Keywords: رابطه فعالیت ساختاری; RAFI; Viral entry; Fusion inhibitors; Biophysical mechanism; HSV; Structure activity relationship;
مقالات ISI رابطه فعالیت ساختاری (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: رابطه فعالیت ساختاری; Bioavailability; Cardioprotective activity; Saponins; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; Mu opioid receptor; Delta opioid receptor; Kappa opioid receptor; Pain; Analgesia; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; CDK; cyclin dependent kinase; CDK4/6; cyclin dependent kinase 4 and 6; cdc; cell division cycle; CDC25C; cell division cycle 25 homolog; Ser/Thr; serine/ threonine; kDa; kilodaltonsâ(molecular weight); Cip/Kip; CDK interacting protein/kinase inhibitory
Keywords: رابطه فعالیت ساختاری; NTM; nontuberculous mycobacteria; Mtb; Mycobacterium tuberculosis; SAR; structure activity relationship; Mbs; Mycobacterium abscessus ATCC 19977; MIC; minimum inhibitory concentration; RHS; right hand side; LHS; left hand side; ADME; absorption, distribut
Keywords: رابطه فعالیت ساختاری; Ionic liquids; Antimicrobial; API-ILs; Structure activity relationship; Membrane modifications; Lipopolysaccharide;
Keywords: رابطه فعالیت ساختاری; Ultrasound irradiation; 1,4-Dihydropyridine derivatives; Anticoagulant activity; Antimicrobial activity; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; COND; conductivity; CT-DNA; calf thymus DNA; CV; cyclic voltammetry; DMF; dimethylformamide; DMSO; dimethylsulfoxide; DPPH; 1,1-diphenyl-2-picrylhydrazyl radical; EA; elemental analysis; EPR; electron paramagnetic resonance; IC50; half maximal inhibitory
Keywords: رابطه فعالیت ساختاری; Nav1.7; Pain; Pharmacophore models; Molecular docking; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; Allosteric inhibition; PEF(S); Calpain-1 inhibitors; Structure-based design; Docking; PEF(S); penta-EF hand calcium binding domain; TNS; p-toluidinylnaphthalene-6-sulfonate; CysPc; calpain-like protease domain; kDa; kilo Dalton; SAR; structure activity re
Keywords: رابطه فعالیت ساختاری; Pyrrole; Anticancer; Antimicrobial; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; data sharing; exposure effect relationship; outcomes research; pharmaceutical enterprise; structure activity relationship; target discovery;
Keywords: رابطه فعالیت ساختاری; Boc; tert-butyloxycarbonyl; Cbz; carboxybenzyl; CC50; half maximal cytoxicity concentration; EC50; half maximal effective concentration; EDC; N-(3-Dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; IBX; 2-iodoxybenzoic acid; Ki; inhibitory constan
Keywords: رابطه فعالیت ساختاری; IC50; 50% inhibitory concentration; MIC; minimum inhibitory concentration; MIC50; 50% minimum inhibitory concentration; SAR; structure activity relationship; MABA; microplate alamar blue assay; Flavonoids; Polyphenols; Oral candidiasis; Drug resistance; A
Keywords: رابطه فعالیت ساختاری; Antimicrobial resistance; Nitrofuran isoxazoline; MRSA; Medicinal chemistry; Antibacterial activity; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; HIV Integrase; 2-pyridinone aminal; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; Albizia julibrissin; Triterpenoid saponins; Cytotoxicity; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; MBC; minimum bactericidal concentration; MIC; minimum inhibitory concentration; CAC; critical aggregation concentration; ARI; antimicrobial-resistant infections; ITC; isothermal titration calorimetry; HLB; hydrophilic lipophilic balance; Triple-headed amp
Keywords: رابطه فعالیت ساختاری; Disulfide-rich peptides; Model membranes; Pain; Rational drug design; Surface plasmon resonance; Sodium channel; Cryo-EM; cryo-electron microscopy; DOPG; 1,2-dioleoyl-sn-glycero-3-phosphoglycerol; DHPC; 1,2-diheptanoyl-sn-glycero-3-phosphocholine; GMT; ga
Keywords: رابطه فعالیت ساختاری; AR; Structure activity relationship; MPTP; 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine; ATP; Adenosine triphosphate; CDEC; Carbamodithioic acid, diethyl-, 2-chloro-2-propenyl ester; OCR; Oxygen consumption rate; Environmental chemicals; Toxicants; Mitoch
