Keywords: گیرنده سیگما; Sigma receptor; Tumor; Radiobromine;
مقالات ISI گیرنده سیگما (ترجمه نشده)
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Keywords: گیرنده سیگما; Sigma receptor; Sodium channel; NMDA; Opioid; Antiviral; Neuroprotection;
Keywords: گیرنده سیگما; Astrocytes; Sigma receptor; BDNF; Neurotrophin; In situ ELISA; 4-PPBP (PubChem CID: 3035672); (+)-SKF10047 (PubChem CID: 13286169); BD1063 (PubChem CID: 574780); NE-100 (PubChem CID: 9841596); Haloperidol (PubChem CID: 3559); Reduced haloperidol (PubChem
Keywords: گیرنده سیگما; Low molecular weight heparin; Ursolic acid; Nanodrugs; Anti-angiogenesis; Combination therapy; Sigma receptor
Keywords: گیرنده سیگما; Sigma receptor; Sigma-1 receptor; ER stress; MAM; Chaperone
Keywords: گیرنده سیگما; Sigma receptor; Tumor; Astatine; Alpha therapy
Keywords: گیرنده سیگما; Sigma receptor; Synthesis; Ligands; Tetrahydroindazole; Affinity;
Keywords: گیرنده سیگما; Sigma receptor; Pulmonary pharmacology; Mouse; Radioligand binding;
Keywords: گیرنده سیگما; Ischemic stroke; Afobazole; Middle cerebral artery occlusion; Sigma receptor; Behavior; Neuroprotection; Oligodendroglia;
Keywords: گیرنده سیگما; Sigma receptor; Tumor; Radiobromine;
Keywords: گیرنده سیگما; Quetiapine; (+)-Pentazocine; Sigma receptor; Depression; FST;
Keywords: گیرنده سیگما; Agmatine; Allodynia; Hyperalgesia; Neuropathic pain; Sigma Receptor; Hippocampus; TNF-α;
Synthesis and pharmacological evaluation of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as sigma-2 receptor ligands
Keywords: گیرنده سیگما; Sigma receptor; Ligands; 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline; Affinity;
Short communicationThe Ï1 receptor agonist (+)-pentazocine increases store-operated Ca2+ entry in MCF7Ï1 and SK-N-SH cell lines
Keywords: گیرنده سیگما; BD1063; 1-[2-(3,4-dichlorophenyl)ethyl]-4-methylpiperazine; PB28; 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine; Ï; Sigma; Endoplasmic reticulum; Neuromodulation; Sigma receptor; (+)-Pentazocine; Cell imaging;
Development of a Sigma-2 Receptor affinity filter through a Monte Carlo based QSAR analysis
Keywords: گیرنده سیگما; QSAR; Sigma receptor; Sigma-2 Receptor; Monte Carlo method; Repurposing; CORAL software; Virtual screening;
Hyphenated 3D-QSAR statistical model-scaffold hopping analysis for the identification of potentially potent and selective sigma-2 receptor ligands
Keywords: گیرنده سیگما; Sigma receptor; Sigma-2 receptor; 3D-QSAR; Scaffold hopping; Virtual screening; Forge and Spark software; Bioisosteric replacements;
Tactics for preclinical validation of receptor-binding radiotracers
Keywords: گیرنده سیگما; Imaging; Validation; Radiopharmaceutical; Radiotracer; Radiopharmacology; Sigma receptor;
Decahydrobenzoquinolin-5-one sigma receptor ligands: Divergent development of both sigma 1 and sigma 2 receptor selective examples
Keywords: گیرنده سیگما; Sigma receptor; CNS; Decahydroquinoline; Radioligand binding; Structure-affinity relationship; Biology-oriented synthesis;
Sigma-1 receptor activation inhibits osmotic swelling of rat retinal glial (Müller) cells by transactivation of glutamatergic and purinergic receptors
Keywords: گیرنده سیگما; Sigma receptor; Estradiol; Cell swelling; Müller cell; Bipolar cell; Retina;
Effects of the psychotomimetic benzomorphan N-allylnormetazocine (SKF 10,047) on prepulse inhibition of startle in mice
Keywords: گیرنده سیگما; Psychotomimetic; Sigma receptor; Prepulse inhibition; Hallucinogen; Dissociative; Kappa receptor; Mice;
Activation of the sigma receptor 1 modulates AMPA receptor-mediated light-evoked excitatory postsynaptic currents in rat retinal ganglion cells
Keywords: گیرنده سیگما; AMPAR; a-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid receptor; BiP; binding immunoglobulin protein; BisIV; bisindolylmaleimide IV; [Ca2+]i; intracellular calcium concentration; DMSO; dimethyl sulfoxide; E-EPSC; electrically evoked excitatory posts
