Keywords: پپتیدهای سیکل; Biphalin; Opioid receptors; MOR/DOR/KOR agonist; Synergistic analgesic effect; Cyclic peptides; Acm; acetamidomethyl; ACN; acetonitrile; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BOP; (benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluoro
مقالات ISI پپتیدهای سیکل (ترجمه نشده)
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Keywords: پپتیدهای سیکل; Crotogossamide; Cyclic peptides; Macrocycles; Oxime resin; Peptide synthesis;
Keywords: پپتیدهای سیکل; Oxytocin; Disulfide bridging; Cyclic peptides; Peptide-based drugs; Increased stability;
Keywords: پپتیدهای سیکل; Protein structures; Similarity/dissimilarity analysis; Contact map matrix; Markov random fields; Cyclic peptides;
Keywords: پپتیدهای سیکل; Cyclic peptides; Cyclotides; Peptide chemistry; Bioactive peptides;
Keywords: پپتیدهای سیکل; Cyclic peptides; Marine organism; Anticancer; Antibacterial; Antifungal;
Keywords: پپتیدهای سیکل; Antimicrobial peptide; Cyclic peptides; Peptide nanotubes; Labaditin; Langmuir monolayers; PM-IRRAS; Large unilamellar vesicles; Staphylococcus aureus;
Keywords: پپتیدهای سیکل; Beyond the rule of 5; Permeability; Conformational shielding; Intramolecular hydrogen bonds; Macrocycles; Cyclic peptides; Efflux transporters; Quantitative structure permeability relationships;
Keywords: پپتیدهای سیکل; Pro-apoptotic agents; Anticancer agents; Cyclic peptides; Peptidomimetics; Nur77; Tubulin; Bcl-2; NMR studies; Molecular modeling; Confocal microscopy; FACS analysis; ADT; AutoDock Tools; COSY; correlation spectroscopy; DBU; 1,8-Diazabicyclo[5.4.0]undec-7
Keywords: پپتیدهای سیکل; Peptides; Translation; Cyclic peptides;
Keywords: پپتیدهای سیکل; Cyclic peptides; Microwave assisted synthesis; Lactam-bridge cyclic peptides; SHU9119; MTII; MWA-SPPS; microwave-assisted solid phase peptide synthesis; MBHA; methylbenzhydryl; MCR; melanocortin receptors; NDP; [Nle4, DPhe7]-αMSH; MTII; melanotan-II; RP-
Keywords: پپتیدهای سیکل; Solid phase peptide synthesis; Cyclic peptides; Opioid receptors; Receptor binding; Calcium mobilization; Hot-plate test;
Keywords: پپتیدهای سیکل; Conotoxins; Peptides; Cyclic peptides; Regulation; Select agents;
Keywords: پپتیدهای سیکل; Mass spectral library; Cyclic peptides; Microcystins; Chemical identification; Rates of qualitative analysis; Cyanobacterial strains
Keywords: پپتیدهای سیکل; Implicit water models; Structure prediction; Cyclic peptides;
Solid-phase synthesis of homodetic cyclic peptides from Fmoc-MeDbz-resin
Keywords: پپتیدهای سیکل; Cyclic peptides; Cyclactive cleavage; MeDbz linker; Solid-phase peptide synthesis;
Improving oral bioavailability of cyclic peptides by N-methylation
Keywords: پپتیدهای سیکل; Bioavailability; Cyclic peptides; N-Methylation; Peptide-based drugs; Caco-2; Peptidomimetics; Membrane transport; Cyclosporin A;
Antimicrobial activity of simplified mimics of celogentin C
Keywords: پپتیدهای سیکل; Celogentin; Antimicrobial peptides; Stapled peptides; Cyclic peptides;
Facile solid-phase synthesis of head-side chain cyclothiodepsipeptides through a cyclative cleavage from MeDbz-resin
Keywords: پپتیدهای سیکل; Solid-phase peptide synthesis; Cyclic peptides; Thiopeptides; Thiolactone; On resin cyclization;
Cyclic tetrapeptide HDAC inhibitors as potential therapeutics for spinal muscular atrophy: Screening with iPSC-derived neuronal cells
Keywords: پپتیدهای سیکل; Spinal muscular atrophy; HDAC inhibitor; iPSC; Neurons; Cyclic peptides;
Diastereoselective synthesis of the 5-hydroxy-pyrrolidinone amino acid of the microsclerodermins and model studies for an end-game strategy for microsclerodermin B
Keywords: پپتیدهای سیکل; Amino acids; Cyclic peptides; Stereoselective synthesis; Peptide coupling; Metathesis;
The intramolecular click reaction using 'carbocontiguous' precursors
Keywords: پپتیدهای سیکل; Click chemistry; Cyclic carbohydrates; Cyclic peptides; Dipolar cycloaddition; 1,2,3-Triazole;
Comprehensive profiling and characterization of chemical constituents of rhizome of Anemarrhena asphodeloides Bge.
Keywords: پپتیدهای سیکل; Anemarrhena asphodeloides Bge.; Cyclic peptides; Xanthones; Steroidal saponins; UHPLC-QTOF-MS;
Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues
Keywords: پپتیدهای سیکل; BU72; 17-methyl-3-hydroxy-[5β,7β,3â²,5â²]-pyrrolidino-2â²[S]-phenyl-7α-methyl-6,14-endoetheno morphinan; CHO; Chinese hamster ovary; DPDPE; [D-Ala2-N-Me-Phe4-Gly-ol] enkephalin; EM-2; endomorphin-2; NMe; N-methyl; Opioid receptors; N-Methylated amin
Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1
Keywords: پپتیدهای سیکل; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; ACN; acetonitrile; BSA; bovine serum albumin; (bt)-VEGF165; biotinylated-VEGF165; 6-Cl-HOBt; 6-chloro-1-hydroxybenzotriazole dihydrate; DIPEA; N,N-diisopropylethylamine; DMEM;
Glycosidase- and β-lactamase-like activity of dinuclear copper(II) patellamide complexes
Keywords: پپتیدهای سیکل; Cyclic peptides; Copper(II) complexes; Ascidian; Prochloron; Glycosidase; Lactamase
Synthesis and biological evaluation of analogues of the potent ADAM8 inhibitor cyclo(RLsKDK) for the treatment of inflammatory diseases and cancer metastasis
Keywords: پپتیدهای سیکل; ADAM8 inhibitors; Cancer metastasis; Cyclic peptides; Peptidomimetics; SAR study
Azide-alkyne cycloaddition-mediated cyclization of phosphonopeptides and their evaluation as PTP1B binders and enrichment tools
Keywords: پپتیدهای سیکل; Protein tyrosine phosphatases; Azide-alkyne click chemistry; Pull-down baits; Cyclic peptides; PTP1B and TCPTP;
Efficient synthesis of trypsin inhibitor SFTI-1 via intramolecular ligation of peptide hydrazide
Keywords: پپتیدهای سیکل; Cyclic peptides; Protein chemical synthesis; SFTI-1; Peptide hydrazides;
An efficient synthesis of a novel analog of octreotide with an unnatural l-lysine-like tetrazolyl amino acid
Keywords: پپتیدهای سیکل; XUAURGHUNZKOHJ-DXAXHBCISA-N; KSSNYHFBDHCJLF-FQEVSTJZSA-N; Unnatural amino acid; 1H-Tetrazole; l-Lysine; Cyclic peptides; Somatostatin analogs;
Jatrophidin I, a cyclic peptide from Brazilian Jatropha curcas L.: Isolation, characterization, conformational studies and biological activity
Keywords: پپتیدهای سیکل; Jatropha curcas; Euphorbiaceae; Cyclic peptides; Protease inhibition activity;
Synthesis and biological evaluation of the osteoblast proliferating cyclic peptides dianthins G and H
Keywords: پپتیدهای سیکل; Cyclic peptides; Dianthin G; Osteoblast proliferation; Macrolactamisation;
Synthesis of the unusual α-amino acid component of some novel histone deacetylase inhibiting cyclic peptides
Keywords: پپتیدهای سیکل; α-Amino acid; Cyclic peptides; Cross-metathesis; Histone deacetylase inhibitor; Chiral pool;
Predicting cyclic peptide chemical shifts using quantum mechanical calculations
Keywords: پپتیدهای سیکل; Macrocycles; NMR; Chemical shift prediction; Cyclic peptides;
Synthetic studies of cyclic peptides stephanotic acid methyl ester, celogentin C, and moroidin
Keywords: پپتیدهای سیکل; Total synthesis; Cyclic peptides; Natural product; Tandem reaction;
Metal-binding and redox properties of substituted linear and cyclic ATCUN motifs
Keywords: پپتیدهای سیکل; ATCUN; Catalysis; Copper; Cyclic peptides; Metallopeptides; Nickel
