دانلود مقالات ISI درباره Sar + ترجمه فارسی

Discovery of potent inhibitors of interleukin-2 inducible T-cell kinase (ITK) through structure-based drug design

Keywords: Kinase; Structure-based drug design; ITK; Tec kinase; SAR; Inhibitor; Benzimidazole

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

M3 muscarinic acetylcholine receptor antagonists: SAR and optimization of bi-aryl amines

Keywords: Muscarinic acetylcholine receptor; M3 mAChR; Antagonists; SAR; Sub-type selectivity; COPD; Asthma; Bi-aryl amines

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and SAR studies of 1,4-diazabicyclo[3.2.2]nonane phenyl carbamates – subtype selective, high affinity α7 nicotinic acetylcholine receptor agonists

Keywords: Alpha 7; Nicotinic acetylcholine receptor; nAChR; SAR; 1,4-Diazabicyclo[3.2.2]nonane phenyl carbamate; Agonist

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and SAR of 2-phenyl-1-sulfonylaminocyclopropane carboxylates as ADAMTS-5 (Aggrecanase-2) inhibitors

Keywords: SAR; ADAMTS-5 (Aggrecanase-2) inhibitors; 2-Phenyl-1-sulfonylaminocyclopropanecarboxylates

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Structure–activity relationship (SAR) studies of 3-(2-amino-ethyl)-5-(4-ethoxy-benzylidene)-thiazolidine-2,4-dione: Development of potential substrate-specific ERK1/2 inhibitors

Keywords: ERK1/2; Substrate-specific inhibitor; Synthesis; SAR; Thiazolidine-2,4-dione; Rational design; Molecular modeling

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B

Keywords: Maslinic acid; Protein tyrosine phosphatase 1B; Inhibitor; SAR; Diabetes

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Discovery of 4-anilino-N-methylthieno[3,2-d]pyrimidines and 4-anilino-N-methylthieno[2,3-d]pyrimidines as potent apoptosis inducers

Keywords: Apoptosis inducers; Anticancer agents; HTS; SAR; In vivo activity

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Hit-to-lead optimization of pyrrolo[1,2-a]quinoxalines as novel cannabinoid type 1 receptor antagonists

Keywords: CB1 receptor; Rimonabant; Hit-to-lead; SAR; Pyrrolo[1,2-a]quinoxaline

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Discovery and SAR of benzyl phenyl ethers as inhibitors of bacterial phenylalanyl-tRNA synthetase

Keywords: Phenylalanyl-tRNA synthetase; PheRS; FRS; Aminoacyl-tRNA synthetase; Benzyl phenyl ether; Antibacterial; SAR

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

A simplified SAR protocol for TT-OSL

Keywords: Quartz; Thermally-transferred OSL; SAR; Dating

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Efficacy of fungicides and a systemic acquired resistance activator (acibenzolar-S-methyl) against tobacco blue mould

Keywords: Acrobat; Actigard; Azoxystrobin; Blue mould; Dimethomorph; Disease control; Dithane; Forum; Fungicides; Mancozeb; Nicotiana tabacum; Peronospora tabacina; Quadris; SAR; Tobacco

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Tetrahydroquinoline derivatives as CRTH2 antagonists

Keywords: CRTH2; PGD2; Antagonists; GPCR; Allergic diseases; Tetrahydroquinoline; SAR; Lead optimization;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Structure-Activity Relationship of novel phenylacetic CXCR1 inhibitors

Keywords: GPCRs; Allosteric modulators; SAR; Conformational analysis;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Evaluation of structurally diverse neuronal nicotinic receptor ligands for selectivity at the α6∗ subtype

Keywords: Neuronal nicotinic receptor; NNR; Alpha 6; a3b4; SAR; Pyrimidine; Nicotinic acetylcholine receptor; Smoking cessation; Nicotine addiction; Dopamine release; Parkinson's disease;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Structure-activity relationship (SAR) of parthenin analogues with pro-apoptotic activity: Development of novel anti-cancer leads

Keywords: Cytotoxicity; Apoptosis; Topoisomerase-II; Telomerase; SAR; Parthenin;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2009 سفارش ترجمه

Luminescence characteristics of quartz and feldspar from tectonically uplifted terraces in Kashmir Basin, Jammu and Kashmir, India

