Keywords: ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid)diammonium salt; BSA; bovine serum albumin; (bt)-VEGF165; biotinylated-VEGF165; 6-Cl·HOBt; 6-chloro-1-hydroxybenzotriazole dehydrate; DIPEA; N,N-diisopropylethylamine; ELISA; enzyme-linked imm
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Keywords: AM251; 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(1-piperidyl)pyrazo-le-3-carboxamide; BSA; bovine serum albumin; DAMGO; [d-Ala2, N-MePhe4, Gly-ol]-enkephalin; DIEA; diisopropylethylamine; DMF; dimethylformamide; EGTA; ethylene glycol-bis(2-amino
Keywords: Abz; ortho-aminobenzoic acid; EDDnp; N-(2,4-dinitrophenyl)-ethylenediamine; FRET; fluorescence resonance energy transfer; hMIP; human mitochondrial intermediate peptidase; HOBt; hydroxybenzotriazole; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethylur
Keywords: Diversity-oriented synthesis; Imidazoheterocyclic; Groebke-Blackburn-Bienayme reaction; Fused imidazole; Lewis acid; Ugi type; Ac; acetyl; Aq; aqueous; Ar; aryl; Bn; benzyl; Boc; tert-butoxycarbonyl; BDMS; bromodimethylsulfonium bromide; CDK; cyclin-d
Keywords: AgOTf; silver triflate; BBB; blood-brain barrier; CDMT; 2-chloro-4,6-bis[3-(perfluorohexyl)propyloxy]-1,3,5-triazine; CNS; central nervous system; DMF; dimethylformamide; EM-2; endomorphin-2; Fmoc; N-(9-fluorenylmethyloxycarbonyl); GPI assay; guinea pig
Selenoprotein L-inspired nano-vesicular peroxidase mimics based on amphiphilic diselenides
Keywords: Cys; l-cysteine; DAN; 2,3-diaminonaphtalene; GPx; glutathione peroxidase; GSH; glutathione in the reduced form; MALDI TOF-MS; matrix-assisted laser desorption ionization time of flight-mass spectrometry; NADPH; nicotinamide adenine dinucleotide phosphate;
DNA sequence-specific ligands. XVII. Synthesis, spectral properties, virological and biochemical studies of fluorescent dimeric bisbenzimidazoles DBA(n)
Keywords: topo-I; DNA topoisomerase I; DMT; DNA methyltransferase; HSV-1; herpes simplex virus type 1; CMV; cytomegalovirus; scDNA; supercoiled DNA; b.p.; base pairs; MABs; monoclonal antibodies; ACV; acyclovir; PBS; phosphate buffered saline; PFU/cells; plaque for
Cathepsin B inhibitors: Further exploration of the nitroxoline core
Keywords: Abz; 2-aminobenzoyl; AMC; 7-amido-4-methylcoumarin; catB; cathepsin B; DIPEA; N,N-diisopropylethylamine; DMSO; dimethyl sulfoxide; ECM; extracellular matrix; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,
Novel aromatic sulfonyl naphthalene-based boronates as 20S proteasome inhibitors
Keywords: TEA; triethylamine; THF; tetrahydrofuran; Py; pyridine; DIPEA; N,N-diisopropylethylamine; TBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium tetrafluoroborate; DCM; dichloromethane; TPLM; (1R)-(S)-pinanediol-1-ammonium trifluoroacetate-3-methylbut
Lactam hybrid analogues of solonamide B and autoinducing peptides as potent S. aureus AgrC antagonists
Keywords: Autoinducing peptides; Anti-virulence therapy; Solonamide; Quorum-sensing system; Staphylococcus aureus; AIP; autoinducing peptide; CA-MRSA; community-associated; Dap; (S)-2,3-diaminopropamoic acid; Fmoc; fluoren-9-ylmethoxycarbonyl; hLeu; homoleucine; HO
Continuous assays for meprin alpha and beta using prolyl tripeptidyl aminopeptidase (PtP) from Porphyromonas gingivalis
Keywords: Astacins; Auxiliary enzyme; Continuous assay; Meprin α/β; Prolyl tripeptidyl aminopeptidase (PtP); AMC; 7-amido-4-methylcoumarin; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DMF; dimethylformamide; DTE; Dithioerythritol; HIC-EBA; hydrophobic inter
Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
Keywords: Neuropilin-1; VEGF165; Neuropilin/VEGF165 binding inhibition; Structure-activity relationship; Peptide biostability; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; Ahp; 7-aminoheptanoic acid; Aun; 11-aminoundecanoic acid;
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity
Keywords: Antibacterial; DNA gyrase; GyrB; Inhibitor; N-phenylpyrrolamide; ParE; Topoisomerase IV; ATCC; American type culture collection; ATR; attenuated total reflectance; CDI; 1,1â²-carbonyldiimidazole; CFU; colony-forming unit; CLSI; Clinical and Laboratory St
Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1
Keywords: ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; ACN; acetonitrile; BSA; bovine serum albumin; (bt)-VEGF165; biotinylated-VEGF165; 6-Cl-HOBt; 6-chloro-1-hydroxybenzotriazole dihydrate; DIPEA; N,N-diisopropylethylamine; DMEM;
