دانلود مقالات ISI درباره رابطه ساختار-فعالیت + ترجمه فارسی

One-pot synthesis and biological evaluation of 2-pyrrolidinyl-4-amino-5-(3′,4′,5′-trimethoxybenzoyl)thiazole: A unique, highly active antimicrotubule agent

Keywords: رابطه ساختار-فعالیت; Microtubules; Structure-activity relationship; Thiazole; In vivo and in vitro activity; Tubulin

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis of N-substituted 2-[(1E)-alkenyl]-4-(1H)-quinolone derivatives as antimycobacterial agents against non-tubercular mycobacteria

Keywords: رابطه ساختار-فعالیت; Antimycobacterial; Lipophilicity; N-Substituted-2-[(1E)-alkenyl]-4-(1H)-quinolone; Structure-activity relationship;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2011 سفارش ترجمه

l-Proline anchored multicomponent synthesis of novel pyrido[2,3-a]carbazoles; investigation of in vitro antimicrobial, antioxidant, cytotoxicity and structure activity relationship studies

Keywords: رابطه ساختار-فعالیت; Pyrido[2,3-a]carbazoles; Antibacterial; Antifungal; Antioxidant; Cytotoxicity; Structure-activity relationship;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis and antiproliferative activity of indolizine derivatives incorporating a cyclopropylcarbonyl group against Hep-G2 cancer cell line

Keywords: رابطه ساختار-فعالیت; Indolizine derivatives; Antiproliferative activities; Hep-G2 cell line; EGFR; Structure-activity relationship; Docking simulations

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2010 سفارش ترجمه

Comparative effects of β-carbolines on platelet aggregation and lipid membranes

Keywords: رابطه ساختار-فعالیت; β-carbolines; antiplatelet effects; human platelet aggregation; membrane interaction; structure-activity relationship

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2010 سفارش ترجمه

α-Glucosidase and α-amylase inhibitory activities of guava leaves

Keywords: رابطه ساختار-فعالیت; Guava leaves; α-Glucosidase and α-amylase inhibitor; Flavonoid compounds; Structure-activity relationship; Diabetes

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2010 سفارش ترجمه

Synthesis and structure-activity relationship study of 8-hydroxyquinoline-derived Mannich bases as anticancer agents

Keywords: رابطه ساختار-فعالیت; Clioquinol; 8-Hydroxyquinoline; Mannich-type reaction; Structure-activity relationship

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2010 سفارش ترجمه

Structural features of prostanoid analogues involved in hepatocytes protection against CCl4-induced injury

Keywords: رابطه ساختار-فعالیت; CCl4, carbon tetrachloride; LDH, lactic dehydrogenase; PG, prostaglandin; DMEM, Dulbecco's modified Eagle medium; SAR, structure-activity relationshipProstaglandins; CCl4; Cytoprotection; Rat liver hepatocytes; Structure-activity relationship

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2010 سفارش ترجمه

Synthesis, biological activity, and evaluation of the mode of action of novel antitubercular benzofurobenzopyrans substituted on A ring

Keywords: رابطه ساختار-فعالیت; Antimycobacterials; 3,3-Dimethyl-3H-benzofuro[3,2-f][1]benzopyran; Structure-activity relationship; Mycolates

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2010 سفارش ترجمه

Superhydrophilicity of anodic aluminum oxide films: From “honeycomb” to “bird's nest”

Keywords: رابطه ساختار-فعالیت; Superhydrophilicity; Anodic aluminum oxide films; Structure-activity relationship

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2009 سفارش ترجمه

Role of V in supported V–Sb–O catalysts for the ammoxidation of propane to acrylonitrile: Multilayered VOx/SbOx/Al2O3 catalysts

Keywords: رابطه ساختار-فعالیت; V–Sb–Al; V–Sb–O; Oxidation; Ammoxidation; Propane; Acrylonitrile; Structure-activity relationship; In situ Raman; XRD

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligands

Keywords: رابطه ساختار-فعالیت; Dopamine receptors; Antipsychotics; Structure-activity relationship; Benzolactams; Arylpiperazines

