Keywords: رابطه ساختار-فعالیت; Anionic porphyrins; ROS production; Structure-activity relationship; TBY-2 cells; pH effect;
مقالات ISI رابطه ساختار-فعالیت (ترجمه نشده)
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Keywords: رابطه ساختار-فعالیت; Ecteinascidin pentacyclic skeleton; Synthesis; Cytotoxicity; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; 1,3,4-Oxadiazole derivatives; Intermediate derivatization method; Rice sheath blight; Sorghum anthracnose; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Biphalin; Opioid receptors; MOR/DOR/KOR agonist; Synergistic analgesic effect; Cyclic peptides; Acm; acetamidomethyl; ACN; acetonitrile; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BOP; (benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluoro
Keywords: رابطه ساختار-فعالیت; Plasminogen activator inhibitor-1 (PAI-1); PAI-1 inhibitor; N-Acylanthranilic acid derivatives; Oral bioavailability; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Essential oil; Antimicrobial; Structure-activity relationship; Escherichia coli; Staphylococcus aureus;
Keywords: رابطه ساختار-فعالیت; d-Amino acid oxidase; Open-lid conformation; Virtual screening; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Tuberculosis; MTB H37Rv; MDR-MTB; 3,5-Dinitrobenzamides; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Ciprofloxacin; Isatin; Hybrids; Antimicrobial; Antibacterial; Antimycobacterial; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; AmB; amphotericin B; ATCC; American Type Culture Collection; CAS; caspofungin; CLSI; Clinical and Laboratory Standards Institute; FBS; fetal bovine serum; FLC; fluconazole; KANB; kanamycin B; mRBCs; murine red blood cells; PI; propidium iodide; SAR; struc
Keywords: رابطه ساختار-فعالیت; PAL inhibitors; Aminophosphonates; Molecular modeling; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; SMP; starfish myorelaxant peptide; SAR; structure-activity relationships; PP; pedal peptide; OK; orcokinin; ACh; acetylcholine; TFA; trifluoroacetic acid; RP; reversed-phase; HOBT; 1-hydroxybenzotriazole; DIPCI; N,N-diisopropylcarbodimide; ASW; artificial
Keywords: رابطه ساختار-فعالیت; ABC; ATP-binding cassette; AKT; V-Akt murine thymoma viral oncogene homolog; ALDH1; aldehyde dehydrogenase 1; AR; androgen receptor; Bad; Bcl-2-associated death promoter; Bak; Bcl-2 homologous antagonist killer; Bax; Bcl-2-associated X protein; Bcl-2; B-c
Keywords: رابطه ساختار-فعالیت; Drug discovery; Structure-activity relationship; Target; Nuclear receptor; Drug repositioning; Antihypertensive drugs;
Keywords: رابطه ساختار-فعالیت; QPA; quaternary protoberberine alkaloid; TF; transcriptional factor; UC; ulcerative colitis; IEC-6; intestinal epithelial cell-6; XBP1; X-box-binding protein 1; MIC; minimal inhibitory concentration; SAR; structure-activity relationship; SASP; Sulfasalazi
Keywords: رابطه ساختار-فعالیت; GCGR; glucagon receptor; cAMP; cyclic-adenosine monophosphate; T2DM; type 2 diabetes mellitus; SGLT-2; sodium-glucose cotransporter-2; HGP; hepatic glucose production; GPCRs; G-protein coupled receptors; SAR; structure-activity relationship; Ser; Serine;
Keywords: رابطه ساختار-فعالیت; Fluoroquinolones; Ciprofloxacin; Antibacterial; Hybrid compounds; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Matrix metalloproteinase 13; Structure-property relationship; Structure-activity relationship; Microsomal stability; Solubility; Permeability; In vitro and in vivo pharmacokinetics;
Keywords: رابطه ساختار-فعالیت; Benzofuran-isatin hybrids; Anti-mycobacterial; Anti-tubercular; Multi-drug resistant; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; 2-Phenol-4,6-dichlorophenyl-pyridines; Anti-proliferative activity; Topoisomerase inhibitor; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Larotaxel; Toxoids; Structure-activity relationship; Semi-synthesis; Drug-resistant; Cytotoxicity;
Keywords: رابطه ساختار-فعالیت; 2-Thio-5-amino substituted benzoquinones; Anti-tumor activity; Synthesis; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; DPPH; 2,2-diphenyl-1-picrylhydrazyl; FRAP; ferric reducing antioxidant power; HCA; hierarchical cluster analysis; HPSEC; high performance size-exclusion chromatography; LRPs; lotus root polysaccharides; MLR; multiple linear regression; NO; nitrogen oxide;
