دانلود مقالات ISI درباره Sar + ترجمه فارسی

1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents

Keywords: Tumor cell inhibitor; Hemaopoietic cell lines; BJAB; G0/G1 cell cycle; B-cell lymphoma; SAR; 1-Thiazol-2-yl-N-3-methyl-1H-pyrazole-5-carboxylic acid;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2017 سفارش ترجمه

Comparison of object-based and pixel-based Random Forest algorithm for wetland vegetation mapping using high spatial resolution GF-1 and SAR data

Keywords: Wetland vegetation mapping; Image fusion; Random Forest classifier; GF-1; SAR; Northeast China;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of pentacyclic triterpene 3β-ester derivatives as a new class of cholesterol ester transfer protein inhibitors

Keywords: CETP inhibitor; Pentacyclic triterpenes; Non-HDL-C; Dyslipidemia; CVDs; cardiovascular diseases; CETP; cholesteryl ester transfer protein; HDL-C; high density lipoprotein-cholesterol; LDL-C; low density lipoprotein-cholesterol; VLDL; very-low-density lipo

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2017 سفارش ترجمه

Mapping axonal density and average diameter using non-monotonic time-dependent gradient-echo MRI

Keywords: Axon density; Axon diameter; Susceptibility; Gradient echo; Multi-gradient echo; T2∗; Magnetic resonance imaging (MRI); Ultrahigh field MRI; CNS; Central Nervous System; dCST; dorsal corticospinal tract; DTI; Diffusion Tensor Imaging; EPI; Echo Planar I

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2017 سفارش ترجمه

Novel anti-prostate cancer scaffold identified by the combination of in silico and cell-based assays targeting the PI3K-AKT-mTOR pathway

Keywords: AKT; protein kinase B; AR; androgen receptor; mTOR; mammalian target of rapamycin; PI3K; phosphatidylinositol-3-kinase; S6; ribosomal protein S6 kinase; SAR; structureactivity relationship; SBVS; structure-based virtual screening; In silico screening; Pro

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2017 سفارش ترجمه

Oxadiazole-substituted naphtho[2,3-b]thiophene-4,9-diones as potent inhibitors of keratinocyte hyperproliferation. Structure−activity relationships of the tricyclic quinone skeleton and the oxadiazole substituent

Keywords: Antiproliferative activity; HaCaT cells; Quinone; Redox activation; Superoxide radical; 7-AAD; 7-aminoactinomycin D; CPR; NADPH-cytochrome P450 oxidoreductase; DCC; N,N'-dicyclohexylcarbodiimide; DHE; dihydroethidium; DMAP; 4-(dimethylamino)pyridine; DTPA

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2017 سفارش ترجمه

Efficacy of a series of alpha-pyrone derivatives against Leishmania (L.) infantum and Trypanosoma cruzi

Keywords: Alpha-pyrones; Leishmania; Trypanosoma cruzi; SAR; Phenotypic screening; AJCLHNYQRKPYFQ-UHFFFAOYSA-N; ADCLDRLWUWHAKC-UHFFFAOYSA-N; ULJWSSHLAKGIKW-UHFFFAOYSA-N; YTMDDHDOCBVTHT-UHFFFAOYSA-N; JRSGUWWIBIQYEB-UHFFFAOYSA-N; SQFXKUVOJMLOFO-UHFFFAOYSA-N; ZGKWGZIF

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2017 سفارش ترجمه

Importance of 5/6-aryl substitution on the pharmacological profile of 4ʹ-((2-propyl-1H-benzo[d]imidazol-1-yl)methyl)-[1,1ʹ-biphenyl]-2-carboxylic acid derived PPARγ agonists

Keywords: Peroxisome proliferator-activated receptor γ; Pharmacological profile; Coactivator recruitment; Transactivation assay; Molecular modeling; H; helix; LBD; ligand binding domain; PDB; Protein Data Bank; PPAR; peroxisome proliferator-activated receptor; PPR

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2017 سفارش ترجمه

Pyrrolizines: Design, synthesis, anticancer evaluation and investigation of the potential mechanism of action

Keywords: ALK1; activin receptor-like kinase; CDCl3; deuterated chloroform; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide; DSV; discovery studio visualizer; DYRK3; dual specificity tyrosine phosphorylation-regulated kinase; CDK2; cyclin-depende

