Keywords: HIV-1 انتگرال; HIV-1 integrase; Strand-transfer inhibitors; Molecular docking; Flow chemistry;
مقالات ISI HIV-1 انتگرال (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
The discovery and preclinical evaluation of BMS-707035, a potent HIV-1 integrase strand transfer inhibitor
Keywords: HIV-1 انتگرال; HIV-1 integrase; Strand transfer inhibitors; INSTI; Pyrimidinone carboxamides; Antiviral activity; Pharmacokinetics;
Novel secondary mutations C56S and G149A confer resistance to HIV-1 integrase strand transfer inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Strand transfer inhibitor; Cabotegravir; Secondary mutations;
1-Hydroxypyrido[2,3-d]pyrimidin-2(1H)-ones as novel selective HIV integrase inhibitors obtained via privileged substructure-based compound libraries
Keywords: HIV-1 انتگرال; HIV-1; CuAAC; HIV-1 integrase; HIV-1 RNase H; “Privileged structure”-guided scaffold reposition;
An effective HIV-1 integrase inhibitor screening platform: Rationality validation of drug screening, conformational mobility and molecular recognition analysis for PFV integrase complex with viral DNA
Keywords: HIV-1 انتگرال; HIV-1 integrase; Molecular docking; Molecular dynamics simulation; Binding free energy; Drug design;
Discovery of novel 3-hydroxypicolinamides as selective inhibitors of HIV-1 integrase-LEDGF/p75 interaction
Keywords: HIV-1 انتگرال; HIV-1 integrase; Allosteric inhibitor; LEDGF/p75; Dimerization; 3-Hydroxypicolinamide;
Exploring the binding of d(GGGT)4 to the HIV-1 integrase: An approach to investigate G-quadruplex aptamer/target protein interactions
Keywords: HIV-1 انتگرال; Aptamer T30695; G-quadruplex; HIV-1 integrase; Microscale thermophoresis; Circular dichroism; NMR;
2-hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4
Keywords: HIV-1 انتگرال; HIV-1 integrase; Two-metal binding pharmacophore; Antiretroviral; 2-hydroxyisoquinoline-1,3(2H,4H)-diones; AZT; azidothymidine; CPE; cytopathic effect; CYP; cytochrome P450; FC; fold-change in EC50 relative to wild-type strain of HIV-1; FDA; food and drug
Investigation on the sucrose binding pocket of HIV-1 Integrase by molecular dynamics and synergy experiments
Keywords: HIV-1 انتگرال; HIV-1 Integrase; Sucrose; Protein–protein interaction; Molecular dynamics
Anti-HIV-1 integrase diterpenoids from Dichrocephala benthamii
Keywords: HIV-1 انتگرال; Asteraceae; Dichrocephala benthamii; Clerodane diterpenoids; HIV-1 integrase;
Design and synthesis of N-methylpyrimidone derivatives as HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibitors; N-Methylpyrimidone; Synthesis;
Novel furocoumarins as potential HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; Furocoumarins; HIV-1 integrase; Strand-transfer inhibitors; Rational design
1,4-Bis(5-(naphthalen-1-yl)thiophen-2-yl)naphthalene, a small molecule, functions as a novel anti-HIV-1 inhibitor targeting the interaction between integrase and cellular Lens epithelium-derived growth factor
Keywords: HIV-1 انتگرال; HIV-1 integrase; Lens epithelium-derived growth factor (LEDGF/P75); Molecular docking
Nuclear trafficking of the HIV-1 pre-integration complex depends on the ADAM10 intracellular domain
Keywords: HIV-1 انتگرال; ADAM10; ADAM15; γ-Secretase; HIV-1 replication; Macrophages; CD4+ T lymphocytes; HIV-1 pre-integration complex (PIC); HIV-1 integrase;
Discovery of a novel HIV-1 integrase inhibitor from natural compounds through structure based virtual screening and cell imaging
Keywords: HIV-1 انتگرال; HIV-1 integrase; Lens epithelium-derived growth factor (LEDGF/P75); Virtual screening;
Consensus HIV-1 subtype A integrase and its raltegravir-resistant variants: Design and characterization of the enzymatic properties
Keywords: HIV-1 انتگرال; HIV-1 integrase; Subtype A; Consensus; Catalytic activity; Raltegravir; Drug resistance;