Novel platinum(IV) complexes conjugated with a wogonin derivative as multi-targeted anticancer agents
Keywords: TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium tetrafluoroborate; DCM; dichloromethane; TEA; triethylamine; DMF; N/Nâ²-dimethylformamide; DMSO; dimethylsulfoxide; PBS; phosphate buffer solution; SGC7901; human gastric carcinoma cell line; H
Effect of TLR ligands co-encapsulated with multiepitopic antigen in nanoliposomes targeted to human DCs via Fc receptor for cancer vaccines
Keywords: AAA; amino acid analysis; C18; octadecylsilica; DIEA; N,N-diisopropyl-ethylamine; DIPCDI; N,N'-Diisopropylcarbodiimide; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide Fmoc, 9-fluorenylmethoxycarbonyl; HOAt; 1-hydroxy-7-azabenzotriazole (3-hydroxy-
Synthesis and binding characteristics of [3H]neuromedin N, a NTS2 receptor ligand
Keywords: BH; Bolton-Hunter; Bmax; maximal number of the binding sites; BSA; bovine serum albumin; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; EC50; half maximal effective concentration; Emax; maximal stimulation (Efficacy); GDP; guanosine 5â²-
Novel internally quenched substrate of the trypsin-like subunit of 20S eukaryotic proteasome
Keywords: 20S Eukaryotic proteasome; Internally quenched peptides; Fluorescence; UPS; ubiquitin-proteasome system; ACC; 7-amino-4-carbamoylmethylcoumarin; AMC; 7-amino-4-methylocoumarin; FRET; fluorescent resonance energy transfer; ABZ; 2-aminobenzoic acid; Tyr(3
Discovery of antitumor anthra[2,3-b]furan-3-carboxamides: Optimization of synthesis and evaluation of antitumor properties
Keywords: Anthra[2,3-b]furan-3-carboxamides; DNA ligands; Topoisomerase inhibitors; Protein kinase inhibitors; Cytotoxicity; Circumvention of multidrug resistance; Antitumor activity; CDI; 1,1â²-carbonyldiimidazole; DCC; N,Nâ²-dicyclohexylcarbodiimide; EDC; 1-eth
Locking PDK1 in DFG-out conformation through 2-oxo-indole containing molecules: Another tools to fight glioblastoma
Keywords: PDK1 inhibitors; Kinase inhibitors; Oxindole derivatives; Pyridonyl derivatives; Glioblastoma; GBM stem cells; OXIDs; 2-oxindole derivatives; TBTU; N,N,Nâ²,Nâ²-Tetramethyl-O-(benzotriazol-1-yl)uronium tetrafluoroborate; DIPEA; N,N-Diisopropylethylamine;
Novel S1P1 receptor agonists - Part 4: Alkylaminomethyl substituted aryl head groups
Keywords: S1P1 receptor agonist; Immunomodulator; Lymphocyte count; Aminomethyl pyridine; Aminomethyl benzene; Aminomethyl thiophene; Phototoxicity; BuLi; n-butyl lithium; CC; column chromatography; DCM; dichloromethane; DIPEA; diisopropylethylamine; DEAD; diethyl
A novel synthetic luteinizing hormone-releasing hormone (LHRH) analogue coupled with modified β-cyclodextrin: Insight into its intramolecular interactions
Keywords: BOP; benzotriazole-1-yl-oxy-tris-(dimethylamino)-phosphonium hexafluorophosphate; CLTR-Cl; 2-chlorotrityl chloride; DCC; N,Nâ²-dicyclohexylcarbodiimide; DMA; dimethylacetamide; DIC; N,Nâ²-diisopropylcarbodiimide; DIEA; diisopropylethylamine; DMF; N,N-di
The synthesis of indolo[2,3-b]quinoline derivatives with a guanidine group: Highly selective cytotoxic agents
Keywords: Neocryptolepine; Antiproliferative activity; Antifungal activity; Biofilm; Guanidine group; Mechanism of action; Apoptosis; Hemolytic activity; Boc; tert-butyloxycarbonyl group; BSTU; N,Nâ²-bis-Boc-thiourea; DIPEA; N,N-diisopropylethylamine; DMF; dimethy
Microwave-assisted guanidinylation in solid phase peptide synthesis: comparison of various reagents
Keywords: Boc; tert-butyloxycarbonyl; Dab; 2,4-diaminobutyric acid; Dap; 2,3-diaminopropionic acid; Dap(g); 3-guanidino-2-aminopropionic acid; DIC; 1,3-diisopropylcarbodiimide; DIEA; diisopropylethylamine; hArg(g); 2,6-diguanidinohexanoic acid; MW; microwave; TBTU;
Synthetically modified l-histidine-rich peptidomimetics exhibit potent activity against Cryptococcus neoformans
Keywords: AA; amino acid; Boc; tert-butoxycarbonyl; DIC; 1,3-diisopropylcarbodiimide; DIEA; N,N-diisopropylethylamine; EYPC; egg yolk l-a-phosphatidylcholine; DMF; N,N-dimethylformamide; EYPG; egg yolk l-a-phosphatidyl-dl-glycerol; TBTU; O-(benzotriazol-1-yl)-N,N,N
The interactions of glycated decapeptide, the Amadori product, with copper(II) ions - A possible effect on the oxidative stress induced aggregation?
