Keywords: حمل و نقل کاتیونی آلی; ABC; ATP-binding cassette; ASBT; apical sodium-dependent bile acid transporter; Bamet-UD2; cisplatin-ursodeoxycholic acid derivative; CCA; cholangiocarcinoma; DHMEQ; dehydroxymethyl epoxyquinomicin; EGFR; epidermal growth factor receptor; 5-FU; 5-fluorour
مقالات ISI حمل و نقل کاتیونی آلی (ترجمه نشده)
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Keywords: حمل و نقل کاتیونی آلی; ABC; ATP-binding cassette; AHUI; aqueous humor uptake index; AUC; area under the curve; BAB; blood-aqueous barrier; BBB; blood-brain barrier; BCRP; breast cancer resistance protein; BRB; blood-retinal barrier; BUI; brain uptake index; MATE1; multidrug and
Keywords: حمل و نقل کاتیونی آلی; ARV; antiretroviral; CHO; Chinese Hamster Ovary; CID; collision-induced dissociation; DMEM/F12; Dulbecco's Modified Eagle's Medium: Ham's F12 Medium; DMF; dimethylformamide; DMSO; dimethylsulfoxide; GGT; γ-glutamyltransferase; HIV; human immunodefi
Keywords: حمل و نقل کاتیونی آلی; cilostazol; hepatic transport; OATP 1B1/1B3; biliary excretion; efflux transporter; AP; apical; BL; basolateral; DMEM; Dulbecco's modified Eagle's medium; EGCG; (-)-epigallocatechin gallate; HEK293 cells; human embryonic kidney cells; MDCKII cells; Madi
Keywords: حمل و نقل کاتیونی آلی; basic drug; blood-brain barrier; organic cation transporter; varenicline;
Keywords: حمل و نقل کاتیونی آلی; organic cation transporters (OCTs); renal clearance; hepatic transport; hepatocytes; elderly; AUC; area under the curve; CKD; chronic kidney disease; CVD; cardiovascular disease; FMO3; flavin-containing monooxigenase 3; HEK; human embryonic kidney; HK; h
Keywords: حمل و نقل کاتیونی آلی; absorption; computational ADME; efflux pumps; in vitro models; organic cation transporters; P-glycoprotein; peptide transporters; pulmonary delivery/absorption; ABC transporters; organic anion-transporting polypeptide transporters; BAL; bronchoalveolar l
Keywords: حمل و نقل کاتیونی آلی; in silico modeling; QSAR; transporters; computational ADME; high-throughput technologies; AUC; area under the curve; BCRP; breast cancer resistance protein; DDI; drug-drug interaction; fup; protein unbound fraction in plasma; ITC; International Transpor
Keywords: حمل و نقل کاتیونی آلی; Intracellular drug concentration; Pharmacodynamics; OCT; MATE; PMAT; Drug transporter; ABC; ATP-binding cassette; ACC; acetyl-CoA carboxylase; AMP; adenosine monophosphate; AMPK; AMP-activated protein kinase; AUC; area under the concentration time curve;
Keywords: حمل و نقل کاتیونی آلی; intestinal absorption; intestinal epithelia; transporters; organic cation transporter; drug transport; metformin;
Keywords: حمل و نقل کاتیونی آلی; 3Rs; reduce, refine, replace; A; apical; ABC; ATP-binding cassette; B; basal; BCF; bioconcentration factor; BTA; bi-directional transport assay; CETA; concentration equilibrated transport assay; Ci; Curie; Dpm; disintegrations per minute; Kow; octanol-w
Keywords: حمل و نقل کاتیونی آلی; 3D; three-dimensional; c log P; the calculated log octanol/water partition coefficient; DNA; deoxyribonucleic acid; ATP; adenosine triphosphate; HPT1; intestinal peptide-associated transporter 1; PEPT1; peptide transporter 1; OCT; organic cation transpo
Keywords: حمل و نقل کاتیونی آلی; Steviol glucuronide; OAT3; Uptake transport; Food-drug interaction; BCRP; breast cancer resistant protein; MATE; multidrug and toxin extrusion protein; MRP; multidrug resistant protein; OAT; organic anion transporter; OATP; organic anion transport protein
Keywords: حمل و نقل کاتیونی آلی; hOCT, human organic cation transporter; MDCK, Madin-Daby canine kidney; 5-HT, serotonin; NE, norepinephrine; MPP+, 1-methyl-4- phenylpyridinium; LC-MS/MS, liquid chromatography-tandem mass spectrometryAntidepressant; Berberine; Organic cation transporter
Keywords: حمل و نقل کاتیونی آلی; active transport; blood-brain barrier; drug transport; in vitro models; membrane transporter; microdialysis; organic cation transporter; tramadol;