N-phenylpropyl-Nâ²-substituted piperazines occupy sigma receptors and alter methamphetamine-induced hyperactivity in mice
Keywords: گیرنده سیگما; Behavior; Methamphetamine; Locomotor activity; Mouse; Dopamine transporter; Receptor occupancy; Sigma receptor;
Associate editor: S. EnnaPharmacology of dextromethorphan: Relevance to dextromethorphan/quinidine (Nuedexta®) clinical use
Keywords: گیرنده سیگما; NMDA receptors; Pseudobulbar affect; Serotonin transporter; Nicotinic receptor; Sigma receptor; Pharmacokinetics; 5-HT; 5-hydroxytryptamine (serotonin); ACh; acetylcholine; BD1047; [2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(diamino)ethylamine; BD1063; 1-[2
Mild, Pd-catalyzed stannylation of radioiodination targets
Keywords: گیرنده سیگما; Stannylation; Radioiodination; Opioid; Sigma receptor; Radioligand binding
From NMDA receptor antagonists to discovery of selective Ï2 receptor ligands
Keywords: گیرنده سیگما; Glutamate; GluN2B/NMDA; Sigma receptor; Indoles; Ifenprodil;
SN79, a sigma receptor antagonist, attenuates methamphetamine-induced astrogliosis through a blockade of OSMR/gp130 signaling and STAT3 phosphorylation
Keywords: گیرنده سیگما; Sigma receptor; Methamphetamine neurotoxicity; Glia; Astrocyte; Neuroinflammation;
Effects of N-phenylpropyl-Nâ²-substituted piperazine sigma receptor ligands on cocaine-induced hyperactivity in mice
Keywords: گیرنده سیگما; Behavior; Cocaine; Locomotor activity; Mouse; Sigma receptor;
SN79, a sigma receptor ligand, blocks methamphetamine-induced microglial activation and cytokine upregulation
Keywords: گیرنده سیگما; Methamphetamine; Sigma receptor; Microglial activation; Cytokine; Neurotoxicity;
N-substituted 8-aminopentacyclo[5.4.0.02,6.03,10.05,9]undecanes as Ï receptor ligands with potential neuroprotective effects
Keywords: گیرنده سیگما; CNS; central nervous system; DTG; 1,3-di-o-tolylguanidine; DA; dopamine; DAT; dopamine transporter; HEK; human embryonic kidney; 5-HT; 5-hydroxytryptamine; IP3; inositol-1,4,5-triphosphate; LPS; lipopolysccharide; MAM; mitochondria-associated endoplasmic
Exploration of ring size in a series of cyclic vicinal diamines with Ï1 receptor affinity
Keywords: گیرنده سیگما; Sigma receptor; Piperazine; Imidazolidine; Diazepane; Diamine;
Neuropharmacology and analgesiaSigma receptor antagonists attenuate acute methamphetamine-induced hyperthermia by a mechanism independent of IL-1β mRNA expression in the hypothalamus
Keywords: گیرنده سیگما; Hyperthermia; Hypothalamus; Interleukin-1β; Methamphetamine; Sigma receptor;
CM156, a sigma receptor ligand, reverses cocaine-induced place conditioning and transcriptional responses in the brain
Keywords: گیرنده سیگما; ANOVA; analysis of variance; CM156; 3-(4-(4-cyclohexylpiperazin-1-yl)butyl)benzo[d]thiazole-2(3H)-thione; CPP; conditioned place preference; Ct; threshold cycle; malat1; metastasis associated lung adenocarcinoma transcript 1; MAS 5.0.; Affymetrix microarr
Evaluation of sigma (σ) receptors in the antidepressant-like effects of ketamine in vitro and in vivo
Keywords: گیرنده سیگما; Antidepressant; Depression; Ketamine; Neurite outgrowth; NMDA receptor; Sigma receptor
Anisamide-targeted cyclodextrin nanoparticles for siRNA delivery to prostate tumours in mice
Keywords: گیرنده سیگما; Non-viral vector; PEGylation; Anisamide; Sigma receptor; RNAi; Prostate cancer
The effect of substance P1–7 amide on nociceptive threshold in diabetic mice
Keywords: گیرنده سیگما; Antinociception; Diabetes; Substance P fragment substance P1–7; Opioid receptors; Substance P1–7 amide; Sigma receptor
Sigma-1 receptor ligand PRE-084 reduced infarct volume, neurological deficits, pro-inflammatory cytokines and enhanced anti-inflammatory cytokines after embolic stroke in rats
Keywords: گیرنده سیگما; Sigma receptor; Inflammation; Cytokine; Neuroprotection; Embolic stroke
Sigma (Ï) receptor ligand, AC927 (N-phenethylpiperidine oxalate), attenuates methamphetamine-induced hyperthermia and serotonin damage in mice
Keywords: گیرنده سیگما; Hyperthermia; Methamphetamine; Serotonin; Sigma Receptor;
