Keywords: ایمیدازپیریدین; Imidazopyridine; Triazoles; Tubulin; Apoptosis; Lung cancer;
مقالات ISI ایمیدازپیریدین (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: ایمیدازپیریدین; Aldosterone; CYP11B2; Hypertension; Imidazopyridine; Heart failure;
Keywords: ایمیدازپیریدین; Imidazopyridine; Ortho-haloaminopyridine; C-N coupling; Imidazopyrazine; Purine;
Keywords: ایمیدازپیریدین; Imidazopyridine; IR and Raman spectra
Keywords: ایمیدازپیریدین; Ionic liquid; Imidazopyridine; Heterocyclization; Room temperature; Mild reaction conditions;
Iron(III)-catalyzed synthesis of 3-aroylimidazo[1,2-a]pyridines from 2-aminopyridines and ynals
Keywords: ایمیدازپیریدین; Iron-catalyzed; Imidazopyridine; Aminopyridine; Ynal; Cyclization;
Identification of an imidazopyridine scaffold to generate potent and selective TYK2 inhibitors that demonstrate activity in an in vivo psoriasis model
Keywords: ایمیدازپیریدین; TYK2; Kinase; Psoriasis; Imidazopyridine; IL-23;
Development of 1-aryl-3-furanyl/thienyl-imidazopyridine templates for inhibitors against hypoxia inducible factor (HIF)-1 transcriptional activity
Keywords: ایمیدازپیریدین; Hypoxia inducible factor (HIF)-1; Imidazopyridine; CH direct arylation; Microwave;
Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-PI3 kinases that are efficacious in a mouse xenograft model
Keywords: ایمیدازپیریدین; Cancer; Lipid kinases; PI3K; Pan-PI3 kinases; Pan-PI3 kinase inhibitor; Imidazopyridine; Dihedral angle
Composés á structure imidazopyridinyl-arylpropénone, nouveaux agents anti-infectieux potentiels
Keywords: ایمیدازپیریدین; Imidazopyridine; Arylpropenone; Antiplasmodial; Nematicidal; Anti-Candida albicans; Imidazopyridine; Arylpropénone; Antiplasmodial; Nématocide; Anticandidosique;
Design, syntheses, and anti-tuberculosis activities of conjugates of piperazino-1,3-benzothiazin-4-ones (pBTZs) with 2,7-dimethylimidazo [1,2-a]pyridine-3-carboxylic acids and 7-phenylacetyl cephalosporins
Keywords: ایمیدازپیریدین; Tuberculosis; Benzothiazinones; Imidazopyridine; Cephalosporin;
Synthesis and biological evaluation of imidazopyridinyl-1,3,4-oxadiazole conjugates as apoptosis inducers and topoisomerase IIα inhibitors
Keywords: ایمیدازپیریدین; Imidazopyridine; Oxadiazole; Cytotoxicity; Topoisomerase; Molecular docking;
Discovery of potent 1H-imidazo[4,5-b]pyridine-based c-Met kinase inhibitors via mechanism-directed structural optimization
Keywords: ایمیدازپیریدین; c-Met tyrosine kinase; Small molecule inhibitor; Imidazonaphthyridinone; Imidazopyridine; Binding mode; Pyridone-3-carboxamide; Cyclopropane-1,1-dicarboxamide
Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability
Keywords: ایمیدازپیریدین; PDE10A inhibitor; Schizophrenia; Benzimidazole; Imidazopyridine; Metabolic stability;
Imidazo[4,5-b]pyridine inhibitors of B-Raf kinase
Keywords: ایمیدازپیریدین; B-Raf; Imidazopyridine; Scaffold hopping; DFG-in; αC-helix out;
Synthesis of 2-substituted 3-ethyl-3H-imidazo[4,5-b]pyridines catalyzed by Al3+-exchanged K10 clay as solid acids
Keywords: ایمیدازپیریدین; Al3+-exchanged on K10 clay; Imidazopyridine; Heterogeneous catalysis; Solid acids; Heterocycles;
Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K
Keywords: ایمیدازپیریدین; Cancer; Lipid kinase; PI3 kinase inhibitor; Imidazopyridine; Structure-guided drug design; Scaffold morphing
Design, synthesis and biological evaluation of novel imidazopyridines as potential antidiabetic GSK3β inhibitors
Keywords: ایمیدازپیریدین; Glycogen synthase kinase 3; Imidazopyridine; Type 2 diabetes mellitus; Oral glucose tolerance test;
Bridging homogeneous and heterogeneous catalysis with MOFs: Cu-MOFs as solid catalysts for three-component coupling and cyclization reactions for the synthesis of propargylamines, indoles and imidazopyridines
Keywords: ایمیدازپیریدین; Cu-MOF catalysis; Three-component coupling; Indole; Imidazopyridine;
Discovery and optimization of potent and selective imidazopyridine and imidazopyridazine mTOR inhibitors
Keywords: ایمیدازپیریدین; mTOR; Kinase inhibitor; Oncology; Imidazopyridine; Imidazopyridazine
Arylazolyl(azinyl)thioacetanilides. Part 10: Design, synthesis and biological evaluation of novel substituted imidazopyridinylthioacetanilides as potent HIV-1 inhibitors
Keywords: ایمیدازپیریدین; HIV; NNRTIs; Heterocycle; Synthesis; Anti-HIV-1 activity; SAR; Imidazopyridine; Scaffold hopping;
Synthesis of 5-bromo-6-methyl imidazopyrazine, 5-bromo and 5-chloro-6-methyl imidazopyridine using electron density surface maps to guide synthetic strategy
