Keywords: شیمی ترکیبی; Combinatorial chemistry; Iron; Hydrogel; Ligands; Colorimetric; Sensor; Water quality;
مقالات ISI شیمی ترکیبی (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: شیمی ترکیبی; Multicomponent reaction; Benzofuran; Microwave; Combinatorial chemistry;
Keywords: شیمی ترکیبی; In vitro selection; SELEX; RNA aptamer; Combinatorial chemistry; Biotechnology;
Keywords: شیمی ترکیبی; SECM tip; Approach curve; Generation/collection mode; Combinatorial chemistry; Feedback mode; Rapid screening of catalysts
Keywords: شیمی ترکیبی; Fluorous Fmoc reagent; Protecting groups; Large scale synthesis; Combinatorial chemistry; Peptides;
Keywords: شیمی ترکیبی; 5-Carbamoyl-thiazole; Solid-phase synthesis; Combinatorial chemistry; Traceless support; Heterocycles;
Keywords: شیمی ترکیبی; Peptidomimetics; Oligoheterocyclic peptidomimetics; Solid-phase synthesis; Combinatorial chemistry; Opioid receptors
Keywords: شیمی ترکیبی; Thiophene-3-carbonitrile; Solid-phase synthesis; Combinatorial chemistry; Heterocycles;
Keywords: شیمی ترکیبی; 2-Aminothioazoles; Multicomponent reactions; Combinatorial chemistry; Privileged structures; Parallel solution-phase synthesis;
Keywords: شیمی ترکیبی; Solid phase synthesis; Combinatorial chemistry; Substituted piperazines; Antitubercular
Selective, C-3 Friedel-Crafts acylation to generate functionally diverse, acetylated Imidazo[1,2-a]pyridine derivatives
Keywords: شیمی ترکیبی; Imidazo[1,2-a]pyridine; Combinatorial chemistry; Friedel-Crafts acylation; Drug discovery; Library generation;
Combinatorial screening of photoanode materials - Uniform platform for compositional arrays and macroscopic electrodes
Keywords: شیمی ترکیبی; Scanning photoelectrochemical microscopy; Solar water splitting; Combinatorial chemistry; Material printing; Transition metal oxides; Oxygen evolution; XPS; Raman spectroscopy;
Synthesis of (3S,4S,5S)-trihydroxylpiperidine derivatives as enzyme stabilizers to improve therapeutic enzyme activity in Fabry patient cell lines
Keywords: شیمی ترکیبی; Iminosugar; Trihydroxylated piperidine; Fabry disease; Enzyme stabilizer; Combinatorial chemistry; Lysosomal α-galactosidase;
Rapid preparation of (3R,4S,5R) polyhydroxylated pyrrolidine-based libraries to discover a pharmacological chaperone for treatment of Fabry disease
Keywords: شیمی ترکیبی; Azasugar; Polyhydroxylated pyrrolidine; Fabry disease; Pharmacological chaperone; Combinatorial chemistry; Lysosomal α-galactosidase;
Recent advances on the encoding and selection methods of DNA-encoded chemical library
Keywords: شیمی ترکیبی; DNA-encoded library; Drug discovery; High throughput screening; Combinatorial chemistry; Dynamic combinatorial library;
Tryptophan tags and de novo designed complementary affinity ligands for the expression and purification of recombinant proteins
Keywords: شیمی ترکیبی; Affinity tag; Affinity ligand; Combinatorial chemistry; Ugi reaction; Green fluorescent protein; Recombinant proteins; Affinity chromatography;
Identification of selective covalent inhibitors of platelet activating factor acetylhydrolase 1B2 from the screening of an oxadiazolone-capped peptoid–azapeptoid hybrid library
Keywords: شیمی ترکیبی; Peptoid; Serine hydrolase; PAFAH1B2; Combinatorial chemistry; High throughput screening
Discovery of 1,3-dihydro-2,1,3-benzothiadiazole 2,2-dioxide analogs as new RORC modulators
Keywords: شیمی ترکیبی; Virtual screening; Combinatorial chemistry; Crystal structure; Retinoid orphan receptor
Synthetic derivatives of the SUMO consensus sequence provide a basis for improved substrate recognition
Keywords: شیمی ترکیبی; Combinatorial chemistry; Conjugation; Enzymes; Peptide mimics; SUMO;
Synthesis, anti-mycobacterial activity and DNA sequence-selectivity of a library of biaryl-motifs containing polyamides