Euryjanicins E-G, poly-phenylalanine, and poly-proline cyclic heptapeptides from the Caribbean sponge Prosuberites laughlini
Keywords: پپتیدهای سیکل; Prosuberites laughlini; Cyclic peptides; Caribbean sponge; Cytotoxicity; Peptides;
Cyclic peptides containing tryptophan and arginine as Src kinase inhibitors
Keywords: پپتیدهای سیکل; Arginine; Cyclic peptides; Src; Tryptophan; Tyrosine kinase
A comparative protease stability study of synthetic macrocyclic peptides that mimic two endocrine hormones
Keywords: پپتیدهای سیکل; Cyclic peptides; Peptide pharmaceuticals; Head-to-tail cyclization; Protease stability; Drug design
Simultaneous determination of 24 constituents in Cortex Lycii using high-performance liquid chromatography–triple quadrupole mass spectrometry
Keywords: پپتیدهای سیکل; HPLC–ESI-MS/MS; Cortex Lycii; Quantification; Cyclic peptides; Phenolic amides; Principal component analysis
Design, synthesis and efficacy of novel G protein-coupled receptor kinase 2 inhibitors
Keywords: پپتیدهای سیکل; GRK2 inhibitors; Cardiovascular system; Cyclic peptides; NMR conformational analysisDPC, dodecylphosphocholine; SAR, structure–activity relationship; DCM, dichloromethane; DIPEA, N,N-diisopropylethyl-amine; DMF, N,N-dimethylformamide; Pr3SiH or TIS, triis
Inhibition of platelet adhesion by peptidomimetics mimicking the interactive β-hairpin of glycoprotein Ibα
Keywords: پپتیدهای سیکل; Platelets; Platelet receptor GPIbα; von Willebrand factor; Cyclic peptides;
New cyclic peptides with osteoblastic proliferative activity from Dianthus superbus
Keywords: پپتیدهای سیکل; Dianthus superbus L.; Caryophyllaceae; Cyclic peptides; Osteoblastic proliferative activity;
Cyclization of conotoxins to improve their biopharmaceutical properties
Keywords: پپتیدهای سیکل; Conotoxins; Cyclization; Cyclic peptides; Drug design; Cyclotides; Marine toxins
Pharmacodynamic synergy strictly dependent on the co-operative aggregation of enantiomers of cyclic peptides in the bacterial cell membrane
Keywords: پپتیدهای سیکل; Antimicrobial peptides; Synergy; Enantiomers; Cyclic peptides;
Isolation and characterization of cytotoxic cyclotides from Viola philippica
Keywords: پپتیدهای سیکل; Cyclotides; Cyclic peptides; Violaceae; Viola philippica; Cytotoxic activity; Viphi A-H;
Cyclopeptide alkaloids from Scutia buxifolia Reiss
Keywords: پپتیدهای سیکل; Scutia buxifolia; Rhamnaceae; Cyclopeptide alkaloids; Cyclic peptides; Stereochemistry; X-ray diffraction;
Diabetic nephropathy-related active cyclic peptides from the roots of Brachystemma calycinum
Keywords: پپتیدهای سیکل; Brachystemma calycinum; Caryophyllaceae; Cyclic peptides; Cytokines; Collagen IV; ROS
Perthamides C-F, potent human antipsoriatic cyclopeptides
Keywords: پپتیدهای سیکل; Marine compounds; Cyclic peptides; Theonella swinhoei; Anti-Inflammatory activity;
The arginine mimicking β-amino acid β3hPhe(3-H2N-CH2) as S1 ligand in cyclotheonamide-based β-tryptase inhibitors
Keywords: پپتیدهای سیکل; Mast cells; Cyclic peptides; Serine proteases; Structure-activity relationship; Solid phase peptide synthesis;