Keywords: پنتامیدین; Arrhythmia; Pentamidine; PA-6; Effective refractory period; Inward rectifier; Diastolic variance; Andersen syndrome;
مقالات ISI پنتامیدین (ترجمه نشده)
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Keywords: پنتامیدین; Pentamidine; Accuracy profiles; μSPE; UPLC; Benzamidines
Keywords: پنتامیدین; Aquaporin; Water; Glycerol; Antimonials; Pentamidine; Parasite;
Keywords: پنتامیدین; Pyrimidine; Chalcone; Pentamidine; Anti-leishmanial activity; Anti-malarial activity;
High-potency block of Kir4.1 channels by pentamidine: Molecular basis
Keywords: پنتامیدین; Kir4.1; Pentamidine; PA-6; Molecular modeling; Mutagenesis;
Full length articlePentamidine antagonizes the benznidazole's effect in vitro, and lacks of synergy in vivo: Implications about the polyamine transport as an anti-Trypanosoma cruzi target
Keywords: پنتامیدین; Trypanosoma cruzi; Chagas disease; Pentamidine; Benznidazole; Polyamine transport;
Safety pharmacology studies using EFP and impedance
Keywords: پنتامیدین; CardioExcyte 96; Dofetilide; E4031; EAD-like; Extracellular field potential; Impedance; Isoproterenol; Nifedipine; Pentamidine; Safety pharmacology;
Zoonotic trypanosomes in South East Asia: Attempts to control Trypanosoma lewisi using human and animal trypanocidal drugs
Keywords: پنتامیدین; Trypanosoma lewisi; Trypanocidals; Fexinidazole; Trypanosoma evansi; Efficacy; Rats; Suramin; Pentamidine; Eflornitine; Nifurtimox; Benznidazole;
Chimerization at the AQP2–AQP3 locus is the genetic basis of melarsoprol–pentamidine cross-resistance in clinical Trypanosoma brucei gambiense isolates
Keywords: پنتامیدین; Human African trypanosomiasis; Sleeping sickness; Trypanosoma brucei gambiense; Drug resistance; Melarsoprol; Pentamidine; Aquaporin; Reverse genetics
Pentamidine analogs as inhibitors of [3H]MK-801 and [3H]ifenprodil binding to rat brain NMDA receptors
Keywords: پنتامیدین; Pentamidine; NMDA receptor; Ifenprodil; Polyamine; Bisbenzamidine; Alkylation; Coupling; Radioligand binding; Rat brain; Molecular docking;
Pentamidine exerts in vitro and in vivo anti Trypanosoma cruzi activity and inhibits the polyamine transport in Trypanosoma cruzi
Keywords: پنتامیدین; Trypanosoma cruzi; Chagas' disease; Polyamine transport; Pentamidine;
In vivo SPECT imaging of [123I]-labeled pentamidine pro-drugs for the treatment of human African trypanosomiasis, pharmacokinetics, and bioavailability studies in rats
Keywords: پنتامیدین; Pentamidine; Pro-drug; SPECT-imaging; Bioavailibility;
Synthesis of 2-methoxybenzoylhydrazone and evaluation of their antileishmanial activity
Keywords: پنتامیدین; 2-Methoxybenzoylhydrazone; Antileishmanial activity; Pentamidine; Leishmania promestigotes
In situ potentiometric method to evaluate bacterial outer membrane-permeabilizing ability of drugs: Example using antiprotozoal diamidines
Keywords: پنتامیدین; K+-selective electrode; Tyrocidine A; Bacterial outer membrane permeabilizer; Diminazene; Pentamidine; DAPI;
Pentamidine sensitizes chronic myelogenous leukemia K562 cells to TRAIL-induced apoptosis
Keywords: پنتامیدین; Pentamidine; TRAIL; Leukemia; Apoptosis;
Effect of cimetidine on pentamidine induced hyperglycemia in rats
Keywords: پنتامیدین; Pentamidine; Cimetidine; Hyperglycemia; Organic cation transporter; Drug interaction; Rat;
