Keywords: مهارکننده رنین; Fragment-based drug discovery (FBDD); High-throughput synthetic chemistry; Structure-based drug design (SBDD); Renin inhibitor; Crystal structure;
مقالات ISI مهارکننده رنین (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهارکننده رنین; Renin inhibitor; MM-GB/SA; 3D-QSAR; In silico modeling; MD simulation;
Keywords: مهارکننده رنین; Aliskiren; Renin inhibitor; Formalin; Hot plate test; Post-operative pain; Neuropathic pain;
Discovery of benzimidazole derivatives as orally active renin inhibitors: Optimization of 3,5-disubstituted piperidine to improve pharmacokinetic profile
Keywords: مهارکننده رنین; BA; bioavailability; RAAS; renin-angiotensin-aldosterone system; BP; blood pressure; Ang I; angiotensin I; ACE; Angiotensin-converting enzyme; Ang II; angiotensin II; AT1; Ang II type I receptor; DRI; direct renin inhibitor; TPSA; topological polar surfac
Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors
Keywords: مهارکننده رنین; AcOH; acetic acid; Ang I; angiotensin I; Ang II; angiotensin II; AUC; area under the blood concentration-time curve; C5min; concentration in plasma 5Â min after administration; CLtotal; total clearance; Cmax; maximum concentration in plasma; DIEA; N,N-d
Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhexanamides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor
Keywords: مهارکننده رنین; HR; heart rate; PR; PR interval; QRS; QRS width; QTc; corrected QT interval; Renin inhibitor; Ketopiperazine; Plasma renin activity; Hypertension; Na channel;
Effect of SPP 635, a renin inhibitor, on intraocular pressure in glaucomatous monkey eyes
Keywords: مهارکننده رنین; SPP 635; renin inhibitor; renin-angiotensin system; intraocular pressure; glaucoma monkey;
Chronic Direct Renin Inhibition With Aliskiren Prevents the Development of Hypertension in Cyp1a1-Ren2 Transgenic Rats With Inducible ANG II-Dependent Hypertension
Keywords: مهارکننده رنین; Kidney; Renin-angiotensin system; Renin inhibitor; Renal hemodynamics; Sodium excretion;
Design and optimization of novel (2S,4S,5S)-5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxy-2-isopropylhexanamides as renin inhibitors
Keywords: مهارکننده رنین; Renin inhibitor; Hypertension; Ketopiperazine; Structure-based drug design; X-ray crystallography
Direct Renin Inhibition With Aliskiren Normalizes Blood Pressure in Cyp1a1-Ren2 Transgenic Rats With Inducible Angiotensin II-Dependent Malignant Hypertension
Keywords: مهارکننده رنین; Kidney; Renin-angiotensin system; Malignant hypertension; Renin inhibitor; Renal hemodynamics;
Piperidine-based renin inhibitors: Upper chain optimization
Keywords: مهارکننده رنین; Hypertension; Renin angiotensin aldosterone system; Renin inhibitor; Piperidine
New classes of potent and bioavailable human renin inhibitors
Keywords: مهارکننده رنین; Renin inhibitor; Rational design; Double transgenic rat (TGR) model
Treating hypertension while protecting the vulnerable islet in the cardiometabolic syndrome
Keywords: مهارکننده رنین; Antihypertensive treatment; islet amyloid; insulin resistance; renin inhibitor
Discovery of 6-ethyl-2,4-diaminopyrimidine-based small molecule renin inhibitors
Keywords: مهارکننده رنین; Renin inhibitor; Hypertension; 2,4-Diaminopyrimidine; Structure based drug design; Renin–angiotensin system; RAS; Conformational overlap; Scaffold hopping
Aliskiren, an Orally Effective Renin Inhibitor, Provides Antihypertensive Efficacy Alone and in Combination With Valsartan
Keywords: مهارکننده رنین; Blood pressure; combination; hypertension; plasma renin activity; randomized controlled trial; renin inhibitor;
Aliskiren, the First Renin Inhibitor for Treating Hypertension: Reactive Renin Secretion May Limit Its Effectiveness
Keywords: مهارکننده رنین; Aliskiren; renin inhibitor; renin; renin-angiotensin; clinical trial; hypertension; renovascular hypertension; malignant hypertension; angiotensin-converting enzyme inhibitor; angiotensin II type 1 receptor blocker; diuretic;
Ketopiperazine-based renin inhibitors: Optimization of the “C” ring
Keywords: مهارکننده رنین; Renin inhibitor; Hypertension; Ketopiperazine; CYP3A4;
Benzyl ether structure–activity relationships in a series of ketopiperazine-based renin inhibitors
Keywords: مهارکننده رنین; Renin inhibitor; Hypertension; Topliss tree
Equipotent activity in both enantiomers of a series of ketopiperazine-based renin inhibitors
Keywords: مهارکننده رنین; Renin inhibitor; Ketopiperazine
Discovery of novel non-peptidic ketopiperazine-based renin inhibitors
Keywords: مهارکننده رنین; Renin–angiotensin system; Renin inhibitor; Ketopiperazinone; Double transgenic mouse model; Blood pressure
Analogs of 1α,25-dihydroxyvitamin D3 as novel inhibitors of renin biosynthesis
Keywords: مهارکننده رنین; Vitamin D; Vitamin D analogs; Gemini compounds; Renin; Renin-angiotensin system; Renin inhibitor; As4.1 cells;