دانلود مقالات ISI درباره Sar + ترجمه فارسی

Design and synthesis of novel potent anticoagulant and anti-tyrosinase pyranopyrimidines and pyranotriazolopyrimidines: Insights from molecular docking and SAR analysis

Keywords: Pyranopyrimidines; Pyranotriazolopyrimidines; Anticoagulant; Anti-tyrosinase; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 39 صفحه سال انتشار : 2019 سفارش ترجمه

Experimental and numerical analysis of Y-shaped split and recombination micro-mixer with different mixing units

Keywords: SAR; split and recombination micro-mixer; YSSAR; Y-shaped straight split and recombination micro-mixer; YRSAR; Y-shaped rhombus split and recombination micro-mixer; YCSAR; Y-shaped circular split and recombination micro-mixer; YRCSAR; Y-shaped rhombus and

دانلود رایگان متن کامل مقاله ISI 41 صفحه سال انتشار : 2019 سفارش ترجمه

Assessment of geothermal water quality for industrial and irrigation purposes in the Unai geothermal field, Gujarat, India

Keywords: LSI; Langelier Saturation Index; RSI; Ryznar Stability Index; PSI; Puckorius or Practical Scaling Index (PSI); LS; Larson-Skold Index; EC; Electrical Conductivity; TDS; Total Dissolved Salts; SAR; Sodium Absorption Ratio; KR; Kelly's Ratio; RSC; Residual

دانلود رایگان متن کامل مقاله ISI 45 صفحه سال انتشار : 2019 سفارش ترجمه

Identification of a 4-fluorobenzyl l-valinate amide benzoxaborole (AN11736) as a potential development candidate for the treatment of Animal African Trypanosomiasis (AAT)

Keywords: Benzoxaborole; Trypanosomiasis; Cattle; SAR; Lead optimisation; Protozoan;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2018 سفارش ترجمه

SAR for gastro-intestinal absorption and blood-brain barrier permeation of pesticides

Keywords: SAR; Pesticide; OECD principle; Binary classification; Monte Carlo method; CORAL software;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2018 سفارش ترجمه

Progress in antischistosomal N,N′-diaryl urea SAR

Keywords: N,N′-Diaryl urea; Antischistosomal; SAR;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis and biological evaluation of anti-cancer agents that selectively inhibit Her2 over-expressed breast cancer cell growth via down-regulation of Her2 protein

Keywords: Her2; Breast cancer; Lead optimization; SAR;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2018 سفارش ترجمه

Feasibility of aortic valve planimetry at 7 T ultrahigh field MRI: Comparison to aortic valve MRI at 3 T and 1.5 T

Keywords: SAR; specific absorption rate; UHF; ultrahigh field; Aortic valve imaging; Planimetry; Aortic valve opening area; 7 T ultrahigh field MRI; Cardiovascular magnetic resonance imaging;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2018 سفارش ترجمه

Antinociceptive effect of neo-clerodane diterpenes obtained from Baccharis flabellata

Keywords: Baccharis flabellata; Furan neoclerodane; Diene-acid clerodane dimer; Agonists of kappa receptors; AMSL; Above mean sea level; i.p.; Administered via the intraperitoneal route; ANMAT; Administración Nacional de Medicamentos, Alimentos y Tecnología Médi

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis of novel (−)-epicatechin derivatives as potential endothelial GPER agonists: Evaluation of biological effects

Keywords: Epi; (−)-epicatechin; eNOS; endothelial nitric oxide synthase; NO; nitric oxide; GPER; G-protein coupled estrogen receptor; BCAEC; bovine coronary artery endothelial cells; GPCRs; G-protein coupled receptors; EPI-COLUMN; affinity column with Epi covalen

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2018 سفارش ترجمه

Evaluation of analogues of furan-amidines as inhibitors of NQO2

Keywords: NQO2 inhibitors; Furan-amidines; Isosteres; Anti-cancer; Malaria; SAR;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2018 سفارش ترجمه

Design and synthesis of a series of bioavailable fatty acid synthase (FASN) KR domain inhibitors for cancer therapy

Keywords: FASN; Fatty acid synthase; LRS; lipid-reduced serum; NADPH; nicotinamide adenine dinucleotide phosphate; KR; ketoreductase domain; ER; enoylreductase domain; ψME; pseudo-methyltransferase domain; ψKR; pseudo-ketoreductase domain; Fatty acid synthase; En

