Keywords: هیستون deacetylases; AMPK; AMP-activated protein kinase; CamKKβ; calmodulin-dependent kinase kinase β (CamKKβ); DARPP-32; dopamine-and cAMP-regulated phosphoprotein of Mr 32 kDa; ERK; extracellular signal-regulated kinase; HDACs; histone deacetylases; MAO-A; monoamine oxi
مقالات ISI هیستون deacetylases (ترجمه نشده)
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Keywords: هیستون deacetylases; ECMs; extracellular matrix; α-SMA; α-smooth muscle actin; TGF-β1; transforming growth factor-β1; Ang-II; angiotension II; DNMTs; DNA methyltransferases; 5-Aza-dC; 5-Aza-2â²-deoxycytidine; EZH2; Enhancer of zeste homolog 2; HDAC; histone deacetylases;
Keywords: هیستون deacetylases; BLA; basolateral amygdala; CBP; CREB binding protein; CREB; cyclic AMP-responsive element binding factor; DG; dentate gyrus; Dnmt; DNA methyl transferase; GR; glucocorticoid receptor; HAT; histone acetyltransferase; HDACs; histone deacetylases; LTD; long-
Keywords: هیستون deacetylases; FOXO; forkhead box O; GC; glucocorticoids; MuRF-1; muscle RING-finger protein-1; mTOR; mammalian target of rapamycin; IGF-I; Insulin-like Growth Factor-I; eIF4E; eukaryotic translation initiation factor 4E; S6K1; ribosomal protein kinase 1; 4E-BP1; eukary
Keywords: هیستون deacetylases; Cognitive enhancer; Histone deacetylases; Epigenetic; Chromatin; Acetylation; CREB; AcH4K12; acetylated histone H4 lysine 12; AcH3K9; acetylated histone lysine 9; Bdnf; brain-derived neurotrophic factor; CRE; cAMP response element; CREB; cAMP response ele
Histone deacetylases inhibition: a potential diagnostic and therapeutic target for cancers
Keywords: هیستون deacetylases; Histone deacetylases; Carcinogenesis; Hepatocellular carcinoma; Pancreatic cancer;
CD36 mediates lipid accumulation in pancreatic beta cells under the duress of glucolipotoxic conditions: Novel roles of lysine deacetylases
Keywords: هیستون deacetylases; CD36; Caspase 3; Glucolipotoxicity; Histone deacetylases; Pancreatic beta cells;
The cross roles of sphingosine kinase 1/2 and ceramide glucosyltransferase in cell growth and death
Keywords: هیستون deacetylases; Sphingosine kinases 1 and 2; Sphingosine; S1P; Ceramide; Ceramide glucosyltransferase; Cell cycle; Anti-cancer; SK1; sphingosine kinases 1; SK2; sphingosine kinases 2; PCNA; proliferating cell nuclear antigen; GSL; glycosphingolipids; Cer; Ceramide; Sph;
SET promotes H2Ak9 acetylation by suppressing HDAC1 in trichloroethylene-induced hepatic cytotoxicity
Keywords: هیستون deacetylases; TCE; trichloroethylene; TCA; trifluoroacetic acid; DMSO; dimethyl sulphoside; SET; (Su (var)3-9, Enhancer-of-zeste, Trithorax); GAPDH; glyceraldehyde-3-phosphate dehydrogenase; TAU-PAGE; triton-acetic acid-urea-polyacrylamide gel electrophoresis; Trichl
Polyphenolic derivatives from mango (Mangifera Indica L.) modulate fecal microbiome, short-chain fatty acids production and the HDAC1/AMPK/LC3 axis in rats with DSS-induced colitis
Keywords: هیستون deacetylases; AMPK; AMP-activated protein kinase; ATCC; American Type Culture Collection; Atgs; autophagy-related genes; DSS; dextran sodium sulfate; GAE; gallic acid equivalent; GAPDH; glyceraldehyde-3-phosphate dehydrogenase; GC-MS; gas chromatography-mass spectr
Low-dose hydrocortisone prolongs survival in a lethal sepsis model in adrenalectomized rats
Keywords: هیستون deacetylases; Hydrocortisone; Sepsis; Adrenalectomy; Tumor necrosis factor; Histone deacetylases; DNA methytransferases;