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of orally bioavailable cyclohexanol-based NR2B-selective NMDA receptor antagonists with analgesic activity utilizing a scaffold hopping approach

Keywords: AcOEt; ethyl acetate; chloramine-T; N-chloro 4-methylbenzenesulfonamide sodium salt; DMAP; N,N-4-dimethylaminopyridine; DMF; N,N-dimethylformamide; hERG; human Ether-a-go-go Related Gene; HOBt; 1-hydroxybenzotriazole; IBX; o-iodoxybenzoic acid; LDA; lithi

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2017 سفارش ترجمه

Using multi-polarization C- and L-band synthetic aperture radar to estimate biomass and soil moisture of wheat fields

Keywords: Biomass; Soil moisture; Multi-polarization; SAR; Wheat;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis of selective 11β-HSD1 inhibitors based on dammarane scaffold

Keywords: 11β-HSD1 inhibitor; Hupehenols; Dammarane; SAR;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2017 سفارش ترجمه

Characterizing hydrologic changes of the Great Dismal Swamp using SAR/InSAR

Keywords: Great Dismal Swamp; Peatlands; Groundwater level changes; SAR; InSAR; Soil moisture; SMAP;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2017 سفارش ترجمه

Chronology of the Upper Pleistocene loess sequence of Havrincourt (France) and associated Palaeolithic occupations: A Bayesian approach from pedostratigraphy, OSL, radiocarbon, TL and ESR/U-series data

Keywords: Loess; Palaeosols; Northern France; Optical dating; SAR; Quartz; ESR/U-series dating; Periglacial processes; Middle and Upper Palaeolithic; Weichselian;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2017 سفارش ترجمه

K-Ras and its inhibitors towards personalized cancer treatment: Pharmacological and structural perspectives

Keywords: Personalized medicine; Inhibitors; K-Ras; Cancer; SAR; Signaling pathways;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis and evaluation of (E)-2-(5-phenylpent-2-en-4-ynamido)cyclohex-1-ene-1-carboxylate derivatives as HCA2 receptor agonists

Keywords: LDL; low-density lipoprotein; HDL; high-density lipoprotein; cAMP; 3′-5′-cyclic adenosine monophosphate; SAR; structure-activity relationship; RLB; radioligand binding; GPCR; G-protein coupled receptor; BSA; bovine serum albumin; DCM; dichloromethane;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2017 سفارش ترجمه

Structural modifications of diarylpyrimidines (DAPYs) as HIV-1 NNRTIs: Synthesis, anti-HIV activities and SAR

Keywords: AIDS; Anti-HIV; Diarylpyrimidines; Nonnucleoside reverse transcriptase inhibitors; SAR;

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2017 سفارش ترجمه

Diverse amide analogs of sulindac for cancer treatment and prevention

Keywords: NSAID; non-steroidal anti-inflammatory drug; COX; cyclooxygenase; SSA; sulindac sulfide amide; SAR; structure-activity relationship; AA; amino acid; ALL; acute lymphoblastic leukemia; CPC; choroid plexus carcinoma; TPSA; topological polar surface area; Li

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2017 سفارش ترجمه

Targeting Wnt-driven cancers: Discovery of novel tankyrase inhibitors

Keywords: Tankyrase inhibitors; PARP family; Wnt/β-catenin signaling pathway; Wnt pathway disruption; Wnt-driven cancers; APC; adenomatous polyposis coli gene product; ARTD; ADP-ribosyltransferases; CK1; casein kinase 1; DMPK; drug metabolism and pharmacokinetics;

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2017 سفارش ترجمه

A mangrove forest map of China in 2015: Analysis of time series Landsat 7/8 and Sentinel-1A imagery in Google Earth Engine cloud computing platform

Keywords: ETM+/OLI; SAR; NDVI; Greenness; Canopy coverage; Tidal inundation;

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2017 سفارش ترجمه

Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies

Keywords: Coumarins; Sulfonates; Inhibitory activity; Alkaline phosphatase; SAR; Docking studies;

