
A pharmacological assessment of agonists and modulators at α4β2γ2 and α4β2δ GABAA receptors: The challenge in comparing apples with oranges
Keywords: GABAAR; γ-amino butyric acid receptor type A; DS1 and DS2; Delta selective agents 1 and 2; ECD; extracellular domain; ICL; intracellular loop between TM3 and TM4; PAM; positive allosteric modulator; TMD; transmembrane domain; wt.; wild-type; GABAA recept