Combined ligand and structure-based approaches on HIV-1 integrase strand transfer inhibitors
Keywords: HIV-1 انتگرال; 3D-QSAR; HIV-1 integrase; Pharmacophore; QPLD; Strand transfer inhibitor;
Molecular dynamics study of carbon nanotube as a potential dual-functional inhibitor of HIV-1 integrase
Keywords: HIV-1 انتگرال; HIV-1 integrase; Integrase inhibitor; Carbon nanotube; Drug delivery; Molecular dynamics simulation;
Reduced HIV-1 integrase flexibility as a mechanism for raltegravir resistance
Keywords: HIV-1 انتگرال; HIV-1 integrase; Drug resistance; Raltegravir; Molecular dynamics; NAMD;
New scaffolds of natural origin as Integrase-LEDGF/p75 interaction inhibitors: Virtual screening and activity assays
Keywords: HIV-1 انتگرال; HIV-1 Integrase; LEDGF/p75; Protein-protein interaction inhibitors; LEDGINs; Natural products; Virtual screening; AIDS; acquired immunodeficiency syndrome; CCD; catalytic core domain; HIV-1; human immunodeficiency virus type 1; IBD; integrase binding do
Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase-LEDGF/p75 interaction
Keywords: HIV-1 انتگرال; IN; HIV-1 integrase; LEDGF/p75; lens epithelium-derived growth factor/p75; HBD; hydrogen bond donor; HBA; hydrogen bond acceptor; IC50; 50% inhibitory concentration; EC50; 50% effective concentration; CC50; 50% cytotoxic concentration; CCID50; cell cultur
Synthesis, docking, and biological studies of phenanthrene β-diketo acids as novel HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1; HIV-1 integrase; Phenanthrene β-diketo acids; ST inhibitors; Docking
6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibit; Raltegravir; Sulfonamide;
Discovery of small molecule HIV-1 integrase dimerization inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Dimerization; AlphaScreen; Protein-protein interactions;
Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 Integrase; Inhibitor; 1,3-Diketo; Polyhydroxylated aromatics; Strand transfer;
A new fluorometric assay for the study of DNA-binding and 3â²-processing activities of retroviral integrases and its use for screening of HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; 3â²-end fluorescein-labeled oligonucleotides; Fluorescence-base assay; 3â²-Processing inhibitors;
Multiple sites of the cleavage of 17- and 19-mer encephalytogenic oligopeptides corresponding to human myelin basic protein (MBP) by specific anti-MBP antibodies from patients with systemic lupus erythematosus
Keywords: HIV-1 انتگرال; Ab; antibody; Abz; abzyme; AD; autoimmune disease; MBP; human myelin basic protein; HIV-1; human immunodeficiency virus type 1; IN; HIV-1 integrase; MCA; 4-methylcoumaryl-7-amine; OP; oligopeptide; RPhC; reverse-phase chromatography; PAGE; polyacrylamide
Development of tricyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibit; Raltegravir; Cycloaddition
4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process
Keywords: HIV-1 انتگرال; HIV-1 integrase; INSTI; IN-LEDGF/p75; Dual inhibitor;
Natural polymorphisms of HIV-1 CRF01_AE integrase coding region in ARV-naïve individuals in Cambodia, Thailand and Vietnam: An ANRS AC12 working group study
Keywords: HIV-1 انتگرال; HIV-1 integrase; Resistance mutations; Antiretroviral naïve; South East Asia
Binding modes of diketo-acid inhibitors of HIV-1 integrase: A comparative molecular dynamics simulation study
Keywords: HIV-1 انتگرال; HIV-1 integrase; Diketo acid inhibitors; Molecular dynamics; Ion-pair interaction; Catalytic loop;
HIV-1 integrase strand-transfer inhibitors: Design, synthesis and molecular modeling investigation
Keywords: HIV-1 انتگرال; HIV-1 integrase; INSTIs; PFV-IN/DNA; Benzylindoles; Molecular dockingINSTIs, integrase strand transfer inhibitors; PFV, prototype foamy virus; DKAs, diketo acids; IFD, induced-fit docking
Active site binding modes of dimeric phloroglucinols for HIV-1 reverse transcriptase, protease and integrase
