Keywords: Conditioning; Pelleting; Reactive lysine; Maillard reaction products; Carboxymethyllysine; Dogs; AGE; advanced glycation end-products; CML; É-N-carboxymethyllysine; DM; dry matter; FL; fructoselysine; HMF; (5-hydroxymethyl)-2-furfural; LAL; lysinoalanine
مقالات ISI (ترجمه نشده)
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Keywords: DMEM; Dulbecco's Modified Eagle Medium; DMSO; Dimethylsulfoxide; Dox; Doxorubicin; RSV; Resveratrol; MCF-7/adr; Doxorubicin-resistant MCF-7; ABC transporter; ATP-binding cassette transporter; MDR; Multi-drug resistance; MRP; Multi-drug resistance associat
Keywords: APAP; acetaminophen; ALT; alanine aminotransferase; CCl4; carbon tetrachloride; CFB; clofibrate; i.p.; intraperitoneal; Fmo3; flavin-containing monooxygenase 3; Lgals3; galectin-3; H202; hydrogen peroxide; MAT1A; methionine adenosyl transferase-1 alpha; M
Keywords: 3D Cell culture; Hepatocyte; Multicellular spheroids; Cell differentiation; Nanocellulose; Organotypic; 2D; two-dimensional; 3D; three-dimensional; ABC transporter; ATP-binding cassette transporter; ALB; Albumin; Calcein-AM; calcein-acetoxymethyl ester; C
Keywords: DCP; decentralised procedure; Eur. Com.; European Commission; EDQM; European Directorate for Quality of Medicines; EFTA; The European Free Trade Association; EMA; European Medicines Agency; EU; European Union; HMP; herbal medicinal product(s); HMPC; Commi
Keywords: Biofortification; Gluten-free; Minor grains; Phytochemicals; ABC; ATP-binding cassette; ABS; Africa biofortified sorghum; ACE; angiotensin-1 converting enzyme; DDGS; distillers dried grain and solubles; FAN; free amino nitrogen; GM; genetically modified;
Keywords: Aged; Exercise; Interleukin-6; Rehabilitation; Women; ANOVA; analysis of variance; CG; control group; IL-6; interleukin 6; MRP; muscle resistance program; sTNFr1; soluble tumor necrosis factor receptor-1; 10MWT; 10-meter walk test; TNF-α; tumor necrosis
Keywords: AA; amino acid; GE; glandular epithelium; IFNT; interferon-Ï; IRF; interferon regulatory factor; ISG; interferon-stimulated gene; LE; luminal epithelium; MRP; maternal recognition of pregnancy; P4; progesterone; PCA; principal component analysis; PG; pro
Keywords: APC; apparent partition coefficient; BCRP; breast cancer resistance protein; CH; cholate; cLPM; canalicular liver plasma membrane; DC; deoxycholate; GC; glycocholate; GDC; glycodeoxycholate; HNAP; hydroxy-2-naphthoic acid; Mw; molecular weight; MATE; mult
Keywords: AML; acute myeloid leukemia; CAM-DR; cell adhesion-mediated drug resistance; CCP; charge-conversion polymer; CLL; chronic lymphocytic leukemia; CNS; central nervous system; CSC; cancer stem cell; EGFR; epidermal growth factor receptor; EPR; enhanced perme
Keywords: Nanomedicine; Drug targeting; Multidrug resistance; MDR; Drug efflux pumps; ABC transporters; Pgp; MRP; Pluronics; siRNA;
Keywords: Coarse woody debris; Soil chemistry; Lignin; Brown-rot fungi; White-rot fungi; WEOC; water-extractable organic carbon; POC; Particulate organic carbon; SUVA280; Specific ultraviolet absorbance at 280Â nm; MRP; Molybdenum-reactive phosphorus;
Keywords: Scheduling; MRP; Advanced Planning and Scheduling; Mixed integer programming
Shikonin upregulates the expression of drug-metabolizing enzymes and drug transporters in primary rat hepatocytes
Keywords: AhR; aryl hydrocarbon receptor; AP1; activating protein 1; ARE; antioxidant-response element; CAR; constitutive androstane receptor; CYP; cytochrome P450; DREs; dioxin-responsive elements; EMSA; electromobility gel shift assay; FBS; fetal bovine serum; GS
Quantification of membrane transporter proteins in human lung and immortalized cell lines using targeted quantitative proteomic analysis by isotope dilution nanoLC-MS/MS
Keywords: BCRP; breast cancer resistant protein; BEAS; bronchial epithelium and adenovirus; MDCK; madin darby canine kidney; MDR1; multidrug resistance protein 1 (also known as P-gp); MRM; multiple reaction monitoring; MRP; multidrug resistance-associated protein;
Significance of A-to-I RNA editing of transcripts modulating pharmacokinetics and pharmacodynamics