Keywords: رابطه فعالیت ساختاری; CA; Chromosome aberrations; CBZ; 3-methyl-2-thioxo-4-imidazoline-1-carboxylate (carbimazole); CMBZT; 5-chloro-2-mercaptobenzothiazole; dppm; 1,1-bis(diphenylphosphino)methane; E. coli; Escherichia coli; H2stsc; {(2-HO-C6H4)(H)C2Â =Â N3-N2H-C1(=Â S)N
Keywords: رابطه فعالیت ساختاری; DOHQPHWDPCNACE-UHFFFAOYSA-N; ACh; acetylcholine; AChE; acetylcholinesterase; eelAChE; electric eel acetylcholinesterase; BuCh; butyrylcholine; BuChE; butyrylcholinesterase; eqBuChE; equine serum butyrylcholinesterase; ChE; cholinesterase; AD; Alzheimer'
Keywords: رابطه فعالیت ساختاری; Liver cancer; Progenitor cells; Thalidomide; Analogues; Lenalidomide; Sorafenib; Apoptosis; Mitosis; LPCs; liver progenitor cells; HCC; hepatocellular carcinoma; FDA; Federal Drug Administration; SAR; structure activity relationship; BMOL; bipotential mou
Keywords: رابطه فعالیت ساختاری; Hybrid molecules; Anti-fungal; Anti-tubercular; Anti-malarial; anti-inflammatory; ACTs; artemesinin based combination therapy; CQ; chloroquine; CC50; concentration required to reduce growth by 50%; EC50; half maximal effective concentration; Fqa; ferroqui
Keywords: رابطه فعالیت ساختاری; Safety evaluation; Leachables; Extractables; Permitted daily exposure; Safety threshold; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; Purine; Cancer; Kinases; Cell lines; Structure activity relationship; Design strategies;
Keywords: رابطه فعالیت ساختاری; 8-Aminoquinoline; Pyrazolopyrimidine; Plasmodium falciparum; Structure activity relationship; Hybridization;
Keywords: رابطه فعالیت ساختاری; Antiplasmodial agents; Adamantane; Plasmodium falciparum; Structure activity relationship;
Keywords: رابطه فعالیت ساختاری; calorimetry (DSC); oxidation; protein structure; proteins; stability; structure activity relationship; structure property relationship;
Keywords: رابطه فعالیت ساختاری; 3OH-Heli; 3-hydroxy-helichrysetin; 3OH-XNH; 3-hydroxy-xanthohumol H; 3OMe-XNH; 3-methoxy-xanthohumol H; 4Ac-XN; 4-O-acetyl-xanthohumol; 4Me-XN; 4-O-methyl-xanthohumol; 4â²Me-XN; 4â²-O-methyl-xanthohumol; C; cardamonin; dhFKC; dihydro-flavokawain C; dhHe
Keywords: رابطه فعالیت ساختاری; Isatin-ferrocene conjugates; Click chemistry; Structure activity relationship; Antimalarial evaluation; Cytotoxicity;
Keywords: رابطه فعالیت ساختاری; Natural products; Structure activity relationship; Monocytes; Cell death; Cytotoxicity
Keywords: رابطه فعالیت ساختاری; DCM; dichloromethane; E(1); one-electron reduction potential; FCS; foetal calf serum; FRT; fractionated radiotherapy; HCR; hypoxic cytotoxicity ratio; NCS; N-chlorosuccinimide; SAR; structure activity relationship; SBRT; stereotactic body radiotherapy; Ni
Keywords: رابطه فعالیت ساختاری; Algal drugs; Enzyme inhibitors; Dementia; Diabetes; Drug likeness; Inflammation; Structure activity relationship
Keywords: رابطه فعالیت ساختاری; DFT; density functional theory; B3LYP; Becke, three-parameter, Lee-Yang-Parr; BDE; bond dissociation energy; IP; ionization potential; ZPE; zero point energy; NBO; natural bond orbital; IC50; the half-maximal inhibitory concentration; DPPH; 2,2-diphen
Keywords: رابطه فعالیت ساختاری; Natural products; High throughput screening; Structure activity relationship; Targeted cancer therapy; Chemo-resistance; Drug formulation;
Structure activity relationships and antinociceptive activity of two novel dammarane-type sapogenins with notable anticancer effect
Keywords: رابطه فعالیت ساختاری; Ginseng sapogenins; Ginseng saponins; Antinociceptive activity; Animal models; Structure activity relationship;
An SAR study of hydroxy-trifluoromethylpyrazolines as inhibitors of Orai1-mediated store operated Ca2+ entry in MDA-MB-231 breast cancer cells using a convenient Fluorescence Imaging Plate Reader assay