Keywords: HIV-1 انتگرال; HIV-1 reverse transcriptase; HIV-1 integrase; HIV-1 protease; Dimeric phloroglucinols; Docking;
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor
Keywords: HIV-1 انتگرال; HIV-1 integrase; LEDGF/p75; Protein–protein interactions; Molecular docking; GRID
Crystal structure of the HIV-1 integrase core domain in complex with sucrose reveals details of an allosteric inhibitory binding site
Keywords: HIV-1 انتگرال; Anti-HIV drug; Ligand binding; HIV-1 integrase; X-ray crystallography
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action
Keywords: HIV-1 انتگرال; HIV-1 integrase; Induced-fit docking; Integrase strand-transfer inhibitors; Microwave-assisted organic synthesis;
1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 position
Keywords: HIV-1 انتگرال; HIV-1 integrase; Integration; Two-metal chelation
3-Hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylates—A new class of HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibitor; Spread assay; Pyridopyrimidine; Oxalamide
Dihydroxy-pyrimidine and N-methylpyrimidone HIV-integrase inhibitors: Improving cell based activity by the quaternarization of a chiral center
Keywords: HIV-1 انتگرال; HIV-1 integrase; Pyrimidines; N-Methylpyrimidones; PAMPA
Cellular protein TTRAP interacts with HIV-1 integrase to facilitate viral integration
Keywords: HIV-1 انتگرال; TTRAP; HIV-1 integrase; Lentivirus; Integration
A docking study of l-chicoric acid with HIV-1 integrase
Keywords: HIV-1 انتگرال; l-Chicoric acid; HIV-1 integrase; Ligand binding; α,β-Unsaturated ester; Conformational analysis; AM1; Ab initio
HIV-1 integrase-hydrolyzing antibodies from sera of HIV-infected patients
Keywords: HIV-1 انتگرال; Human blood antibodies; HIV-infected patients; Catalytic IgGs; Hydrolysis of HIV integrase; Ab; antibody; Abz; abzyme; AI; autoimmune; GL; generalized lymphoadenopathy; IN; HIV-1 integrase; pIgG; polyclonal IgG; RT; HIV-1 reverse transcriptase; SDS-PAGE;
Multivariate QSAR study of 4,5-dihydroxypyrimidine carboxamides as HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; QSAR; 4,5-Dihydroxypyrimidine carboxamides; HIV-1 integrase; OPS; PLS3′P, 3′-processing; 5CITEP, 1-(5-chloroindol-3-yl)-3-hydroxy-3-(2H-tetrazol-5-yl)-propenone; AIDS, acquired immunodeficiency syndrome; AM1, Austin Model 1; ARE, average relative error; B
Diketoacid-genre HIV-1 integrase inhibitors containing enantiomeric arylamide functionality
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibit; Enantiomer; Arylamide; Diketoacid
Site-specific integration of retroviral DNA in human cells using fusion proteins consisting of human immunodeficiency virus type 1 integrase and the designed polydactyl zinc-finger protein E2C
Keywords: HIV-1 انتگرال; Designed polydactyl zinc-finger protein; E2C; Gene therapy; HIV-1 integrase; IN fusion proteins; Insertional mutagenesis; Quantitative PCR; Retroviral vectors; Retroviral DNA integration; Site-directed integration
Docking-based 3D-QSAR study of HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; HIV-1 integrase; Docking; CoMFA; CoMSIA
Analysis of binding parameters of HIV-1 integrase inhibitors: Correlates of drug inhibition and resistance
Keywords: HIV-1 انتگرال; HIV-1 integrase; Inhibitors; Raltegravir; Elvitegravir; Autodock; Resistance;
Daxx interacts with HIV-1 integrase and inhibits lentiviral gene expression
Keywords: HIV-1 انتگرال; Daxx; HIV-1 integrase; Lentivirus; Gene expression; Histone deacetylases (HDACs)
Synthesis of trans-caffeate analogues and their bioactivities against HIV-1 integrase and cancer cell lines
Keywords: HIV-1 انتگرال; Caffeate analogues; HIV-1 integrase; Antitumor
4-Hydroxy-5-pyrrolinone-3-carboxamide HIV-1 integrase inhibitors
Keywords: HIV-1 انتگرال; AIDS; HIV-1 integrase; Diketoacids; Pyrimidines; Pyrrolinones