Keywords: Ach; acetylcholine; ADHD; attention-deficit hyperactivity disorder; BDNF; brain-derived neurotrophic factor; BEND; beta-endorphin; BFNA; beta-funaltrexamine; Ca(2+); calcium; CAMK; calmodulin-dependent protein kinase II; cAMP; cyclic adenosine monophospha
مقالات ISI (ترجمه نشده)
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Keywords: ACC; anterior cingulate; ACSF; artificial cerebrospinal fluid; AI; agranular region; DAMGO; [D-Ala2,N-Me-Phe4,Gly5-ol]-Enkephalin acetate salt; DPDPE; [D-Pen2,5]-Enkephalin hydrate; FS; fast-spiking; IC; insular cortex; Pyr; pyramidal; uIPSCs; unitary inh
Keywords: Ach; acetylcholine; ACTH; adrenocorticotrophic hormone; BDNF; brain-derived neurotrophic factor; BEND; beta-endorphin; BFNA; beta-funaltrexamine; BNST; bed nucleus of the stria terminalis; Ca(2+); calcium; CaMKII; calcium/calmodulin-dependent protein kina
Keywords: BBB; blood-brain barrier; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CNS; central nervous system; DAMGO; H-Tyr-d-Ala-Gly-NMePhe-Gly-ol; DCM; dichloromethane; DIEA; N,N-diisopropylethylamine; DOR; δ-opioid receptor; DPDPE; Tyr-c(d
Keywords: Ach; acetylcholine; AchE; acetylcholine esterease; ACTH; adrenocorticotrophic hormone; ADHD; attention deficit/hyperactivity disorder; AIDS; autoimmune deficiency syndrome; AMSH; alpha-melanocyte-stimulating hormone; BAM; bovine adrenal medulla peptide; B
Amniotic-fluid ingestion enhances central δ-opioid-induced hypoalgesia in rats in the cold-water tail-flick assay in a repeated-measures design
Keywords: Cold-water tail-flick assay; DPDPE; Opioids; Pain; Placental Opioid-Enhancing Factor; Repeated-measures design;
Can crosstalk between DOR and PARP reduce oxidative stress mediated neurodegeneration?
Keywords: Oxidative stress (OS); Delta opioid receptor (DOR); Poly (ADP-ribose)-polymerase1 (PARP1); Neuroprotection; Attenuation; OS; Oxidative stress; DOR; Delta opioid receptor; PARP; Poly (ADP-ribose)-polymerase; AD; Alzheimer's disease; PD; Parkinson's disease
Pharmacological characterization of novel synthetic opioids (NSO) found in the recreational drug marketplace
Keywords: Analgesia; Butyrylfentanyl; Mu-opioid receptor; MT-45; U-47700; DAMGO; [D-Ala2,N-MePhe4,Gly-ol]-enkephalin; DPDPE; [D-Pen2, D-Pen5]-enkephalin; DOR-1; delta-opioid receptor; GTPγS; guanosine 5â²-O-[gamma-thio]triphosphate; KOR-1; kappa-opioid receptor;
Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues
Keywords: BU72; 17-methyl-3-hydroxy-[5β,7β,3â²,5â²]-pyrrolidino-2â²[S]-phenyl-7α-methyl-6,14-endoetheno morphinan; CHO; Chinese hamster ovary; DPDPE; [D-Ala2-N-Me-Phe4-Gly-ol] enkephalin; EM-2; endomorphin-2; NMe; N-methyl; Opioid receptors; N-Methylated amin
The antinociceptive effects of a δ-opioid receptor agonist in mice with painful diabetic neuropathy: Involvement of heme oxygenase 1
Keywords: CoPP; cobalt protoporphyrin IX; CORM-2; tricarbonyldichlororuthenium(II) dimer; DOR; δ-opioid receptor; DPDPE; [d-Pen(2),d-Pen(5)]-Enkephalin; HO-1; inducible heme oxygenase; MOR; μ-opioid receptor; SnPP; tin protoporphyrin IX; STZ; streptozotocin; Anal
Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of replacement of the 3-hydroxyphenyl group with pyridine or thiophene bioisosteres
Keywords: [35S]GTPγS; sulfur-35 guanosine-5â²-O-(3-thio)triphosphate; DAMGO; [D-Ala2,MePhe4,Gly-ol5]enkephalin; DPDPE; [D-Pen2,D-Pen5]enkephalin; U69,593; (5α,7α,8β)-(â)-N-methyl-N-[7-(1-pyrrolidinyl)-1-oxaspiro[4,5]dec-8-yl]benzeneacetamide; JDTic; Opioids;
Design and synthesis of novel bivalent ligands (MOR and DOR) by conjugation of enkephalin analogues with 4-anilidopiperidine derivatives
Keywords: ACN; Acetonitrile; Boc; tert-butyloxycarbonyl; CHO; Chinese hamster ovary; DCM; Dichloromethane; DIPEA; N,N-Diisopropylethylamine; DALEA; [D-Ala2, Leu5] enkephalin amide; DAMGO; [D-Ala2,NMePhe4,Gly5-ol]enkephalin; Dmt; 2,6-dimethyltyrosine; DPDPE; c[D-Pen
