Keywords: گیرنده mGlu5; Cross-species translation; Drug discovery; Major depressive disorder; mGlu5 receptor; Negative allosteric modulator; Substance use disorder;
مقالات ISI گیرنده mGlu5 (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: گیرنده mGlu5; mGlu5 receptor; Cocaine; Learning; Extinction; Reinforcement; Mice
ADX-47273, a mGlu5 receptor positive allosteric modulator, attenuates deficits in cognitive flexibility induced by withdrawal from 'binge-like' ethanol exposure in rats
Keywords: گیرنده mGlu5; Ethanol; Barnes maze; Reversal learning; mGlu5 receptor; NMDA receptor;
Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators
Keywords: گیرنده mGlu5; mGlu5 receptor; Negative allosteric modulator; 4-amino-3-arylsulfonyl-quinolines; Parallel synthesis; Optimization;
DSR-98776, a novel selective mGlu5 receptor negative allosteric modulator with potent antidepressant and antimanic activity
Keywords: گیرنده mGlu5; mGlu5 receptor; Major depressive disorder; Mania; Bipolar disorder; Negative allosteric modulator
Implication of mGlu5 receptor in the enhancement of morphine-induced hyperlocomotion under chronic treatment with zolpidem
Keywords: گیرنده mGlu5; mGlu5 receptor; GABAA receptor; Nucleus accumbens; Morphine; Zolpidem; Drug dependence;
Chronic Metabotropic Glutamate Receptor 5 Inhibition Corrects Local Alterations of Brain Activity and Improves Cognitive Performance in Fragile X Mice
Keywords: گیرنده mGlu5; Amygdala; CTEP; Fmr1 KO mice; fMRI; fragile x syndrome (FXS); mGlu5 receptor
Discovery of (1R,2R)-N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide, a potent and orally efficacious mGlu5 receptor negative allosteric modulator
Keywords: گیرنده mGlu5; mGlu5 receptor; Negative allosteric modulator; Receptor occupancy; Formalin model; Rotorod test;
The mGlu5 positive allosteric modulator LSN2463359 differentially modulates motor, instrumental and cognitive effects of NMDA receptor antagonists in the rat
Keywords: گیرنده mGlu5; mGlu5 receptor; Potentiator; Glutamate; NMDA receptor antagonist; Schizophrenia; Psychosis; Behaviour; Reversal learning; ADX47273; [S-(4-fluoro-phenyl)-{3-[3-(4-fluoro-phenyl)-[1,2,4]-oxadiazol-5-yl]-piperidin-1-yl}-methanone]; ANCOVA; analysis of covari
Potentiation of mGlu5 receptors with the novel enhancer, VU0360172, reduces spontaneous absence seizures in WAG/Rij rats
Keywords: گیرنده mGlu5; Absence epilepsy; WAG/Rij rats; mGlu5 receptor; VU0360172; MTEP;
MPEP, an mGlu5 receptor antagonist, reduces the development of l-DOPA-induced motor complications in de novo parkinsonian monkeys: Biochemical correlates
Keywords: گیرنده mGlu5; mGlu5 receptor; Dyskinesia; l-DOPA; MPTP-lesioned monkey; MPEP;
mGlu2/3 and mGlu5 receptors: Potential targets for novel antidepressants
Keywords: گیرنده mGlu5; mGlu2/3 receptor; mGlu5 receptor; Depression; Ketamine;
In vitro characterisation of the novel positive allosteric modulators of the mGlu5 receptor, LSN2463359 and LSN2814617, and their effects on sleep architecture and operant responding in the rat
Keywords: گیرنده mGlu5; mGlu5 receptor; Glutamate; NMDA receptor antagonist; Schizophrenia; Psychosis; ADX47273; [S-(4-fluorophenyl)-{3-[3-(4-fluorophenyl)-[1,2,4]-oxadiazol-5-yl]-piperidin-1-yl}-methanone]; ANCOVA; analysis of covariance; ANOVA; analysis of variance; CDPPB; 3-C
Is the mGlu5 receptor a possible target for new antidepressant drugs?