Keywords: IRSL dating; SAR; Kashmir Valley; Anomalous fading

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Syntheses and opioid receptor binding properties of carboxamido-substituted opioids

Keywords: Opioids; SAR

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

N-Hydroxy-1,2-disubstituted-1H-benzimidazol-5-yl acrylamides as novel histone deacetylase inhibitors: Design, synthesis, SAR studies, and in vivo antitumor activity

Keywords: HDAC inhibitor; Benzimidazole; Hydroxamic acid; SAR; Anticancer

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Discovery of 3-aryl-5-aryl-1,2,4-oxadiazoles as a new series of apoptosis inducers. 2. Identification of more aqueous soluble analogs as potential anticancer agents

Keywords: Apoptosis inducers; Anticancer agents; HTS; SAR;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Discovery of a novel class of 2-mercaptohexanoic acid derivatives as highly active PPARα agonists

Keywords: PPAR; 2-Mercaptohexanoic acid; SAR; PPARα agonists;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Identification of PDE4B Over 4D subtype-selective inhibitors revealing an unprecedented binding mode

Keywords: Lead optimisation; Ligand docking; Induced fit; SAR

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and biological evaluation of new 4-carboxyl quinoline derivatives as cyclooxygenase-2 inhibitors

Keywords: Cyclooxygenase-2 inhibition; 4-Carboxyl quinolines; SAR

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Shoreline changes and vertical displacement of the 2 April 2007 Solomon Islands earthquake Mw 8.1 revealed by ALOS PALSAR images

Keywords: Solomon Islands; SAR; Shoreline; Displacement;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Reuse of laundry greywater as affected by its interaction with saturated soil

Keywords: Greywater; Hydraulic conductivity; Irrigation; Laundry greywater; SAR; Water retention

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Design and synthesis of ten biphenyl-neolignan derivatives and their in vitro inhibitory potency against cyclooxygenase-1/2 activity and 5-lipoxygenase-mediated LTB4-formation

Keywords: Honokiol derivatives; Cyclooxygenase; Lipoxygenase; Anti-inflammatory; SAR

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Highly efficacious factor Xa inhibitors containing α-substituted phenylcycloalkyl P4 moieties

Keywords: Factor Xa inhibitors; α-Substituted phenylcyclopropyls; SAR; Pharmacokinetic; Rabbit arterio-venous shunt

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

The discovery of the potent aurora inhibitor MK-0457 (VX-680)

Keywords: Aurora; Kinase inhibitor; SAR

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Design, synthesis and structure–activity relationships of antiproliferative 1,3-disubstituted urea derivatives

Keywords: Urea derivatives; Antiproliferative; K562 cell line; KB cell line; Morpholine ring; SAR

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and structure–activity relationships of cassiarin A as potential antimalarials with vasorelaxant activity

Keywords: Cassiarin A; Cassia siamea; Plasmodium falciparum; Antimalarial activity; Vasorelaxant activity; Nitric oxide; SAR

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Towards development of a broadly-applicable SAR TT-OSL dating protocol for quartz

Keywords: Thermally transferred OSL; Chinese loess; Quartz; Dating; SAR

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Jasmonate signaling in plant interactions with resistance-inducing beneficial microbes

Keywords: BTH; benzothiadiazole; ET; ethylene; ETI; effector triggered immunity; ISR; induced systemic resistance; JA; jasmonic acid; LPS; lipopolysaccharides; MAMPs; microbe-associated molecular patterns; MAPKs; mitogen activated protein kinases; PAMPs; pathogen a

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Salicylic acid-induced resistance to Fusarium oxysporum f. sp. lycopersici in tomato

Keywords: Fusarium oxysporum f. sp. lycopersici; Hydroponics; Induced resistance; Leaf yellowing wilting; Peroxidase; Phenylalanine ammonia lyase; Salicylic acid; Solanum lycopersicum; Systemic acquired resistance; Vascular browning; Fol; Fusarium oxysporum f. sp.