Keywords: Boc2O; di-tert-butyl dicarbonate; DMF; N,N-dimethylformamide; Fru; aminofructose moiety; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium tetrafluoroborate; TFA; trifluoroacetic acid; TIS; triisopropylsilane; Coordination chemistry; Copper(II)
Peptides that activate the 20S proteasome by gate opening increased oxidized protein removal and reduced protein aggregation
Keywords: ALS; amyotrophic lateral sclerosis; AMC; 7-amido-4-methylcoumarin; z-ARR-AMC; z-Ala-Arg-Arg-amido-4-methylcoumarin; ChT-L; chymotrypsin-like proteasomal activity; DMF; N,N-dimethyl formamide; DMSO; dimethyl sulfoxide; DNPH; 2,4-dinitrophenylhydrazine; DTT
New chiral derivatives of xanthones: Synthesis and investigation of enantioselectivity as inhibitors of growth of human tumor cell lines
Keywords: Chiral derivatives of xanthones; Enantiomerically pure; TBTU; Antitumor; Enantioselectivity;
Differences in the inhibition of coagulation factor XIII-A from animal species revealed by Michael Acceptor- and thioimidazol based blockers
Keywords: Abz; ortho-aminobenzoic acid; CAD; cadaverine; DNP; 2,4-dinitrophenyl; tBu; tert-butyl ester; Trt; trityl; Fmoc; Fluorenylmethyloxycarbonyl; DMF; Dimethylformamide; TBTU; O-(Benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; HOBt; Hydroxyb
Novel state-dependent voltage-gated sodium channel modulators, based on marine alkaloids from Agelas sponges
Keywords: Agelas; Marine; Clathrodin; Sodium channel modulator; DMF; N,N-dimethylformamide; DRG; dorsal root ganglia; TBTU; O-benzotriazol-1-yl-N,N,Nâ²,Nâ²-tetramethyluronium tetrafluoroborate; THF; tetrahydrofuran; VGSC; voltage-gated sodium channel;
Proteasome inhibitors for cancer therapy
Keywords: BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DMSO; dimethyl sulfoxide; HMPA; hexamethyl phosphoramide; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; DMF; N,N-dimethyformamide; LDA; lithium diisopropylamide; THF;
The role of endocytosis on the uptake kinetics of luciferin-conjugated cell-penetrating peptides
Keywords: CPP; Cell-penetrating peptide; siRNA; Short interfering ribonucleic acid; EGF; Epidermal growth factor; EGFR; Epidermal growth factor receptor; CME; Clathrin-mediated endocytosis; SPPS; Solid phase peptide synthesis; t-Boc; tert-Butyloxycarbonyl; HOBt; Hy
Synthesis of new chiral xanthone derivatives acting as nerve conduction blockers in the rat sciatic nerve
Keywords: Chiral xanthone derivatives; TBTU; Sciatic nerve; Hypotonic haemolysis; Local anaesthetic-like properties; Action potential blockade
Synthesis, anticonvulsant activity, and neuropathic pain-attenuating activity of N-benzyl 2-amino-2-(hetero)aromatic acetamides
Keywords: AED; antiepileptic drug; ASP; Anticonvulsant Screening Program; B:P; brain-to-plasma; Cbz; carboxybenzyl; DBU; 1,8-diazabicycloundec-7-ene; DIPEA; N,N-diisopropylethylamine; DMTMM; 4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride; ED50;
Substrate specificity of kallikrein-related peptidase 13 activated by salts or glycosaminoglycans and a search for natural substrate candidates
Keywords: Kinin; Protease; Histatins; Kosmotropic salts; Myelin basic protein; Q-EDDP; (glutamyl-N-[ethylenediamine] 2,4-dinitrophenyl); Abz; ortho-aminobenzoic acid; HOBt; N hydroxybenzotriazole; TBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethylaminium tetrafluo
