دانلود مقالات ISI درباره Sar + ترجمه فارسی

Chemotography for multi-target SAR analysis in the context of biological pathways

Keywords: GPCR; G-protein coupled receptor; LGIC; ligand-gated ion channel; SAR; structure-activity relationship; Chemical space; Color; Visualization; Molecular fingerprints; Chemogenomics; Systems pharmacology; Molecular pathways;

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2012 سفارش ترجمه

Inhibition of thioredoxin reductase by a novel series of bis-1,2-benzisoselenazol-3(2H)-ones: Organoselenium compounds for cancer therapy

Keywords: TrxR; thioredoxin reductase; Trx; thioredoxin; GR; glutathione reductase; SAR; structure-activity relationship; DTNB; 5,5′-dithiol-bis-2-nitrobenzoic acid; Log Pcal; calculated Log P; BIAM; biotin-conjugated iodoacetamide; Organoselenium compound; T

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2012 سفارش ترجمه

Spatial and temporal soil moisture estimation from RADARSAT-2 imagery over Flevoland, The Netherlands

Keywords: Soil moisture; SAR; IEM; Change detection

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Optically stimulated luminescence dating of glaciofluvial sediments on the Canterbury Plains, South Island, New Zealand

Keywords: OSL; Coarse-grained quartz; SAR; Canterbury Plains; LGM; Braided river

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

SAR observations of internal solitary waves generated at the Estremadura Promontory off the west Iberian coast

Keywords: Iberia coast; Portugal; Estremadura Promontory; Internal tides; Internal solitary waves; SAR; Refraction

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

The design, synthesis and biological evaluations of C-6 or C-7 substituted 2-hydroxyisoquinoline-1,3-diones as inhibitors of hepatitis C virus

Keywords: IN; integrase; RNH; ribonuclease H; HCV; hepatitis C virus; peg-INF; pegylated interferon; RBV; ribavirin; SVR; sustained virological response; DAA; direct-acting antiviral; NNI; nonnucleoside inhibitor; DKA; diketoacid; Luc; luciferase; 2 mA; 2′-C-met

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Design, synthesis, and biological evaluation of 4-phenylpyrrole derivatives as novel androgen receptor antagonists

Keywords: PC; prostate cancer; AR; androgen receptor; GnRH; gonadotropin-releasing hormone; CAB; combined androgen blockade; PSA; prostate-specific antigen; WT; wild-type; DHT; dihydrotestosterone; SAR; structure-activity relationship; DIBAL; diisobutylaluminium

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Geomorphological, chemical and physical study of “calanchi” landforms in NW Sicily (southern Italy)

Keywords: Calanchi fronts; Chemical and physical properties; SAR; Microforms; Mineralogy;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis and evaluation of antimicrobial activity of 4H-pyrimido[2,1-b]benzothiazole, pyrazole and benzylidene derivatives of curcumin

Keywords: Antimicrobial activity; SAR; Cytotoxicity; Pyrazoles; Benzylidene; 4H-Pyrimido[2,1-b]benzothiazole derivatives of curcumin;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Identification of novel benzimidazole derivatives as inhibitors of leukotriene biosynthesis by virtual screening targeting 5-lipoxygenase-activating protein (FLAP)

Keywords: AA; arachidonic acid; cPLA2; cytosolic phospholipase A2; FLAP; 5-lipoxygenase-activating protein; 5-HpETE; 5-hydroperoxyeicosatetraenoic acid; 5-LO; 5-lipoxygenase; LT; leukotriene; PGC buffer; phosphate-buffered saline pH 7.4 containing 1 mg/mL glucose

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

Structure-activity relationships for the binding of polymyxins with human α-1-acid glycoprotein

Keywords: ANS; 1-anilino-8-naphthalene sulfonic acid; AO; Auramine O; AGP; human α-1-acid glycoprotein; CAPs; cationic antimicrobial peptides; CMS; colistin methanesulfonate; Fmoc; fluorenylmethyloxycarbonyl; Dab; diaminobutyric-acid; ITC; isothermal titration cal

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

t-Butylsarcosinedithiocarbamato gold(III)-based anticancer agents: Design, in vitro biological evaluation and interaction with model biomolecules

Keywords: BrdU; bromodeoxyuridine; BSA; bovine serum albumin; dAMP; 2′-deoxyadenosine-5′-monophosphate; dGMP; 2′-deoxyguanosine-5′-monophosphate; DMSO; methyl sulfoxide; DSC; differential scanning calorimetry; dtc; dithiocarbamate; ELISA; enzyme-linked immu

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis, anticonvulsant activity, and neuropathic pain-attenuating activity of N-benzyl 2-amino-2-(hetero)aromatic acetamides

