Keywords: مهار رقابت; Mushroom tyrosinase; Inhibitor; Thiazolidine derivatives; Competitive inhibition;
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Keywords: مهار رقابت; Resveratrol; Neurosteroid; Steroid 5α-reductase 1; 3α-Hydroxysteroid dehydrogenase; Retinol dehydrogenase 2; Competitive inhibition;
Keywords: مهار رقابت; Competitive inhibition; Local and global asymptotic stability; Lyapunov techniques; Chemostat model; Coexistence;
Keywords: مهار رقابت; Chalcone oximes; Competitive inhibition; Tyrosinase; Docking;
Keywords: مهار رقابت; AAC; mitochondrial ADP/ATP carrier; CiC; mitochondrial citrate carrier; DIC; mitochondrial dicarboxylate carrier; GSH; glutathione; GSSG; glutathione disulphide; NEM; N-ethylmaleimide; OGC; mitochondrial 2-oxoglutarate carrier; TBS; Tris-buffered saline;
Keywords: مهار رقابت; Binding constant; Competitive inhibition; Surface plasmon resonance; Charged gel matrix; Electrostatic interaction; Donnan potential; Mass-transport-induced dissociation;
Keywords: مهار رقابت; Diabetes mellitus; Dianthus basuticus; Antioxidant; Competitive inhibition
Characterization of l-aspartate oxidase from Arabidopsis thaliana
Keywords: مهار رقابت; DE; dicarboxylic exchangers; FAD; flavin adenine dinucleotide; FADH2; FAD hydroquinone form; GST; glutathione S-transferase; iminoasp.; iminoaspartate; IPTG; isopropyl thio-β-d-galactoside; LASPO; l-aspartate oxidase; NAD+; nicotinamide adenine dinucleot
GAPDH with NAD+-binding site mutation competitively inhibits the wild-type and affects glucose metabolism in cancer
Keywords: مهار رقابت; GAPDH; NAD+-binding; glycolysis; cancer metabolism; competitive inhibition;
Antagonistic effects of Lactobacillus plantarum 0612 on the adhesion of selected foodborne enteropathogens in various colonic environments
Keywords: مهار رقابت; Probiotic; Caco-2â¯cells; Adherence; Competitive inhibition; Foodborne pathogens; Colonic condition;
An in vitro investigation of the inhibitory mechanism of β-galactosidase by cinnamaldehyde alone and in combination with carvacrol and thymol
Keywords: مهار رقابت; Cinnamaldehyde; β-Galactosidase; Competitive inhibition; Molecular modeling; Synergistic effect;
Gossypol enantiomers potently inhibit human placental 3β-hydroxysteroid dehydrogenase 1 and aromatase activities
Keywords: مهار رقابت; Steroids; Testosterone; Competitive inhibition; 3β-hydroxysteroid dehydrogenase 1; Aromatase; JEG-3 cells
Structure-activity relationships of phthalates in inhibition of human placental 3β-hydroxysteroid dehydrogenase 1 and aromatase
Keywords: مهار رقابت; Steroids; Progesterone; Competitive inhibition; 3β -hydroxysteroid dehydrogenase 1; Aromatase;
Selective inhibitory effects of machilin A isolated from Machilus thunbergii on human cytochrome P450 1A and 2B6
Keywords: مهار رقابت; Machilus thunbergii; Competitive inhibition; Cytochromes P450; Human liver microsomes; Machilin A
Expression and characterization of a cytosolic glucose 6 phosphate dehydrogenase isoform from barley (Hordeum vulgare) roots
Keywords: مهار رقابت; G6PDH; Barley; Pentose phosphate pathway; Anion exchange chromatography; pET3d; NADPH; Competitive inhibition;
Inhibitory effect of ephedrannins A and B from roots of Ephedra sinica STAPF on melanogenesis
Keywords: مهار رقابت; α-MSH; melanin stimulating hormone; l-DOPA; l-3,4-dihydroxyphenylalaninine; ECG; epicathechin-3-O-gallate; DMEM; Dulbecco's modified Eagle's medium; FBS; Fetal bovine serum; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; DMSO; dimethy
Competitive Inhibition of AQP7-mediated Glycerol Transport by Glycerol Derivatives
Keywords: مهار رقابت; aquaporin 7; facilitative carrier; glycerol; glycerol derivatives; competitive inhibition; substrate specificity
Anti-amylolytic activity of fresh and cooked okra (Hibiscus esculentus L.) pod extract
Keywords: مهار رقابت; Okra pod; Cooking; Antihyperglycemic activity; Competitive inhibition; Mixed inhibition;
