Discovery and SAR of pyrrolo[2,1-f][1,2,4]triazin-4-amines as potent and selective PI3Kδ inhibitors

Discovery and SAR of pyrrolo[2,1-f][1,2,4]triazin-4-amines as potent and selective PI3Kδ inhibitors

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 26, Issue 17, 1 September 2016, Pages 4256-4260

Rajeev S. Bhide, James Neels, Lan-Ying Qin, Zheming Ruan, Sylwia Stachura, Carolyn Weigelt, John S. Sack, Kevin Stefanski, Xiaomei Gu, Jenny H. Xie, Christine B. Goldstine, Stacey Skala, Donna L. Pedicord, Stefan Ruepp, T.G. Murali Dhar, Percy H. Carter,