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2018 سفارش ترجمه

Identification of tagitinin C from Tithonia diversifolia as antitrypanosomal compound using bioactivity-guided fractionation

Keywords: 1D and 2D NMR; One and two-dimensional nuclear magnetic resonance; BALB//3T3; Mouse fibroblasts; CH2Cl2/MeOH; Methylene chloride/Methanol; DMSO; Dimethylsulfoxide; HAT; Human African Trypanosomiasis; NTDs; Neglected tropical diseases; SAR; Structure-activ

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Non-monotonicity in the influence of nanoparticle concentration on SAR in magnetic nanoparticle hyperthermia

Keywords: Magnetic hyperthermia; Magnetic nanoparticles; Specific absorption rate; SAR; Specific loss power; SLP; Concentration; Silicone;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Wind resource assessment using SODAR and meteorological mast - A case study of Pakistan

Keywords: NREL); National Renewable Energy Laboratory; Research and Development; R&D; Light Detection and Ranging; LiDAR; Sound Detection and Ranging; SODAR; Wind Atlas Analysis and Application Program; WAsP; Synthetic Aperture Radar; SAR; Pakistan Meteorological D

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, molecular docking study and thymidine phosphorylase inhibitory activity of 3-formylcoumarin derivatives

Keywords: Synthesis; 3-formylcoumarin; Molecular docking study; Thymidine phosphorylase inhibition; SAR;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

A small diversity library of α-methyl amide analogs of sulindac for probing anticancer structure-activity relationships

Keywords: NSAID; non-steroidal anti-inflammatory drug; COX; cyclooxygenase; PG; prostaglandin; FAP; familial adenomatous polyposis; SSA; sulindac sulfide amide; SAR; structure-activity relationship; qHTS; quantitative high-throughput screen; CPC; choroid plexus car

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Assessment of MRI issues at 1.5 T for the Temperature Logger Implant

Keywords: PCB; Printed Circuit Board; EEPROM; Electrically Erasable Programmable Read-Only Memory; MEMS; Microelectromechanical Systems (MEMS); ASTM; American Society of Testing and Materials; SAR; Specific Absorption Rate; GRE; Gradient Echo Pulse Sequence; UAF; U

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Design, synthesis, in vitro and in vivo evaluation, and structure-activity relationship (SAR) discussion of novel dipeptidyl boronic acid proteasome inhibitors as orally available anti-cancer agents for the treatment of multiple myeloma and mechanism stud

Keywords: SAR; structureactivity relationship; UPP; ubiquitinproteasome pathway; FDA; Food and Drug Administration; ATP; Adenosine triphosphate; CP; core particle; RP; regulatory proteasome; C-L; caspase-like; T-L; trypsin-like; CT-L; chymotrypsin-like; EDCI; 1-eth

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, α-glucosidase inhibition and molecular docking study of coumarin based derivatives

Keywords: Synthesis; Coumarin; α-Glucosidase inhibition; Molecular docking study; SAR;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2018 سفارش ترجمه

An SAR study of hydroxy-trifluoromethylpyrazolines as inhibitors of Orai1-mediated store operated Ca2+ entry in MDA-MB-231 breast cancer cells using a convenient Fluorescence Imaging Plate Reader assay

Keywords: FLIPR; Fluorescence Imaging Plate Reader; STIM1; stromal interaction molecule 1; ER; endoplasmic reticulum; TNBC; triple negative breast cancer; SAR; structure activity relationship; LHS; left hand side; RHS; right hand side; THF; tetrahydrofuran; i-PrOH;

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2018 سفارش ترجمه

Structure characteristics for intestinal uptake of flavonoids in Caco-2 cells

Keywords: CU; cellular uptake of flavonoid without verapamil; CUV; cellular uptake of flavonoid with verapamil; SAR; structure activity relationship; QSAR; quantitative structure absorption relationship; MRP; multidrug resistance-associated protein; P-gp; P-glycopr

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2018 سفارش ترجمه

Discovery of 1-(4-((3-(4-methylpiperazin-1-yl)propyl)amino)benzyl)-5-(trifluoromethyl)pyridin-2(1H)-one, an orally active multi-target agent for the treatment of diabetic nephropathy

