Metabolic responses in Candida tropicalis to complex inhibitors during xylitol bioconversion
Keywords: بازدارنده; Metabolomics; Xylitol; Inhibitor; Hemicellulose hydrolysate; GC/MS;
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Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
Keywords: بازدارنده; Rhodesain; Dipeptide-like; 3-Bromo isoxazoline; Inhibitor; Molecular modeling
4-Dechloro-14-deoxy-oxacyclododecindione and 14-deoxy-oxacylododecindione, two inhibitors of inducible connective tissue growth factor expression from the imperfect fungus Exserohilum rostratum
Keywords: بازدارنده; CTGF; Inhibitor; Fibrosis; β-Resorcylic acid lactones
Effect of SI-591, a new class of cathepsin K inhibitor with peptidomimetic structure, on bone metabolism in vitro and in vivo
Keywords: بازدارنده; OP; Osteoporosis; CTX-I; C-terminal crosslinking telopeptide of type I collagen; BGP; Bone Gla protein; BMD; Bone mineral density; PTH; Parathyroid hormone; TRAP; Tartrate-resistant acid phosphatase; OVX; Ovariectomized; DEXA; Dual energy X-ray absorptiom
Design, synthesis and evaluation of XZH-5 analogues as STAT3 inhibitors
Keywords: بازدارنده; STAT3; Inhibitor; SARs; SH2; Small organic molecule; Molecular docking
Discovery of bicyclic pyrazoles as class III histone deacetylase SIRT1 and SIRT2 inhibitors
Keywords: بازدارنده; DJSXAFBEVHGPLR-UHFFFAOYSA-N; Sirtuin; SIRT; Inhibitor; Pyrazole; Docking;
In vitro inhibitory effects of ethanol extract of Danshen (Salvia miltiorrhiza) and its components on the catalytic activity of soluble epoxide hydrolase
Keywords: بازدارنده; Danshen (Salvia miltiorrhiza); Soluble epoxide hydrolase (sEH); Inhibitor; Tanshinone IIA; Cryptotanshinone; Salvianolic acid C
Effects of third generation P-glycoprotein inhibitors on the sensitivity of drug-resistant and -susceptible isolates of Haemonchus contortus to anthelmintics in vitro
Keywords: بازدارنده; P-glycoprotein; Inhibitor; Anthelmintic; Resistance; In vitro; Haemonchus contortus;
Theoretical and experimental investigations on corrosion control of 65Cu-35Zn brass in nitric acid by two thiophenol derivatives
Keywords: بازدارنده; Brass; Inhibitor; Corrosion; Adsorption; Quantum chemical study;
Effect of NaCl, methanol and ethylene glycol on the phase equilibrium of methane hydrate in aqueous solutions of tetrahydrofuran (THF) and tetra-n-butyl ammonium bromide (TBAB)
Keywords: بازدارنده; Hydrate; Inhibitor; Phase stability; Tetrahydrofuran; Tetra-n-butyl ammonium bromide
Inhibitors of serine proteases decrease sperm penetration during porcine fertilization in vitro by inhibiting sperm binding to the zona pellucida and acrosome reaction
Keywords: بازدارنده; Serine protease; Inhibitor; Porcine; IVF
Epoxide hydrolase activities and epoxy fatty acids in the mosquito Culex quinquefasciatus
Keywords: بازدارنده; Mosquito; Epoxide hydrolase; Epoxy fatty acid; Eicosanoid; Inhibitor; Signaling moleculeEH, epoxide hydrolase; JH, juvenile hormone; sEH, soluble epoxide hydrolase; JHEH, juvenile hormone epoxide hydrolase; AgEH, epoxide hydrolase from A. gambiae; HsEH, s
Novel pH-dependent regulation of human cytosolic sialidase 2 (NEU2) activities by siastatin B and structural prediction of NEU2/siastatin B complex
Keywords: بازدارنده; Neuraminidase 2; Siastatin B; Docking model; Inhibitor; Chemical chaperone
Inhibitive activities detection of monoamine oxidases (MAO) A and B inhibitors in human liver MAO incubations by UPLC-ESI-MS/MS
Keywords: بازدارنده; MAO-A; MAO-B; 5-HIAA; PAA; Inhibitor; UPLC-ESI MS/MS;
Structures and binding studies of the complexes of phospholipase A2 with five inhibitors
Keywords: بازدارنده; Phospholipase A2; Inflammation; Inhibitor; Binding study; Crystal structure;
Synthesis of mannoheptose derivatives and their evaluation as inhibitors of the lectin LecB from the opportunistic pathogen Pseudomonas aeruginosa
Keywords: بازدارنده; Lectin; Pseudomonas aeruginosa; Inhibitor;