Keywords: شیمی ترکیبی; Distamycin; Antibiotic resistance; Anti-tubercular agents; DNA-minor groove ligands; Whole cell phenotypic evaluation; Combinatorial chemistry;
Substrate specificity of human matriptase-2
Keywords: شیمی ترکیبی; Matriptase-2; Combinatorial chemistry; Fluorogenic substrates; Internally quenched substrates;
Combinatorial discovery of Ni-based binary and ternary catalysts for hydrazine electrooxidation for use in anion exchange membrane fuel cells
Keywords: شیمی ترکیبی; Direct hydrazine hydrate fuel cells; Anion exchange membrane fuel cells; Combinatorial chemistry; Hydrazine oxidation; Ni-based binary and ternary catalysts;
A novel protocol to accelerate dynamic combinatorial chemistry via isolation of ligand-target adducts from dynamic combinatorial libraries: A case study identifying competitive inhibitors of lysozyme
Keywords: شیمی ترکیبی; Drug discovery; Enzyme inhibitors; Combinatorial chemistry; Ligand separation;
AlCl3-NaI assisted cleavage of polymer-bound esters with concomitant amine coupling and azido-reductive cyclization: synthesis of pyrrolobenzodiazepine derivatives
Keywords: شیمی ترکیبی; Pyrrolobenzodiazepines; Solid-phase synthesis; Combinatorial chemistry; AlCl3-NaI; Azido-reductive cyclization; SLE method;
A new proteinase 3 substrate with improved selectivity over human neutrophil elastase
Keywords: شیمی ترکیبی; Neutrophil serine proteases; Intermolecular quenched substrate; Proteinase 3; Combinatorial chemistry;
Combinatorial synthesis with high throughput discovery of protein-resistant membrane surfaces
Keywords: شیمی ترکیبی; Low protein adhesion; Combinatorial chemistry; Amide monomer; High throughput; Atmospheric pressure plasma
Ligand/kappa-opioid receptor interactions: Insights from the X-ray crystal structure
Keywords: شیمی ترکیبی; Kappa-opioid receptor; Tetrapeptide; Molecular modeling; Combinatorial chemistry
Bio-orthogonal and combinatorial approaches for the design of binding growth factors
Keywords: شیمی ترکیبی; Growth factor; Bio-orthogonal chemistry; Combinatorial chemistry; Molecular evolutionary engineering; Protein engineering
Solid phase synthesis of isoxazole and isoxazoline-carboxamides via [2+3]-dipolar cycloaddition using resin-bound alkynes or alkenes
Keywords: شیمی ترکیبی; Isoxazoles; Isoxazolines; Heterocycles; 1,3-Dipolar cycloadditions; Solid phase synthesis; Combinatorial chemistry;
Bicyclic benzofuran and indole-based salicylic acids as protein tyrosine phosphatase inhibitors
Keywords: شیمی ترکیبی; Protein tyrosine phosphatases; Therapeutic target; Salicylic acid; Inhibitor specificity; Bioavailability; Combinatorial chemistry;
Ultrasound-promoted catalyst-free one-pot four component synthesis of 2H-indazolo[2,1-b]phthalazine-triones in neutral ionic liquid 1-butyl-3-methylimidazolium bromide
Keywords: شیمی ترکیبی; 1-Butyl-3-methylimidazolium bromide; Ultrasound; 2H-Indazolo[2,1-b]phthalazine-trione; Catalyst-free reaction; Multi-component reaction; Combinatorial chemistry
Identification of a bladder cancer-specific ligand using a combinatorial chemistry approach
Keywords: شیمی ترکیبی; Bladder cancer; Targeted therapy; Combinatorial chemistry
Diverse combinatorial design, synthesis and in vitro evaluation of new HEPT analogues as potential non-nucleoside HIV-1 reverse transcription inhibitors
Keywords: شیمی ترکیبی; Combinatorial design; Diversity selection HIV-1; NNRTIs HEPT; Antiviral activity; RHHROCXXJZOAGP-UHFFFAOYSA-N; KMCGFILCIRJEHJ-UHFFFAOYSA-N; XXFUGXPQNOZBIR-UHFFFAOYSA-N; OFOHDLYVTOWSFB-UHFFFAOYSA-N; PWAKKEPZIWJVBA-UHFFFAOYSA-N; DTCUBSJAMNGQFU-UHFFFAOYSA-N;
Cerium and bismuth catalysis hand in hand—Synthesis of a eight-membered ring lactam library
