Keywords: AZT; azidothymidine; DSB; double-strand break; dsDNA; double-strand DNA; gDNA; gapped DNA; HR; homologous recombination; HU; hydroxyurea; indel; insertion/deletion; IR; inverted repeats; QP; quasipalindrome; QPM; quasipalindrome-associated mutagenesis; SC
مقالات ISI (ترجمه نشده)
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Keywords: ABC; ATP-binding cassette; AP; absorption potential; API; active pharmaceutical ingredient; ATP; adenosine triphosphate; AZT; azidothymidine; BA/BE; bioavailability/bioequivalence; BCRP; breast cancer resistance protein; BCS; biopharmaceutical classificat
Keywords: meta-analysis; nontuberculous mycobacteria; systematic review; treatment outcome; 6MWT; 6-min walk test; AMX; amikacin; ATS; American Thoracic Society; AZT; azithromycin; BTS; British Thoracic Society; CLARI; clarithromycin; IDSA; Infectious Diseases Soci
Keywords: AIDS; acquired immune deficiency syndrome; ALV; avian leukosis virus; AMV; avian myeloblastosis virus; APOBEC; apolipoprotein B mRNA-editing enzyme-catalytic polypeptide-like; ASLV; avian sarcoma leukosis virus; AZT; 3â² -azido-3â² -deoxythymidine; BIV;
Keywords: 3TC; Lamivudine; ABC; Abacavir; ARV; Antiretroviral; ATV; Atazanavir; AZT; Zidovudine; d4T; Stavudine; DRV; Darunavir; EFV; Efavirenz; FTC; Emtricitabine; L&D; Labor and delivery; LOQ; Limit of quantification; LPV; Lopinavir; M8; NFV hydroxy-tert-butylami
Keywords: Carboranyl pyrimidine nucleoside analog; Thymidine kinase 1 (TK1); Carborane; Boron neutron capture therapy (BNCT); 3CTAs; 3-carboranyl thymidine analogs; 10B; boron-10; ATCC; American type culture collection; AZT; zidovudine; B; boron; BNCT; boron neutro
Keywords: AIM2; absent in melanoma 2; AP-1; activating protein-1; APOBEC; apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like; AZT; azidothymidine; CCCR5; C-C chemokine receptor type 5; CDK1; cyclin-dependent kinase 1; CXCR4; C-X-C chemokine receptor t
Keywords: Aβ peptide; Beta Amyloid peptide; AD; Alzheimer Disease; AFM; Atomic Force Microscopy; AMP; Antimicrobial Peptide; ATR-FTIR; Attenuated Total Reflection Fourier Transform Infrared Spectroscopy; AZT; Azithromycin; BAM; Brewster Angle Microscopy; BM; Big M
Keywords: AA; arachidonic acid; ADP; adenosine diphosphate; AIF; apoptosis-inducing factor; AMPK; AMP-activated protein kinase; ANT; adenine nucleotide translocase; Apaf-1; apoptotic protease activating factor-1; ATP; adenosine triphosphate; ATP-ase; ATP synthase;
Keywords: MAFP (methyl arachidonyl fluoro phosphonate); Progesterone; BMP (bismonoacylglycerophosphate); Sterol transporter NPC-1; PLRP2 (pancreatic lipase-related protein 2); Desmosterol; Cholesterol epoxide; MAFP; methyl arachidonyl fluoro phosphonate; PROG; prog
Keywords: SOD; superoxide dismutase; GPx; glutathione peroxidases; CAT; catalase; GSH; reduced glutathione; GSSG; oxidized glutathione; GST; glutathione S-transferase; GR; glutathione reductase; mtDNA; mitochondrial DNA; DOX; doxorubicin; APAP; acetaminophen; NAPQI
Keywords: nontuberculous mycobacteria; pulmonary disease; treatment outcome; AMX; amikacin; ATS; American Thoracic Society; AZT; azithromycin; CFZ; clofazimine; Clari; clarithromycin; LAI; liposomal AMX for inhalation; MAC; Mycobacterium avium complex; MAC-PD; MAC
Diagnosis and management of neuromyelitis optica spectrum disorders - An update
Keywords: AQP4; aquaporin-4; AQP4 IgG; immunoglobulin G against aquaporin-4; ARR; Annualized Relapse Rates; AZT; azathioprine; BBB; blood-brain barrier; CNS; central nervous system; EDSS; Expanded Disability Status Scale; GFAP; glial fibrillary acid protein; ICAM1;
Spread of multidrug-resistant Escherichia coli harboring integron via swine farm waste water treatment plant
Keywords: AMP; ampicillin; AMC; amoxicillin/clavulanic acid; CZ; cefazolin; FOX; cefoxitin; CTX; cefotaxime; CAZ; ceftazidime; FEP; cefepime; AZT; aztreonam; AK; amikacin; CIP; ciprofloxacin; GN; gentamicin; MDR; multi-drug resistance; ESBL; extended-spectrum β-la
Structural patterns of the human ABCC4/MRP4 exporter in lipid bilayers rationalize clinically observed polymorphisms
Keywords: 6-MP; 6-mercaptopurine; ABC; ATP-binding cassette; ADV; adefovir; AZT; azidothymidine; BLOSUM; blocks substitution matrix; CFTR; cystic fibrosis transmembrane conductance regulator; Chol; cholesterol; cryo-EM; cryo-electronic microscopy; DMAV; dimethylars
Recomendaciones de GESIDA/PETHEMA sobre el diagnóstico y tratamiento de los linfomas en pacientes infectados por el virus de la inmunodeficiencia humana
Keywords: Linfoma no hodgkiniano; Linfoma de Hodgkin; VIH; Sida; Tratamiento antirretroviral; Non-Hodgkin's lymphoma; Hodgkin's lymphoma; HIV; AIDS; Antiretroviral therapy; ABC; abacavir; ABVD; adriamicina, bleomicina, vinblastina y dacarbazina; Ara-C; arabinósido
GESIDA/PETHEMA recommendations on the diagnosis and treatment of lymphomas in patients infected by the human immunodeficiency virus
Keywords: ABC; abacavir; ABVD; adriamycin, bleomycin, vinblastine and dacarbazine; Ara-C; cytosine arabinoside; AZT; zidovudine; BCNU; carmustine; BEACOPP; bleomycin, etoposide, adriamycin, cyclophosphamide, vincristine, procarbazine and prednisone; CDC; Centers fo
Safety profile of AZT derivatives: Organoselenium moieties confer different cytotoxic responses in fresh human erythrocytes during in vitro exposures
Keywords: AZT; 3â²-deoxythymidine or zidovudine; SZ1; 5â²-(4-chlorophenylseleno)zidovudine; SZ2; 5â²-(Phenylseleno)zidovudine; SZ3; 5â²-(4-methylphenylseleno)zidovudine; Se; Selenium; HIV; human immunodeficiency virus; AIDS; Acquired immunodeficiency syndrome;
Effects of Fuzheng Paidu tablet immunization on AIDS BALB/c mice
Keywords: Friend murine leukemia virus; BALB/c mice; AZT;
Dual inhibitors of the human blood-brain barrier drug efflux transporters P-glycoprotein and ABCG2 based on the antiviral azidothymidine
Keywords: Blood-brain barrier; P-glycoprotein; ABCG2; AZT; Inhibition;
Original ArticleWhole body clonality analysis in an aggressive STLV-1 associated leukemia (ATLL) reveals an unexpected clonal complexity
Keywords: STLV-1; Retrovirus; Leukemia/Lymphoma; Therapy; Clonality; LM-PCR; ATLL; Adult T cell Leukemia/Lymphoma; AZT; azidothymidine; CUIS; common unique integration site; HAM/TSP; Associated Myelopathy/Tropical Spastic Paraparesis; HTLV-1; Human T-Lymphotropic V
The Ca2+/CaMKK2 axis mediates the telbivudine induced upregulation of creatine kinase: Implications for mechanism of antiviral nucleoside analogs' side effect
Keywords: LdT; Telbivudine; HBV; hepatitis B virus; CHB; chronic Hepatitis B; CK; creatine kinase; HSKMCs; human skeletal muscle cells; SOD; superoxide dismutase; MDA; malondialdehyde; LPO; lipid peroxide; ROS; reactive oxygen species; CaMKK2; calmodulin-dependent
Azidothymidine-triphosphate impairs mitochondrial dynamics by disrupting the quality control system
Keywords: ATP; adenosine triphosphate; AZT; 3ê-azido-3ê-deoxythymidine; AZT-DP; AZT diphosphate; AZT-MP; AZT monophosphate; AZT-TP; AZT-triphosphate; calcein-AM; calcein acetoxymethyl ester; cDNA; complementary DNA; DHE; dihydroethidium; DMEM; Dulbecco's Modifi
Synthesis and cytotoxic evaluation of novel indenoisoquinoline-substituted triazole hybrids
Keywords: Indenoisoquinolines; Triazole; AZT; Hybrids; Cytotoxic agents
Acrolein enhances epigenetic modifications, FasL expression and hepatocyte toxicity induced by anti-HIV drug Zidovudine
Keywords: AZT; azidothymidine or Zidovudine; ACR; acrolein; ART; antiretroviral therapy; ChIP; chromatin immunoprecipitation; FasL; Fas ligand; H3K9Ac; histone 3 lysine 9 acetylation; H3K4Me3; histone 3 lysine 4 trimethylation; RNA Pol II; RNA polymerase II; TF; tr
2-hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4
Keywords: HIV-1 integrase; Two-metal binding pharmacophore; Antiretroviral; 2-hydroxyisoquinoline-1,3(2H,4H)-diones; AZT; azidothymidine; CPE; cytopathic effect; CYP; cytochrome P450; FC; fold-change in EC50 relative to wild-type strain of HIV-1; FDA; food and drug
Neutralization Takes Precedence Over IgG or IgA Isotype-related Functions in Mucosal HIV-1 Antibody-mediated Protection
Keywords: ADCC; Antibody-dependent cell-mediated cytotoxicity; ARV; Anti-retroviral; AZT; Zidovudine; bnAb; Broadly neutralizing antibody; CD4bs; CD4 binding site; dIgA; Dimeric IgA; FcRn; Neonatal Fc receptor; GalCer; Galactosyl ceramide; GI; Gastrointestinal; GU;
Tetrahedron report 1111Synthesis routes to anti-HIV drugs
Keywords: AIDS; Anti-HIV; Synthesis; FDA; Enantiomeric excess; ABC; abacavir; AIBN; azobisisobutyronitrile; AIDS; acquired immune deficiency syndrome; ARV; antiretroviral; AZT; 3â²-azido-3â²-deoxythymidine; CAPIC; 2-chloro-3-amino-4-picoline; CD4; cluster of diff
SiO2 nanoparticles as platform for delivery of 3′-triazole analogues of AZT-triphosphate into cells
Keywords: SiO2 nanoparticles; Delivery of triphosphate into cells; Substrate properties; 3′-Triazole derivatives of thymidine triphosphates; AZT; ‘Click’ chemistry
Characterization of the enhanced apoptotic response to azidothymidine by pharmacological inhibition of NF-kB
Keywords: Apoptosis; AZT; Bcl-2; Chemotherapy; NF-kB;
Synthesis and cytotoxic evaluation of novel amide-triazole-linked triterpenoid-AZT conjugates
Keywords: Triterpenoids; AZT; Hybrids; Cytotoxic agents;
Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2â²,3â²-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity
Keywords: Pro-nucleotides; AZT; 2â²,3â²-dideoxynucleosides; H-phosphonates; Phosphoramidates; Heteroaryl amines; Anti-HIV; Lipophilicity;
Synthesis and cytotoxic evaluation of novel ester-triazole-linked triterpenoid–AZT conjugates
Keywords: Triterpenoids; AZT; Hybrids; Cytotoxic agents
Synthesis and evaluation of sulfonylethyl-containing phosphotriesters of 3â²-azido-3â²-deoxythymidine as anticancer prodrugs
Keywords: AZT; AZT monophosphate; Sulfonylethyl; Phosphotriester; Pronucleotide; β-Elimination; Prodrugs;
Comparative analysis of genetic toxicity of antiretroviral combinations in somatic cells of Drosophila melanogaster
Keywords: NRTI; nucleoside reverse transcriptase inhibitor; HAART; highly active antiviral therapy; AZT; 3â²-azido-3â²-deoxythymidine; ddI; 2â²,3â²-dideoxyinosine; 3TC; [â] 2â²-deoxy-3â²-thiacytidine; d4T; 3â²-deoxy-2â²,3â²-didehydrothymidine; SMART; som
A protein ballet around the viral genome orchestrated by HIV-1 reverse transcriptase leads to an architectural switch: From nucleocapsid-condensed RNA to Vpr-bridged DNA
Keywords: (â) SSDNA; minus-strand strong-stop DNA; (â) ss-DNA; minus-strand single-stranded DNA; +SSDNA; plus-strand strong-stop DNA; AFM; atomic force microscopy; AZT; azidothymidine; BAF; barrier-to-autointegration factor; bp; base-pairs; CA; capsid; cFlap; c
Bifunctional inhibition of HIV-1 reverse transcriptase: A first step in designing a bifunctional triphosphate
Keywords: HIV-1; human immunodeficiency virus type 1; RT; reverse transcriptase; NRTIs; nucleoside RT inhibitors; NNRTIs; nonnucleoside RT inhibitors; dNTP; deoxynucleoside triphosphate; dNMP; 3â²-deoxynucleoside monophosphate; PPi; pyrophosphate; AZT; β-d-(+)-3â
Expression of P-glycoprotein and multidrug resistance-associated protein on human brain-microvascular endothelial cells with electromagnetic stimulation
Keywords: AZT; azidothymidine; BBB; blood-brain barrier; EMF; electromagnetic field; HA; human astrocyte; HBMEC; human brain-microvascular endothelial cell; HBMEC/HA; HA-regulated HBMECs; MRP; multidrug resistance-associated protein; P-gp; P-glycoprotein; SQV; sa
HIV-1 mother-to-child transmission and drug resistance among Brazilian pregnant women with high access to diagnosis and prophylactic measures
Keywords: HIV-1; human immunodeficiency virus type 1; MTCT; mother-to-child transmission; ARV; antiretroviral; PPPW; Program for the Protection of Pregnant Women; HAART; highly active antiretroviral therapy; NRTI; nucleoside reverse-transcriptase inhibitors; NNRTI;
High frequency of antiviral drug resistance and non-B subtypes in HIV-1 patients failing antiviral therapy in Cuba
Keywords: ART; antiretroviral therapy; CI; confidence interval; NRTI; nucleoside reverse transcriptase inhibitor; NNRTI; non-nucleoside RTI; PI; protease inhibitor; FCR; full-class resistance; CRF; circulating recombinant form; HIV; human immunodeficiency virus; MD
Old plants newly discovered: Cassia sieberiana D.C. and Cassia abbreviata Oliv. Oliv. root extracts inhibit in vitro HIV-1c replication in peripheral blood mononuclear cells (PBMCs) by different modes of action
Keywords: AIDS; Acquired Immunodeficiency Syndrome; ARVs; anti-retroviral drugs; AZT; azidothymidine; HIV; human immunodeficiency virus; STI; sexually transmitted infections; HIV-1c (MJ4); Antiviral; Entry inhibitor; Traditional medicine; Botswana;
A pyrophosphatase activity associated with purified HIV-1 particles
Keywords: Retrovirus; Reverse transcription; Resistance; Excision; Pyrophosphorolysis; HIV-1; human immunodeficiency virus type 1; RT; reverse transcriptase; AZT; 3â²-azido-3â²-deoxythymidine, zidovudine; d4T; 2â²-3â²-didehydro-2â²-3â²-dideoxythymidine; TAM;
Diverse combinatorial design, synthesis and in vitro evaluation of new HEPT analogues as potential non-nucleoside HIV-1 reverse transcription inhibitors
Keywords: Combinatorial design; Diversity selection HIV-1; NNRTIs HEPT; Antiviral activity; RHHROCXXJZOAGP-UHFFFAOYSA-N; KMCGFILCIRJEHJ-UHFFFAOYSA-N; XXFUGXPQNOZBIR-UHFFFAOYSA-N; OFOHDLYVTOWSFB-UHFFFAOYSA-N; PWAKKEPZIWJVBA-UHFFFAOYSA-N; DTCUBSJAMNGQFU-UHFFFAOYSA-N;
Synthesis and anti-HIV activities of bis-(cycloSaligenyl) pronucleotides derivatives of 3â²-fluoro-3â²-deoxythymidine and 3â²-azido-3â²-deoxythymidine
Keywords: Nucleosides; Bis-(cycloSaligenyl); AZT; FLT; Anti-HIV;
Synthesis of 3′-azido-3′-deoxythymidine (AZT)—Cinchona alkaloid conjugates via click chemistry: Toward novel fluorescent markers and cytostatic agents
Keywords: Nucleosides; AZT; Cinchona alkaloids; Click chemistry; Conjugation
Enhancement of Zidovudine Transfer to Molt-4 Cells, a Human T-Cell Model, by Dehydroepiandrosterone Sulfate
Keywords: antiretroviral drug; permeation enhancers; AZT; transporter; drug targeting; distribution; drug interactions
Interferon regulatory factor-4 activates IL-2 and IL-4 promoters in cooperation with c-Rel
Keywords: IRF-4; interferon regulatory factor-4; IFN; interferon; ISRE; IFN-stimulated response element; TCR; T-cell receptor; PMA; phorbol-12-myristate-13-acetate; I; Ionomycin; TAP; tandem affinity purification; IL-4; interleukin-4; HTLV-1; human adult T-cell leu
Highly active antiretroviral therapy drug combination induces oxidative stress and mitochondrial dysfunction in immortalized human blood-brain barrier endothelial cells
Keywords: AZT; 3â²-azido-2â²,3â²-deoxythymidine; BBB; blood-brain barrier; IDV; indinavir; HIV-1; human immunodeficiency virus; HAND; HIV-1-associated neurocognitive disorders; HAART; highly active antiretroviral therapy; GSH; glutathione; MDA; malondialdehyde
Protein overexpression following lentiviral infection of primary mature neutrophils is due to pseudotransduction
Keywords: Lentiviral gene transfer; Neutrophil; Pseudotransduction; AZT; 3â²-azido-3â²-deoxythymidine; CHX; cycloheximide; DAPK2; death-associated protein kinase 2; FCS; fetal calf serum; GM-CSF; granulocyte/macrophage colony-stimulating factor; GFP; green fluore
Moving to tolerance: Clinical application of T regulatory cells
Keywords: APC; antigen presenting cell; ATG; anti thymocyte globulin; aTreg; adaptive T regulatory cell; AZT; 3â²-azido-3â²-deoxythymidine; CNI; calcineurin inhibitor; CyA; cyclosporin A; DC; dendiric cell; DST; donor specific transfusion; GVHD; graft versus host