Synthesis of chiral oxazolidinone derivatives through lipase-catalyzed kinetic resolution

â¿¢Chiral oxazolidinone derivatives were synthesized with excellent enantiopurities.â¿¢Lipase-catalyzed kinetic resolution of two-step, cascade acylation was described.â¿¢Carbonates were used as double acyl donors for lipase-catalyzed cyclizations.