Chronic administration of the anabolic androgenic steroid nandrolone alters neurosteroid action at the sigma-1 receptor but not at the sigma-2 or NMDA receptors
Keywords: گیرنده سیگما; Anabolic androgenic steroids (AAS); Nandrolone; [3H]ifenprodil; NMDA (N-methyl-d-aspartyl) receptor; NR2B subunit; Neurosteroids; Pregnenolone sulphate (PS); Pregnanolone sulphate (3α5βS); Rat brain; Sigma receptor; (+)-SKF 10,047
Activation of the sigma receptor 1 suppresses NMDA responses in rat retinal ganglion cells
Keywords: گیرنده سیگما; ÏR1; NMDA receptor; neurotransmission; retina; ganglion cells; G protein; [Ca2+]i; intracellular Ca2+ concentration; DAG; diacylglycerol; DMSO; dimethyl sulfoxide; GC; ganglion cell; IP3; inositol-1,4,5-triphosphate; IPL; inner plexiform layer; mGluR; me
Oxo-bridged isomers of aza-trishomocubane sigma (σ) receptor ligands: Synthesis, in vitro binding, and molecular modeling
Keywords: گیرنده سیگما; Sigma receptor; Trishomocubane; Hemiaminal; Structure–activity; Molecular modeling; Drug design
Effect of acute topical application of (+)-pentazocine on the mechanical allodynia in diabetic mice
Keywords: گیرنده سیگما; Anti-allodynia; Nitric oxide (NO); Sigma receptor; Sensory nerve; (Diabetic mice)
Radiosynthesis and biological evaluation of a promising σ2-receptor ligand radiolabeled with fluorine-18 or iodine-125 as a PET/SPECT probe for imaging breast cancer
Keywords: گیرنده سیگما; Breast cancer; Molecular imaging; F-18; I-125; Sigma receptor
The sigma agonist 1,3-di-o-tolyl-guanidine directly blocks SK channels in dopaminergic neurons and in cell lines
Keywords: گیرنده سیگما; SK channel; Sigma receptor; DTG; Dopaminergic neuron
Synthesis and characterization of N,N-dialkyl and N-alkyl-N-aralkyl fenpropimorph-derived compounds as high affinity ligands for sigma receptors
Keywords: گیرنده سیگما; Sigma receptor; Cancer; Tumor cell lines; FenpropimorphyERG2, yeast sterol C8–C7 isomerase; CHO-K1, Chinese hamster ovary cells; FAC, focal adhesion contacts; SBDLI, steroid binding domain-like I; SBDLII, steroid binding domain-like II; BD1047, N-[2-(3,4-
Sigma-1 ligands: Tic-hydantoin as a key pharmacophore
Keywords: گیرنده سیگما; Sigma receptor; Hydantoin; TetrahydroisoquinolinePHPLC, Purity determined by HPLC; TLC, Thin-layer chromatography; tR, HPLC retention time; CDI, 1,1′-Carbonyldiimidazole; tCDI, 1,1′-Thiocarbonyldiimidazole; EP, Petroleum ether; AcOEt, Ethyl acetate; Hex,
Expression of sigma receptor 1 mRNA and protein in rat retina
Keywords: گیرنده سیگما; sigma receptor; immunofluorescence double labeling; confocal laser scanning microscopy; amacrine cell; bipolar cell; ACh; acetylcholine; CB; calbindin; ChAT; choline acetyltransferase; DT-PBS; 3% normal donkey serum, 1% bovine serum albumin and 0.2% Trito
The role of dehydroepiandrosterone (DHEA) in drug-seeking behavior
Keywords: گیرنده سیگما; Addiction; AMPA; Cocaine; DHEA; DHEA-S; GABA; Glutamate; Neurosteroid; NMDA; Sigma receptor
Sigma receptors: Potential targets for a new class of antidepressant drug
Keywords: گیرنده سیگما; Antidepressant; Glutamate; Serotonin; Sigma receptor; Signal transduction; Neuroplasticity; NeurogenesisAkt, protein kinase β; AMPA, alpha-amino-3-hydroxy-5-methyl-4-isoxazoleproprionic acid; AP-1, activator protein 1; BD1047, N-[2-(3,4-dichlorophenyl)eth
The C-terminal amidated analogue of the substance P (SP) fragment SP1-7 attenuates the expression of naloxone-precipitated withdrawal in morphine dependent rats
Keywords: گیرنده سیگما; Morphine; Opiate; Substance P (SP); SP1-7 amide; Rat; Withdrawal; Sigma receptor;
Haloperidol disrupts Akt signalling to reveal a phosphorylation-dependent regulation of pro-apoptotic Bcl-XS function
Keywords: گیرنده سیگما; HAL; haloperidol; DTG; 1,3-di-o-tolylguanidine; SUL; sulpiride; PARP; poly(ADP-ribose) polymerase; VDAC; voltage-dependent anion channel.; Bcl-X; Cytochrome c; Mitochondria; VDAC; Dementia; Schizophrenia; Sigma receptor;