دانلود رایگان متن کامل مقاله ISI 19 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis of 3-[4-(dimethylamino)phenyl]alkyl-2-oxindole derivatives and their effects on neuronal cell death

Keywords: Oxindole derivative; SAR; Suppression of neuronal cell death; Oxidative stress;

دانلود رایگان متن کامل مقاله ISI 19 صفحه سال انتشار : 2017 سفارش ترجمه

Evaluation of known and novel inhibitors of Orai1-mediated store operated Ca2+ entry in MDA-MB-231 breast cancer cells using a Fluorescence Imaging Plate Reader assay

Keywords: Calcium signalling; Store-operated calcium entry (SOCE); Pharmacological inhibitors; Pharmacophore modelling; Orai1; Breast cancer; AFU; arbitrary fluorescence units; CPA; cyclopiazonic acid; [Ca2+]CYT; cytosolic free Ca2+; ER; endoplasmic reticulum; FLIP

دانلود رایگان متن کامل مقاله ISI 20 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor

Keywords: BRD4 inhibitor; Kinase; BI-2536; Dihydroquinoxalin-2(1H)-one; PLK1; Polo-like Kinase 1; JAK2; Janus kinase 2; PTMs; post-translational modifications; KAc; acetylated lysine; BET; Bromodomain and Extra-Terminal; P-TEFb; positive transcription elongation fa

دانلود رایگان متن کامل مقاله ISI 20 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis and in vitro evaluation of Ca2 + channel blockers 1,4-dihydropyridines analogues against Trypanosoma cruzi and Leishmania amazonensis: SAR analysis

Keywords: 1,4-dihydropyridines; Leishmanicidal activity; Trypanocidal activity; SAR;

دانلود رایگان متن کامل مقاله ISI 21 صفحه سال انتشار : 2017 سفارش ترجمه

Post-failure evolution analysis of a rainfall-triggered landslide by multi-temporal interferometry SAR approaches integrated with geotechnical analysis

Keywords: Persistent Scatterers Interferometry; SAR; Coherent Pixel Technique-Temporal Sublook Coherence; Small Baseline Subset; Landslide; Crotone province; Slope stability analysis;

دانلود رایگان متن کامل مقاله ISI 22 صفحه سال انتشار : 2017 سفارش ترجمه

Use DAS algorithm to break through the device limitations of switched-capacitor-based DAC in an ADC consisting of pipelined SAR and TDC

Keywords: DAS; Switched capacitor; CMOS process; Energy; Bandwidth; CDAC; ADC; SAR; Pipeline;

دانلود رایگان متن کامل مقاله ISI 22 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis of piperazine sulfonamide analogs as diabetic-II inhibitors and their molecular docking study

Keywords: Synthesis; Piperazine; Sulfonamide; α-Amylase inhibition; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 23 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis and study of the α-amylase inhibitory potential of thiadiazole quinoline derivatives

Keywords: Synthesis; Thiadiazole quinoline; α-Amylase inhibitory potential; SAR;

دانلود رایگان متن کامل مقاله ISI 23 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis, characterization and biological activities of copper(II) complex of 2-Benzimidazolyl-urea and the nitrate salt of 2-Benzimidazolyl-urea

Keywords: Biological inorganic chemistry; Urea derivative; Copper(II) complexes; Cells screening; Crystal structure; SAR;

دانلود رایگان متن کامل مقاله ISI 25 صفحه سال انتشار : 2017 سفارش ترجمه

Large improvement of RF transmission efficiency and reception sensitivity for human in vivo 31P MRS imaging using ultrahigh dielectric constant materials at 7 T

Keywords: MRS; magnetic resonance spectroscopy; CSI; chemical shift imaging; FSW; Fourier series window; RF; radiofrequency; SNR; signal-to-noise ratio; HDC; high dielectric constant; uHDC; ultrahigh dielectric constant; B1+;  RF magnetic transmit field; B1−;  

دانلود رایگان متن کامل مقاله ISI 27 صفحه سال انتشار : 2017 سفارش ترجمه

Substituted methoxybenzyl-sulfonyl-1H-benzo[d]imidazoles evaluated as effective H+/K+-ATPase inhibitors and anti-ulcer therapeutics

Keywords: Benzimidazole; H+/K+-ATPase; Anti-ulcer; SAR; Molecular docking;