Keywords: حمل و نقل کاتیونی آلی; APC; apparent partition coefficient; BCRP; breast cancer resistance protein; CH; cholate; cLPM; canalicular liver plasma membrane; DC; deoxycholate; GC; glycocholate; GDC; glycodeoxycholate; HNAP; hydroxy-2-naphthoic acid; Mw; molecular weight; MATE; mult
Inhibition of organic cation transporter (OCT) activities by carcinogenic heterocyclic aromatic amines
Keywords: حمل و نقل کاتیونی آلی; Drug transporter; Toxicokinetics; Organic cation transporter; Heterocyclic amines; Toxicity;
Herb-drug interaction of Nisha Amalaki and Curcuminoids with metformin in normal and diabetic condition: A disease system approach
Keywords: حمل و نقل کاتیونی آلی; NA; Nisha Amalaki; CE; Curcuminoids; MET; metformin; DDI; drug-drug interactions; HDI; herb-drug interactions; CYPs; cytochrome p450 isoenzymes; IS; internal standard; MWR; Male Wistar rats; STZ; streptozotocin; MNC; mononuclear cells; OCT; organic cation
Significance of A-to-I RNA editing of transcripts modulating pharmacokinetics and pharmacodynamics
Keywords: حمل و نقل کاتیونی آلی; ABC; ATP-binding cassette transporter; ADAR; adenosine deaminase acting on RNA; ADH; alcohol dehydrogenase; AhR; aryl hydrocarbon receptor; AKR; aldo-keto reductase; ALS; amyotrophic lateral sclerosis; AZIN1; antizyme inhibitor 1; AMPA; α-amino-3-hydroxy
Organic solute carrier 22 (SLC22) family: Potential for interactions with food, herbal/dietary supplements, endogenous compounds, and drugs
Keywords: حمل و نقل کاتیونی آلی; Hepatic transport; Nephrotoxicity; Organic anion transporter; Organic cation transporter; Renal transport;
Losartan prevents the imbalance between renal dopaminergic and renin angiotensin systems induced by fructose overload. l-Dopa/dopamine index as new potential biomarker of renal dysfunction
Keywords: حمل و نقل کاتیونی آلی; Ang II; angiotensin II; AT1R; angiotensin II type 1 receptor; CrCl; creatinine clearance; D1R; dopamine sub-type 1 receptor; DA; dopamine; FENa; fractional sodium excretion; FO; fructose overload; GFR; glomerular filtration rate; IR; Insulin resistance; N
Purification and reconstitution of polyspecific H+/organic cation antiporter human MATE1
Keywords: حمل و نقل کاتیونی آلی; MATE; multidrug and toxin extrusion; hMATE1; human MATE1; TEA; tetraethyl ammonium; PQ; paraquat; OC; organic cation; DDTM; n-dodecyl-β-d-thiomaltopyranoside; TM; transmembrane helix; Multidrug and toxic compound extrusion; Organic cation transporter; Pu
Aryl hydrocarbon receptor (AhR) mediated short-term effects of 2,3,7,8-tetrachlorodibenzo-p-dioxin (TCDD) on bile acid homeostasis in mice
Keywords: حمل و نقل کاتیونی آلی; Aryl hydrocarbon receptor; TCDD; Bile acids; Biliary excretion; Taurodeoxycholic acid; Cyp8b1; 1°BAs; Primary bile acids; 2°BAs; Secondary bile acids; 6-OH; 6-hydroxylated (6-OH); 12-OH; 12α-hydroxylated; Abc; ATP-binding cassette; AhR; Aryl hydrocarbo
Imaging techniques to study drug transporter function in vivo
Keywords: حمل و نقل کاتیونی آلی; ABC; ATP-binding cassette; AD; Alzheimer's disease; ADME; absorption, distribution, metabolism and elimination; ATP; adenosine triphosphate; AUC; area under the curve; BBB; blood-brain barrier; BCRP; breast cancer resistance protein; BPND; non-displaceabl
The Polymorphic Variants rs3088442 and rs2292334 in the Organic Cation Transporter 3 (OCT3) Gene and Susceptibility Against Type 2 Diabetes: Role of their Interaction
Keywords: حمل و نقل کاتیونی آلی; Organic cation transporter; OCT3; rs3088442G>A; rs2292334G>A; type 2 diabetes;
Intestinal Drug Interactions Mediated by OATPs: A Systematic Review of Preclinical and Clinical Findings
Keywords: حمل و نقل کاتیونی آلی; drug interaction; inhibition; transporter; organic anion-transporting polypeptide transporters; intestinal absorption; polymorphism; AUC; area under the plasma concentration-time curve; DDIs; drug-drug interactions; EMA; European Medicines Agency; FDA
Expanding the repertoire of L-DOPA's actions: A comprehensive review of its functional neurochemistry
