
Identification of 2-aminopyrimidine derivatives as inhibitors of the canonical Wnt signaling pathway
Keywords: APC; adenomatous polyposis coli; CK1; casein kinase-1; CYP3A4; Cytochrome P450 3A4; FPSA; fractional polar surface area; Fz; frizzled; GSK3; glycogen synthase kinase 3; LEF; lymphoid enhancer-binding factor; LRP; lipoprotein receptor-related protein; MW;