MiR-17-5p enhances pancreatic cancer proliferation by altering cell cycle profiles via disruption of RBL2/E2F4-repressing complexes
Keywords: هیستون deacetylases; miR-17-5p; RBL2; E2F4; Cell cycle; Pancreatic cancer; CRF; Chromatin remodeling factor; DP; Dimerization partner; HDACs; Histone deacetylases; MuvB; Multivulva class B; PDAC; Pancreatic ductal adenocarcinoma; RBL2; Retinoblastoma-like protein2;
HDAC1 localizes to the mitochondria of cardiac myocytes and contributes to early cardiac reperfusion injury
Keywords: هیستون deacetylases; Ischemia reperfusion injury; Histone deacetylases; Mitochondria; Basic science research; Ischemia; Epigenetics; Metabolism; Oxidant stress; HAT; histone acetyltransferase enzyme; HDAC; histone deacetylase enzyme; I/R; ischemia reperfusion injury; dP/dtmax
Repurposing of sodium valproate in colon cancer associated with diabetes mellitus: Role of HDAC inhibition
Keywords: هیستون deacetylases; ACF; aberrant crypt foci; ALP; alkaline phosphatase; ANOVA; one-way analysis of variance; CEA; carcinogenic embryonic antigen; DMH; 1,2 dimethylhydrazine; EDTA; ethylene diamine tetra acetic acid; ELISA; enzyme-linked immunosorbent assay; HbA1c; glycosyla
HDAC inhibitors as epigenetic regulators for cancer immunotherapy
Keywords: هیستون deacetylases; AICD; activation-induced cell death; AML; acute myeloid leukemia; APC; antigen-presenting cells; CAR; coxsackie- and adenovirus receptor; CDKs; cyclin-dependent kinases; CG; cancer germline; DCs; dendritic cells; HAT; histone acetyltransferase; HDAC; hist
Effects of Class II-Selective Histone Deacetylase Inhibitor on Neuromuscular Function and Disease Progression in SOD1-ALS Mice
Keywords: هیستون deacetylases; CMAPs; Compound muscle action potentials; FGFBP; fibroblast growth factor binding protein; HDACs; histone deacetylases; MEF; myocyte enhancer factor; PBS; phosphate-buffered saline; amyotrophic lateral sclerosis; HDAC inhibitor; SOD1G93A mice; skeletal mu
An appraisal on synthetic and pharmaceutical perspectives of pyrazolo[4,3-d]pyrimidine scaffold
Keywords: هیستون deacetylases; A. flavus; Aspergillus flavus; C. albicans; Candida albicans; cAMP; cyclic adenosine monophosphate; CDK; cyclin-dependent kinase; CNS; central nervous system; COX; cyclooxygenase; CRF; corticotropin-releasing hormone; CRK; cdc2-related kinase; CYC6; cycli
Sargassum polysaccharide inhibits inflammatory response in PCV2 infected-RAW264.7 cells by regulating histone acetylation
Keywords: هیستون deacetylases; SP; Sargassum polysaccharide; PCV2; porcine circovirus type 2; HATs; histone acetyltransferases; HDACs; histone deacetylases; H3; histone 3; TNF-α; tumor necrosis factor-α; IL-; interleukin-; MCP; monocyte chemotactic protein; COX-; cyclooxygenase-; PMW
Structural and biological characterization of new hybrid drugs joining an HDAC inhibitor to different NO-donors
Keywords: هیستون deacetylases; Histone deacetylases; Nitric oxide; Multitarget drugs; Muscle differentiation; Vasodilatation;
DACT2 Epigenetic Stimulator Exerts Dual Efficacy for Colorectal Cancer Prevention and Treatment
Keywords: هیستون deacetylases; 5aza; thioguanine and 5-azacytidine; AOM; azoxymethane; CRC; clinical colorectal cancer; DACT2; dishevelled binding antagonist of beta catenin 2; DAI; disease activity index; DNMTs; DNA methyltransferases; DSS; dextran sodium sulfate; HDACs; histone deace
