATP; adenosine triphosphate; CFU; colony forming unit; CLSI; Clinical & Laboratory Standards Institute; CMFDA; 5-chloromethylfluorescein diacetate; CYP; cytochrome P450; CL; card

دانلود رایگان متن کامل مقاله ISI 73 صفحه سال انتشار : 2016 سفارش ترجمه