Keywords: گیرنده mGlu5; antidepressant drugs; ketamine; mGlu5 receptor; MTEP; MPEP; NMDA receptor
Analgesic Effect of a Single Preoperative Dose of the Antibiotic Ceftriaxone in Humans
Keywords: گیرنده mGlu5; Ceftriaxone; analgesia; GLT-1; mGlu5 receptor; postsurgical pain; inflammatory pain
Involvement of mGlu5 and NMDA receptors in the antidepressant-like effect of acamprosate in the tail suspension test
Keywords: گیرنده mGlu5; CDPPB; 3-Cyano-N-(1,3-diphenyl-1H-pyrazol-5-yl) benzamide; NMDA; N-Methyl-d-aspartic acid; Acamprosate; CDPPB; mGlu5 receptor; NMDA; Tail suspension test;
Differential effects of the mGluR5 positive allosteric modulator CDPPB in the cortex and striatum following repeated administration
Keywords: گیرنده mGlu5; mGlu5 receptor; CDPPB; Receptor binding; NMDA receptor subunit phosphorylation; Antipsychotic activity; Sleep;
A model for Ca2+ oscillations stimulated by the type 5 metabotropic glutamate receptor: An unusual mechanism based on repetitive, reversible phosphorylation of the receptor
Keywords: گیرنده mGlu5; Computational model; mGlu5 receptor; Dynamic uncoupling; Protein kinase C; Protein phosphatase; Receptor phosphorylation
Differential effect of the mGlu5 receptor positive allosteric modulator ADX-47273 on early and late hippocampal LTP
Keywords: گیرنده mGlu5; LTP; NMDA; VDCC; mGlu5 receptor; CA1; ADX-47273
Functional interaction of metabotropic glutamate receptor 5 and NMDA-receptor by a metabotropic glutamate receptor 5 positive allosteric modulator
Keywords: گیرنده mGlu5; NMDA(N-methyl-D-aspartate)-receptor; mGlu5 receptor; Metabotropic glutamate receptor 5; Positive allosteric modulator; ADX-47273; Long-term potentiation
Distinct roles of group I mGlu receptors in striatal function
Keywords: گیرنده mGlu5; MGlu1 receptor; MGlu5 receptor; Striatal neurons; Synaptic plasticity; Endocannabinoids; Neostriatum; Interneuron
Face-washing behavior induced by the group I metabotropic glutamate receptor agonist (S)-3,5-DHPG in mice is mediated by mGlu1 receptor
Keywords: گیرنده mGlu5; mGlu1 receptor; mGlu5 receptor; mGlu2/3 receptor; DHPG; Face-washing behavior; Convulsion
Research reportMGlu5 antagonism impairs exploration and memory of spatial and non-spatial stimuli in rats
Keywords: گیرنده mGlu5; mGlu5 receptor; Antagonist; MPEP; Rat; Exploration; Maze learning; Object recognition; Prelimbic cortex;
Synthesis and SAR comparison of regioisomeric aryl naphthyridines as potent mGlu5 receptor antagonists
Keywords: گیرنده mGlu5; mGlu5 receptor; Antagonist; 1,5-Naphthyridine; 1,6-Naphthyridine; 1,8-Naphthyridine; Rat; Osteoarthritis; Pain
mGlu5 receptor and protein kinase C implicated in the development and induction of neuropathic pain following chronic ethanol consumption
Keywords: گیرنده mGlu5; Alcoholic neuropathy; Ethanol; mGlu5 receptor; PKC; Glutamate
Antiaggressive effects of MPEP, a selective antagonist of mGlu5 receptors, in agonistic interactions between male mice
Keywords: گیرنده mGlu5; Aggression; Metabotropic glutamate receptor; mGlu5 receptor; (Mice)
Changes in mGlu5 receptor expression in the basal ganglia of reserpinised rats
Keywords: گیرنده mGlu5; mGlu5 receptor; ‘in situ’ hybridisation; mRNA; [3H]MPEP ligand binding; Reserpine; Rat; Parkinson's disease