Keywords: ACR; albumin-to-creatinine ratio; AUC0-t; area under the curve; BuOH; n-butanol; BUN; blood urea nitrogen; Cmax; peak concentration; C13-NMR; C13-nuclear magnetic resonance; CCr; creatinine clearance rate; CCR2; CCchemkin receptor 2; CDCl3; Deuterotrichlo

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis and molecular docking study of piperazine derivatives as potent inhibitor of thymidine phosphorylase

Keywords: Synthesis; Piperazine; Thymidine phosphorylase; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2018 سفارش ترجمه

Using satellite radar amplitude imaging for monitoring syn-eruptive changes in surface morphology at an ice-capped stratovolcano

Keywords: Explosive volcanism; Radar amplitude; SAR;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Organic matter accumulation and salinity change in open water areas within a saline boreal fen in the Athabasca Oil Sands Region, Canada

Keywords: OM; organic matter; OMAR; organic matter accumulation rate; SAR; sediment accumulation rate; AOSR; Athabasca Oil Sands Region; Organic matter; Salinity; Saline wetlands; Plant macrofossils; Diatoms;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Quantifying the conservation value of Sacred Natural Sites

Keywords: Sacred Natural Sites; SNS; Species Abundance Relationships; SAR; Sacred Natural Sites; Conservation value; Biodiversity; Extinction debt; Beta diversity;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

HPTLC-profiling of eleutherosides, mechanism of antioxidative action of eleutheroside E1, the PAMPA test with LC/MS detection and the structure-activity relationship

Keywords: Eleutherococcus; Eleutheroside E1; Załuski's hypothesis; HPTLC-autography; Antioxidant; PAMPA test; SAR;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Bisindolylmethane thiosemicarbazides as potential inhibitors of urease: Synthesis and molecular modeling studies

Keywords: Synthèsis; Bisindole; Urease inhibition; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis of Bis-indolylmethane sulfonohydrazides derivatives as potent α-Glucosidase inhibitors

Keywords: Synthesis; Bis-indolylmethane; Sulfonohydrazides; α-glucosidase activity; SAR; Molecular docking;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis: Small library of hybrid scaffolds of benzothiazole having hydrazone and evaluation of their β-glucuronidase activity

Keywords: Benzothiazole; Synthesis; β-Glucuronidase activity; SAR;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, in vitro α-glucosidase inhibitory potential and molecular docking study of thiadiazole analogs

Keywords: Synthesis; Thiadiazole; α-Glucosidase; Molecular docking study; SAR;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2018 سفارش ترجمه

Combining Sentinel-1 and Sentinel-2 data for improved land use and land cover mapping of monsoon regions

Keywords: Sentinel-1; Sentinel-2; Random forest; Multi-sensory; SAR; Land use and land cover classification; Cloud-prone; India;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Aim for the core: suitability of the ubiquitin-independent 20S proteasome as a drug target in neurodegeneration

Keywords: 20S; core 20S proteasome; AD; Alzheimer's disease; ALS; amyotrophic lateral sclerosis; ATP; adenosine triphosphate; BBB; blood-brain barrier; DUB; deubiquitinating enzyme; HbYX; hydrophobic-tyrosine-unspecified residue 'X'; IDP; intrinsically disorder

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Combining COSMO-SkyMed satellites data and numerical modeling for the dynamic management of artificial recharge basins

Keywords: Groundwater; Artificial recharge basin; Infiltration; Remote sensing; SAR; Clogging;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

An approach for flood monitoring by the combined use of Landsat 8 optical imagery and COSMO-SkyMed radar imagery

Keywords: SAR; Water extraction; Support vector machine; Active contour; Inundation analysis;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Stoichiometry dependent inhibition of rat α3β4 nicotinic acetylcholine receptor by the ribbon isomer of α-conotoxin AuIB

Keywords: ACh; acetylcholine; AChBP; acetylcholine-binding protein; ECD; extracellular domain; gAuIB; globular AuIB; ICD; intracellular domain; nAChR; nicotinic acetylcholine receptor; rAuIB; ribbon AuIB; SAR; structure-activity relationship; TMD; transmembrane dom

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Exposure to GSM 900-MHz mobile radiation impaired inhibitory avoidance memory consolidation in rat: Involvements of opioidergic and nitrergic systems