Keywords: ABC; ATP-binding cassette transporter; ADAR; adenosine deaminase acting on RNA; ADH; alcohol dehydrogenase; AhR; aryl hydrocarbon receptor; AKR; aldo-keto reductase; ALS; amyotrophic lateral sclerosis; AZIN1; antizyme inhibitor 1; AMPA; α-amino-3-hydroxy
Cellular Pharmacokinetic Model-Based Analysis of Genistein, Glyceollin, and MK-571 Effects on 5 (and 6)-Carboxy-2â²,7â²-Dichloroflourescein Disposition in Caco-2 Cells
Keywords: active transport; Caco-2 cells; drug transport; efflux pumps; intestinal secretion/transport; membrane transport; pharmacokinetics; transcellular transport; transporters; ABCC2; ATP binding cassette sub-family C, member 2; ABCC3; ATP binding cassette sub-
Chrysin: Sources, beneficial pharmacological activities, and molecular mechanism of action
Keywords: Passifloraceae; Passiflora caerulea; Chrysin; Pharmacological activities; Bioavailability; Molecular docking; AC; adenylyl cyclase; AGEs; advanced glycation end products; ACR; acrylamide; AHR; aryl hydrocarbon receptor; AMPK; AMP-activated protein kinase;
PDZ domain containing protein 1 (PDZK1), a modulator of membrane proteins, is regulated by the nuclear receptor THRβ
Keywords: Thyroid hormones; Scaffold protein; PDZ-domain; Gene regulation; Thyroid hormone receptors; 5-HT2A; Serotonin 2A receptor; ABC; ATP-binding cassette transporter; AhR; Transcription factor aryl hydrocarbon receptor; BCRP; Breast cancer resistance protein;
Digital gene expression analysis in the gills of Ruditapes philippinarum exposed to short- and long-term exposures of ammonia nitrogen
Keywords: DGE; Digital gene expression technology; UIA; un-ionized ammonia nitrogen; NMDA; N-Methyl-d-aspartic acid; DEG; differentially expressed genes; Nr; NCBI non-redundant protein sequences; Nt; NCBI non-redundant nucleotide sequences; Pfam; Protein family; KO
Allergen-Specific Low Zone Tolerance Is Independent of MRP8/14-, TLR4-, TLR7-, and TLR9-Mediated Immune Processes
Keywords: CHS; contact hypersensitivity; KO; knockout; LZT; low zone tolerance; MRP; myeloid-related protein; TLR; toll-like receptor;
Phytic acid transport in Phaseolus vulgaris: A new low phytic acid mutant in the PvMRP1 gene and study of the PvMRPs promoters in two different plant systems
Keywords: lpa; low phytic acid; Ins; myo-inositol; InsPs; inositol phosphates; InsP6; phytic acid; PtdIns; phosphatidylinositol; MRP; multidrug resistance protein; ABC; ATP-binding cassette; EMS; ethyl methane sulfonate; GUS; β-glucuronidase; P; phosphorous; Pi; i
Platelet-Derived MRP-14 Induces Monocyte Activation in Patients With Symptomatic Peripheral Artery Disease
Keywords: macrophages; monocytes; peripheral artery disease; platelet-monocyte aggregates; platelets; CAS; carotid artery stenosis; CLI; critical limb ischemia; LPA; leukocyte-platelet aggregate(s); MACLE; major adverse cardiovascular and limb events; MPA; mono
Cigarette smoke condensate alters Saccharomyces cerevisiae efflux transporter mRNA and activity and increases caffeine toxicity
Keywords: ABC transporter; Pdr5; Snq2; Cigarette smoke; Caffeine; Saccharomyces cerevisiae; ABC; ATP-binding cassette; AαC; 2-amino-9H-pyrido[23-b]indole; 4- ABP; 4-aminobiphenyl; BaP; benzo(a)pyrene; BLAST; Basic local alignment search tool; BCRP; breast cancer r
Aryl hydrocarbon receptor (AhR) mediated short-term effects of 2,3,7,8-tetrachlorodibenzo-p-dioxin (TCDD) on bile acid homeostasis in mice
Keywords: Aryl hydrocarbon receptor; TCDD; Bile acids; Biliary excretion; Taurodeoxycholic acid; Cyp8b1; 1°BAs; Primary bile acids; 2°BAs; Secondary bile acids; 6-OH; 6-hydroxylated (6-OH); 12-OH; 12α-hydroxylated; Abc; ATP-binding cassette; AhR; Aryl hydrocarbo
Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site
Keywords: Tubulin inhibitor; Colchicine binding site; Combretastatin A-4; Pyrazole analogue; Anti-tumour; Co-crystal structure; ABC; ATP-binding cassette; P-gp; P-glycoprotein; MRP; multidrug resistant proteins; CA-4; combretastatin A-4; SARs; structure-activity re
Imaging techniques to study drug transporter function in vivo
Keywords: ABC; ATP-binding cassette; AD; Alzheimer's disease; ADME; absorption, distribution, metabolism and elimination; ATP; adenosine triphosphate; AUC; area under the curve; BBB; blood-brain barrier; BCRP; breast cancer resistance protein; BPND; non-displaceabl
In vitro and in vivo experimental models employed in the discovery and development of antiepileptic drugs for pharmacoresistant epilepsy
Keywords: CNS; central nervous system; COX; cyclooxygenase; EEG; electroencephalography; ED50; median effective dose; MAM; methylazoxymethanol; MES; maximal electroshock; MRP; multidrug resistance-associated protein; PTZ; pentylenetetrazole; scPTZ; subcutaneous pen
Clinical benefits and pharmacology of scutellarin: A comprehensive review
Keywords: Aβ; β-amyloid peptide; ACE; angiotensin-converting enzyme; AD; Alzheimer's disease; ADE; adverse drug effect; ADR; adverse drug reaction; AIF; apoptosis-inducing factor; Akt; protein kinase B or PKB; ALS; amyotrophic lateral sclerosis; AMPK; AMP-activat
The transepithelial transport mechanism of polybrominated diphenyl ethers in human intestine determined using a Caco-2 cell monolayer
Keywords: ABC transporters; ATP-binding cassette transporters; AP; apical; BCRP; breast cancer resistance protein; BL; basolateral; DMSO; dimethyl sulphoxide; EDTA; ethylenediamine tetraacetic acid; GC/MS; gas chromatography/mass spectrometry; MEM; minimum essentia
Effects of Adjuvant-Induced Inflammation on Disposition of Diclofenac and Its Metabolites in Perfused Rat Liver
Keywords: biliary excretion; disposition; metabolism; MRP; transporters;
Gender-specific expression of ATP-binding cassette (Abc) transporters and cytoprotective genes in mouse choroid plexus
Keywords: CP; choroid plexus; BBB; blood-brain barrier; CSF; cerebrospinal fluid; Mrp; multidrug resistance-associated protein; Abc; ATP binding cassette; MTX; methotrexate; Mrp4; multidrug resistance-associated protein 4; BCSFB; blood-cerebrospinal fluid barrier;
Zuotai and HgS differ from HgCl2 and methyl mercury in Hg accumulation and toxicity in weanling and aged rats
Keywords: Mrp; Multidrug resistance-associated protein; Mdr1b; multidrug resistance gene 1b; OAT; organic anion transporter; OATP; organic anion-transporting polypeptides; OCT; organic cation transporters; Zuotai and HgS; HgCl2 and MeHg; Weanling and aged rats; Hg
RNA sequencing indicates that atrazine induces multiple detoxification genes in Daphnia magna and this is a potential source of its mixture interactions with other chemicals
Keywords: Gene expression; Mixture model; Nuclear receptor; Aquatic toxicology; Induction; Concentration-dependent; ADH; Alcohol dehydrogenase; AUC; Area under the curve; ABC transporter; ATP-binding cassette transporter; BPA; Bisphenol A; CATAM; Computational Appr
The interrelationship between bile acid and vitamin A homeostasis
Keywords: ATGL; Adipose triglyceride lipase; ADH; Alcohol dehydrogenase; ALD; Alcoholic liver disease; atRA; All-trans retinoic acid; ASBT/SLC10A2; Apical sodium-dependent bile salt transporter; ABCA1; ATP-binding cassette transporter member 1; BCMO1; Beta-carotene
Anti-cancer effect of oncolytic adenovirus-armed shRNA targeting MYCN gene on doxorubicin-resistant neuroblastoma cells
Keywords: Neuroblastoma; MDR; Doxorubicin; MYCN; MRP; Oncolytic adenovirus;
Terminology of elemental speciation - An IUPAC perspective
Keywords: DMA; dimethylarsinic acid; DMT; divalent metal transporter; DNA; deoxyribonucleic acid; IUPAC; International Union of Pure and Applied Chemistry; MMA; methylarsonic acid; MRP; multidrug resistance protein; RNA; ribonucleic acid; SAM; S-adenosylmethionine;
ATP-dependent activity and mitochondrial localization of drug efflux pumps in doxorubicin-resistant breast cancer cells
Keywords: BSA; Bovine serum albumin; BCRP; breast cancer resistance protein; FCCP; Carbonyl cyanide 4-(trifluoromethoxy)phenylhydrazone; CSI; Confocal multispectral imaging; DOX; Doxorubicin; LCSM; Laser scanning confocal microscopy; MRP; Multidrug resistance-assoc
Ipratropium is 'luminally recycled' by an inter-play between apical uptake and efflux transporters in Calu-3 bronchial epithelial cell layers
Keywords: a-b; apical to basolateral; ALI; air-liquid interface; b-a; basolateral to apical; FITC; fluorescein isothiocyanate; HBSS; Hank's Balanced Salt Solution; IPRL; isolated perfused rat lungs; MATE; multidrug and toxin extrusion transporters; MRP; Multidrug
Information processing structures and decision making delays in MRP and JIT
Keywords: Production control system; Information processing structure; Decision making delay; MRP; JIT;
Quantitative Analyses of the Influence of Parameters Governing Rate-Determining Process of Hepatic Elimination of Drugs on the Magnitudes of Drug-Drug Interactions via Hepatic OATPs and CYP3A Using Physiologically Based Pharmacokinetic Models
Keywords: cytochrome P450; drug interaction; hepatic clearance; mathematical model; organic anion-transporting polypeptide transporters; pharmacokinetics; AUC; area under the plasma concentration-time curve; CL; clearance; CLint,all; overall hepatic intrinsic cle
Comparative study of CYP2B1/2 induction and the transport of bilirubin and taurocholate in rat hepatocyte-mono- and hepatocyte-Kupffer cell co-cultures
Keywords: B; bilirubin; Bsep; bile salt export pump; CYP; cytochrome P-450; GdCl3; gadolinium(III) chloride; H/KC; hepatocyte-Kupffer-cell co-culture; HBSS; Hanks' balanced salt solution; HPLC; high-performance liquid chromatography; KC; Kupffer-cell; LPS; lipopoli
Dual role of LRRC8A-containing transporters on cisplatin resistance in human ovarian cancer cells
Keywords: A2780WT; drug-sensitive human ovarian cancer cells; A2780CisR; cisplatin resistant A2780 cells; ABC; ATP-binding cassette; Ano6; Anoctamin 6; Apaf-1; apoptotic protease activating factor 1; Atox1; Antioxidant 1 copper chaperone; AP; alkaline phosphatase;
Dioscin protects against ANIT-induced cholestasis via regulating Oatps, Mrp2 and Bsep expression in rats
Keywords: ALT; alanine amiotransferase; ANIT; alpha-naphthylisothiocyanate; AST; aspartate transaminase; BIL; bilirubin; Bsep; bile salt export pump; CMC-Na; carboxymethylcellulose sodium; E3S; estrone-3-sulfate; FXR; Farnesoid X receptor; IS; hydrochlorothiazide;
Selective GPR55 antagonism reduces chemoresistance in cancer cells
Keywords: GPR55; G protein-coupled receptor 55; MNF; (R,R⿿)-4⿲-methoxy-1-naphthylfenoterol; Pgp; P-glycoprotein; BCRP; breast cancer resistance protein; PancCa; pancreatic adenocarcinoma; MRP; multidrug resistance-related protein; AM251; 1-(2,4-dichlorophenyl)-
CT imaging of bone and bone marrow infiltration in malignant melanoma-Challenges and limitations for clinical staging in comparison to 18FDG-PET/CT
Keywords: 18F-FDG-PET/CT; 18F-fluododeoxyglucose positron emission tomography/computed tomography; AJCC; American Joint Committee on Cancer; BM; bone marrow; BMA; bone marrow attenuation; CECT; contrast-enhanced computed tomography; CT; computed tomography; HU; hou
An overview of chemical inhibitors of the Nrf2-ARE signaling pathway and their potential applications in cancer therapy
Keywords: AA; Ascorbic acid; AEM1; ARE expression modulator 1; AEG1; Astrocyte elevated gene-1; Akt; Protein kinase B; AMPK; AMP-activated protein kinase; APL; Acute promyelocytic leukemia; ARE; Antioxidant response element; ATO; Arsenic trioxide; Bach; BTB and CNC
Targeting tumor microenvironment with PEG-based amphiphilic nanoparticles to overcome chemoresistance
Keywords: ABCs; ATP-binding cassette superfamily; AUC; area under the curve; BBB; blood brain barrier; BCRP; breast cancer resistance protein; CMC; critical micellar concentration; CT; computed tomography; CUR; curcumin; DOX; doxorubicin; DSPE-PEG; 1,2-distearoyl-s
Asp residues of βDELSEED-motif are required for peptide binding in the Escherichia coli ATP synthase
Keywords: MRP; melittin related peptide; AMP; anti-microbial peptide; membrane; membrane bound F1Fo ATP synthase; F1Fo ATP synthase; ATPase; Peptide; Enzyme inhibition; βDELSEED;
Multixenobiotic resistance efflux activity in Daphnia magna and Lumbriculus variegatus
Keywords: ABC protein; ATP-binding cassette transfer protein; Ca-AM; calcein-AM; MDR; multidrug resistance protein; MRP; multidrug resistance related protein; MXR; multixenobiotic resistance (protein); NBD; nucleotide binding domain; P-gp; permeability glycoprotein