Co-targeting of BET proteins and HDACs as a novel approach to trigger apoptosis in rhabdomyosarcoma cells
Keywords: هیستون deacetylases; Apoptosis; Cell death; Mitochondria; HDAC; BET proteins; Rhabdomyosarcoma; JQ1; ARMS; alveolar rhabdomyosarcoma; BRD; bromodomain; BET protein; bromo- and extra-Terminal protein; CI; combination index; ERMS; embryonal rhabdomyosarcoma; EV; empty vector; F
Aflatoxin B1 induced multiple epigenetic modulators in human epithelial cell lines
Keywords: هیستون deacetylases; Aflatoxin B1; DNMTs; HAT; HDACs; Polycomb repressor complex; DNMTs; DNA methyltransferases; HATs; histone acetyltransferases; HDACs; histone deacetylases; PcG; polycomb group proteins; PRC; polycomb repressive complex; EZH2; enhancer of zeste homolog 2; S
Diarylcyclopropane hydroxamic acid inhibitors of histone deacetylase 4 designed by combinatorial approach and QM/MM calculations
Keywords: هیستون deacetylases; Huntington's disease; Histone deacetylases; Inhibitors of HDAC4; Computer-assisted drug design; QM/MM approach; B3LYP; hybrid gradient-corrected exchange-correlation functional of electron density; CADD; computer-assisted drug design; DCHA; trans-(2R,3R)-
Class I histone deacetylases in retinal progenitors and differentiating ganglion cells
Keywords: هیستون deacetylases; Histone deacetylases; HDACs; Mouse; Murine; Retina; Progenitors; Retinal ganglion cells;
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups
Keywords: هیستون deacetylases; BRD4; BI2536; Indoline; WPF binders; c-Myc; PD-L1; BCPs; Bromodomain-containing proteins; BET; bromodomain and extra-terminal; BRD4-BD1; first bromodomain of BRD4; CREB; cyclic-AMP response element binding protein; FA; fluorescence anisotropy; FBDD; fragm
Design, synthesis and biological evaluation of novel histone deacetylase inhibitors incorporating 4-aminoquinazolinyl systems as capping groups
Keywords: هیستون deacetylases; Histone deacetylases; 4-aminoquinazolinyl; Selectivity; Antiproliferative activity; Synthesis;
The role of SIRT1 in diabetic cardiomyopathy
Keywords: هیستون deacetylases; SIR2; Silent Information Regulator2; HDACs; histone deacetylases; NAD +; nicotinamide adenine dinucleotide; DM; diabetes mellitus; CAD; coronary artery disease; HF; heart failure; DCP; diabetic cardiomyopathy; MRI; magnetic resonance imaging; MAPK; mitoge
ReviewThe microbial epigenome in metabolic syndrome
Keywords: هیستون deacetylases; Firmicutes/Bacteroidetes ratio; SCFAs; DNA methylation; Obesity; BHB; beta-hydroxybutyrate; BMI; body mass index; CNS; central nervous system; GF; germ-free; GPRs; G-protein coupled receptors; HDAC; histone deacetylases; IECs; intestinal epithelial cells;
Steroid receptor coactivators present a unique opportunity for drug development in hormone-dependent cancers
Keywords: هیستون deacetylases; SRCs; steroid receptor coactivators; NR; nuclear receptor; PR; progesterone receptor; HATs; histone acetyltransferases; CBP; CREB-binding protein; HDACs; histone deacetylases; HMTs; histone methyltransferases; BRDs; bromodomains; bHLH-PAS; basic helix-loo
Research articleThe histone deacetylase inhibitor sodium butyrate protects against noise-induced hearing loss in Guinea pigs
Keywords: هیستون deacetylases; 3-NT; 3-nitrotyrosine; DAPI; 4â²,6-diamidino-2-phenylindole; ABR; auditory brainstem response; HATs; histone acetyltransferases; HDACs; histone deacetylases; H3-AcK9; acetyl-histone H3 (Lys9); HC; hair cell; IHC; inner hair cell; NIHL; noise-induced hear