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Discovery and functional evaluation of diverse novel human CB1 receptor ligands

Keywords: CB1; cannabinoid receptor, subtype 1; CB2; cannabinoid receptor, subtype 2; CNS; central nervous system; FFA; free fatty acids; GPCR; G-protein coupled receptor; MMFF; Merck molecular force-field; NA; not available; NSB; non-specific binding; SAR; structu

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and evaluation of anticancer activity of 2-arylamino-6-trifluoromethyl-3-(hydrazonocarbonyl)pyridines

Keywords: Hydrazones; Anticancer activity; SAR

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and in vitro anti-HIV evaluation of a new series of 6-arylmethyl-substituted S-DABOs as potential non-nucleoside HIV-1 reverse transcriptase inhibitors

Keywords: NNRTIs; S-DABOs; Antiviral activity; In vitro; SAR; HIV-1; HIV-2CDI, 1,1′-carbonyldiimidazole; DABO, 2-alkoxyl-6-benzyl-3,4-dihydropyrimidin-4(3H)-ones; DDI, 2′,3′-dideoxyinosine; DMF, N,N-dimethylformamide; HEPT, 1-[(2-hydroxyethoxy)methyl]-6-(phenylsulf

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Classification comparisons between dual-pol, compact polarimetric and quad-pol SAR imagery

Keywords: Remote sensing; SAR; Classification

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Rapid mapping of high resolution SAR scenes

Keywords: SAR; Scene interpretation; Textural features; Road extraction

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis, biological evaluation and SAR of sulfonamide 4-methoxychalcone derivatives with potential antileishmanial activity

Keywords: Leishmaniasis; SAR; Sulfonamide 4-methoxychalcones; Antiparasite; Promastigote; Amastigote

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

Flood monitoring in a semi-arid environment using spatially high resolution radar and optical data

Keywords: SAR; Texture analysis; Flood monitoring

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

Novel and potent small-molecule urotensin II receptor agonists

Keywords: Urotensin II; Agonists; SAR; R-SAT; Parallel synthesis

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

Use of multitemporal SAR data for monitoring vegetation recovery of Mediterranean burned areas

Keywords: SAR; Forest monitoring; Fires; Forest biomass

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

InSAR analyses of terrain deformation near the Wieliczka Salt Mine, Poland

Keywords: Subsidence; Monitoring; Remote sensing; SAR; Landslides; Interferometry

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and evaluation of functionalized isoindigos as antiproliferative agents

Keywords: Isoindigo; Antiproliferative activity; CDK2 inhibition; SAR; Molecular modeling

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Ursolic acid derivatives induce cell cycle arrest and apoptosis in NTUB1 cells associated with reactive oxygen species

Keywords: Synthesis; Ursolic acid derivatives; Cytotoxicity; NTUB1; ROS; Cell cycle; Anticancer; Seco-compound; SAR

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Dibenzazecine scaffold rebuilding—Is the flexibility always essential for high dopamine receptor affinities?

Keywords: Dopamine receptor; Azecines; SAR; Heterocyclic compounds

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Natural polyprenylated benzophenones inhibiting cysteine and serine proteases

Keywords: Benzophenones; Proteases; Guttiferone A; Cathepsin G; SAR; Flexible dockingCC, column chromatography; TLC, thin layer chromatography; MAP, mitogen-activated protein; XRD, X-ray diffraction; HPLC, High Performance Liquid Chromatography; Z-FR-AMC, carbobenz

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Autotaxin structure–activity relationships revealed through lysophosphatidylcholine analogs

Keywords: Autotaxin; Lysophosphatidylcholine; Lysophosphatidic acid; LPC; LPA; SAR

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Secreted phospholipases A2: A proinflammatory connection between macrophages and mast cells in the human lung

Keywords: AA; arachidonic acid; Akt; protein kinase B; BA; bronchial asthma; BAL; bronchoalveolar lavage; BBMCs; bone marrow-derived mast cells; COPD; chronic obstructive pulmonary disease; ERK1/2; extracellular-regulated kinase 1/2; HSPG; heparan sulfate proteogly

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and evaluation of a novel series of heterocyclic oleanolic acid derivatives with anti-osteoclast formation activity

Keywords: Oleanolic acid; Heterocyclic derivatives; Osteoclast formation; Inhibitory activity; SAR

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2009 سفارش ترجمه

Estimating the quantity and quality of coarse woody debris in Yellowstone post-fire forest ecosystem from fusion of SAR and optical data

Keywords: Coarse woody debris; Remote sensing; Forest fire; SAR; Data fusion; Yellowstone

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2009 سفارش ترجمه