دانلود مقالات ISI درباره Tert-Butyloxycarbonyl + ترجمه فارسی

سنتز و بررسی بیولوژیکی آمینوتیازول ها در برابر هیستوپلاسما کپسولاتوم و کریپتوکوک نوورفنس

Synthesis and biological evaluation of aminothiazoles against Histoplasma capsulatum and Cryptococcus neoformans

Keywords: Boc; tert-butyloxycarbonyl; DMAP; 4-dimethylaminopyridine; DCM; dichloromethane; DMF; dimethylformamide; DMSO; dimethyl sulfoxide; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HIV; human immunodeficiency virus; HOBt; hydroxybenzotriazole; HR-ESI;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2018 سفارش ترجمه

چارچوب های آلی فلزات برای تبدیل انرژی خورشیدی توسط کاتالیزور نور سنج

Metal-organic frameworks for solar energy conversion by photoredox catalysis

Keywords: 1,4-biyb; 1,4-bis(imidazol-1-ylmethyl)benzene; 2,6-ndc; 2,6-naphthalenedicarboxylate; 2-cmsnH2; 2-carboxymethylsulfanyl nicotinic acid; 3-dpye; N,N′-bis(3-pyridinecarboxamide)-1,2-ethane; 4,4′-bpy; 4,4′-bipyridine; 4,4′-obb; 4,4′-oxybis(benzoate

دانلود رایگان متن کامل مقاله ISI 33 صفحه سال انتشار : 2018 سفارش ترجمه

سنتز شیمیایی بیورفوگین و آنالوگ

Chemical synthesis of febrifugine and analogues

Keywords: Ac; acetyl; AD-mix; asymmetric dihydroxylation mix; ATP; adenosine triphosphate; Bn; benzyl; Boc; tert-butyloxycarbonyl; Bu; butyl (n-Bu, n-butyl; I; isobutyl; sec-Bu; sec-butyl; t-Bu; tert-butyl); Bz; benzoyl; CAL-B; Candida antartcia lipase-B; CAN; ceri

دانلود رایگان متن کامل مقاله ISI 50 صفحه سال انتشار : 2018 سفارش ترجمه

جداسازی انانیتومرو کروماتوگرافی مایع با استفاده از مبدلهای یونی مبدلهای کربنی بر اساس الکلوئیدهای سینچونا

Liquid chromatographic enantiomer separations applying chiral ion-exchangers based on Cinchona alkaloids

Keywords: Ac; acetyl; AcOH; acetic acid; AccQ; 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate; AIDA; 1-aminoindan-1,5-dicarboxylic acid; aq.; aqueous; BA; butylamine; Boc; tert-butyloxycarbonyl; t-BuCQD; t-butylcarbamoylated quinidine-based CSP; t-BuCQN; t-butylca

دانلود رایگان متن کامل مقاله ISI 78 صفحه سال انتشار : 2018 سفارش ترجمه

مطالعه تطبیقی ​​کلاهک های طراحی مهارکننده های پروتئاز سیتی

A comparative study of warheads for design of cysteine protease inhibitors

Keywords: Boc; tert-butyloxycarbonyl; Cbz; carboxybenzyl; CC50; half maximal cytoxicity concentration; EC50; half maximal effective concentration; EDC; N-(3-Dimethylaminopropyl)-N′-ethylcarbodiimide hydrochloride; IBX; 2-iodoxybenzoic acid; Ki; inhibitory constan

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2017 سفارش ترجمه

گلیکولایپید هورمون آزاد کننده گنادوتروپین جدید با فعالیت ضد انعقادی مستقیم و قدرت گنادوتروپین آزاد

New gonadotropin-releasing hormone glycolipids with direct antiproliferative activity and gonadotropin-releasing potency

Keywords: °C; degrees Celsius; ANOVA; analysis of variance; AUC; area under the curve; BBB; blood brain barrier; Boc; tert-butyloxycarbonyl; C12; 2-amino-d,l-dodecanoic acid; CSS; charcoal stripped serum; DHT; dihydrotestosterone; DMEM; Dulbecco's modified Eagle

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2017 سفارش ترجمه

طراحی، سنتز و ارزیابی آنالوگهای اندومورفین جدید با افزایش ضد انعقادی مرکزی پس از تجویز محیطی

Design, synthesis, and evaluation of new endomorphin analogs with enhanced central antinociception after peripheral administration

Keywords: BBB; blood-brain barrier; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CNS; central nervous system; DAMGO; H-Tyr-d-Ala-Gly-NMePhe-Gly-ol; DCM; dichloromethane; DIEA; N,N-diisopropylethylamine; DOR; δ-opioid receptor; DPDPE; Tyr-c(d

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2015 سفارش ترجمه

فنیل متیون سولفونیل فلوراید، مهار کننده پروتئز سرین، سرکوب نابود کننده نالوکسون منتهی به ترک موش های وابسته به مورفین

Phenylmethanesulfonyl fluoride, a serine protease inhibitor, suppresses naloxone-precipitated withdrawal jumping in morphine-dependent mice

Keywords: Boc-; tert-butyloxycarbonyl; -Bz; benzoyl; Phenylmethanesulfonyl fluoride; Tissue plasminogen activator; Plasmin; Protease activated receptor-1; Withdrawal jumping; Intracerebroventricular injection; Morphine-dependent mice;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2013 سفارش ترجمه

تداوم مایکل دیکمن / واکنش کلاسین ارتو-تلوات - حلال استونتون-وینبر

Tandem Michael-Dieckmann/Claisen reaction of ortho-toluates-the Staunton-Weinreb annulation

Keywords: Ac; acetyl; acac; acetylacetonate; 9-BBN; 9-borabicyclo[3.3.1]nonane; Bn; benzyl; Boc; tert-butyloxycarbonyl; BOM; benzyloxymethyl; brsm; based on recovered starting material; Bz; benzoyl; CAN; ammonium cerium(IV) nitrate; Cbz; benzyloxycarbonyl; CD; circ

دانلود رایگان متن کامل مقاله ISI 27 صفحه سال انتشار : 2013 سفارش ترجمه

Continuous assays for meprin alpha and beta using prolyl tripeptidyl aminopeptidase (PtP) from Porphyromonas gingivalis

Keywords: Astacins; Auxiliary enzyme; Continuous assay; Meprin α/β; Prolyl tripeptidyl aminopeptidase (PtP); AMC; 7-amido-4-methylcoumarin; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DMF; dimethylformamide; DTE; Dithioerythritol; HIC-EBA; hydrophobic inter

دانلود رایگان متن کامل مقاله ISI 24 صفحه سال انتشار : 2018 سفارش ترجمه

Development of novel oxazolo[5,4-d]pyrimidines as competitive CB2 neutral antagonists based on scaffold hopping

Keywords: Cannabinoid; CB2 receptor; Neutral antagonist; oxazolo[5,4-d]pyrimidine; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CHO; Chinese hamster ovary cells; CHO-CB2; Chinese hamster ovary cells expressing CB2 receptors; CHO-WT; Chinese ham

دانلود رایگان متن کامل مقاله ISI 44 صفحه سال انتشار : 2018 سفارش ترجمه

Copper(II) complexes of N3O tripodal ligands appended with pyrene and polyamine groups: Anti-proliferative and nuclease activities

Keywords: Boc; tert-ButylOxyCarbonyl; CT; Charge Transfer; CT DNA; Calf Thymus DeoxyriboNucleic Acid; CV; Cyclic Voltammetry; DFT; Density Functional theory; DMEM; Dulbecco's Modified Eagle's Medium; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; DNA; Deoxyri

دانلود رایگان متن کامل مقاله ISI 59 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, cytotoxic evaluation and target identification of thieno[2,3-d]pyrimidine derivatives with a dithiocarbamate side chain at C2 position

Keywords: Thieno[2,3-d]pyrimidine; Dithiocarbamate; Cytotoxicity; Probe; Target identification; Tubulin; Boc; tert-butyloxycarbonyl; CPT; camptothecin; DMF; N,N-dimethylformamide; DMSO; dimethyl sulphoxide; DSB; DNA double-strand break; EDCI; 1-ethyl-3-(3-dimethyla

دانلود رایگان متن کامل مقاله ISI 70 صفحه سال انتشار : 2018 سفارش ترجمه

Smart polymersomes and hydrogels from polypeptide-based polymer systems through α-amino acid N-carboxyanhydride ring-opening polymerization. From chemistry to biomedical applications

Keywords: ADSCs; adipose derived stem cells; AFM; atomic force microscopy; AG; l/dl-allylglycine; AIBN; 2,2′-azobisisobutyronitrile; Ala; alanine; ATR-FTIR; attenuated total reflectance Fourier transform infrared spectroscopy; ATRP; atom transfer radical polymeri

دانلود رایگان متن کامل مقاله ISI 137 صفحه سال انتشار : 2018 سفارش ترجمه

Design and synthesis of novel bivalent ligands (MOR and DOR) by conjugation of enkephalin analogues with 4-anilidopiperidine derivatives

Keywords: ACN; Acetonitrile; Boc; tert-butyloxycarbonyl; CHO; Chinese hamster ovary; DCM; Dichloromethane; DIPEA; N,N-Diisopropylethylamine; DALEA; [D-Ala2, Leu5] enkephalin amide; DAMGO; [D-Ala2,NMePhe4,Gly5-ol]enkephalin; Dmt; 2,6-dimethyltyrosine; DPDPE; c[D-Pen

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2015 سفارش ترجمه

Design of novel 3,6-diazabicyclo[3.1.1]heptane derivatives with potent and selective affinities for α4β2 neuronal nicotinic acetylcholine receptors

Keywords: 3,6-diazabicyclo[3.1.1]heptanes; Synthesis; α4β2 neuronal nicotinic acetylcholine receptors selectivity; Agonism; Antagonism; CNS; central nervous system; nAChRs; nicotinic acetylcholine receptors; ACh; acetylcholine; GABA; gamma amino butyric acid; Trp

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2015 سفارش ترجمه

Synthesis and biological evaluation of new C-10 substituted dithranol pleiotropic hybrids

Keywords: AAPH; 2,2-azobis(2-amidinopropane) dihydrochloride; Boc; tert-butyloxycarbonyl; DPPH; 1,1-diphenyl-2-picrylhydrazyl radical; ET; single electron transfer; FCC; Flash Column Chromatography; HAT; hydrogen atom transfer; LOX; lipoxygenase; MTT; 3-(4,5-dimeth

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

BN/CC isosterism in borazaronaphthalenes towards phosphodiesterase 10A (PDE10A) inhibitors

Keywords: cAMP; cyclic adenosine monophosphate; cGMP; cyclic guanosine monophosphate; Boc; tert-butyloxycarbonyl; THF; tetrahydrofuran; DMF; dimethylformamide; CPME; cyclopentyl methyl ether; TFA; trifluoroacetic acid; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodi

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

Benserazide, the first allosteric inhibitor of Coxsackievirus B3 3C protease

Keywords: CVB3; Cosxackievirus B3; CVB3 3Cpro; Cosxackievirus B3 3C protease; FRET; fluorescence resonance energy transfer; l-DOPA; levodopa; Boc; tert-butyloxycarbonyl; TFA; trifluoroacetic acid; DCM; dichloromethane; IC50; the half maximal inhibitory concentratio

دانلود رایگان متن کامل مقاله ISI 34 صفحه سال انتشار : 2015 سفارش ترجمه

Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives

Keywords: AcOH; acetic acid; Boc; tert-butyloxycarbonyl; CCL2; chemokine ligand 2; CCR2; chemokine receptor 2; DCE; dichloroethane; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMAP; N,N-dimethylaminopyridine; DMSO; dimethylsulfoxide; INCB3344; N-(2-(((3

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Implications of N-capped urea/thiourea and C-capped 3-(1-piperazinyl)-1,2-benzisothiazole with bridging Gly-Val/Phe-Gly-Val-Pro as therapeutic targets

Keywords: Peptides; Conjugation; Antimicrobial; Antiglycation; Urease inhibition; H+/K+-ATPase activity; ANSA; 1-amino-2-naphthol-4-sulphonic acid; Bis-PNPC; bis(4-nitrophenyl)carbonate; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; EGTA; ethylene glycol tetraa

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2014 سفارش ترجمه

Microwave-assisted guanidinylation in solid phase peptide synthesis: comparison of various reagents

Keywords: Boc; tert-butyloxycarbonyl; Dab; 2,4-diaminobutyric acid; Dap; 2,3-diaminopropionic acid; Dap(g); 3-guanidino-2-aminopropionic acid; DIC; 1,3-diisopropylcarbodiimide; DIEA; diisopropylethylamine; hArg(g); 2,6-diguanidinohexanoic acid; MW; microwave; TBTU;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

[Dmt1]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profile

Keywords: Boc; tert-butyloxycarbonyl; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; Dmp; 2′,6′-dimethylphenylalanine; Dmt; 2′,6′-dimethyltyrosine; [Dmt1]DALDA; H-Dmt-d-Arg-Phe-Lys-NH2; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH; EDT; 1,2-ethanediol; Emp; 2′-ethyl-6â