In vitro inhibition of fatty acid synthase by 1,2,3,4,6-penta-O-galloyl-β-d-glucose plays a vital role in anti-tumour activity
Keywords: مهار رقابت; C; competitive inhibition; N; noncompetitive inhibition; U; uncompetitive inhibition; 1,2,3,4,6-Penta-O-galloyl-β-d-glucose (PGG); Fatty acid synthase (FAS); Anti-tumour;
Physiologically based pharmacokinetic modeling of CYP3A4 induction by rifampicin in human: Influence of time between substrate and inducer administration
Keywords: مهار رقابت; Drug–drug interaction (DDI); Auto-induction; Competitive inhibition; Dynamic simulation; Physiologically based pharmacokinetic (PBPK) modeling; Study design recommendations
Inhibition of soluble epoxide hydrolase by fulvestrant and sulfoxides
Keywords: مهار رقابت; Soluble epoxide hydrolase; Epoxy-eicosatrienoic acids; Fulvestrant; Competitive inhibition; X-ray structure;
In vivo evidence that Agxt2 can regulate plasma levels of dimethylarginines in mice
Keywords: مهار رقابت; ADMA; asymmetric dimethylarginine; AGXT2; alanine-glyoxylate aminotransferase 2; BAIB; beta-aminoisobutyrate; DDAH; dimethylarginine dimethylaminohydrolase; DMGV; α-keto-δ-(N(G),N(G)-dimethylguanidino)valeric acid; SDMA; symmetric dimethylarginine; AD
Synthesis of new heterocyclic hybrids based on pyrazole and thiazolidinone scaffolds as potent inhibitors of tyrosinase
Keywords: مهار رقابت; Thiazolidinone scaffolds; Tyrosinase inhibitors; Competitive inhibition; Heterocyclic hybrids
Inhibition of monoamine oxidase by selected C6-substituted chromone derivatives
Keywords: مهار رقابت; Chromone; Monoamine oxidase; Reversible inhibition; Competitive inhibition; Molecular docking; Structure–activity relationship
The dehaloperoxidase paradox
Keywords: مهار رقابت; Peroxidase; Competitive inhibition; Hemoglobin; Phenol; Marine; Enzyme;
Kinetics of nitrate and perchlorate removal and biofilm stratification in an ion exchange membrane bioreactor
Keywords: مهار رقابت; Ion exchange membrane bioreactor; Drinking water; Nitrate and perchlorate; Competitive inhibition; Biofilm stratification; FISH
Asparagus racemosus competitively inhibits in vitro the acetylcholine and monoamine metabolizing enzymes
Keywords: مهار رقابت; Asparagus racemosus; Saponins; Cholinesterase; Monoamine oxidase; Competitive inhibition;
The 184th residue of β-glucosidase Bgl1B plays an important role in glucose tolerance
Keywords: مهار رقابت; β-Glucosidase; Competitive inhibition; GH1; Glucose tolerance; Mutation
Synthesis, biological assay in vitro and molecular docking studies of new Schiff base derivatives as potential urease inhibitors
Keywords: مهار رقابت; Competitive inhibition; Docking studies; Electrostatic potential; Schiff base; Thiourea derivatives; Urease inhibition;
Validation of a four-primer real-time PCR as a diagnostic tool for single and mixed Plasmodium infections
Keywords: مهار رقابت; Competitive inhibition; malaria; mixed infections; Plasmodium; real-time PCR
Autohydrogenotrophic perchlorate reduction kinetics of a microbial consortium in the presence and absence of nitrate
Keywords: مهار رقابت; Perchlorate; Nitrate; Hydrogen; Kinetics; Competitive inhibition; Biological treatment
Effect of temperature and benzalkonium chloride on nitrate reduction
Keywords: مهار رقابت; Benzalkonium chloride; Competitive inhibition; Nitrate reduction; Sorption; Temperature;
Inhibition of monoamine oxidase by selected C5- and C6-substituted isatin analogues
Keywords: مهار رقابت; Monoamine oxidase; Reversible inhibition; Selectivity; Competitive inhibition; Isatin; Molecular docking;
Mode of inhibition of acetylcholinesterase by monoterpenoids and implications for pest control
Keywords: مهار رقابت; Acetylcholinesterase; Competitive inhibition; Mixed inhibition; Monoterpenoids; Fenchone; S-carvone; Linalool; Sitophilus oryzae; Rhyzopertha dominica; Cryptolestes pusillus
Effect of enzyme processivity on the efficacy of a competitive chitinase inhibitor