C-(2-Deoxy-d-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors
Keywords: بازدارنده; C-Glycosyl compounds; d-Glucal; Oxadiazoles; Glycogen phosphorylase; Inhibitor;
Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1,5-dihydro-pyrrol-2-one
Keywords: بازدارنده; ASK1; apoptosis signal-regulating kinase 1; MAPK; mitogen-activated protein kinase; ER; endoplasmic reticulum; TNF-α; tumor necrosis factor-alpha; AIP-1; ASK1-interacting protein 1; VEGF; vascular endothelial growth factor; Aβ; amyloid beta; CK2; protei
A high throughput screening assay for identifying glycation inhibitors on MALDI-TOF target
Keywords: بازدارنده; Screening assay; Glycation; MALDI-TOF; Reaction on target; Inhibitor
PTEN inhibitors: An evaluation of current compounds
Keywords: بازدارنده; Phosphatase; Enzyme; Inhibitor; Drug; PI 3-Kinase; PTEN; Phosphoinositide;
FAITH - Fast Assembly Inhibitor Test for HIV
Keywords: بازدارنده; Retrovirus; HIV; Assembly; Assay; Inhibitor; High-throughput screening; Capsid; CA;
Phosphatidylinositol 4-kinases: Function, structure, and inhibition
Keywords: بازدارنده; Phosphatidylinositol 4-kinase; Inhibitor; Crystal structure; Virus
Les inhibiteurs du goût sucré : perspectives thérapeutiques
Keywords: بازدارنده; Goût; Récepteur; Ãdulcorant; Inhibiteur; Obésité; Diabète; Taste; Receptor; Sweetener; Inhibitor; Obesity; Diabetes;
A potent and selective 11β-hydroxysteroid dehydrogenase type 1 inhibitor, SKI2852, ameliorates metabolic syndrome in diabetic mice models
Keywords: بازدارنده; 11β-hydroxysteroid dehydrogenase type 1; Inhibitor; Type 2 diabetes; Glucocorticoid; Gluconeogenesis; Insulin resistance
Novel fatty acid binding protein 4 (FABP4) inhibitors: Virtual screening, synthesis and crystal structure determination
Keywords: بازدارنده; FABP4; Inhibitor; Diabetes; Virtual screening; Crystal structure
Synthesis and in-vitro evaluation of 2-amino-4-arylthiazole as inhibitor of 3D polymerase against foot-and-mouth disease (FMD)
Keywords: بازدارنده; Foot-and-mouth disease virus (FMDV); Antiviral; Inhibitor; 3D polymerase (3Dpol); 2-Amino-4-arylthiazole
Development of fluorescent peptide substrates and assays for the key autophagy-initiating cysteine protease enzyme, ATG4B
Keywords: بازدارنده; VWBVATUTVWMVIR-LJAQVGFWSA-N; ATG4B; autophagin 1; FRET; fluorescence resonance energy transfer; HTS; high throughput screening; LC3B; microtubule-associated protein 1 A/B light chain 3B; NEM; N-ethylmaleimide; LC-MS; liquid chromatography coupled mass s
Discovery of 4-(dihydropyridinon-3-yl)amino-5-methylthieno[2,3-d]pyrimidine derivatives as potent Mnk inhibitors: synthesis, structure-activity relationship analysis and biological evaluation
Keywords: بازدارنده; eIF4E; Mnk; Inhibitor; Structure-activity relationship; Thieno[2,3-d]pyrimidine derivatives;
Identification of 6-benzyloxysalicylates as a novel class of inhibitors of 15-lipoxygenase-1
Keywords: بازدارنده; Lipoxygenase; Expression; Inhibitor; Enzyme kinetics; Salicylate; QZMBYVCXVKIUFL-UHFFFAOYSA-N; CNMBMLGUWXDQDM-UHFFFAOYSA-N; RHUIESSPNHQDMS-UHFFFAOYSA-M; JKVJFXHBGZSZIR-GMUIIQOCSA-M; WLNHIKPHHAWGLS-UHFFFAOYSA-N; ZXAHUQRHXLVQED-UHFFFAOYSA-N; JKVJFXHBGZSZIR-
Discovery of novel spiro 1,3,4-thiadiazolines as potent, orally bioavailable and brain penetrant KSP inhibitors
Keywords: بازدارنده; Kinesin spindle protein; Inhibitor; Anti-proliferation; Spirocycles; 1,3,4-Thiadiazolines;
Discovery of novel N-(5-(tert-butyl)isoxazol-3-yl)-Nâ²-phenylurea analogs as potent FLT3 inhibitors and evaluation of their activity against acute myeloid leukemia in vitro and in vivo
Keywords: بازدارنده; FMS-like tyrosine kinase 3 (FLT3); Inhibitor; Acute myeloid leukemia; N-(5-(tert-Butyl)isoxazol-3-yl)-Nâ²-phenylurea;
Structure-activity studies in the development of a hydrazone based inhibitor of adipose-triglyceride lipase (ATGL)