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

A total synthesis of a highly N-methylated cyclodepsipeptide [2S,3S-Hmp]-aureobasidin L using solid-phase methods

Keywords: Aureobasidin; N-Methylated cyclodepsipeptide; Depsidipeptide; Fmoc-based solid-phase peptide synthesis; Boc; tert-butyloxycarbonyl; BTC; bis-(trichloromethyl)-carbonate; 13C NMR; carbon-13 nuclear magnetic resonance; COSY; correlation spectroscopy; DBU; 1

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that block the transmission of malaria to mosquitoes

Keywords: Plasmodium falciparum; PfCDPK4; PfCDPK1; Pyrazolopyrimidine; Exflagellation; ACT; artemisinin combination therapy; ATP; adenosine triphosphate; Boc; tert-butyloxycarbonyl; CAMKII; Ca2+/calmodulin-dependent protein kinase II; CDPK1; calcium-dependent prote

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2014 سفارش ترجمه

N-terminal guanidinylation of TIPP (Tyr-Tic-Phe-Phe) peptides results in major changes of the opioid activity profile

Keywords: BBB; blood-brain barrier; Boc; tert-butyloxycarbonyl; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DAMGO; H-Tyr-D-Ala-Gly-Phe(NMe)-Gly-ol; DIC; 1,3-diisopropylcarbodiimide; DIPP; H-Dmt-Tic-Phe-Phe-OH; DIPP-NH2; H-Dmt-Tic-Phe-Phe-NH2; DIPP-NH2[Ψ]; H-Dmt-Ti

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2013 سفارش ترجمه

Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists

Keywords: Boc; tert-butyloxycarbonyl; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; DIC; 1,3-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DPDPE; H-Tyr-c[d-Pen-Gly-Phe-D-Pen]OH; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2012 سفارش ترجمه

Anthelmintic PF1022A: stepwise solid-phase synthesis of a cyclodepsipeptide containing N-methyl amino acids

Keywords: ACN; acetonitrile; Boc; tert-butyloxycarbonyl; BOPCl; N,N′-bis(2-oxo-3-oxazolidinyl)phosphinic chloride; DCM; dichloromethane; DEAD; diethylazodicarboxylate; DHP; 3,4-dihydro-2H-pyrane; DIC; N,N′-diisopropylcarbodiimide; DIEA; diisopropylethylamine; D

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2012 سفارش ترجمه

The role of endocytosis on the uptake kinetics of luciferin-conjugated cell-penetrating peptides

Keywords: CPP; Cell-penetrating peptide; siRNA; Short interfering ribonucleic acid; EGF; Epidermal growth factor; EGFR; Epidermal growth factor receptor; CME; Clathrin-mediated endocytosis; SPPS; Solid phase peptide synthesis; t-Boc; tert-Butyloxycarbonyl; HOBt; Hy

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2012 سفارش ترجمه

Interpolymer radical coupling: A toolbox complementary to controlled radical polymerization

Keywords: acac; acetylacetonato; AGET; activator generated by electron transfer; ARGET; activator regenerated by electron transfer; AIBN; azobisisobutyronitrile; AN; acrylonitrile; ATNRC; atom transfer nitroxide radical coupling; ATRC; atom transfer radical couplin

دانلود رایگان متن کامل مقاله ISI 27 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis of a-factor peptide from Saccharomyces cerevisiae and photoactive analogues via Fmoc solid phase methodology

Keywords: Boc; tert-butyloxycarbonyl; Br-BC5; [(E)-(3-((4-bromo-2-methylbut-2-enyloxy)methyl)phenyl)-(phenyl)methanone]; Br-BC10; [(3-(((2E,6E)-8-bromo-2,6-dimethylocta-2,6-dienyloxy)methyl)-phenyl)(phenyl)methanone]; t-Bu; tert-butyl; CLEAR; cross-linked ethoxylat

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2011 سفارش ترجمه

Protection against malaria is conferred by passive transferring rabbit F(ab)2′ antibody fragments, induced by Plasmodium falciparum MSP-1 site-directed designed pseudopeptide-BSA conjugates assessed in a rodent model

Keywords: F(ab)′2; antibody fragment for antigen binding; HABP; high activity binding peptide; ψ-[CH2NH]; reduced amide isoster bond; MHC; major histocompatibility complex; TCR; T-cell receptor; TCC; T-cell clone; APC; antigen presenting cell; CDR; complimentari