Keywords: ANOVA; analysis of variance; EMF; electromagnetic field; GSM; global system for mobile communications; Hz; hertz; h; hour; IA; inhibitory avoidance; i.c.v.; intracerebroventricular; i.p.; intraperitoneal; LTP; long term potentiation; L-NAME; NG-Nitro-L-ar

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Structure-activity relationships of rationally designed AMACR 1A inhibitors

Keywords: α-Methylacyl-CoA racemase (AMACR, P504S); Drug lipophilicity; Enzyme inhibitors; Rational drug design; Structure-activity relationships; AMACR; α-methylacyl-CoA racemase; CDI; carbonyldiimidazole; DAST; (Diethylamino)sulfur trifluoride; DCC; Dicyclohexy

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, molecular docking study and in vitro thymidine phosphorylase inhibitory potential of oxadiazole derivatives

Keywords: Synthesis; Oxadiazole; Thymidine phosphorylase; Molecular docking; SAR;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Biological sand filter system treating winery effluent for effective reduction in organic load and pH neutralisation

Keywords: WWW; winery wastewater; WW; wastewater; HRT; hydraulic retention time; CW(s); constructed wetland; OMWW; olive mill wastewater; COD; chemical oxygen demand; BSF(s); biological sand filter; k; hydraulic conductivity; VOA(s); volatile organic acid; AAC; ace

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2018 سفارش ترجمه

Simultaneous ocean surface current and wind vectors retrieval with squinted SAR interferometry: Geophysical inversion and performance assessment

Keywords: Ocean surface current vector; Ocean wind vector; Doppler; Scatterometer; SAR; Along-track interferometry;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Quantitative mapping of groundwater depletion at the water management scale using a combined GRACE/InSAR approach

Keywords: CFE; Comisión Federal de Electricidad; CONAGUA/CNA; Comisión Nacional del Agua; DDK; Deccorelation filter for GRACE data created by J. Kusche (GFZ, Posdam, Germany); GLDAS; Global Land Data Assimilation System (LSM output dataset); GRACE; Gravity Recove

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Locally distributed ground deformation in an area of potential phreatic eruption, Midagahara volcano, Japan, detected by single-look-based InSAR time series analysis

Keywords: SAR; Ground deformation; Phreatic eruption, Midagahara volcano;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

The evaluation of potent antitumor activities of shikonin coumarin-carboxylic acid, PMMB232 through HIF-1α-mediated apoptosis

Keywords: HIF-1α; hypoxia-inducible factor alpha 1; DMAP; 4 dimethyamino- pyridine; DCC; N, N' dicyclohexylcarbodiimide; DMEM; Dulbecco's modified Eagle's medium; MTT; 3-(4 5-dimethyl-2-thiazolyl)-2 5-diphenyl-2-H-tetrazolium bromide; IC50; Half of maximal i

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Hit optimization studies of 3-hydroxy-indolin-2-one analogs as potential anti-HIV-1 agents

Keywords: AIDS; Reverse transcriptase; Toxicity; Virtual screening; SAR; Docking;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists

Keywords: GPR52; G protein-coupled receptor 52; SAR; structure-activity relationship; cAMP; 3′,5′-cyclic adenosine monophosphate; EC50; half maximal effective concentration; MAP; methamphetamine; NMDA; N-methyl-d-aspartate; PK; pharmacokinetic; CHO; Chinese h

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II

Keywords: Cdk1; Cyclin-dependent kinase 1; EFS; embryonal FYN-associated substrate; (6-FAM); 6-carboxyfluorescein; FL; full-length; FP; fluorescence polarization; FPIA; fluorescence polarization based immunoassay; KD; kinase domain; PKIS; protein kinase inhibitor s

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Impacts of an ice-free Northeast Passage on LNG markets and geopolitics

Keywords: AMSA; Arctic Marine Shipping Assessment; BP; British Petroleum; CNPC; China National Petroleum Corporation; EIA; U.S. Energy Information Administration; E&P; Exploration and Production; FID; Final Investment Decision; FSU; Former Soviet Union; GECF; Gas E

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, SAR elucidations and molecular docking study of newly designed isatin based oxadiazole analogs as potent inhibitors of thymidine phosphorylase

Keywords: Isatin; Oxadiazole; Synthesis; TP inhibition; SAR; Molecular docking;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه