
Tricyclic pyrazoles. Part 8. Synthesis, biological evaluation and modelling of tricyclic pyrazole carboxamides as potential CB2 receptor ligands with antagonist/inverse agonist properties
Keywords: Tricyclic pyrazoles; Synthesis; Cannabinoid receptors; CB2 antagonism; Molecular modelling; Î9-THC; Î9-Tetrahydrocannabinol; 2-AG; 2-Arachidonoylglycerol; CB1; cannabinoid receptor type 1; CB2; cannabinoid receptor type 2; CNS; Central nervous system; T