Keywords: رابطه ساختار-فعالیت; Peptides; Peptidomimetics; Biofilm; Antibiofilm; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Boron; Glycaemia; Diabetes; Structure-activity relationship; Inflammation;
Keywords: رابطه ساختار-فعالیت; Antitubercular activity; Diphenyl ether; Enzyme inhibition; InhA; Structure-activity relationship; Triclosan;
Keywords: رابطه ساختار-فعالیت; Chiral pesticide; Lead optimization; Drimane; Oxazinone; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Fluoroquinolones; Anti-mycobacterial; Anti-tubercular; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; bioequivalence; dose-response; glycoprotein; glycosylation; in vitro-in vivo correlations; pharmacokinetics; pharmacodynamics; structure-activity relationship; regulatory science;
Keywords: رابطه ساختار-فعالیت; Amino-substituted 1H-phenalen-1-ones; Anti-leishmanial activity; Structure-activity relationship; Mitochondrial membrane potential; IYOABNFVEYPDRP-UHFFFAOYSA-N; KAIWDUKYQHSVPW-UHFFFAOYSA-N; ORPSFAGNVFPTPF-UHFFFAOYSA-N; KKWCGVRETPEFLX-UHFFFAOYSA-N; VOJLSGF
Keywords: رابطه ساختار-فعالیت; Silver nanoparticles; Phenolic acids; Structure-activity relationship; Antioxidant activity;
Keywords: رابطه ساختار-فعالیت; Morita-Baylis-Hillman bromides; Palladium-catalyzed coupling; Phosphonic acids; Enzyme inhibitors; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Fluorocyclopentenyl nucleoside; Structure-activity relationship; Fluorination; Phosphorylation; Prodrug; Anticancer;
Keywords: رابطه ساختار-فعالیت; Quinolone; Fluoroquinolone; Hybrids; Gram-positive pathogens; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; 1,2,3-triazoles; Cytotoxicity; Neurotoxicity; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Antiplatelet; Preclinical studies; Structure-activity relationship (SAR) studies; Pharmacokinetic parameters; Safety profile; AA; arachidonic acid; ADP; adenosine diphosphate; ATP; adenosine triphosphate; CNS; central nervous system; COX-1; cyclooxygenase
Keywords: رابطه ساختار-فعالیت; Antiplasmodial; Antimalarial; Quinolone; Fluoroquinolone; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Imidazole; Nitroimidazole; Hybrids; Anti-mycobacterial; Anti-tubercular; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Antioxidative efficacies; Antibacterial activities; Aqueous ethanol extracts; Berries; Leaves; Phenolic compounds; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Sophoridine derivatives; Anticancer; Structure-activity relationship; Apoptosis; Tumor xenograft;
Keywords: رابطه ساختار-فعالیت; Tubulin; Microtubule-stabilizing agents; Chemotherapy; Paclitaxel; Taccalonolide; Epothilone; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Quinolone amides; Trypanosoma brucei brucei; Structure-activity relationship; Fluorine walk; Metabolism; Blood-brain barrier; Autoradiography;
Keywords: رابطه ساختار-فعالیت; Quinolone derivatives; Hybrid compounds; Antibacterial; Escherichia coli; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; ADME; Absorption, Distribution, Metabolism, Excretion; AOPs; adverse outcome pathways; AUC; Area under the Curve; AEs; assessment elements; AOs; assessment options; BMDL; benchmark dose lower bound; CAAT; Center for Alternatives to Animal Testing; Cefic-L
Keywords: رابطه ساختار-فعالیت; Quinazoline; Structure-activity relationship; Drug design and development; Therapeutic agents; Pharmacological significance;
Keywords: رابطه ساختار-فعالیت; Anti-diabetes; Molecular targets; Structure-activity relationship; Type-II diabetes;
Synthesis and biological evaluation of 4-methyl-1,2,3-thiadiazole-5-carboxaldehyde benzoyl hydrazone derivatives
Keywords: رابطه ساختار-فعالیت; 1,2,3-Thiadiazole; Benzoyl hydrazone; Synthesis; Fungicidal activity; Curative activity against TMV; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Co-graft starch-based flocculant; Charge density; Average graft chain length; Flocculation performance; Flocculation mechanism; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Photodynamic therapy; Phthalocyanine; Chlorambucil; Structure-activity relationship; Anticancer;
Keywords: رابطه ساختار-فعالیت; Chiral pesticide; Lead optimization; Natural products; Mixed synthesis; Structure-activity relationship;