Keywords: مهارکننده توبولین; Anticancer activity; Tubulin inhibitor; Chalcone; Naphthalene;
مقالات ISI مهارکننده توبولین (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهارکننده توبولین; Dolastatin 10; Tubulin inhibitor; Cytotoxicity;
Keywords: مهارکننده توبولین; Silybin; Ring disjunctive natural product lead optimization; (E)-3-(3-(benzyloxy)phenyl)-1-phenylprop-2-en-1-one; Tubulin inhibitor; Chemoprevention;
Keywords: مهارکننده توبولین; Trypanosomiasis; Tubulin inhibitor; Selective index; Drug development;
Keywords: مهارکننده توبولین; Coscinamides; Bisindoles; Ketohydrazide-hydrazones; Cytotoxicity; Apoptosis; Tubulin inhibitor;
Keywords: مهارکننده توبولین; 2-Alkylthio-4,5-diaryl-thiazole; Tubulin inhibitor; Cytotoxicity; Cell cycle analysis; Molecular docking;
Synthesis and biological evaluation of benzo[b]furo[3,4-e][1,4]diazepin-1-one derivatives as anti-cancer agents
Keywords: مهارکننده توبولین; Podophyllotoxin; Benzo[b]furodiazepin-1-ones; Anti-cancer; Cytotoxic; Synthesis; Apoptosis; Tubulin inhibitor;
Pharmacodynamic and pharmacokinetic characteristics of YMR-65, a tubulin inhibitor, in tumor-bearing mice
Keywords: مهارکننده توبولین; UPLC-MS/MS; ultra-performance liquid chromatography-tandem mass spectrometer; IS; internal standard; Cmax; maximum concentration of plasma; t1/2; half-life; AUC; area under the curve; Vd; apparent volume of distribution; MRT; Mean Retention Time; CL; clea
Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site
Keywords: مهارکننده توبولین; Tubulin inhibitor; Colchicine binding site; Combretastatin A-4; Pyrazole analogue; Anti-tumour; Co-crystal structure; ABC; ATP-binding cassette; P-gp; P-glycoprotein; MRP; multidrug resistant proteins; CA-4; combretastatin A-4; SARs; structure-activity re
Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents
Keywords: مهارکننده توبولین; Anticancer agents; Tubulin inhibitor; Intra-molecular hydrogen bonding; Colchicine binding site; RYRVKOAZGRXPLW-UHFFFAOYSA-N; MHEDZIYFQFWRMO-UHFFFAOYSA-N; QBNMSKFVSPKNSV-UHFFFAOYSA-N; YMIQVUIBWOJUPW-UHFFFAOYSA-N; HKFGTRWTMQYJOL-UHFFFAOYSA-N; ZBJRJZBGMBEVH
Design and synthesis of cis-restricted benzimidazole and benzothiazole mimics of combretastatin A-4 as antimitotic agents with apoptosis inducing ability
Keywords: مهارکننده توبولین; Tubulin inhibitor; Combretastatin A-4; Benzimidazole; Benzothiazole; Apoptosis
Methylene versus carbonyl bridge in the structure of new tubulin polymerization inhibitors with tricyclic A-rings
Keywords: مهارکننده توبولین; Tubulin inhibitor; Phenothiazine; Azaphenothiazine; Phenoxazine; Iminodibenzyl; 9(10H)Acridone; Antitumor agent;
Synthesis and structure-activity relationship studies of cytotoxic vinorelbine amide analogues
Keywords: مهارکننده توبولین; Vinorelbine; C-22 amide analogues; Tubulin inhibitor; Structure-activity relationship (SAR); Cytotoxicity;
Identification of selective tubulin inhibitors as potential anti-trypanosomal agents
Keywords: مهارکننده توبولین; Trypanosomiasis; Tubulin inhibitor; Sulfonamide; Drug development;
Isolation and identification of five impurities of ALB 109564(a) drug substance
Keywords: مهارکننده توبولین; ALB 109564(a); Tubulin inhibitor; Impurities; Structure elucidation; Capillary NMR;
Discovery of substituted N′-(2-oxoindolin-3-ylidene)benzohydrazides as new apoptosis inducers using a cell- and caspase-based HTS assay
Keywords: مهارکننده توبولین; Apoptosis inducer; Anticancer agent; HTS; SAR; Tubulin inhibitor
Synthesis and SAR of vinca alkaloid analogues
Keywords: مهارکننده توبولین; Vinca alkaloids; Vinblastine; Vincristine; Vinorelbine; Tubulin inhibitor; Anticancer; HeLa; MCF7; P388; Palladium
Discovery of 5-(4-hydroxy-6-methyl-2-oxo-2H-pyran-3-yl)-7-phenyl-(E)-2,3,6,7-tetrahydro-1,4-thiazepines as a new series of apoptosis inducers using a cell- and caspase-based HTS assay
Keywords: مهارکننده توبولین; Apoptosis inducer; HTS assay; Tubulin inhibitor
Phase I study of continuous weekly dosing of dimethylamino benzoylphenylurea (BPU) in patients with solid tumours
Keywords: مهارکننده توبولین; Tubulin inhibitor; Pharmacokinetics; Accelerated titration introduction
Total synthesis and biological evaluation of ustiloxin natural products and two analogs
Keywords: مهارکننده توبولین; Ustiloxins D and F; Tubulin inhibitor; Phomopsin; Total synthesis; Biological evalution; Antimitotic agent
Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors
Keywords: مهارکننده توبولین; Tubulin inhibitor; Tubulin polymerization; 1,2,4-Triazole; Vascular disrupting agent; Tumor vasculature; Antimitotic