Keywords: رابطه فعالیت ساختاری; FLIPR; Fluorescence Imaging Plate Reader; STIM1; stromal interaction molecule 1; ER; endoplasmic reticulum; TNBC; triple negative breast cancer; SAR; structure activity relationship; LHS; left hand side; RHS; right hand side; THF; tetrahydrofuran; i-PrOH;
Structure characteristics for intestinal uptake of flavonoids in Caco-2 cells
Keywords: رابطه فعالیت ساختاری; CU; cellular uptake of flavonoid without verapamil; CUV; cellular uptake of flavonoid with verapamil; SAR; structure activity relationship; QSAR; quantitative structure absorption relationship; MRP; multidrug resistance-associated protein; P-gp; P-glycopr
Novel autophagy modulators: Design and synthesis of (+)-epogymnolactam analogues and structure-activity relationship
Keywords: رابطه فعالیت ساختاری; Epogymnolactam; Autophagy inducer; Autophagy inhibitor; Structure activity relationship; NIH3T3 cells;
DN604: A platinum(II) drug candidate with classic SAR can induce apoptosis via suppressing CK2-mediated p-cdc25C subcellular localization in cancer cells
Keywords: رابطه فعالیت ساختاری; SAR; structure activity relationship; CBDC; 1,1-cyclobutanedicarboxylate; OCBDC; 3-oxocyclobutane-1,1-dicarboxylate; CDKs; cyclin-dependent kinases; MPF; M-phase-promoting factor; Pt; Potassium tetrachloroplatinate; ICP-MS; inductively coupled plasma mass
In vitro secondary pharmacological profiling: An IQ-DruSafe industry survey on current practices
Keywords: رابطه فعالیت ساختاری; AUC; Area Under the Curve; CRO; Contract Research Organization; CTA; Clinical Trial Authorization; GLP; Good Laboratory Practice; hERG; human ether-a-go-go-related gene; ICH; International Conference on Harmonization; IND; Investigational New Drug; IQ; In
Mechanism of action of cytotoxic compounds from the seeds of Euphorbia lathyris
Keywords: رابطه فعالیت ساختاری; Euphorbia lathyris; Euphorbia factor; Cytotoxicity; Collateral sensitivity; Multidrug resistance (MDR); EFL1-21; euphorbia factors L1-L21; MDR; multidrug resistance; P-gp; P-glycoprotein; ABC; ATP-binding cassette; SAR; structure activity relationship
Theoretical insights into the surface structure of In2O3(1â¯1â¯0) surface and its effect on methanol synthesis from CO2 hydrogenation
Keywords: رابطه فعالیت ساختاری; In2O3; Methanol synthesis; Surface structure; Structure activity relationship; DFT; Atmostic thermodynamics;
Design, synthesis and bioevalucation of novel 2,3-dihydro-1H-inden-1-amine derivatives as potent and selective human monoamine oxidase B inhibitors based on rasagiline
Keywords: رابطه فعالیت ساختاری; hMAO-B; Isoform selectivity; Fragment-based drug design; Structure activity relationship;
Heterocyclic Schiff bases as non toxic antioxidants: Solvent effect, structure activity relationship and mechanism of action
Keywords: رابطه فعالیت ساختاری; Schiff base; Antioxidant activity; DPPH; ABTS; Solvent effect; Structure activity relationship;
New developments in non-quinolone-based antibiotics for the inhibiton of bacterial gyrase and topoisomerase IV
Keywords: رابطه فعالیت ساختاری; Bacterial gyrase; Topoisomerase IV; Drug resistance; Binding sites; Potency; DNA; deoxyribonucleic acid; ATP; adenosine triphosphate; GyrA; gyrase A subunit; GyrB; gyrase B subunit; ParC; topoisomerase IV C subunit; ParE; topoisomerase IV E subunit; PDB;
Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
Keywords: رابطه فعالیت ساختاری; Neuropilin-1; VEGF165; Neuropilin/VEGF165 binding inhibition; Structure-activity relationship; Peptide biostability; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; Ahp; 7-aminoheptanoic acid; Aun; 11-aminoundecanoic acid;
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: رابطه فعالیت ساختاری; Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
Activity of mefloquine and mefloquine derivatives against Echinococcus multilocularis
Keywords: رابطه فعالیت ساختاری; Alveolar echinococcosis; Treatment; Anti-malaria; HPLC; Drug repurposing; Structure activity relationship;