Enquête sur l'utilisation des nébulisations de pentamidine en pédiatrie
Keywords: پنتامیدین; Pentamidine; Aérosolthérapie; Nébuliseur; Prophylaxie; Pneumocystose; Enfant; Pentamidine; Aerosol therapy; Nebulizer; Prophylaxis; Pneumocystis; Children;
Pharmaceutical nanotechnologyInsights into the multi-equilibrium, superstructure system based on β-cyclodextrin and a highly water soluble guest
Keywords: پنتامیدین; Supramolecular complex; β-cyclodextrin; Pentamidine; Multi-equilibrium; Leishmaniasis; In vivo experiments;
Comparative modeling of HGPRT enzyme of L. donovani and binding affinities of different analogs of GMP
Keywords: پنتامیدین; HGPRT; hypoxanthine-guanine phosphoribosyl transferase; HPRT; hypoxanthine phosphoribosyltransferase; CL; cutaneous leishmaniasis; MCL; muco-cutaneous leishmaniasis; VL; visceral leishmaniasis; PKDL; post-kala-azar dermal leishmaniasis; BLAST; basic local
Fatal bilateral pneumothoraces following administration of aerosolised pentamidine
Keywords: پنتامیدین; Pentamidine; Adverse effects; Pneumothorax; Human immunodeficiency virus; Autopsy
Synthesis and biological evaluation of l-valine-amidoximeesters as double prodrugs of amidines
Keywords: پنتامیدین; Benzamidine; Biotransformation; Pentamidine; Prodrug; Valine;
Inhibition of lysosomal degradation rescues pentamidine-mediated decreases of KIR2.1 ion channel expression but not that of Kv11.1
Keywords: پنتامیدین; Pentamidine; KIR2.1; hERG; Potassium ion channel; Trafficking; Lysosome
Pentamidine reduces expression of hypoxia-inducible factor-1α in DU145 and MDA-MB-231 cancer cells
Keywords: پنتامیدین; Hypoxia-inducible factor-1α; Pentamidine; Protein translation
Three optimized and validated (using accuracy profiles) LC methods for the determination of pentamidine and new analogs in rat plasma
Keywords: پنتامیدین; Pentamidine; Validation; Accuracy profiles; SPE; LC; Benzamidines;
Novel pentamidine derivatives: Synthesis, anti-tumor properties and polynucleotide-binding activities
Keywords: پنتامیدین; Dibenzamidine; 2,5-Furandicarboxamide; Pentamidine; Antitumor evaluation; Polynucleotide binding
Treatment of visceral leishmaniasis with intravenous pentamidine and oral fluconazole in an HIV-positive patient with chronic renal failure — a case report and brief review of the literature
Keywords: پنتامیدین; Visceral leishmaniasis; HIV; Fluconazole; Pentamidine; Miltefosine; Renal failure
Pharmacophore model for pentamidine analogs active against Plasmodium falciparum
Keywords: پنتامیدین; Pharmacophore; GALAHAD; Pentamidine; P. falciparum; Malaria; Molecular modeling
Structural binding evidence of the trypanocidal drugs Berenil® and Pentacarinate® active principles to a serine protease model
Keywords: پنتامیدین; β-Trypsin; Binding; Diminazene; Pentamidine; Protein crystallography; Thermodynamics
Evidence for the presence of R250G mutation at the ATPase domain of topoisomerase II in an arsenite-resistant Leishmania donovani exhibiting a differential drug inhibition profile
Keywords: پنتامیدین; Leishmania donovani; Topoisomerase II; Novobiocin; Pentamidine; Doxorubicin; Actinomycin D
Two novel nucleobase/pentamidine transporters from Trypanosoma brucei