Keywords: حمل و نقل کاتیونی آلی; AADC; aromatic L amino acid decarboxylase; COMT; catechol-O-methyl-transferase; CSF; cerebrospinal fluid; 6-OHDA; 6-hydroxydopamine; DBH; dopamine β-hydroxylase; DOPAC; 3,4-dihydroxyphenylacetic acid; 3-MT; 3-methoxytyramine; DA; dopamine; DAT; dopamine
Different Involvement of OAT in Renal Disposition of Oral Anticoagulants Rivaroxaban, Dabigatran, and Apixaban
Keywords: حمل و نقل کاتیونی آلی; drug interactions; solute transporters; organic anion transporters (OAT); pharmacokinetics/pharmacodynamics; renal transport; BCRP; breast cancer resistance protein; CCK8; cholecystokinin-8; E217βG; estradiol 17β-D-glucuronide; E-sul; estrone 3-sulfate;
Involvement of organic cation transporter 3 (Oct3/Slc22a3) in the bioavailability and pharmacokinetics of antidiabetic metformin in mice
Keywords: حمل و نقل کاتیونی آلی; Metformin; OCT3; Transporter; Intestinal absorption; Bioavailability; Mouse; AUC; area under the plasma concentration-time curve; CL; clearance; Cmax; maximum concentration; OCT/Oct; organic cation transporter; SLC; solute carrier; tmax; time to maximum
Localization of organic cation transporter 2 (OCT2) in monoaminergic and cholinergic axon terminals of the mouse brain
Keywords: حمل و نقل کاتیونی آلی; Organic cation transporter; Neurotransmitter transporter; Monoamine; Acetylcholine; Neurotransmitter reuptake;
Prostaglandin transporter (OATP2A1/SLCO2A1) contributes to local disposition of eicosapentaenoic acid-derived PGE3
Keywords: حمل و نقل کاتیونی آلی; NSAIDs; non-steroidal anti-inflammatory drugs; EPA-E; eicosapentaenoic acid ethyl ester; AA; arachidonic acid; PGE2; prostaglandin E2; PGE3; prostaglandin E3; EP; PGE receptor; OATP; organic anion transporting polypeptide; OAT; organic anion transporter;
Dual role of LRRC8A-containing transporters on cisplatin resistance in human ovarian cancer cells
Keywords: حمل و نقل کاتیونی آلی; A2780WT; drug-sensitive human ovarian cancer cells; A2780CisR; cisplatin resistant A2780 cells; ABC; ATP-binding cassette; Ano6; Anoctamin 6; Apaf-1; apoptotic protease activating factor 1; Atox1; Antioxidant 1 copper chaperone; AP; alkaline phosphatase;
Immuno-detection of OCTN1 (SLC22A4) in HeLa cells and characterization of transport function
Keywords: حمل و نقل کاتیونی آلی; TEA; tetraethylammonium; PLP; pyridoxal 5-phosphate; MTSEA; 2-aminoethyl methanethiosulfonate; VAChT; vesicular acetylcholine transporter; OCT; organic cation transporter; OCTN; organic cation transporter novel; ChT; choline transporter; Transporters; Pro
The variant organic cation transporter 2 (OCT2)-T201M contribute to changes in insulin resistance in patients with type 2 diabetes treated with metformin
Keywords: حمل و نقل کاتیونی آلی; HOMA-BCF; HOMA-IR; Metformin; OCT2-T201M; Organic cation transporter; Type 2 diabetes;
Short term uptake and transport process for metformin in roots of Phragmites australis and Typha latifolia
Keywords: حمل و نقل کاتیونی آلی; Pharmaceuticals; Root; Pitman chamber; Inhibitor; Organic cation transporter;
The involvement of selected membrane transport mechanisms in the cellular uptake of 177Lu-labeled bombesin, somatostatin and gastrin analogues
Keywords: حمل و نقل کاتیونی آلی; Megalin; Nephrotoxicity; Organic anion transporter; Organic cation transporter; Fluid phase endocytosis; Peptides
Carrier-Mediated Transport of Nicotine Across the Inner Blood–Retinal Barrier: Involvement of a Novel Organic Cation Transporter Driven by an Outward H+ Gradient
Keywords: حمل و نقل کاتیونی آلی; blood–retinal barrier; nicotine; organic cation transporter; membrane transport; transporters; membrane transporter; drug transport; in vitro models; TR-iBRB2 cells
Evidence for organic cation transporter-mediated metformin transport and 5â²-adenosine monophosphate-activated protein kinase activation in rat skeletal muscles
Keywords: حمل و نقل کاتیونی آلی; MET; metformin; AMPK; 5â²-adenosine monophosphate-activated protein kinase; OCT; organic cation transporter; PCr; phosphocreatine, T2DM, type 2 diabetes mellitus; KRB; Krebs-Ringer bicarbonate buffer; DNP; 2,4-dinitrophenol; AICAR; 5-aminoimidazole-4-c
Role of organic cation transporters (OCTs) in the brain
