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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Acknowledgements to Reviewers
Fulltext Access 4 Pages 2007
Evaluation of native and modified forms of Pennisetum glaucum (millet) starch as disintegrant in chloroquine tablet formulations
Fulltext Access 4 Pages 2007
Improvement of dissolution rate of arbidol hydrochloride from solid dispersion prepared with PEG system by fusion method
Fulltext Access 4 Pages 2007
Design and evaluation of a floating ranitidine tablet as a drug delivery system for oral application
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Elastic positively-charged liposomes for topical administration of acyclovir
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EUFEPS and EAPB announcment on Monoclonal AntiBodies (MABW) Workshop
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EUFEPS and EAPB announcment on Monoclonal AntiBodies (MABW) Workshop
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Film/tablet adhesion, film thickness, internal stresses and bridging of the intagliations—A unified model with practical implications
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EUFEPS and EAPB Workshop on Monoclonal Antibodies
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De nouvelles stratégies thérapeutiques pour le cancer du rein
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Suppression de l'arsenal thérapeutique de spécialités déremboursées au CHRU de Lille
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Meetings Calendar
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The effect of suction during die fill on a rotary tablet press
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Novel possibility for protein absorption in the blood through the digestive system
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In vitro erythemal UV-A protection factors of inorganic sunscreens distributed in aqueous media using carnauba wax–decyl oleate nanoparticles
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HCV research and anti-HCV drug discovery: Toward the next generation
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Thank you to reviewers
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Author Index Volume 122 (2007)
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Blood–brain barrier delivery of protein and non-viral gene therapeutics with molecular Trojan horses
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Author Index Volume 117 (2007)
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Topical iodine facilitates transdermal delivery of insulin
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Synthesis, in vitro antibacterial and antifungal evaluations of 2-amino-4-(1-naphthyl)-6-arylpyrimidines
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Graphical contents list
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Graphical contents list
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High selective leishmanicidal activity of 3-hydroxy-2-methylene-3-(4-bromophenyl)propanenitrile and analogous compounds
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Antinociceptive activity and chemical composition of constituents from Caragana microphylla seeds
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Depigmenting activity of new kojic acid derivative obtained as a side product in the synthesis of cinnamate of kojic acid
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Mixtures of triblock copolymers E62P39E62 and E137S18E137: Potential for drug delivery from in situ gelling micellar formulations
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The effect of a high-fat meal on the pharmacodynamics of a model lipophilic compound that binds extensively to triglyceride-rich lipoproteins
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Surface activity of a non-micelle forming compound containing a surface-active impurity
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Accumulation of cadmium and its effects on liver and kidney functions in rats given diet containing cadmium-polluted radish bulb
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Author Index/Subject Index
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No effect of a traditional Chinese medicine, Hochu-ekki-to, on antibody titer after influenza vaccination in man: A randomized, placebo-controlled, double-blind trial
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An extract of Pelargonium sidoides (EPs 7630) inhibits in situ adhesion of Helicobacter pylori to human stomach
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Isolation of pure compound R/J/3 from Pluchea indica (L.) Less. and its anti-amoebic activities against Entamoeba histolytica
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Cytotoxic and antiprotozoal activity of flavonoids from Lonchocarpus spp.
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Upregulation of PBR mRNA expression in human neuroblastoma cells by flavonoids
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In vitro antidrepanocytary actvity (anti-sickle cell anemia) of some congolese plants
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Relationship between quantum-chemical descriptors of proton dissociation and experimental acidity constants of various hydroxylated coumarins. Identification of the biologically active species for xanthine oxidase inhibition
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Antileishmanial activity of indole alkaloids from Aspidosperma ramiflorum
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Ginkgo biloba in dyslexia: A pilot study
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Lipid peroxidation, cyclooxygenase enzyme and tumor cell proliferation inhibitory compounds in Cornus kousa fruits
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Ergosterol peroxides as phospholipase A2 inhibitors from the fungus Lactarius hatsudake
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EPs® 7630-solution – an effective therapeutic option in acute and exacerbating bronchitis
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EPs® 7630, an extract from Pelargonium sidoides roots inhibits adherence of Helicobacter pylori to gastric epithelial cells
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Pharmacokinetic properties of crocin (crocetin digentiobiose ester) following oral administration in rats
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Pharmacological studies on the sedative and hypnotic effect of salidroside from the Chinese medicinal plant Rhodiola sachalinensis
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Comparison of Echinacea alkylamide pharmacokinetics between liquid and tablet preparations
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Mixed micelles made of Pluronic and PEG-PE for solubilization of poorly soluble anticancer drug paclitaxel
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Bioavailability of metoclopramide from a new chewing gum device
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Bivalent peptides as PDZ domain ligands
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Catalysis of imido group hydrolysis in a maleimide conjugate
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Potent oxindole based human β3 adrenergic receptor agonists
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2-(2-Chloro-6-fluorophenyl)acetamides as potent thrombin inhibitors
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Synthesis of novel anilinoquinolines as c-fms inhibitors
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In vitro characterization of the Gd complex of [2,6-pyridinediylbis(methylene nitrilo)] tetraacetic acid (PMN-tetraacetic acid) and of its Eu analogue, suitable bimodal contrast agents for MRI and optical imaging
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Pyrazolo[1,5-a]pyrimidines as orally available inhibitors of cyclin-dependent kinase 2
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Versatile templates for the development of novel kinase inhibitors: Discovery of novel CDK inhibitors
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Geometry of GPPE binding to picrate and to the urokinase type plasminogen activator
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NMR detection of adventitious xylose binding to the quorum-sensing protein SdiA of Escherichia coli
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The discovery of indole-derived long acting β2-adrenoceptor agonists for the treatment of asthma and COPD
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Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1
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Biphenyls as potent vitronectin receptor antagonists. Part 3: Squaric acid amides
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Androstene-3,5-dienes as ER-β selective SERMs
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Investigating the antiproliferative activity of quinoline-5,8-diones and styrylquinolinecarboxylic acids on tumor cell lines
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3,5-Bis(3′-indolyl)pyrazoles, analogues of marine alkaloid nortopsentin: Synthesis and antitumor properties
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Binding of an aptamer to the N-terminal fragment of VCAM-1
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Novel synthetic ligands for targeted PET imaging and radiotherapy of copper
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Modifications of the chemical structure of terpenes in antiplasmodial and antifungal drug research
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Discovery of novel 8-azoniabicyclo[3.2.1]octane carbamates as muscarinic acetylcholine receptor antagonists
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Microbial transformation of three bufadienolides by Nocardia sp. and some insight for the cytotoxic structure–activity relationship (SAR)
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Inhibitory effects of phloridzin dihydrate on the activity of mushroom (Agaricus bisporus) tyrosinase
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Antimalarial activity of 1-aryl-3,3-dialkyltriazenes
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Graphical contents list
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Synthesis of chlorogenic acid derivatives with promising antifungal activity
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RNAi gene silencing using cerasome as a viral-size siRNA-carrier free from fusion and cross-linking
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Synthesis and antigenotoxic activity of some naphtho[2,1-b]pyrano[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine derivatives
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Graphical contents list
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Synthesis of 7-thiaarachidonic acid as a mechanistic probe of prostaglandin H synthase-2
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Structure–activity relationships of bioisosteres of a carboxylic acid in a novel class of bacterial translation inhibitors
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Inhibition of IGF-1R and lipoxygenase by nordihydroguaiaretic acid (NDGA) analogs
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Ferulic acid and benzothiazole dimer derivatives with high binding affinity to β-amyloid fibrils
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The discovery of long acting β2-adrenoreceptor agonists
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Cyclic benzamidines as orally efficacious NR2B-selective NMDA receptor antagonists
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SAR of the arylpiperazine moiety of obeline somatostatin sst1 receptor antagonists
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Discovery of inhibitors of the pentein superfamily protein dimethylarginine dimethylaminohydrolase (DDAH), by virtual screening and hit analysis
Fulltext Access 4 Pages 2007
New syntheses of tetrazolylmethylphenylalanine and O-malonyltyrosine as pTyr mimetics for the design of STAT3 dimerization inhibitors
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Design and synthesis of a new, conformationally constrained, macrocyclic small-molecule inhibitor of STAT3 via ‘click chemistry’
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Structure–activity relationships of novel N-acyloxy-1,4-dihydropyridines as P-glycoprotein inhibitors
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Synthesis and biological evaluation of l-cysteine derivatives as mitotic kinesin Eg5 inhibitors
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Inhibitory effect of 2-arylbenzofurans from Erythrina addisoniae on protein tyrosine phosphatase-1B
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3-Arylamino-2H-1,2,4-benzothiadiazin-5-ol 1,1-dioxides as novel and selective CXCR2 antagonists
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4-Phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives as non-peptidic selective δ-opioid agonists with potential anxiolytic/antidepressant properties. Part 2
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A high-throughput assay for O-GlcNAc transferase detects primary sequence preferences in peptide substrates
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In vitro cytotoxicity study on platinum (II) complexes with epoxysuccinates as leaving groups
Fulltext Access 4 Pages 2007
A multigram chemical synthesis of the γ-secretase inhibitor LY411575 and its diastereoisomers
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Effects of quinones on free-radical processes of oxidation and fragmentation of hydroxyl-containing organic compounds
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Effect of varying the 4″-position of arbekacin derivatives on antibacterial activity against MRSA and Pseudomonas aeruginosa
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Some new acyclic nucleotide analogues as antiviral prodrugs: Synthesis and bioactivities in vitro
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Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase
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