Keywords: مهار رقابت; Glycoside hydrolase; Chitin; Chitosan; Processivity; Competitive inhibition
Investigating the interaction of McN-A-343 with the M2 muscarinic receptor using its nitrogen mustard derivative
Keywords: مهار رقابت; M2 muscarinic receptor; McN-A-343; Allosterism; Competitive inhibition; Irreversible binding;
Conserved extracellular cysteines differentially regulate the inhibitory effect of ethanol in rat P2X4 receptors
Keywords: مهار رقابت; P2X; P2X4 receptor; Cysteine; Disulfide bond; Mutation; Ethanol; Competitive inhibition; Noncompetitive inhibition
Kinetic evidence for an anion binding pocket in the active site of nitronate monooxygenase
Keywords: مهار رقابت; NMO, nitronate monooxygenase; FMN, flavin mononucleotide2-Nitropropane dioxygenase; Nitronate monooxygenase; Anion inhibition; Alkyl nitronates; Competitive inhibition; Hansenula mrakii; Neurospora crassa; Substrate specificity
The (+)- and (â)-gossypols potently inhibit both 3β-hydroxysteroid dehydrogenase and 17β-hydroxysteroid dehydrogenase 3 in human and rat testes
Keywords: مهار رقابت; Steroids; Testosterone; Competitive inhibition; Hydroxysteroid dehydrogenase;
Inhibition of monoamine oxidase B by N-methyl-2-phenylmaleimides
Keywords: مهار رقابت; Monoamine oxidase B; Reversible inhibitors; Competitive inhibition; Maleimide; Hydrolysis;
Spectroscopic study on the interaction of celecoxib with human carbonic anhydrase II: Thermodynamic characterization of the binding process
Keywords: مهار رقابت; Human carbonic anhydrase II; Celecoxib; Competitive inhibition; Fluorescence quenching; Binding study; Protein surface hydrophobicity
Mechanism of bis(7)-tacrine inhibition of GABA-activated current in cultured rat hippocampal neurons
Keywords: مهار رقابت; GABAA receptor; Acetylcholinesterase inhibitor; Competitive inhibition; pA2; KineticsACh, acetylcholine; AChE, acetylcholinesterase; AD, Alzheimer's disease; ANOVA, analysis of variance; Bis(7)-tacrine, 1,7-N-heptylene-bis-9,9′-amino-1,2,3,4-tetrahydroacr
Theoretical analysis of inhibition effect on steady states of enzymatic membrane reactor with substrate and product retention for reaction producing weak acid
Keywords: مهار رقابت; Enzymatic membrane reactor; Reactor performance; Enzyme activity; Competitive inhibition; Uncompetitive inhibition; Structure of steady state; Bifurcation
Simulating calcium influx and free calcium concentrations in yeast
Keywords: مهار رقابت; Calcium homeostasis; Calcium signaling; Response curve; Competitive inhibition
Competitive and product inhibition-based α-amylase activity analysis method
Keywords: مهار رقابت; α-amylase; Competitive inhibition; Product inhibition; Enzyme activity; Gal-G2-CNP
Heavy metal effects on fermentative hydrogen production using natural mixed microflora
Keywords: مهار رقابت; Chromium; Clostridium; Competitive inhibition; Copper; Heavy metal; Hydrogen production; Sucrose; Volatile fatty acid; Zinc
Exploring the possibility of predicting CALB activity in liquid organic medium, with the aid of intrinsic kinetic parameters and intrinsic solvent effect data obtained in solid/gaz reactor
Keywords: مهار رقابت; Lipase B from Candida antarctica; Alcoholysis; Organic solvent; Solid/gas biocatalysis; Competitive inhibition
Kinetics of a chlorate-accumulating, perchlorate-reducing bacterium
Keywords: مهار رقابت; Perchlorate; Chlorate; Kinetics; Competitive inhibition; Smin
Human mevalonate diphosphate decarboxylase: Characterization, investigation of the mevalonate diphosphate binding site, and crystal structure
Keywords: مهار رقابت; Human mevalonate diphosphate decarboxylase; Isoprenoid biosynthesis; Mevalonate pathway; Competitive inhibition; Active site function; Protein structure
Structure–activity relationships in the inhibition of monoamine oxidase B by 1-methyl-3-phenylpyrroles
Keywords: مهار رقابت; Monoamine oxidase B; Reversible inhibitors; Competitive inhibition; 1-Methyl-3-phenylpyrrole; Structure–activity relationship