دانلود رایگان متن کامل مقاله ISI 27 صفحه سال انتشار : 2017 سفارش ترجمه

Design, synthesis and biological evaluation of new pyrazolyl-ureas and imidazopyrazolecarboxamides able to interfere with MAPK and PI3K upstream signaling involved in the angiogenesis

Keywords: p38MAPK phosphorylation; ERK1/2 phosphorylation; Akt phosphorylation; Migration; Pyrazolylureas; Imidazopyrazole derivatives; HUVECs; Human umbilical vein endothelial cells; BMDCs; bone marrow-derived cells; bFGF; basic fibroblast growth factor; EMT; epit

دانلود رایگان متن کامل مقاله ISI 27 صفحه سال انتشار : 2017 سفارش ترجمه

A new chemotype inhibitor for the human organic cation transporter 3 (hOCT3)

Keywords: OCT3; Phenylguanidines; 3D homology model; In vitro studies; SAR;

دانلود رایگان متن کامل مقاله ISI 28 صفحه سال انتشار : 2017 سفارش ترجمه

Design, synthesis and pharmacological evaluation of 4-hydroxyphenylglycine and 4-hydroxyphenylglycinol derivatives as GPR88 agonists

Keywords: 2-PCCA; (1R,2R)-2-(pyridin-2-yl)cyclopropane carboxylic acid ((2S,3S)-2-amino-3-methylpentyl)-(4′-propylbiphenyl-4-yl)amide; 2-AMPP; (2S)-N-((1R)-2-amino-1-(4-(2-methyl-pentyloxy)phenyl)ethyl)-2-phenylpropanamide; SAR; structure activity relationship; P

دانلود رایگان متن کامل مقاله ISI 28 صفحه سال انتشار : 2017 سفارش ترجمه

Retrieving topsoil moisture using RADARSAT-2 data, a novel approach applied at the east of the Netherlands

Keywords: Soil moisture; C-band; SAR; RADARSAT-2; Vegetation contribution; ADLC; CDF; Signal correction; Oh model; Water Cloud model;

دانلود رایگان متن کامل مقاله ISI 29 صفحه سال انتشار : 2017 سفارش ترجمه

Rapid generation of a novel DPP-4 inhibitor with long-acting properties: SAR study and PK/PD evaluation

Keywords: DPP-4 inhibitor; Type 2 diabetes; SAR; Long-acting; In vivo efficacy;

دانلود رایگان متن کامل مقاله ISI 30 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis and anti-mitotic activity of 6,7-dihydro-4H-isothiazolo[4,5-b]pyridin-5-ones: In vivo and cell-based studies

Keywords: Isothiazoles; Dihydroisothiazolopyridinones; Microtubule destabilization; Sea urchin embryo; Cytotoxicity; CA4P; combretastatin A-4 disodium phosphate; DIP; 6,7-dihydro-4H-isothiazolo[4,5-b]pyridin-5-ones; MDR; multi-drug resistance; Pgp; P-glycoprotein;

دانلود رایگان متن کامل مقاله ISI 32 صفحه سال انتشار : 2017 سفارش ترجمه

Preliminary SAR and biological evaluation of antitubercular triazolothiadiazine derivatives against drug-susceptible and drug-resistant Mtb strains

Keywords: Shikimate dehydrogenase; Antitubercular agent; 3,6-Disubstituted triazolothiadiazine; SAR;

دانلود رایگان متن کامل مقاله ISI 35 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes

Keywords: Quinoline; Fluorination; Phosphodiesterase 5; Radiotracer; Positron emission tomography; AD; alzheimer's disease; AllocCl; allyl chloroformate; ATR; attenuated total reflectance; cAMP; cyclic adenosine 3′,5′-monophosphate; cGMP; cyclic guanosine 3′,

دانلود رایگان متن کامل مقاله ISI 36 صفحه سال انتشار : 2017 سفارش ترجمه

Effects of prenatal exposure to WIFI signal (2.45 GHz) on postnatal development and behavior in rat: Influence of maternal restraint

Keywords: AP; access point; μL; microlitre; ALAT; alanine aminotransferase; ANOVA; analysis of variance; ASAT; aspartate aminotransferase; CAT; catalase; CG; control group; GSH; glutathione; GSH-Px; glutathione peroxidase; GSM; global system of mobile; H2O2; hydro