Keywords: بازدارنده; Adipose triglyceride lipase; Hydrazones; Inhibitor; Lipid metabolism; Triglycerides;
Quantum chemical and experimental investigations on inhibitory behavior of amino–imino tautomeric equilibrium of 2-aminobenzothiazole on steel corrosion in H2SO4 solution
Keywords: بازدارنده; Aminobenzothiazole; Inhibitor; Quantum; QSAR; Langmuir
Design, synthesis and biological evaluation of novel 4-alkynyl-quinoline derivatives as PI3K/mTOR dual inhibitors
Keywords: بازدارنده; PI3K; mTOR; Cancer; Inhibitor; 4-Alkynyl-quinoline
Discovery and SAR study of c-Met kinase inhibitors bearing an 3-amino-benzo[d]isoxazole or 3-aminoindazole scaffold
Keywords: بازدارنده; c-Met kinase; Inhibitor; 3-Amino-benzo[d]isoxazole; 3-Aminoindazole; Non-small cell lung cancer
Fused-ring structure of decahydroisoquinolin as a novel scaffold for SARS 3CL protease inhibitors
Keywords: بازدارنده; SARS 3CL protease; Inhibitor; Decahydroisoquinolin; Hydrophobic interaction;
1,3-Disubstituted and 1,3,3-trisubstituted adamantyl-ureas with isoxazole as soluble epoxide hydrolase inhibitors
Keywords: بازدارنده; Soluble epoxide hydrolase; Inhibitor; Adamantane; Isocyanate; Urea; Isoxazole;
Associate editor: B. TeicherEpigenetic targets and drug discovery Part 2: Histone demethylation and DNA methylation
Keywords: بازدارنده; Histone demethylation; DNA methylation; Inhibitor; Chemical probe; Drug discovery; LSD; lysine-specific histone demethylase; HDAC; histone deacetylase; REST; REST corepressor; DNMT; DNA methyltransferase; MAO; monoamine oxidase; AML; acute myeloid leukemi
Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action
Keywords: بازدارنده; Carbonic anhydrase; Inhibitor; Sulfocoumarin; Tumor-associated enzyme;
Discovery of substituted 1,4-dihydroquinolines as novel class of ABCB1 modulators
Keywords: بازدارنده; Drug discovery; Structure-activity data; Multidrug resistance (MDR); Inhibitor; Efflux pump inhibition;
Synthesis and biological evaluation of 6-substituted indolizinoquinolinediones as catalytic DNA topoisomerase I inhibitors
Keywords: بازدارنده; Indolizinoquinolinedione; DNA topoisomerase; Inhibitor; Anticancer;
Design, synthesis and preliminary bioactivity evaluations of substituted quinoline hydroxamic acid derivatives as novel histone deacetylase (HDAC) inhibitors
Keywords: بازدارنده; Quinoline; Hydroxamic acid; HDAC; Inhibitor; Anti-proliferative;
Resveratrol compounds inhibit human holocarboxylase synthetase and cause a lean phenotype in Drosophila melanogaster
Keywords: بازدارنده; Grapes; Fat mass; Drosophila; Holocarboxylase synthetase; Inhibitor; Resveratrol compounds;
Pyrrolo[2,3-b]pyridine derivatives as potent Bruton's tyrosine kinase inhibitors
Keywords: بازدارنده; BTK kinase; Inhibitor; Pyrrolo[2,3-b]pyridine; SAR;
Evaluation of transition-state mimics in a superior BACE1 cleavage sequence as peptide-mimetic BACE1 inhibitors
Keywords: بازدارنده; BACE 1; Inhibitor; Transition state mimic; Hydroxyethylamine; Hydroxymethylcarbonyl;
New insights into the effect of polyvinylpyrrolidone (PVP) concentration on methane hydrate growth. 1. Growth rate
Keywords: بازدارنده; Clathrate; Methane; Kinetics; Inhibitor; Polyvinylpyrrolidone; Growth;
Development of ssDNA aptamers as potent inhibitors of Mycobacterium tuberculosis acetohydroxyacid synthase
Keywords: بازدارنده; Acetohydroxyacid synthase; Tuberculosis; SELEX; DNA aptamer; Inhibitor;
Identification of novel SIRT2-selective inhibitors using a click chemistry approach
Keywords: بازدارنده; Sirtuin; Histone deacetylase; Inhibitor; Isozyme selectivity
Discovery of hybrid Hsp90 inhibitors and their anti-neoplastic effects against gefitinib-resistant non-small cell lung cancer (NSCLC)
Keywords: بازدارنده; Hsp90; Lung cancer; Gefitinib resistance; Inhibitor; Rational design;
UK-1 and structural analogs are potent inhibitors of hepatitis C virus replication
Keywords: بازدارنده; Hepatitis C; NS3; Helicase; Inhibitor;