Keywords: کانال های سدیم; Mutations; Sodium channels; Heart diseases; Heart arrhythmias; Sudden cardiac death; Mutações; Canais de Sódio; Doenças cardÃacas; Arritmias cardÃacas; Morte súbita cardÃaca;
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Keywords: کانال های سدیم; AGAP; anti-tumor analgesic peptide; AMPA; α-amino-3-hydroxy-5methylisoxazole-4-propionic acid; ASICs; acid-sensitive ion channels; ATP; adenosine triphosphate; Bmk; toxin isolated from Chinese scorpion Mesobuthus martensii (previously Buthus martensii Ka
Keywords: کانال های سدیم; Subiculum; Temporal lobe epilepsy; Action potentials; Sodium channels; Electrophysiology; Nav1.6;
Keywords: کانال های سدیم; Voltage clamp fluorometry; Action potential modeling; Sodium channels; Calcium channels; Potassium channels;
Keywords: کانال های سدیم; Pain; Proprioception; Charcot Marie Tooth; Neuropathy; Pain channelopathy; Transcriptomics; Schwann cells; Gene expression; Glia; RNA-Seq; Dorsal root ganglion; Spinal cord; Sodium channels; TRPV1; TRPA1; Inherited peripheral neuropathy; HSAN; Sciatic ner
Keywords: کانال های سدیم; CSF-contacting nucleus; Sodium homeostasis; Sodium channels; Sodium appetite; Serotonin;
Keywords: کانال های سدیم; West syndrome; Dravet syndrome; mTOR; Epilepsy; Cognition; SUDEP; Arx; GABA; Sodium channels; Multiple-hit model; GABA; NMDA; Tetrodotoxin
Keywords: کانال های سدیم; Acid sensing ion channels; ASICs; Pharmacology; In vivo effects; Animal toxins; Sodium channels;
Keywords: کانال های سدیم; Absence seizures; Genetic epilepsy; Sodium channels; Murine AE; Computational analysis;
Keywords: کانال های سدیم; Sodium channels; Myocardium; Immunocytochemistry; Contractility;
Keywords: کانال های سدیم; sodium channels; lamotrigine; glaucoma; electroretinography; neuroprotection; retinal ganglion cell; optic nerve; Nav; voltage gated sodium channel; LTG; lamotrigine; IOP; intraocular pressure; RGC; retinal ganglion cells; ON; optic nerve; ERG; electroret
Keywords: کانال های سدیم; ASIC; Sodium channels; Toxins; Nervous system; Pathophysiology; Pain;
Keywords: کانال های سدیم; Sodium channels; Ventricular myocytes; Localization;
Keywords: کانال های سدیم; Sodium channels; Ion channel block; Mechanism of action; Local anesthetics
Oxaliplatin and neuropathy: A role for sodium channels
Keywords: کانال های سدیم; Oxaliplatin; Excitability; Neurophysiology; Sodium channels;
Assessment of the TRPM8 inhibitor AMTB in breast cancer cells and its identification as an inhibitor of voltage gated sodium channels
Keywords: کانال های سدیم; AMTB; Breast cancer; TRPM8; Sodium channels;
Nature and Action of Antibodies in Myasthenia Gravis
Keywords: کانال های سدیم; Acetylcholine esterases; Acetylcholine receptors; Autoantibodies; Complement; Muscle specific kinase; Neuromuscular transmission; Sodium channels;
Canalopatias cardÃacas: o papel das mutações nos canais de sódio
Keywords: کانال های سدیم; Mutações; Canais de Sódio; Doenças cardÃacas; Arritmias cardÃacas; Morte súbita cardÃaca; Mutations; Sodium channels; Heart diseases; Cardiac arrhythmias; Cardiac sudden death; Ca2+; Ião cálcio; CAV3; Caveolinaâ3; CMD; Cardiomiopatia Dilatada;
Abnormal sodium channel mRNA splicing in hypertrophic cardiomyopathy
Keywords: کانال های سدیم; Sodium channels; Hypertrophic cardiomyopathy; Sudden cardiac death; Human; SCN5A; Perk; Splicing variants;
Elucidation of pyrethroid and DDT receptor sites in the voltage-gated sodium channel
Keywords: کانال های سدیم; BTX; batrachotoxin; DDT1; ,1,1-trichloro-2,2-bis(p-chlorophenyl) ethane; DMT; deltamethrin; GTX; grayanotoxin; PMT; permethrin; TTX; tetrodotoxin; WHO; World Health Organization; Sodium channels; Insecticides; DDT; Pyrethroids;
De novo and inherited SCN8A epilepsy mutations detected by gene panel analysis
Keywords: کانال های سدیم; SCN8A; Sodium channels; Epilepsy; Gene panel analysis;