Keywords: ایمیدازپیریدین; Electron density surface maps; Electrophilic aromatic substitution; Imidazopyrazine; Imidazopyridine;
Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs
Keywords: ایمیدازپیریدین; Oxadiazole; Benzimidazole; Phenyl imidazole; Imidazopyridine; Imidazo[2,1-b][1,3]benzothiazole; Antibacterial; Antifungal
Vibrational spectra and structure of methyl-derivatives of imidazo[4,5-c]pyridine based on DFT quantum chemical calculations and XRD studies
Keywords: ایمیدازپیریدین; Imidazopyridine; Quantum chemical calculations; Crystal and molecular structure; Infrared and Raman spectra; N–H⋯N hydrogen bond
Modulation of carcinogen metabolizing enzymes by new fused heterocycles pendant to 5,6,7,8-tetrahydronaphthalene derivatives
Keywords: ایمیدازپیریدین; Pyrimidinum bromide; Indolizine; Imidazopyridine; Quinoxaline; Imidazotriazole; Imidazobenzimidazole; Carcinogen metabolizing enzymesCyp1A, Cytochrome P-450 1A; GSH, Glutathione; GSTs, Glutathione S-transferases; mEH, Epoxide hydrolase; MMS, Methyl methan
Post Groebke-Blackburn multicomponent protocol: Synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents
Keywords: ایمیدازپیریدین; Oxadiazole; Benzimidazole; Phenyl imidazole; Imidazopyridine; Imidazopyrimidine; Antibacterial agents;
Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors
Keywords: ایمیدازپیریدین; Dipeptidyl peptidase-IV; DPP-4; DPP-IV; Dipeptidyl peptidase 8; DPP-8; DPP-9; Quiescient peptidyl peptidase; QPP; GLP-1; Glucagon-like peptide 1; Benzimidazole; Imidazopyridine; Buchwald coupling; Sitagliptin;
Imidazopyridine-5,6,7,8-tetrahydro-8-quinolinamine derivatives with potent activity against HIV-1
Keywords: ایمیدازپیریدین; CXCR4; HIV; Antiviral; Imidazopyridine; Tetrahydroquinoline
DNA gyrase (GyrB)/topoisomerase IV (ParE) inhibitors: Synthesis and antibacterial activity
Keywords: ایمیدازپیریدین; Antibacterial; Gyrase; Imidazopyridine; Triazolopyridine
Imidazopyridine derivatives as potent and selective Polo-like kinase (PLK) inhibitors
Keywords: ایمیدازپیریدین; PLK1; Polo-like kinase; Imidazopyridine
Imidazopyridines as VLA-4 integrin antagonists
Keywords: ایمیدازپیریدین; VLA-4; Integrin; Imidazopyridine; Phenylalanine
IRAK-4 inhibitors. Part II: A structure-based assessment of imidazo[1,2-a]pyridine binding
Keywords: ایمیدازپیریدین; IRAK; IRAK-4; JNK; Kinase; Kinase inhibitor; IRAK-4 inhibitor; Homology model; Imidazopyridine; Imidazo[1,2-a]pyridine; Binding mode; JNK crystal structure; GASP; Docking; Hinge binder; Hinge region; Bidentate hydrogen bond; β-Turn; Protein modelling; IRA
Imidazolyl benzimidazoles and imidazo[4,5-b]pyridines as potent p38α MAP kinase inhibitors with excellent in vivo antiinflammatory properties
Keywords: ایمیدازپیریدین; p38 MAP kinase; Inflammation; Imidazole; Imidazopyridine
Imidazo[4,5-c]pyridines inhibit the in vitro replication of the classical swine fever virus and target the viral polymerase
Keywords: ایمیدازپیریدین; Antiviral agent; Flaviviridae; Pestivirus; Inhibition of classical swine fever virus; RNA-polymerase; Imidazopyridine
In Vitro Phototoxic Potential and Photochemical Properties of Imidazopyridine Derivative: A Novel 5-HT4 Partial Agonist
Keywords: ایمیدازپیریدین; phototoxicity; photodegradation; oxidative stress; reactive oxygen species; imidazopyridine;
Synthesis and biological activity of imidazopyridine anticoccidial agents: Part II
Keywords: ایمیدازپیریدین; Coccidiosis; Antiparasitic; Antiprotozoal; Kinase; Imidazopyridine
Synthesis and SAR studies of potent imidazopyridine anticoccidial agents
Keywords: ایمیدازپیریدین; Et-PKG; Coccidiosis; Imidazopyridine
Synthesis and biological activity of imidazopyridine anticoccidial agents: Part I
Keywords: ایمیدازپیریدین; Coccidiosis; Antiparasitic; Antiprotozoal; Kinase; Imidazopyridine
Synthesis and SAR studies of very potent imidazopyridine antiprotozoal agents
Keywords: ایمیدازپیریدین; Protein kinase G; Antiprotozoan; Anticoccidial; Imidazopyridine
Stereodynamics of Ar-CO rotation and conformational preferences of 2-amino-3-(2,4-difluorobenzoyl)-imidazo[1,2-a]pyridine
Keywords: ایمیدازپیریدین; Ar-CO rotation; Conformational analysis; Dynamic NMR; Imidazopyridine; CDK inhibitors;
Inhibitors of casein kinase 1 block the growth of Leishmania major promastigotes in vitro
Keywords: ایمیدازپیریدین; Trypanosomatid; Leishmania; Protozoa; Imidazopyridine; Casein kinase 1