Keywords: AED; antiepileptic drug; ASP; Anticonvulsant Screening Program; B:P; brain-to-plasma; Cbz; carboxybenzyl; DBU; 1,8-diazabicycloundec-7-ene; DIPEA; N,N-diisopropylethylamine; DMTMM; 4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride; ED50;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

Mapping pilicide anti-virulence effect in Escherichia coli, a comprehensive structure-activity study

Keywords: SAR; structure activity relationship; QSAR; quantitative structure activity relationship; PLS; partial least squares; OPLS-DA; orthogonal projections to latent structures discriminant analysis; UTI; urinary tract infection; SMD; statistical molecular desi

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2012 سفارش ترجمه

Design, synthesis, and biological evaluation of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonists

Keywords: AR; androgen receptor; CRPC; castration-resistant prostate cancer; CAB; combined androgen blockade; DHT; dihydrotestosterone; SAR; structure-activity relationship; EDC; N-[3-(dimethylamino)propyl]-N′-ethylcarbodiimide hydrochloride; DMT-MM; 4-(4,6-dim

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2012 سفارش ترجمه

A review of the thermally transferred optically stimulated luminescence signal from quartz for dating sediments

Keywords: Review; OSL; Saturation; Age range; Sensitivity change; TT-OSL; SAR; Thermal stability

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2012 سفارش ترجمه

Analysis of bar morphology using multi-temporal and multi-sensor satellite images: Example from the Han Estuary, Korea

Keywords: satellite remote sensing; optical sensors; SAR; bar morphology; estuary; ecology

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2012 سفارش ترجمه

Nonparametric edge detection in speckled imagery

Keywords: Edge detection; Hypothesis testing; Image analysis; Multiplicative noise; Small samples; Speckle; SAR

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2012 سفارش ترجمه

A novel intranasal therapy of azelastine with fluticasone for the treatment of allergic rhinitis

Keywords: Allergic rhinitis; azelastine; fluticasone propionate; MP29-02; moderate-to-severe; ANCOVA; Analysis of covariance; AR; Allergic rhinitis; FP; Fluticasone propionate; iTNSS; Instantaneous total nasal symptom score; QoL; Quality of life; RQLQ; Rhinitis Qua

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2012 سفارش ترجمه

The neurochemical profile quantified by in vivo 1H NMR spectroscopy

Keywords: AD; Alzheimer's disease; ALS; amyotrophic lateral sclerosis; BOLD; blood-oxygen-level dependence; CNS; central nervous system; CSI; chemical shift imaging; CRLB; Cramér-Rao lower bound; fMRI; functional MRI; GABA; γ-aminobutyrate; Glx; glutamate plus gl

دانلود رایگان متن کامل مقاله ISI 21 صفحه سال انتشار : 2012 سفارش ترجمه

Remote-sensing observations of coastal sub-mesoscale eddies in the south-eastern Baltic

Keywords: Coastal currents; Submesoscale eddies; Baltic Sea; Remote sensing; MODIS; SAR; CODAR

دانلود رایگان متن کامل مقاله ISI 24 صفحه سال انتشار : 2012 سفارش ترجمه

Structure-activity relationships of 2-arylamido-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide derivatives as cannabinoid receptor agonists and their analgesic action

Keywords: GPCR; CB2 agonists; HTS; SAR; Inflammatory pain models;

دانلود رایگان متن کامل مقاله ISI 34 صفحه سال انتشار : 2012 سفارش ترجمه

Peptide deformylase inhibitors with non-peptide scaffold: Synthesis and structure-activity relationships

Keywords: PDF; SAR; Antibacterial; Non-peptide;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Volume-averaged SAR in adult and child head models when using mobile phones: A computational study with detailed CAD-based models of commercial mobile phones

Keywords: RF exposure; Dosimetry; SAR; Children

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis of cholestane saponins as mimics of OSW-1 and their cytotoxic activities

Keywords: Steroidal saponin; OSW-1; Synthesis; Cytotoxicity; SAR

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Rigidized 1-aryl sulfonyl tryptamines: Synthesis and pharmacological evaluation as 5-HT6 receptor ligands

Keywords: 5-HT6R antagonist; SAR; NORT; Water maze

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Acylglycinamides as inhibitors of glycine transporter type 1

Keywords: Glycine transporter type 1; GlyT-1; Schizophrenia; Acylglycinamides; SAR

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Discovery of a novel potent GABAB receptor agonist

Keywords: GABAB; Baclofen; SAR; Palladium; Boronate; Functional potency; Pyridylmethyl ether

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

The identification of 4,7-disubstituted naphthoic acid derivatives as UDP-competitive antagonists of P2Y14

Keywords: Pyrimidinergic receptor; P2Y14; GPR105; Competitive antagonist; SAR; Glucuronidation

