Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy
Keywords: آنتاگونیست CCR2; 6,7,8,9-Tetrahydro-5H-pyrido[43-c]azepin-5-one; 3,4-Dihydro-2,6-naphthyridin-1(2H)-one; CCR2 antagonist; Scaffold hopping; Structure-activity relationship; Selectivity of CCR2 over CCR5;