دانلود رایگان متن کامل مقاله ISI 37 صفحه سال انتشار : 2017 سفارش ترجمه

Spider peptide toxin HwTx-IV engineered to bind to lipid membranes has an increased inhibitory potency at human voltage-gated sodium channel hNaV1.7

Keywords: BSA; bovine serum albumin; CHOL; cholesterol; C1P; ceramide-1-phosphate; FLIPRTETRA; fluorescent imaging plate reader; GMT; gating modifier toxin; HBS; HEPES buffered saline; ICK; inhibitory cystine knot; LUV; large unilamellar vesicle; hNaV; human voltag

دانلود رایگان متن کامل مقاله ISI 37 صفحه سال انتشار : 2017 سفارش ترجمه

Application of the automatic seep location estimator (ASLE) with the use of contextual information for estimating offshore oil seeps

Keywords: Automatic classification; ASLE; Oil slicks; Oil seeps; SAR;

دانلود رایگان متن کامل مقاله ISI 38 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement

Keywords: HIV; NNRTIs; Indolylarylsulfones; Antiviral activity; SAR; Molecular modeling; Chemical space; Drug design;

دانلود رایگان متن کامل مقاله ISI 40 صفحه سال انتشار : 2017 سفارش ترجمه

Interactions between salicylic acid and antioxidant enzymes tilting the balance of H2O2 from photorespiration in non-target crops under halosulfuron-methyl stress

Keywords: Phytotoxicity; Secondary target; Halosulfuron-methyl; Reactive oxygen species; Non-target crop; Sulfonylurea herbicide; HSM; halosufuron-methyl; SU; sulfonylurea herbicide; ALS; acetolactate synthase; BCAAs; branched chain amino acids; ROS; reactive oxyge

دانلود رایگان متن کامل مقاله ISI 41 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF1 receptor antagonist

Keywords: CRF; corticotropin-releasing factor; HPA; hypothalamus-pituitary-adrenocortical; ACTH; adrenocorticotropic hormone; SAR; structureactivity-relationship; CDI; N,N′-carbodiimidazole; WSC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt;

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2017 سفارش ترجمه

The replacement of the 2-methoxy substituent of N-((6,6-diphenyl-1,4-dioxan-2-yl)methyl)-2-(2-methoxyphenoxy)ethan-1-amine improves the selectivity for 5-HT1A receptor over α1-adrenoceptor and D2-like receptor subtypes

Keywords: 5-HT1A receptor; α1-Adrenoceptor subtypes; D2-like receptor subtypes; Selective 5-HT1A receptor agonists; Docking studies; Anxiolytic effect; 5-HT; 5-hydroxytriptamine; GPCR; G protein-coupled receptor; TM; transmembrane; ARs; adrenoceptors; SAR; structu

دانلود رایگان متن کامل مقاله ISI 44 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of hepatitis B virus capsid assembly inhibitors leading to a heteroaryldihydropyrimidine based clinical candidate (GLS4)

Keywords: HBV; Capsid assembly inhibitor; SAR; GLS4; Pharmacokinetics; Safety evaluation;

دانلود رایگان متن کامل مقاله ISI 45 صفحه سال انتشار : 2017 سفارش ترجمه

Discovery of selective ATP-competitive eIF4A3 inhibitors

Keywords: RNA helicase; Eukaryotic initiation factor 4A3 (eIF4A3) inhibitors; Exon junction complex (EJC); ATP-competitive type inhibitors; Isothermal titration calorimetry (ITC); Surface plasmon resonance (SPR); BRR2; bad response to refrigeration 2 (an ATP-depend

دانلود رایگان متن کامل مقاله ISI 46 صفحه سال انتشار : 2017 سفارش ترجمه

Synthesis, characterization, molecular docking and in vitro antimalarial properties of new carboxamides bearing sulphonamide

Keywords: Antimalarial; Antioxidant; Carboxamides; Plasmepsin II; SAR; Sulphonamides;

دانلود رایگان متن کامل مقاله ISI 50 صفحه سال انتشار : 2017 سفارش ترجمه