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors

Keywords: Histone deacetylase; Ring closing metathesis reaction; Anticancer drugs; Docking studies; 4-aba; 4-allyloxybenzaldehyde; 4-Pea; 4-pentenoic acid; 6-Epa; 6-eptenoic acid; BAP; borane-pyridine complex; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DIC

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2010 سفارش ترجمه

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

Keywords: All; allyl; AgRP; Agouti-related protein; ASIP; agouti-signaling protein; Boc; tert-butyloxycarbonyl; Fmoc; fluorenylmethoxycarbonyl; CH3CN; acetonitrile; Cl-HOBt; 1-hydroxy-6-chlorobenzotriazole; DCM; dichloromethane; DIPEA; diisopropylethylamine; DMF; N

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2010 سفارش ترجمه

Synthesis of orthogonally protected optically pure ketopiperazine, diketopiperazine, ketodiazepane, and 3-aminopyrrolidone building blocks for peptidomimetic combinatorial chemistry

Keywords: 'Around-the-scaffold' drug optimization; Orthogonal protection; Boc/Fmoc strategy; Reductive alkylation; Solid Phase Organic Chemistry (SPOC); Alloc; allyloxycarbonyl; Boc; tert-butyloxycarbonyl; Cbz; benzyloxycarbonyl; DCM; dichloromethane; DKP; dike

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis of chiral threefold and sixfold functionalized macrocyclic imidazole peptides

Keywords: Amino acids; Cyclization; Imidazoles; Macrocycles; Peptidomimetics; Bn; benzyl; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DMF; N,N-dimethylformamide; NMM; N-methylmorpholine; PhtN; phthalimido; PyBOP; benzotriazole-1-yloxytrispyrrolidinophosphoniu

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

Amino acids as selective acylating agents: regioselective N1-acylation of imidazolidin-4-one derivatives of the antimalarial drug primaquine

Keywords: Acylation; Amino acid; Imidazolidin-4-one; Microwave-assisted synthesis; Primaquine; Regioselectivity; Boc; tert-butyloxycarbonyl; BocAAOH; Nα-Boc-protected amino acid; DCCI; N,N′-dicyclohexylcarbodiimide; DCM; dichloromethane; DIEA; N-ethyl-N,N-diisop

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2008 سفارش ترجمه

Structures of cytotoxic bicyclic hexapeptides, RA-XIX, -XX, -XXI, and -XXII, from Rubia cordifolia L.

Keywords: RA-XIX; RA-XX; RA-XXI; RA-XXII; Rubia cordifolia; Bouvardin; Cytotoxicity; Boc; tert-butyloxycarbonyl; Cbz; benzyloxycarbonyl; DIEA; diisopropylethylamine; DMF; N,N-dimethylformamide; DPPA; diphenylphosphoryl azide; EDC·HCl; N-ethyl-N′-(3-dimethylamino

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2008 سفارش ترجمه

Designed modification of partial agonist of ORL1 nociceptin receptor for conversion into highly potent antagonist

Keywords: Boc; tert-butyloxycarbonyl; Bpa; p-benzoyl-l-phenylalanine; BSA; bovine serum albumin; DMF; N,N-dimethylformamide; GPCR; G protein coupled receptor; HBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; HOBt; 1-hydroxybenzotriazo

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2008 سفارش ترجمه

Identification of ETA and ETB binding domains using ET-derived photoprobes

Keywords: Endothelin; ETA; ETB; Photolabeling; Binding domains; ACN; acetonitrile; Boc; tert-butyloxycarbonyl; BOP; benzotriazol-1-yl-oxy-tris(dimethylamino)phosphonium hexafluorophosphate; Bpa; p-benzoyl-phenylalanine; BSA; bovine serum albumine; CHO cells; Chines

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2008 سفارش ترجمه

Segment coupling to a highly hindered N-terminal, alamethicin-related α-aminoisobutyric acid (Aib) residue

Keywords: Aib; α-aminoisobutyric acid residue; Boc; tert-butyloxycarbonyl; DCC; dicyclohexylcarbodiimide; DB(DMAP); 2,6-di-t-butyl-4-(dimethylamino)pyridine; DCM; dichloromethane; DIC; N,N′-diisopropylcarbodiimide; DIEA; N,N-diisopropylethylamine; DMF; N,N-dimet

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2007 سفارش ترجمه

Effect of the antimicrobial peptide gomesin against different life stages of Plasmodium spp.