Synthesis and characterization of degradable multivalent cationic lipids with disulfide-bond spacers for gene delivery
Keywords: Boc; tert-butoxycarbonyl; CL; cationic liposome; DEAD; diethylazodicarboxylate; DIEA; N,N-diisopropylethylamine; DLS; dynamic light scattering; DOB; 3,4-di(oleyloxy)benzoic acid; DOPC; 1,2-dioleoyl-sn-glycero-3-phosphatidylcholine; DOTAP; 2,3-dioleoyloxyp
A convergent approach to synthesis of bortezomib: the use of TBTU suppresses racemization in the fragment condensation
Keywords: Bortezomib; PS-341; TBTU; Convergent synthesis; Peptide coupling; Racemization;
Evaluation of new leptin fragments on food intake and body weight of normal rats
Keywords: 2-Cl-Z; 2-chloro-benzyloxycarbonyl; AAA; amino acid analysis; BOP; benzotriazol-1-yl-oxy-tris(dimethylamino) phosphonium hexafluorophosphate; Bzl; benzyl; CD; circular dichroism; CH3CN; acetonitrile; CHO; Formyl; CSF; Cerebrospinal fluid; DCM; dichloromet
Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin αvβ3 and αvβ5 ligands
Keywords: All; allyl; DIC; N,Nâ²-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,N-dimethylformamide; Fmoc; 9H-fluoren-9-yl-methyloxycarbonyl; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; Pbf; 2,2,4,6,7-pe
PS-IIDQ: a supported coupling reagent for efficient and general amide bond formation
Keywords: Coupling reagent; Polymer-supported reagent; Immobilized reagent; IIDQ; Parallel synthesis; Amide bond formation; Amidation; Amide; BOP; benzotriazolyl-N-oxytrisdimethylaminophosphonium hexafluorophosphate; BOP-Cl; N,Nâ²-bis(2-oxo-3-oxazolidinyl)-phosphi
Introduction of the Aib-Pro unit into peptides by means of the 'azirine/oxazolone method' on solid phase
Keywords: α-Aminoisobutyric acid; Azirine/oxazolone method; Peptaibols; Peptide synthesis; Photocleavable linker; Aib; α-aminoisobutyric acid; DIPEA; N,N-diisopropylethylamine; HOBt; 1-hydroxybenzotriazole; PyBOP; (1H-benzotriazol-1-yloxy)tripyrrolidinophosphoniu
Broader cross-reactivity after conjugation of V3 based multiple antigen peptides to HBsAg
Keywords: AA; amino acid; AcOH; acetic acid; Boc; t-butyloxycarbonyl; BSA; bovine serum albumin; DCM; dichoromethane; DIPC; 1,3-diisopropylcarbodiimide; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; HF; hydrogen fluoride; HOBT; 1-hydroxybenzotriazole; P
Explosive properties of 1-hydroxybenzotriazoles
Keywords: 1-Hydroxybenzotriazoles; HOBt; 6-Cl-HOBt; TBTU; HOAt; Explosive properties;
Hemolytic activity of new linear surfactin analogs in relation to their physico-chemical properties
Keywords: CHCA; α-cyano 4-hydroxy cinnamic acid; CMC; critical micellar concentration; DCM; dichloromethane; DIEA; di-isopropyl ethylamine; DMSO; dimethyl sulfoxide; HC50; concentration inducing 50% of hemolysis; HOBt; n-hydroxybenzotriazole; NMP; N-methyl-pyrroli
Potentiation of bradykinin actions by analogues of the bradykinin potentiating nonapeptide BPP9α
Keywords: AA; arachidonic acid; ABA; 4-azidobenzoic acid; ACE; angiotensin I-converting enzyme; Aloc; allyl oxycarbonyl; ASA; 4-azidosalicylic acid; BK; bradykinin; BKR; bradykinin receptor; BKR-B1; bradykinin B1 receptor; BKR-B2; bradykinin B2 receptor; Boc; tert-