Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: Identification of an efficient lead for potent inhibitors of GABA transports
Keywords: بالا به همراه پیچ و خم; ANOVA; analysis of variance; BGT; betaine-GABA transporter; CHO; Chinese hamster ovary; CNS; central nervous systems; EPM; elevated plus maze; GABA; γ-aminobutyric acid; GAT; GABA transporter; LE; ligand efficiency; PTZ; pentylenetetrazole; SNAP; 1-(2-[t