RGS2 and RGS4 proteins: New modulators of the κ-opioid receptor signaling
Keywords: 293Â F; cell line of human embryonic kidney origin; 6ÃÂ His; hexahistidine; aa; amino acids; AC; adenylyl cyclase; AR; adrenergic receptors; AT1; Angiotensin Receptor 1; CT; carboxyl terminus; ÎÎRGS4; RGS4 lacking its N-terminal domain; DAMGO; [d-Ala2,
Blood-brain transfer and antinociception of linear and cyclic N-methyl-guanidine and thiourea-enkephalins
Keywords: Blood-brain barrier (BBB) transport (influx/efflux); Antinociceptive activity; Linear/cyclic enkephalin analogs; In vivo mouse models; AUC; area under the curve; Alloc; allyloxycarbonyl; BBB; blood-brain barrier; Boc; tertButyloxycarbonyl; BSA; bovine
μ-Opioid receptor 6-transmembrane isoform: A potential therapeutic target for new effective opioids
Keywords: MOR; μ-opioid receptor; 6TM MOR; six transmembrane helices μ-opioid receptor; 7TM MOR; seven transmembrane helices μ-opioid receptor; OIH; opioid induced hyperalgesia; VGCC; voltage-gated Ca2 + channels; cAMP; cyclic adenosine monophosphate; AC; adeny
LY2456302 is a novel, potent, orally-bioavailable small molecule kappa-selective antagonist with activity in animal models predictive of efficacy in mood and addictive disorders
Keywords: Opioid receptors; Kappa opioid antagonist; Antidepressant; Addiction; Alcohol dependence; Dynorphin; CREB; cyclic adenosine monophosphate-response element binding protein; DAMGO; [D-Ala2, N-MePhe4, Gly-ol]-enkephalin; DPDPE; [d-Pen2,d-Pen5]-enkephalin; ER
Accumbal core: Essential link in feed-forward spiraling striato-nigro-striatal in series connected loop
Keywords: ANOVA; analysis of variance; CTOP; D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Phe-Thr-NH2; DAMGO; [D-Ala2,N-Me-Phe4,Gly5-ol]-enkephalin; deltorphin II; [D-Ala2,Glu4]-deltorphin; DPDPE; [D-Pen2,5]-enkephalin; DS; dorsal subregion of the neostriatum; Nacc; nucleus accumbe
Endogenous opiates and behavior: 2012
Keywords: Ach; acetylcholine; ACTH; adrenocorticotrophic hormone; ANG; angiotensin; ATP; adenosine triphosphate; BAM22; bovine adrenal medulla 22; BDNF; brain-derived neurotrophic factor; BEND; beta-endorphin; BFNA; beta-funaltrexamine; BNST; bed nucleus of the str
Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists
Keywords: Boc; tert-butyloxycarbonyl; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; DIC; 1,3-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DPDPE; H-Tyr-c[d-Pen-Gly-Phe-D-Pen]OH; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH;
Decabromodiphenyl ethane and decabromodiphenyl ether in Swedish background air
Keywords: Brominated flame retardants; DPDPE; BDE-209; Atmospheric transport
Ãarrestin1-biased agonism at human δ-opioid receptor by peptidic and alkaloid ligands
Keywords: hDOR; human delta-opioid receptor; DPDPE; D-Penicillamine(2,5)-enkephalin; Deltorphin I; Tyr-D-Ala-Phe-Asp-Val-Val-Gly.NH2; δ-opioid receptor; Ãarrestin; G protein-coupled receptor; Peptidic and alkaloid ligands;
Influence of corticostriatal δ-opioid receptors on abnormal involuntary movements induced by L-DOPA in hemiparkinsonian rats
Keywords: AIMs; abnormal involuntary movements; DPDPE; [d-Pen2, d-Pen5]-enkephalin; EDTA; ethylenediaminetetraacetic acid; 6-OHDA; hydroxydopamine hydrochloride, HPLC, high performance liquid chromatography; l-DOPA; l-3,4-dihydroxyphenylalanine + benserazide; LID
Selective interactions of spinophilin with the C-terminal domains of the δ- and μ-opioid receptors and G proteins differentially modulate opioid receptor signaling
Keywords: GPCR; G protein-coupled receptors; RGS; Regulators of G protein Signaling; ÎÎRGS4; RGS4 lacking its N-terminal domain; 6xHis; hexahistidine; aa; amino acids; GEFs; Guanine nucleotide exchange factors; AC; adenylyl cyclase; DAMGO; [D-Ala2,N-MePhe4,Gly5-o