Keywords: حمل و نقل کاتیونی آلی; Organic cation transporter; Monoamines; Clearance; Anxiety; Stress; Antidepressants5-HT, serotonin; D22, decynium22; DA, dopamine; DAT, dopamine transporter; FST, forced-swim test; NE, norepinephrine; NET, norepinephrine transporter; OCT, organic cation t
Functional characterization of the organic cation transporters (OCTs) in human airway pulmonary epithelial cells
Keywords: حمل و نقل کاتیونی آلی; ALI; air-liquid interface culture; EBSS; Earle's Balanced Salt Solution; MPP+; 1-methyl-4-phenylpyridinium; OCT; organic cation transporter; PBS; phosphate-buffered saline solution; PGE2; prostaglandine E2; TEER; transepithelial electrical resistance; P
Expression of xenobiotic transporters in the human renal proximal tubule cell line RPTEC/TERT1
Keywords: حمل و نقل کاتیونی آلی; 4-Di-1-ASP; 4-(4-(Dimethylamino)styryl)-N-Methylpyridinium Iodide; CsA; Cyclosporine A; primary hPT; human primary proximal tubule cells; MATE; multidrug and toxin extrusion proteins; OAT; organic anion transporter; OATP; organic anion polypeptide transpo
Quantitative in vitro to in vivo extrapolation of tissues toxicity
Keywords: حمل و نقل کاتیونی آلی; ADME; absorption, distribution, metabolism, and excretion; ARE; antioxidant responses elements; BBB; blood brain barrier; CsA; cyclosporine A; CYP; cytochrome P450; EPA; Environmental Protection Agency; GCL; glutamate cysteine ligase; GCLC; glutamate cyst
In vitro interaction of clopidogrel and its hydrolysate with OCT1, OCT2 and OAT1
Keywords: حمل و نقل کاتیونی آلی; Organic cation transporter; Organic anion transporter; Clopidogrel; Clopidogrel carboxylate; Drug-drug interactions; Inhibition;
Klotho has dual protective effects on cisplatin-induced acute kidney injury
Keywords: حمل و نقل کاتیونی آلی; acute kidney injury; cisplatin; glucuronidase; Klotho; nephrotoxicity; organic cation transporter;
Update on the pharmacology of selective inhibitors of MAO-A and MAO-B: Focus on modulation of CNS monoamine neurotransmitter release
Keywords: حمل و نقل کاتیونی آلی; Enzyme active site structure; Presynaptic inhibition; Exocytotic and non-exocytotic release; Neuroprotection; Parkinson's disease; Affective disorders; MAO; monoamine oxidase; MAO-A; monoamine oxidase isoform A; MAO-B; monoamine oxidase isoform B; COMT; c
Functional expression of choline transporter-like protein 1 (CTL1) in small cell lung carcinoma cells: A target molecule for lung cancer therapy
Keywords: حمل و نقل کاتیونی آلی; ACh; acetylcholine; AChE; acetylcholinesterase; BuChE; butyrylcholinesterase; ChAT; choline acetyltransferase; CHT1; high-affinity choline transporter 1; CTL1; choline transporter-like protein 1; 4-DAMP; 4-diphenylacetoxy-N-methylpiperidine methiodide; D-
Precise comparison of protein localization among OCT, OAT, and MATE in human kidney
Keywords: حمل و نقل کاتیونی آلی; active transport; renal excretion; membrane transporter; drug transport; organic anion transporter; organic cation transporter; elimination; renal clearance; multidrug and toxin extrusion
Organic cation transporter 2 (SLC22A2), a low-affinity and high-capacity choline transporter, is preferentially enriched on synaptic vesicles in cholinergic neurons
Keywords: حمل و نقل کاتیونی آلی; Ach; acetylcholine; AchR; acetyl choline receptors; BTX; alpha-bungarotoxin; CA; central autonomic cells; CC; central canal; ChAT; choline acetyltransferase; CNS; central nervous system; Co; cortex; DAB; 3,3â²-diaminobenzidine; DMEM; Dulbecco's modifie
Involvement of Carnitine/Organic Cation Transporter OCTN1/SLC22A4 in Gastrointestinal Absorption of Metformin
Keywords: حمل و نقل کاتیونی آلی; oral absorption; organic cation transporter; pharmacokinetics; ADME; drug transport; renal excretion
Propranolol Transport Across the Inner Blood–Retinal Barrier: Potential Involvement of a Novel Organic Cation Transporter
Keywords: حمل و نقل کاتیونی آلی; inner blood–retinal barrier; propranolol; organic cation transporter; diabetic retinopathy; glaucoma; membrane transport; drug transport; in vitro models; TR-iBRB2 cells; blood-brain barrier