Leptin regulation of inward membrane currents, electrical activity and LH release in isolated bovine gonadotropes
Keywords: کانال های سدیم; Action potential; Calcium channels; Gonadotropes; Leptin; Sodium channels;
Clinical ObservationsSCN8A Epileptic Encephalopathy: Detection of Fetal Seizures Guides Multidisciplinary Approach to Diagnosis and Treatment
Keywords: کانال های سدیم; fetal seizures; SCN8A; early infantile epileptic encephalopathy; arthrogryposis; sodium channels; ultrasonography;
Lacosamide diminishes dryness-induced hyperexcitability of corneal cold sensitive nerve terminals
Keywords: کانال های سدیم; Dry eye; Cold thermoreceptors; Hyperexcitability; Sodium channels; Lacosamide;
Antinociceptive properties of the mastoparan peptide Agelaia-MPI isolated from social wasps
Keywords: کانال های سدیم; Mastoparan; Agelaia-MP I; Antinociception; Pain; Sodium channels
The cardiac connexome: Non-canonical functions of connexin43 and their role in cardiac arrhythmias
Keywords: کانال های سدیم; Cx43; Gap junctions; Sodium channels; Desmosomes; Intercalated disc;
Fast-onset lidocaine block of rat NaV1.4 channels suggests involvement of a second high-affinity open state
Keywords: کانال های سدیم; Sodium channels; Local anesthetic; Open-channel block; Voltage-clamp; Xenopus oocytes; Markov models
Pharmacological targeting of ion channels for cancer therapy: In vivo evidences
Keywords: کانال های سدیم; Calcium-permeable channels; Potassium channels; Sodium channels; Anion channels; In vivo cancer models; Pharmacological targeting;
A novel NaV1.5 voltage sensor mutation associated with severe atrial and ventricular arrhythmias
Keywords: کانال های سدیم; NaV1.5; sodium channels; VCF; voltage clamp fluorometry; F-V; voltage sensor movement; VSD; voltage sensing domain; ECG; electrocardiogram; CPR; cardiopulmonary resuscitation; AED; automated external defibrillators; HEK; human embryonic kidney; EGFP; enha
Distinct modulating effects of TipE-homologs 2–4 on Drosophila sodium channel splice variants
Keywords: کانال های سدیم; Auxiliary subunit; Sodium channels; Drosophila melanogaster; TipE; TipE-homologous proteins
Genetic background modulates impaired excitability of inhibitory neurons in a mouse model of Dravet syndrome
Keywords: کانال های سدیم; Dravet Syndrome; Sodium channels; Epilepsy; NaV1.1; Interneuron; Action potential threshold; Excitatory post synaptic potential amplification;
Voltage-gated sodium (NaV) channel blockade by plant cannabinoids does not confer anticonvulsant effects per se
Keywords: کانال های سدیم; AED; antiepileptic drug; CBD; cannabidiol; CBG; cannabigerol; CHL; Chinese hamster lung; CHO; Chinese hamster ovary; IFF; instantaneous spike firing frequency; NaV; voltage-gated Na+ channels; PTZ; pentylenetetrazole; Epilepsy; Cannabinoid; Seizure; Sodiu
Paroxysmal itch caused by gain-of-function Nav1.7 mutation
Keywords: کانال های سدیم; Itch; Neuropathic pain; Sodium channels; SCN9A; Small nerve fiber; Burning pain; Paroxysmal;
Functional characterization of two novel scorpion sodium channel toxins from Lychas mucronatus
Keywords: کانال های سدیم; Sodium channels; Lychas mucronatus; LmαTX3; LmαTX5; Expression and purification; Pharmacological profile;
Myotonic dystrophy type 1 mimics and exacerbates Brugada phenotype induced by Nav1.5 sodium channel loss-of-function mutation
Keywords: کانال های سدیم; BrS, Brugada syndrome; DM1, myotonic dystrophy type 1; PCR, polymerase chain reaction; WT, wild-typeMyotonic dystrophy cardiomyopathy; Brugada syndrome; Sodium channels; Cardiac arrhythmia; Ajmaline challenge
Modulation of peripheral Na+ channels and neuronal firing by n-butyl-p-aminobenzoate
Keywords: کانال های سدیم; AP, action potential; BAB, n-butyl-p-aminobenzoate; VGSCs, voltage gated Na+ channels; OS, Overshoot; TTXr, TTX-resistant; TTXs, TTX-sensitiveDorsal root ganglia; Sodium channels; Nociception; Butamben; NavButamben (PubChem CID: 2482)