A comprehensive study on the putative δ-opioid receptor (sub)types using the highly selective δ-antagonist, Tyr-Tic-(2S,3R)-β-MePhe-Phe-OH
Keywords: Bmax; receptor density; BNTX; 7-benzylidenenaltrexone; DADLE; [d-Ala2,d-Leu5]enkephalin; deltorphin II; Tyr-d-Ala-Phe-Glu-Val-Val-Gly-NH2; DOR-1; δ-opioid receptor; DOR-KO; δ-opioid receptor knock-out; DPDPE; Tyr-c[d-Pen-Gly-Phe-d-Pen]-OH; DSLET; Tyr-d-
Inhibition of spontaneous excitatory transmission induced by codeine is independent on presynaptic K+ channels and novel voltage-dependent Ca2+ channels in the guinea-pig nucleus tractus solitarius
Keywords: EPSC; second-order NTS neuron; codeine; Ca2+ channel; K+ channel; aCSF; artificial cerebrospinal fluid; CNQX; 6-cyano-7-nitroquinoxaline-2,3-dione disodium; CTAP; H-D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2; DAMGO; Tyr-D-Ala-Gly-N-methyl-Phe-Gly-ol; DPDPE;
Peripheral delta opioid receptors require priming for functional competence in vivo
Keywords: DPDPE; Hindpaw; Prostaglandin; Bradykinin; Allodynia
Activation of mu, delta or kappa opioid receptors by DAMGO, DPDPE, U-50488 or U-69593 respectively causes antinociception in the formalin test in the naked mole-rat (Heterocephalus glaber)
Keywords: Formalin test; Naked mole-rat; Nociception; Antinociception; DAMGO; DPDPE; U-50488; U-69593
Pharmacological characterization of the nociceptin/orphanin FQ receptor non peptide antagonist Compound 24
Keywords: N/OFQ; Nociceptin/orphanin FQ; NOP; N/OFQ peptide receptor; Compound 24; 1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4â²-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide; CHO; Chinese hamster ovary; DPN; diprenorphine; DPDPE; [d-Pen2,d-Pen5]enkephalin; BSA;
Role of the opioid system in incentive downshift situations
Keywords: Opioid system; Incentive contrast; Consummatory successive negative contrast; Appetitive extinction; Naloxone; Naltrindole; DPDPE; Rats
Delta opioid receptors mediate chemotaxis in bone marrow-derived dendritic cells
Keywords: MOR; μ-opioid receptor; DOR; δ-opioid receptor; KOR; κ-opioid receptor; DC; dendritic cell; CMFDA; 5-chloromethylfluorescein diacetate; DPDPE; [D-Pen2,5]-Enkephalin; β-CNA; β-Chlornaltrexamine dihydrochloride; Opioids; Chemotaxis; Dendritic cells;
Cellular neurosciencePresynaptic actions of opioid receptor agonists in ventromedial hypothalamic neurons in estrogen- and oil-treated female mice
Keywords: VMH; opioid receptor; patch-clamp; arousal; lordosis; ACSF; artificial cerebrospinal fluid; CTAP; d-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2; DAMGO; [d-Ala2, N-Me-Phe4, Gly5-ol]-enkephalin; DPDPE; [d-Pen2,d-Pen5]-enkephalin; E; 17β-estradiol; GPCRs; G-prote
Neuroprotection and functional recovery conferred by administration of kappa- and delta1-opioid agonists in a rat model of global ischemia
Keywords: Global ischemia; U50; 488H; Neuronal protection; Hippocampus; CA1; Spatial memory; DPDPE; Behavioral hyperactivity; Rats
μ-Opioid agonists inhibit the enhanced intracellular Ca2+ responses in inflammatory activated astrocytes co-cultured with brain endothelial cells
Keywords: astrocyte; calcium; endothelial cells; inflammatory activators; opioids; pain-transmitting peptides; BBB; blood-brain barrier; BSA; bovine serum albumin; [Ca2+]i; intracellular free calcium; CGRP; calcitonin gene-related peptide; DAMGO; [d-Ala2,NMe-Phe4
Anti-allodynic effects of peripheral delta opioid receptors in neuropathic pain
Keywords: Chronic constriction injury; Deltorphin II; DPDPE; Morphine; Dorsal root ganglia; Pain
Influence of glial cells in the dopamine releasing effect resulting from the stimulation of striatal δ-opioid receptors
Keywords: microdialysis; DPDPE; glutamate release; striatum; gliotoxin; l-α-aminoadipateANOVA, analysis of variance; A/P, antero-posterior; AUC, area under the curve; DOPAC, 3,4-dihydroxyphenylacetic acid; DPDPE, [d-Pen2, d-Pen5]-enkephalin; D/V, deep vertical; GMH