Keywords: Antimicrobial peptide; Gomesin; Malaria; Mosquito; Ookinete; Oocyst; Exflagellation; GFP; green fluorescent protein; P. berghei; Plasmodium berghei; P. falciparum; Plasmodium falciparum; An. stephensi; Anopheles stephensi; RPMI-1640; Roswell Park Memorial

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2007 سفارش ترجمه

Synthesis and evaluation of chloromethyl sulfoxides as a new class of selective irreversible cysteine protease inhibitors

Keywords: ESI-MS; electrospray ionization mass spectrometry; Boc; tert-butyloxycarbonyl; BOP; (1H-benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DTT, dithiothreitol; DiPEA; N,N-diisopropylethylamine

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2007 سفارش ترجمه

'Bis-ornithine' (2,2-bis(aminopropyl)glycine): a new tetravalent template for assembling different functional peptides

Keywords: Ac; acetyl; Alloc; allyloxycarbonyl; bisOrn; bis-ornithine; Boc; tert-butyloxycarbonyl; Cbz; benzyloxycarbonyl; 2-BrCbz; 2-bromobenzyloxycarbonyl; 2-ClCbz; 2-chloro benzyloxycarbonyl; DIEA; diisopropylethylamine; DMAP; N,N-dimethylaminopyridine; DMF; N,N-

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2006 سفارش ترجمه

Synthetic applications of fluorous solid-phase extraction (F-SPE)

Keywords: Fluorous; Light fluorous; Fluorous silica gel; Fluorous solid-phase extraction (F-SPE); Reverse F-SPE; Plate-to-plate SPE; Parallel synthesis; High-throughput synthesis; Solution-phase synthesis; Separation; Reagents; Reactants; Catalysts; Chiral auxiliar

دانلود رایگان متن کامل مقاله ISI 29 صفحه سال انتشار : 2006 سفارش ترجمه

Synthesis of amino- and diaminoconduritols and their applications

Keywords: Conduritols; Conduramines; Diaminoconduritols; Asymmetric synthesis; Ac; acetyl; aq; aqueous; AIBN; 2,2′-azobis(isobutyronitrile); Bn; benzyl; Boc; tert-butyloxycarbonyl; n-Bu; n-butyl; s-Bu; sec-butyl; t-Bu; tert-butyl; Bz; benzoyl; CAN; ceric ammonium

دانلود رایگان متن کامل مقاله ISI 36 صفحه سال انتشار : 2006 سفارش ترجمه

Importance of the central region of lamprey gonadotropin-releasing hormone III in the inhibition of breast cancer cell growth

Keywords: lGnRH-III; lamprey gonadotropin-releasing hormone III; GnRH; gonadotropin-releasing hormone; Fmoc; 9-fluorenylmethoxycarbonyl; tBu; tert-butyl; Trt; trytil; Boc; tert-butyloxycarbonyl; HOBt; 1-hydroxybenzotriazole; HBTU; benzotriazolyl-tetramethyluronium

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2005 سفارش ترجمه

Differential effects of N-peptidyl-O-acyl hydroxylamines on dynorphin-induced antinociception in the mouse capsaicin test

Keywords: Boc-; tert-butyloxycarbonyl; Z-; benzyloxycarbonyl; Bz; benzoyl; Dynorphins; Cysteine proteases; N-peptidyl-O-acyl hydroxylamines; Capsaicin test; Intrathecal administration; Mouse;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2005 سفارش ترجمه

Specific negative charges in cysteine protease isoforms of Leishmaniamexicana are highly influential on the substrate binding and hydrolysis

Keywords: Abz; ortho-amino-benzoyl; AMC; 7-amino-4-methylcoumarin; t-Boc; tert-butyloxycarbonyl; DMF; dimethylformamide; DTT; dithiothreitol; EDDnp; N-[2,4-dinitrophenyl]-ethylenediamine; EDTA; ethylenediaminetetraacetic acid; FRET; fluorescence resonance energy tr

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2005 سفارش ترجمه

Synthesis and evaluation of eight-membered cyclic pseudo-dipeptides

Keywords: Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DIBAL; diisobutyl aluminium hydride; DIEA; diisopropyl ethyl amine; EtOAc; ethyl acetate; HATU; O-(7-azabenzotriazol-1-yl)-N,N,N′,N′-tetra-methyluronium hexafluorophosphate; HOBt; hydroxybenzotriazole;

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2005 سفارش ترجمه