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

The design, synthesis and structure–activity relationships of novel isoindoline-based histone deacetylase inhibitors

Keywords: HDAC; hERG; Cancer; Histone deacetylase; Isoindoline; SAR

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X7 antagonists

Keywords: P2X7; Antagonists; Pain; SAR

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Discovery of non-peptide, small molecule antagonists of α9α10 nicotinic acetylcholine receptors as novel analgesics for the treatment of neuropathic and tonic inflammatory pain

Keywords: α9α10 nAChR; SAR; Analgesic; Pain

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Pyridazine-derived γ-secretase modulators

Keywords: SAR; γ-secretase; Modulator; AD; GSI; GSM; Pyridazine; Amyloid-beta

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Pyridine-derived γ-secretase modulators

Keywords: γ-Secretase inhibitor; γ-Secretase modulator; SAR; Pyridine

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2011 سفارش ترجمه

Identification and optimization of tetrahydro-2H-3-benzazepin-2-ones as squalene synthase inhibitors

Keywords: Squalene synthase; Inhibitor; SAR; Atherosclerosis; 3-Benzazepin-2-ones

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

A concise synthesis and antimicrobial activities of 3-polyamino-23,24-bisnorcholanes as steroid–polyamine conjugates

Keywords: Steroid–polyamine conjugate; SAR; Reductive amination; Antimicrobial activity

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Substituted indole-1-acetic acids as potent and selective CRTh2 antagonists—discovery of AZD1981

Keywords: CRTh2; DP2; Prostaglandin; Inflammation; Asthma; Candidate drug; Optimization; SAR

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

A novel class of dual mPGES-1/5-LO inhibitors based on the α-naphthyl pirinixic acid scaffold

Keywords: Inflammation; Arachidonic acid cascade; SAR; mPGES-1; 5-LO

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis of some novel 3-(1-(1-substitutedpiperidin-4-yl)-1H-1,2,3-triazol-4-yl)-5-substituted phenyl-1,2,4-oxadiazoles as antifungal agents

Keywords: Amidoxime; 1,2,4-Oxadiazole; 1,2,3-Triazole; Piperidine; Antifungal activity; MIC values; SAR

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis and SAR of new pyrazolo[4,3-h]quinazoline-3-carboxamide derivatives as potent and selective MPS1 kinase inhibitors

Keywords: MPS1; TTK; Anticancer; Kinase selectivity; SAR

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Identification of 4H,6H-[2]benzoxepino[4,5-c][1,2]oxazoles as novel squalene synthase inhibitors

Keywords: Squalene synthase inhibitor; SAR; Atherosclerosis; 4H,6H-[2]Benzoxepino[4,5-c][1,2]oxazole

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

SAR studies on a series of N-benzyl-4-heteroaryl-1-(phenylsulfonyl)piperazine-2-carboxamides: Potent inhibitors of the polymerase enzyme (NS5B) of the hepatitis C virus

Keywords: HCV; NS5B; Allosteric inhibitors; SAR

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis and biological evaluation of (±)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors

Keywords: HIV; NNRTIs; Benzophenone derivatives; Benzhydrol; SAR;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Discovery of highly potent agents against influenza A virus

Keywords: Hit-to-lead optimization; Influenza A virus; SAR study; M2; matrix-2 protein; SAR; structure-activity relationship;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure-activity relationships

Keywords: Thiazolidione; Staphylococcus epidermidis; Antibiofilm activity; Inhibitors; IMDs; in-dwelling medical devices; TCS; two-component system; PAADs; phenoxy acetic acid derivatives; SAR; structure-activity relationship; MTDLs; multitarget-directed ligands;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

From benzimidazole to indole-5-carboxamide Thumb Pocket I inhibitors of HCV NS5B polymerase. Part 1: Indole C-2 SAR and discovery of diamide derivatives with nanomolar potency in cell-based subgenomic replicons

Keywords: Hepatitis C virus; Antiviral; HCV; NS5B; Polymerase; Inhibitor; SAR

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Optimization of triazoles as novel and potent nonphlorizin SGLT2 inhibitors

Keywords: Noncompetitive SGLT2 inhibitors; Triazoles; SAR; Solubility; Benzooxazinone head groups; Indane tail group

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Local SAR enhancements in anatomically correct children and adult models as a function of position within 1.5 T MR body coil

Keywords: Magnetic resonance imaging; Children; Pregnant; Fetus exposure; Local field enhancement; SAR; Safety

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Ground settlement monitoring based on temporarily coherent points between two SAR acquisitions

Keywords: SAR; Monitoring; Statistics; Change detection; Comparison

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Novel hybrid D/A structures for high-resolution SAR ADCs—analysis, modeling and realization

Keywords: Analog-to-digital converter; SAR; D/A conversion; CMOS integrated circuits; High-resolution

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه