Keywords: بنزن سولفونامید; Anticancer; Apoptosis; Benzenesulfonamide; Isatin; Tumor-associated hCA IX and XII;
مقالات ISI بنزن سولفونامید (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: بنزن سولفونامید; Fluorescent thermal shift assay; Benzenesulfonamide; Carbonic anhydrase; Inhibitor; Structure-thermodynamics relationships; X-ray crystallography;
Keywords: بنزن سولفونامید; Phenothiazine; Benzenesulfonamide; Anticancer; Aromatase inhibitors; Apoptosis;
Keywords: بنزن سولفونامید; Carbonic anhydrase inhibitors; Isatin; Benzenesulfonamide; Anticancer; Apoptosis;
Dual EGFR/HER2 inhibitors and apoptosis inducers: New benzo[g]quinazoline derivatives bearing benzenesulfonamide as anticancer and radiosensitizers
Keywords: بنزن سولفونامید; Benzo[g]quinazoline; Acetamide; Benzenesulfonamide; EGFR; HER2;
Design and synthesis of novel benzenesulfonamide containing 1,2,3-triazoles as potent human carbonic anhydrase isoforms I, II, IV and IX inhibitors
Keywords: بنزن سولفونامید; 1,2,3-Triazoles; Benzenesulfonamide; Carbonic anhydrase isoforms I, II, IV, IX; Acetazolamide; Enaminones;
Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors
Keywords: بنزن سولفونامید; Carbonic anhydrase inhibitors; Isoforms I, II, IV, IX; Benzenesulfonamide; 1,2,3-Triazole; CA; Carbonic anhydrase; hCA; human carbonic anhydrase; CAIs; Carbonic anhydrase inhibitors; AAZ; Acetazolamide; Ki; Inhibition constant; nM; nanomolar; μM; micromo
Synthesis of novel isoindoline-1,3-dione-based oximes and benzenesulfonamide hydrazones as selective inhibitors of the tumor-associated carbonic anhydrase IX
Keywords: بنزن سولفونامید; Isoindoline-1,3-dione; Oxime; Hydrazone; Benzenesulfonamide; Carbonic anhydrase inhibition; Carbonic anhydrase IX; Anti-tumor;
Synthesis and biological evaluation of cyclic imides incorporating benzenesulfonamide moieties as carbonic anhydrase I, II, IV and IX inhibitors
Keywords: بنزن سولفونامید; Cyclic imide; Benzenesulfonamide; Carbonic anhydrase; Inhibitor;
Synthesis and carbonic anhydrase inhibition of polycyclic imides incorporating N-benzenesulfonamide moieties
Keywords: بنزن سولفونامید; Polycyclic imides; Benzenesulfonamide; Carbonic anhydrase; Inhibitor;
Synthesis, characterization and antimicrobial activity of some new 4-(4-(2-isonicotinoylhydrazinyl)-6-((aryl)amino)-1,3,5-triazin-2-ylamino)-N-(pyrimidin-2-yl) benzenesulfonamides
Keywords: بنزن سولفونامید; 1,3,5-Triazine; Pyrimidine; Isoniazid; Benzenesulfonamide; Antimicrobial activity; MIC;
Synthesis and molecular docking against dihydrofolate reductase of novel pyridin-N-ethyl-N-methylbenzenesulfonamides as efficient anticancer and antimicrobial agents
Keywords: بنزن سولفونامید; Benzenesulfonamide; Pyridine; Anticancer; Antimicrobial; Molecular docking;
Discovery of non-zwitterionic aryl sulfonamides as Nav1.7 inhibitors with efficacy in preclinical behavioral models and translational measures of nociceptive neuron activation
Keywords: بنزن سولفونامید; Benzenesulfonamide; Nav1.7 inhibitor; Membrane permeability; Neuropathic and inflammatory pain; Translational electromyogram; Nociceptive flexion reflex (NFR);
Discovery of Benzo[g]quinazolin benzenesulfonamide derivatives as dual EGFR/HER2 inhibitors
Keywords: بنزن سولفونامید; Benzo[g]quinazolin; Acetamide; Benzenesulfonamide; EGFR; HER2;
Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors
Keywords: بنزن سولفونامید; Imidazothiadiazoles; Thiazolotriazoles; Benzenesulfonamide; Carbonic anhydrase isoforms I, II, IX, XII; Acetazolamide;
Synthesis, characterization and antimicrobial activity of some novel 4-(4-(arylamino)-6-(piperidin-1-yl)-1,3,5-triazine-2-ylamino)-N-(pyrimidin-2-yl)benzenesulfonamides
Keywords: بنزن سولفونامید; Antimicrobial activity; Benzenesulfonamide; Cyanuric chloride; Piperidine; Pyrimidine; 1,3,5-Triazine;
Improvement of solid material for affinity resins by application of long PEG spacers to capture the whole target complex of FK506
Keywords: بنزن سولفونامید; Affinity resins; PEG; Target identification; Carbonic anhydrase II; FKBP12; Benzenesulfonamide; FK506; Calcineurin; Target complex
The discovery of benzenesulfonamide-based potent and selective inhibitors of voltage-gated sodium channel Nav1.7
Keywords: بنزن سولفونامید; Benzenesulfonamide; Sodium channel; Nav1.7; Pain
4-Functionalized 1,3-diarylpyrazoles bearing benzenesulfonamide moiety as selective potent inhibitors of the tumor associated carbonic anhydrase isoforms IX and XII
Keywords: بنزن سولفونامید; Pyrazole; Benzenesulfonamide; Carbonic anhydrase isoforms I, II, IX, XII; Acetazolamide
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties
Keywords: بنزن سولفونامید; CA; carbonic anhydrase; hCA; human carbonic anhydrase; CAI; carbonic anhydrase inhibitor; SAR; structure-activity relationship; Zn; zinc; AZM; acetazolamide; MZA; methazolamide; EZA; ethoxzolamide; DCP; dibromophenamide; DZA; dorzolamide; BRZ; brinzolam
Benzenesulfonamide bearing 1,2,4-triazole scaffolds as potent inhibitors of tumor associated carbonic anhydrase isoforms hCA IX and hCA XII
Keywords: بنزن سولفونامید; Triazoles; Benzenesulfonamide; Carbonic anhydrase isoforms I, II, IX, XII; Acetazolamide
Molecular design, synthesis and biological evaluation of cyclic imides bearing benzenesulfonamide fragment as potential COX-2 inhibitors. Part 2
Keywords: بنزن سولفونامید; Cyclic imides; Benzenesulfonamide; COX-2 inhibitors; Anti-inflammatory activities; Molecular docking;
Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety
Keywords: بنزن سولفونامید; Human carbonic anhydrase inhibitors; Benzenesulfonamide; 4,5,6,7-Tetrachloro-1,3-dioxoisoindolin-2-yl benzenesulfonamide; Structure-activity relationship;
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety
Keywords: بنزن سولفونامید; CA; carbonic anhydrase; hCA; human carbonic anhydrase; CAI; carbonic anhydrase inhibitor; SAR; structure-activity relationship; Zn; zinc; AZM; acetazolamide; MZA; methazolamide; EZA; ethoxzolamide; DCP; dibromophenamide; DZA; dorzolamide; BRZ; brinzolam
Structural effect of phenyl ring compared to thiadiazole based adamantyl-sulfonamides on carbonic anhydrase inhibition
Keywords: بنزن سولفونامید; Carbonic anhydrase; Benzenesulfonamide; Adamantyl; X-ray crystallography; Isoform-selective inhibitor
Design and synthesis of novel 4-(4-oxo-2-arylthiazolidin-3-yl)benzenesulfonamides as selective inhibitors of carbonic anhydrase IX over I and II with potential anticancer activity
Keywords: بنزن سولفونامید; Benzenesulfonamide; Thiazolidin-4-one; Carbonic anhydrase IX; Anticancer; Cell lines; Daltion's lymphoma ascitesCA, carbonic anhydrase; HIF-1, hypoxia-inducible transcription factor-1; DLA, Dalton's lymphoma ascites; DCC, N,N-dicyclohexylcarbodiimide; MTT
Superacid synthesis of halogen containing N-substituted-4-aminobenzene sulfonamides: New selective tumor-associated carbonic anhydrase inhibitors
Keywords: بنزن سولفونامید; Hypoxic tumors; Superacid; Fluorine chemistry; Benzenesulfonamide; Halogen effect
Enthalpies of combustion and formation of benzenesulfonamide and some of its derivatives
Keywords: بنزن سولفونامید; Rotating-bomb calorimeter; Combustion energies; Formation enthalpies; Benzenesulfonamide; o-Toluenesulfonamide; p-Toluenesulfonamide; 2-Aminobenzenesulfonamide; 4-Aminobenzenesulfonamide
Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells
Keywords: بنزن سولفونامید; Kynurenine; Tryptophan; Indoleamine 2,3-dioxygenase (IDO); Signal transducer and activator of transcription 1 (STAT1); Benzenesulfonamide;
Benzenesulfonamide attenuates monocrotaline-induced pulmonary arterial hypertension in a rat model
Keywords: بنزن سولفونامید; Monocrotaline; Pulmonary arterial hypertension; LASSBio-965; (N-[2-(34-dimethoxyphenyl) ethyl]-; benzenesulfonamide; Phosphodiesterase; Rhokinase;
Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures (II)
Keywords: بنزن سولفونامید; Carbonic anhydrase; Benzenesulfonamide; Dispersion interaction; Fragment molecular orbital (FMO); Hammett Ï; Hydrophobic constant Ï; Linear expression by representative energy terms (LERE); Quantitative structure-activity relationship (QSAR);
Synthesis and biological evaluation of some 4-functionalized-pyrazoles as antimicrobial agents
Keywords: بنزن سولفونامید; 4-Functionalizedpyrazoles; Carboxylic acids; Carbothioamides; Antibacterial activity; Antifungal activity; Benzenesulfonamide
Structure-activity relationships of various amino-hydroxy-benzenesulfonic acids and sulfonamides as tyrosinase substrates
Keywords: بنزن سولفونامید; Tyrosinase activity; Active site; Benzenesulfonic acid; Benzenesulfonamide; Phenoxazinone;
Selective elution of target protein from affinity resins by a simple reductant with a thiol group
Keywords: بنزن سولفونامید; Affinity resins; Target identification; Carbonic anhydrase II; FKBP12; Benzenesulfonamide; FK506; 2-Mercaptethanol (2ME); AquaFirmus
New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors
Keywords: بنزن سولفونامید; BSA; benzenesulfonamide; HPM; hydroxypyrimidinone; CA; carbonic anhydrase; MMP; matrix metalloproteinase; ZBG; zinc-binding group; HA; hydroxamic acid; Hydroxypyrimidinones; Carbonic anhydrase inhibitors; Sulfonamides; MMP inhibitors;
4-[N-(Substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII
Keywords: بنزن سولفونامید; Carbonic anhydrase isozymes I, II, VII, and XIII; Isothermal titration calorimetry; Thermal shift assay; ThermoFluor®; Benzenesulfonamide; Pyrimidine
Carbonic anhydrase inhibitors: Two-prong versus mono-prong inhibitors of isoforms I, II, IX, and XII exemplified by photochromic cis-1,2-α-dithienylethene derivatives
Keywords: بنزن سولفونامید; Carbonic anhydrase; Isozymes; Tumor-associated enzymes; Benzenesulfonamide; Photochromism; 1,2-Dithienylethene
Selective COX-2 inhibitors. Part 2: Synthesis and biological evaluation of 4-benzylideneamino- and 4-phenyliminomethyl-benzenesulfonamides
Keywords: بنزن سولفونامید; Selective COX-2 inhibitors; Anti-inflammatory; Benzenesulfonamide; Benzylideneamino; Phenyliminomethyl; Resveratrol; Isosterism; SAR
A versatile method of identifying specific binding proteins on affinity resins
Keywords: بنزن سولفونامید; Affinity resins; Competition method; Target identification; Nonspecific binding proteins; FKBP12; Carbonic anhydrase II; Dihydrofolate reductase; FK506; Benzenesulfonamide; Methotrexate