Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice

Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 27, Issue 10, 15 May 2017, Pages 2087-2093

Anthony J. Roecker, Melissa Egbertson, Kristen L.G. Jones, Robert Gomez, Richard L. Kraus, Yuxing Li, Amy Jo Koser, Mark O. Urban, Rebecca Klein, Michelle Clements, Jacqueline Panigel, Christopher Daley, Jixin Wang, Eleftheria N. Finger, John Majercak,