Keywords: شیمی ترکیبی; Bismuth; Cerium; Catalysis; Combinatorial chemistry; 1,4-Diketones; Heterocycles; Lactams
Peptoid ligands that bind selectively to phosphoproteins
Keywords: شیمی ترکیبی; Phosphorylation; Combinatorial chemistry; Peptoid; Screening;
Serendipitous discovery of a new class of agonists for the melanocortin 1 and 4 receptors and a new class of cyclophanes
Keywords: شیمی ترکیبی; Melanocortin receptor 4; Agonist; Cyclophane; Combinatorial chemistry; Obesity
Antibody-free peptide substrate screening of serine/threonine kinase (protein kinase A) with a biotinylated detection probe
Keywords: شیمی ترکیبی; Ser/Thr kinase; Combinatorial chemistry; Peptide library; Phospho-peptide; β-Elimination
On resin amino acid side chain attachment strategy for the head to tail synthesis of new glutamine containing gramicidin-S analogs and their antimicrobial activity
Keywords: شیمی ترکیبی; Solid-phase synthesis; Gramicidin-S; Gramicidin analogs; Antimicrobial; Combinatorial chemistry; Parallel synthesis
Synthesis of novel 7-imino-2-thioxo-3,7-dihydro-2H-thiazolo [4,5-d] pyrimidine derivatives as adenosine A2A receptor antagonists
Keywords: شیمی ترکیبی; Adenosine; A2AR; Combinatorial chemistry; GPCR; Radioligand binding; Parkinson’s disease; Thiazolopyrimidines
Luminescence optimization of MBO3:Eu3+ (M=Y, Gd, Al) red phosphor by spray pyrolysis using combinatorial chemistry
Keywords: شیمی ترکیبی; Luminescence; Phosphor; Spray pyrolysis; Combinatorial chemistry
Substrate specificity and inhibitory study of human airway trypsin-like protease
Keywords: شیمی ترکیبی; Human airway trypsin-like protease; Combinatorial chemistry; FRET peptide; Chromogenic substrate; Inhibitors; Peptidomimetic;
Discovery of novel quinolinone adenosine A2B antagonists
Keywords: شیمی ترکیبی; A2B receptor; Adenosine; Antagonist; Combinatorial chemistry; Quinolinone
Direct grafting of alkoxide promoters on vanadium hydrogen phosphate precursors: Improved catalysts for the selective oxidation of n-butane
Keywords: شیمی ترکیبی; Selective oxidation of n-butane; Maleic anhydride; Vanadyl phosphate; Grafted catalysts; High throughput synthesis; Combinatorial chemistry
Structure–activity relationship in binding ligands to library of artificial receptors: The search for biocompatible sensor
Keywords: شیمی ترکیبی; Artificial receptor; Combinatorial chemistry; Biosensor; Triazine; Indicator
Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands
Keywords: شیمی ترکیبی; Arylpiperazines; Microwave irradiation; Combinatorial chemistry; Serotonin
Identification of a potent and noncytotoxic inhibitor of melanin production
Keywords: شیمی ترکیبی; YOYXSQKGMBWPGK-UHFFFAOYSA-N; Biaryl amide library; Combinatorial chemistry; Depigmenting agents; Laplacian-modified naïve Bayesian; Structure-activity relationships;
Glycopeptide dendrimer colchicine conjugates targeting cancer cells
Keywords: شیمی ترکیبی; Dendrimers; Peptides; Drug delivery; Colchicine; Combinatorial chemistry; On-bead screening; Cytotoxicity; Targeting
Combinatorial investigation of Pt–Ru–Sn alloys as an anode electrocatalysts for direct alcohol fuel cells
Keywords: شیمی ترکیبی; Combinatorial chemistry; Pt–Ru–Sn; Direct alcohol fuel cells
Discovering novel chemotherapeutic drugs for the third millennium
Keywords: شیمی ترکیبی; contemporary drug discovery; novel molecular targets; small molecule mechanism-based drugs; high throughput bioscience assays; combinatorial chemistry; drug design and screening; molecular pharmacodynamics and imaging; hypothesis-testing clinical trials
Synthesis of 2-amino-5-benzoyl-4-(2-furyl)thiazoles as adenosine A2A receptor antagonists
Keywords: شیمی ترکیبی; Adenosine; GPCR; Aminothiazole; Parkinson’s disease; Combinatorial chemistry; ECLiPSTM