Intrarenal ghrelin receptors regulate ENaC-dependent sodium reabsorption by a cAMP-dependent pathway
Keywords: کانال های سدیم; ghrelin; hypertension; kidney; obesity; sodium; sodium channels;
HCN2/SkM1 Gene Transfer Into Canine Left Bundle Branch Induces Stable, Autonomically Responsive Biological Pacing at Physiological Heart Rates
Keywords: کانال های سدیم; gene therapy; HCN channels; heart block; pacemakers; sodium channels; AC1; adenylyl cyclase 1; AP; action potential; HCN2; hyperpolarization-activated cyclic nucleotide-gated channel 2; hMSC; human mesenchymal stem cell; HRV; heart rate variability; Kir
Voltage-gated sodium channels contribute to the b-wave of the rodent electroretinogram by mediating input to rod bipolar cell GABAc receptors
Keywords: کانال های سدیم; retina; electroretinogram; tetrodotoxin; GABAc receptors; sodium channels; bipolar cells; amacrine cells; retinal circuits; CNQX; 6-Cyano-7-nitroquinoxaline-2,3-dion; ERG; electroretinogram; GABA; gamma-aminobutyric acid; Nav; voltage-gated sodium channel
Painful Na-channelopathies: an expanding universe
Keywords: کانال های سدیم; channelopathy; pain; sodium channels
Expanding chemical diversity of conotoxins: Peptoid–peptide chimeras of the sodium channel blocker μ-KIIIA and its selenopeptide analogues
Keywords: کانال های سدیم; μ-Conotoxins; KIIIA; Peptomers; Selenocysteine; Diselenide; Sodium channels; Electrophysiology
Synthesis and biological properties of new N-Mannich bases derived from 3-methyl-3-phenyl- and 3,3-dimethyl-succinimides. Part V
Keywords: کانال های سدیم; Anticonvulsant activity; Mannich bases; Succinimides; 3,3-Disubstituted-pyrrolidine-2,5-diones; In vivo studies; In vitro studies; Sodium channels; Vibrio harveyi assay
AMPK: An emerging target for modification of injury-induced pain plasticity
Keywords: کانال های سدیم; Chronic pain; mTOR; AMPK; ERK; Sodium channels; Plasticity;
Inhibition of NaV1.6 sodium channel currents by a novel series of 1,4-disubstituted-triazole derivatives obtained via copper-catalyzed click chemistry
Keywords: کانال های سدیم; Sodium channels; Patch clamp electrophysiology; 1,4-Triazoles; rNaV1.6; Click chemistry
Ion solvation and structural stability in a sodium channel investigated by molecular dynamics calculations
Keywords: کانال های سدیم; Sodium channels; Molecular dynamics; Structural stability; Ion hydration;
The discovery of aminopyrazines as novel, potent Nav1.7 antagonists: Hit-to-lead identification and SAR
Keywords: کانال های سدیم; Nav1.7; Analgesia; Sodium channels; Aminopyrazine;
Characterization of selectivity and pharmacophores of type 1 sea anemone toxins by screening seven Nav sodium channel isoforms
Keywords: کانال های سدیم; CGTX-II; cangitoxin-II; VGSC; voltage-gated sodium channels; Sea anemone; Bunodosoma cangicum; Sodium channels; Inactivation process; Patch-clamp; Toxins selectivity;
Alterations of 3,4-dihydroxyphenylethylamine and its metabolite 3,4-dihydroxyphenylacetic produced in rat brain tissues after systemic administration of saxitoxin
Keywords: کانال های سدیم; Saxitoxin; Dopamine; DOPAC; Sodium channels; Brain regions; Experimental periods;
Anticonvulsant activity of BmK AS, a sodium channel site 4-specific modulator
Keywords: کانال های سدیم; BmK AS; Sodium channels; Epilepsy; Pentylenetetrazole; Pilocarpine; Scorpion neurotoxin;
l-pGlu-(2-propyl)-l-His-l-ProNH2 attenuates 4-aminopyridine-induced epileptiform activity and sodium current: a possible action of new thyrotropin-releasing hormone analog for its anticonvulsant potential
Keywords: کانال های سدیم; action potential; epilepsy; patch clamp; sodium channels; subiculum; TRH analogCBZ, carbamazepine; nACSF, normal artificial cerebrospinal fluid; NP-647, l-pGlu-(2-propyl)-l-His-l-ProNH2; PDS, paroxysmal depolarization shift; RMP, resting membrane potentia