G-quadruplex-based fluorometric biosensor for label-free and homogenous detection of protein acetylation-related enzymes activities
Keywords: هیستون deacetylases; Histone acetyltransferases; Histone deacetylases; G-quadruplexes; Thioflavin T; Label-free fluorescent method;
Species Differences in the Binding of Sodium 4-Phenylbutyrate to Serum Albumin
Keywords: هیستون deacetylases; albumin; protein binding; protein structure; distribution; molecular modeling; ER; endoplasmic reticulum; HDACs; histone deacetylases; M-PB; methyl 4-phenylbutyrate; PA; phenylacetic acid; PB; sodium 4-phenylbutyrate; PC; 6-phenylcaproic acid; PH; 7-pheny
MTA1 expression in human cancers - Clinical and pharmacological significance
Keywords: هیستون deacetylases; MTAs; metastasis associated proteins; EMT; epithelial to mesenchymal transition; NuRD; nuclear remodeling and deacetylation complex; HDAC1 or HDAC2; histone deacetylases; MBD; methylated CpG binding domain proteins; RbAb46/48; retinoblastoma associated pr
Design, virtual screening, molecular docking and molecular dynamics studies of novel urushiol derivatives as potential HDAC2 selective inhibitors
Keywords: هیستون deacetylases; HDAC; histone deacetylases; HDACIs; histone deacetylases inhibitors; HDLP; histone deacetylases - like protein; MDS; molecular dynamics simulation; MD; molecular dynamics; RMSD; root mean square deviations; RMSF; root mean squared fluctuation; Urushiol de
ReviewHistone modifications: A review about the presence of this epigenetic phenomenon in carcinogenesis
Keywords: هیستون deacetylases; Histone deacetylases; Histone acetyltransferases; Genes; Review;
Hyaluronate synthase-2 overexpression alters estrogen dependence and induces histone deacetylase inhibitor-like effects on ER-driven genes in MCF7 breast tumor cells
Keywords: هیستون deacetylases; Hyaluronan; Hyaluronate synthase 2; Estrogen signaling; Histone deacetylases; Breast cancer; AP1; activating protein -1; CD44; cluster of differenciation 44; DMEM; Dulbelcoo's modified Eagle's Medium; E2; 17β-estradiol; ER; estrogen receptor; ERE; estrog
Original ArticleHDAC4 and HDAC6 sustain DNA double strand break repair and stem-like phenotype by promoting radioresistance in glioblastoma cells
Keywords: هیستون deacetylases; HDAC4; HDAC6; Glioblastoma; Radiotherapy; Radioresistance; GBM; glioblastoma; TMZ; temozolomide; RT; radiotherapy; HDACs; Histone deacetylases; HATs; Histone acetyltransferases; DSBs; DNA double-strand breaks; OS; Overall survival; shRNA; short hairpin RN
HMBA is a putative HSP70 activator stimulating HEXIM1 expression that is down-regulated by estrogen
Keywords: هیستون deacetylases; HEXIM1; hexamethylene bis-acetamide inducible protein 1; HMBA; hexamethylene bis-acetamide; HSP70; heat shock protein 70; SAHA; suberanilohydroxamic acid; HDAC; histone deacetylases; SDS/PAGE; sodium dodecyl sulfate polyacrylamide gel electrophoresis; FBS
Epigenetic regulation of pro-inflammatory cytokine secretion by sphingosine 1-phosphate (S1P) in acute lung injury: Role of S1P lyase
Keywords: هیستون deacetylases; Acute lung injury; S1P signaling; Histone acetylation; S1P lyase; Sphingosine kinases; Hexadecenal; Histone deacetylases;
Original ArticleDoxorubicin anti-tumor mechanisms include Hsp60 post-translational modifications leading to the Hsp60/p53 complex dissociation and instauration of replicative senescence
