کد مقاله کد نشریه سال انتشار مقاله انگلیسی نسخه تمام متن
2500727 1556893 2015 9 صفحه PDF دانلود رایگان
عنوان انگلیسی مقاله ISI
Thieno[2,3-d]pyrimidine based derivatives as kinase inhibitors and anticancer agents
موضوعات مرتبط
علوم پزشکی و سلامت داروسازی، سم شناسی و علوم دارویی علوم دارویی
پیش نمایش صفحه اول مقاله
Thieno[2,3-d]pyrimidine based derivatives as kinase inhibitors and anticancer agents
چکیده انگلیسی

Thienopyrimidines are fused heterocyclic ring systems; structurally resemble purines, exerting pharmacological potential in different aspects. They are known to play a crucial role in various disease conditions. Thieno[2,3-d]pyrimidine derivatives have been explored for their inhibitory activities towards various protein kinase enzymes. The present review is a compilation on chemical synthesis and biological anticancer significance, via inhibition of specific protein kinase enzymes, including structure–activity relationships of thieno[2,3-d]pyrimidines derivatives reported to date.

ناشر
Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Future Journal of Pharmaceutical Sciences - Volume 1, Issue 2, December 2015, Pages 33–41
نویسندگان
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