Keywords: پنتامیدین; BF; bloodstream form; PF; procyclic form; TM; transmembrane domain; ENT; equilibrative nucleoside transporter; qRT-PCR; quantitative real time polymerase chain reaction; GFP; green fluorescent protein; 3HA; triple hemagglutinin epitope tag; ORF; open read
Novel bisbenzimidazoles with antileishmanial effectiveness
Keywords: پنتامیدین; Bisbenzamidine; Bisbenzimidazole; Pentamidine; Pneumocystis carinii pneumonia; Human African trypanosomiasis; Leishmaniasis
Characterization of Leishmania (Leishmania) amazonensis promastigotes resistant to pentamidine
Keywords: پنتامیدین; ABC, ATP-binding cassette; DAPI, 4′,6′-diamidino-2-phenylindole; kb, kilobase; Mb, megabase; PATH, potassium antimonyl tartrate trihydrate; PRP1, pentamidine resistance protein 1; Leishmania; Pentamidine; Drug resistance; ABC transporter
Design, synthesis and in vitro antiprotozoal activity of benzimidazole-pentamidine hybrids
Keywords: پنتامیدین; Antiprotozoal; Benzimidazole; Pentamidine; Giardia; Trichomonas; Entamoeba; Bioisosteric replacement
Mucosal leishmaniasis: Current scenario and prospects for treatment
Keywords: پنتامیدین; American tegumentary leishmaniasis; Leishmania; Leishmania (Viannia) braziliensis; Pentavalent antimonial; Amphotericin B; Pentamidine; Mucosal leishmaniasis; Lipid formulations of amphotericin B; Miltefosine
Melarsoprol- and pentamidine-resistant Trypanosoma brucei rhodesiense populations and their cross-resistance
Keywords: پنتامیدین; Resistance; Cross-resistance; Trypanosome; Furamidine; Melarsoprol; Pentamidine; Trypanosoma brucei rhodesiense; TbAT1 gene;
Leishmania panamensis: Comparative inhibition of nuclear DNA topoisomerase II enzymes from promastigotes and human macrophages reveals anti-parasite selectivity of fluoroquinolones, flavonoids and pentamidine
Keywords: پنتامیدین; Leishmania panamensis; DNA topoisomerase II; Enzyme inhibition; Fluoroquinolone; Pentamidine; Flavonoid; Protoberberine; Bis-benzimidazole;
Clinical presentation and treatment outcome of sleeping sickness in Sudanese pre-school children
Keywords: پنتامیدین; African trypanosomiasis; Sleeping sickness; Children; Pentamidine; Melarsoprol; Adverse events
Cutaneous leishmaniasis treatment
Keywords: پنتامیدین; Leishmaniasis, cutaneous; Anti infective agents, topical; Injections, intralesional; Antimony; Pentamidine; Amphotericin B
In vitro activity of dicationic compounds against a North American foxhound isolate of Leishmania infantum
Keywords: پنتامیدین; Leishmania infantum; Aromatic diamidines; In vitro; Antileishmanial activity; Pentamidine
Induction of apoptosis-like cell death by pentamidine and doxorubicin through differential inhibition of topoisomerase II in arsenite-resistant L. donovani
Keywords: پنتامیدین; Leishmania; Arsenite-resistance; Topoisomerase II; Apoptosis; Pentamidine; Doxorubicin
Drugs and drug resistance in African trypanosomiasis
Keywords: پنتامیدین; Sleeping sickness; Trypanosomiasis; Trypanosoma brucei; chemotherapy; Drug resistance; Pentamidine; Melarsoprol; Nifurtimox
Derivatives of pentamidine designed to target the Leishmania lipophosphoglycan
Keywords: پنتامیدین; Boronate drug targeting; Pentamidine; Leishmania;
Sleep structure: a new diagnostic tool for stage determination in sleeping sickness
Keywords: پنتامیدین; Human African trypanosomiasis; Stage determination; Polysomnography; Angola; Melarsoprol; Pentamidine; SOREMP;