Presynaptic modulation of 5-HT release in the rat septal region
Keywords: lateral septum; medial septum; diagonal band; 5-HT1B; α2-adrenoceptor; opioid receptors; ACh; acetylcholine; ANOVA; analysis of variance; CGP-56,999A; 3-([1-(R)-(3-carboxyphenyl)ethylamino]2-(S)-hydroxy-propyl)-cyclohexyl-methyl-phosphinic acid (lithium
The role of progestin receptors and the mitogen-activated protein kinase pathway in δ opioid receptor facilitation of female reproductive behaviors
Keywords: Lordosis; Progesterone; δ Opioid receptors; MAPK; PD98059; DPDPE; RU486
δ-opioid receptor-mediated actions on rostral ventromedial medulla neurons
Keywords: ACSF; artificial cerebrospinal fluid; BSA; bovine serum albumin; DAMGO; [d-Ala2, NMe-Phe4, Gly-ol5]-enkephalin; deltorphin-II; [d-Ala2]-deltorphin II; DPDPE; [d-Pen2; d-Pen5]-enkephalin; RVM; rostral ventromedial medulla; TPH; tryptophan hydroxylase; TPH-
μ-opioid-mediated inhibition of glutamate synaptic transmission in rat central amygdala neurons
Keywords: phospholipase A2; 4AP-sensitive potassium channel; reward; analgesia; AP5; 2-amino-5-phosphonovaleric acid; BLA; basolateral nucleus of the amygdala; CeA; central nucleus of the amygdala; CNQX; 6-cyano-7-nitroquinoxaline-2,3-dione; DAMGO; [d-Ala2,N-MePhe4
Leishmania donovani amastigote component-induced colony-stimulating factor production by macrophages: modulation by morphine
Keywords: Morphine; Leishmania donovani; Colony-stimulating factors; Macrophages; CDMEM; complete DMEM; CM; conditioned media; CSFs; colony-stimulating factors; DAGO; (d-Al2, N-Me-Phe4, Gly5-ol)-enkephalin acetate salt; DMEM; Dulbecco's modified Eagle's medium;
Localization of opioid receptor antagonist [3H]-LY255582 binding sites in mouse brain: Comparison with the distribution of mu, delta and kappa binding sites
Keywords: AcbC; nucleus accumbens,core; BLA; basolateral nucleus of the amygdala; CA3; CA3 region of the hippocampus; cl; claustrum; CG; central gray; CI, 977; (â)-N-methyl-N-[7-(1-pyrrolidinyl)-1-oxaspiro[4,5]dec-8-yl]-4-benzofuranacetamide; CPu; caudate; CTR; c
The non-peptidic delta opioid receptor agonist TAN-67 enhances dopamine efflux in the nucleus accumbens of freely moving rats via a mechanism that involves both glutamate and free radicals
Keywords: TAN-67; dopamine; nucleus accumbens; microdialysis; glutamate; free radical; ANOVA; analysis of variance; deltorphin-II; [d-Ala2,Glu4]-deltorphin; DPDPE; d-[Pen2,5]-enkephalin; EDTA; ethylendiaminetetraacetic acid; α-methyl-para-tyrosine; α-methyl-para-
Interactions among mu- and delta-opioid receptors, especially putative delta1- and delta2-opioid receptors, promote dopamine release in the nucleus accumbens
Keywords: opioid receptors; receptor interaction; nucleus accumbens; dopamine release; rats; ANOVA; analysis of variance; BNTX; (E)-7-benzylidenenaltrexone; CTOP; d-Phe-Cys-Tyr-d-Trp-Orn-Thr-Phe-Thr-NH2; DAMGO; [d-Ala2,N-Me-Phe4,Gly5-ol]-enkephalin; DPDPE; [d-Pen2,
N-methyl-d-aspartate receptors and large conductance calcium-sensitive potassium channels inhibit the release of opioid peptides that induce μ-opioid receptor internalization in the rat spinal cord
Keywords: dorsal horn; dynorphin; enkephalin; internalization; mu-opioid receptor; opioid; aCSF; artificial cerebrospinal fluid; ANOVA; analysis of variance; AP-5; dl-2-amino-5-phosphonopentanoic acid; BK(Ca2+); large conductance Ca2+-sensitive K+ channels; CCK; ch
Intracerebroventricular d-Pen2, d-Pen5-enkephalin administration soon after stressor imposition influences behavioral responsivity to a subsequent stressor encounter in CD-1 mice
Keywords: Opioid; Footshock; Horizontal locomotion; Rearing; Dose; DPDPE; Contextual learning; Cues; Memory; Sensitization;