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2009 سفارش ترجمه

The effects of twelve representative flavonoids on tissue factor expression in human monocytes: Structure-activity relationships

Keywords: رابطه ساختار-فعالیت; TF; tissue factor; PCA; procoagulation activity; LPS; lipopolysaccharide; TNF-α; tumor necrosis factor-α; HBSS; hank's balanced salt solution; PPSB; prothrombin complex; SARs; structure-activity relationships; Flavonoids; Tissue factor; Structure-activi

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

Regulation of neurosteroid allopregnanolone biosynthesis in the rat spinal cord by glycine and the alkaloidal analogs strychnine and gelsemine

Keywords: رابطه ساختار-فعالیت; steroidogenesis in nerve cells; steroids and nervous system; glycinergic system; structure-activity relationship; neurosteroidogenesis regulator; neurosteroid and neurotransmitterANOVA, analysis of variance; DCM, dichloromethane; GABAA receptor, GABA type

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2008 سفارش ترجمه

A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitors

Keywords: رابطه ساختار-فعالیت; Diabetes; Pharmacophore; CATALYST; Structure-activity relationship; Dipeptidyl peptidase IV

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2008 سفارش ترجمه

Studies directed towards a mechanistic evaluation of inactivation of aromatase by the suicide substrates androsta-1,4-diene-3,17-diones and its 6-ene derivatives: Aromatase inactivation by the 19-substituted derivatives and their enzymic aromatization

Keywords: رابطه ساختار-فعالیت; Aromatase inhibitor; 19-Substituted androsta-1,4-diene-3,17-dione; Time-dependent inactivation; Structure-activity relationship; Aromatization; Gas chromatography–mass spectrometry

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2007 سفارش ترجمه

Theoretical evaluation of flavonoids as multipotent agents to combat Alzheimer's disease

Keywords: رابطه ساختار-فعالیت; Alzheimer's disease; Flavonoids; Inhibitor; Multipotent agent; Xanthones; Docking; Aβ; amyloid-βpeptide; ACh; acetylcholine; AChE; acetylcholinesterase; AD; Alzheimer's disease; BChE; butyrylcholinesterase; IHB; intramolecular hydrogen bond; MAO; monoam

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2006 سفارش ترجمه

Role of pharmacologically active metabolites in drug discovery and development

Keywords: رابطه ساختار-فعالیت; Pharmaceutical Science; Drug Discovery; Pharmacology; EndocrinologyRole; formation; structure-activity relationship; detection of pharmacologically active metabolites

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2006 سفارش ترجمه

Active dimer of Epratuzumab provides insight into the complex nature of an antibody aggregate

Keywords: رابطه ساختار-فعالیت; adduct; glycoprotein; physical stability; preformulation; protein aggregation; protein formulation; protein structure; solvation; structure-activity relationship;

دانلود رایگان متن کامل مقاله ISI 20 صفحه سال انتشار : 2006 سفارش ترجمه

Ligand efficiency indices as guideposts for drug discovery

Keywords: رابطه ساختار-فعالیت; Drug Discovery; Pharmaceutical Science; Pharmacokinetics; Structure-activity relationship; Molecular weight; Polar surface area; Ligand-binding efficiency;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2005 سفارش ترجمه

Relationship between cucurbitacins reversed-phase high-performance liquid chromatography hydrophobicity index and basal cytotoxicity on HepG2 cells

Keywords: رابطه ساختار-فعالیت; Cucurbitacin; Chromatographic hydrophobicity index; CHI; HepG2; IC50; Cytotoxicity; Structure-activity relationship; SAR; log P; C log P; RP-HPLC;

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2005 سفارش ترجمه

Cryogenically cooled probes-a leap in NMR technology

Keywords: رابطه ساختار-فعالیت; NMR (Nuclear Magnetic Resonance); Cryogenic probe technology; Sensitivity; Signal-to-noise ratio; 1D; 1-dimensional; 2D; 2-dimensional; 3D; 3-dimensional; ASTM; American Society for Testing and Materials; BPTI; bovine pancreatic trypsine inhibitor; CDCl3;

دانلود رایگان متن کامل مقاله ISI 25 صفحه سال انتشار : 2005 سفارش ترجمه