Keywords: هیستون deacetylases; Doxorubicin; Hsp60; Acetylation; Ubiquitination; p53; Replicative senescence; DMSO; dimethylsulfoxide; ELISA; enzyme linked immunosorbent assay; GAPDH; glyceraldehyde-3-phosphate dehydrogenase; GUSB; betaglucuronidase; HDAC; histone deacetylases; H2AX; H2
Anti-androgenic mechanisms of Bisphenol A involve androgen receptor signaling pathway
Keywords: هیستون deacetylases; AR; androgen receptor; BPA; Bisphenol A; EDCs; endocrine-disrupting chemicals; DHT; dihydrotestosterone; AREs; androgen response elements; N/C; amino- and carboxyl-terminal regions; SRC-1; steroid receptor coactivator-1; SMRT; silencing mediator of retino
Complexity of the Wnt/βâcatenin pathway: Searching for an activation model
Keywords: هیستون deacetylases; APC; adenomatous polyposis coli; BCL-9; B-cell lymphoma 9; BMPs; bone morphogenetic proteins; CARM; coactivator-associated arginine methyltransferase; CBP; CREB-binding protein; CK1α; casein kinase 1α; CRD; Cysteine-Rich Domain; DIX; Dishevelled interac
Functional relevance of miRNAs in premature ageing
Keywords: هیستون deacetylases; CRP; C-reactive protein; DDR; DNA damage response; DSB; double-strand breaks; HATs; histone acetyltransferases; HDACs; histone deacetylases; hMSCs; human mesenchymal stem cells; HRR; homologous recombination repair; MEFs; mouse embryonic fibroblast; ROS;
The thermodynamic signature of ligand binding to histone deacetylase-like amidohydrolases is most sensitive to the flexibility in the L2-loop lining the active site pocket
Keywords: هیستون deacetylases; Thermodynamic signatures; Protein-ligand binding; Histone deacetylases; Binding mechanism; Conformational flexibility;
Insights into inner ear-specific gene regulation: Epigenetics and non-coding RNAs in inner ear development and regeneration
Keywords: هیستون deacetylases; bps; base pairs; DHS; DNase Hypersensitive sites; TFBS; transcription factor binding sites; PTMs; post-translational modifications; HDACs; histone deacetylases; H3K4me3; histone 3 lysine 4 tri-methylation; H3K27me3; histone 3 lysine 27 tri-methylation; Ch
Design and synthesis of tranylcypromine derivatives as novel LSD1/HDACs dual inhibitors for cancer treatment
Keywords: هیستون deacetylases; Lysine-specific demethylase 1; Histone deacetylases; Dual inhibitor; Synthesis;
Synthesis of a selective HDAC6 inhibitor active in neuroblasts
Keywords: هیستون deacetylases; Histone deacetylases; Isoform selectivity; HDAC6; PAMPA; Neuroblastoma cells;
Cross metathesis with hydroxamate and benzamide BOC-protected alkenes to access HDAC inhibitors and their biological evaluation highlighted intrinsic activity of BOC-protected dihydroxamates
Keywords: هیستون deacetylases; Metathesis; Histone deacetylases; Cancer; Tubulin
Dissecting structure–activity-relationships of crebinostat: Brain penetrant HDAC inhibitors for neuroepigenetic regulation
Keywords: هیستون deacetylases; Cognitive enhancer; Nootropic; Histone deacetylases; Epigenetic; Chromatin; Acetylation; CREB; Neuroepigenetic
Associate editor: B. TeicherBenefits of short-chain fatty acids and their receptors in inflammation and carcinogenesis
Keywords: هیستون deacetylases; GPR41; G protein-coupled receptor 41; GPR43; G protein-coupled receptor 43; GPR109A; G protein-coupled receptor 109A; HDAC; Histone deacetylases; DSS; dextran sulfate sodium; AOM; azoxymethane; APC; adenomatous polyposis; DC; dendritic cell; Treg; T regul