Keywords: مقاومت چنددارویی; Microtubule-stabilizing agent; Paclitaxel; Epothilone; Cancer therapy; Natural productMDA, Microtubule-destabilizing agent; MDR, Multidrug resistance; MSA, Microtubule-stabilizing agent; P-gp, P-glycoprotein; SAR, Structure–activity relationship
مقالات ISI مقاومت چنددارویی (ترجمه نشده)
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Keywords: مقاومت چنددارویی; ABC transporter, ATP-binding cassette transporter; MDR, multidrug resistance; MRP, multidrug resistance-associated protein; cMOAT, canalicular multispecific organic anion transporter; BCRP, breast cancer resistance protein; MXR, mitoxantrone resistance pr
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; IC50, 50% inhibition concentration; MDR, multidrug resistance; NCI, National Cancer Institute; (P-gp), P-glycoproteinABC transporters; Chemotherapy; Multidrug resistance; Natural products; Pharmacogenomics; Phytotherapy
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; MDR, multidrug resistance; P-gp, P-glycoprotein; DHP, dihydropyridine; CCB, calcium channel blocking; MTT, thiazolyl blue tetrazolium bromide; Rh123, rhodamine 123.1,4-Dihydropyridine (CID 104822); Multidrug resistance; Cytotoxi
Keywords: مقاومت چنددارویی; CNTN-1; MDR; Cisplatin; Apoptosis; Invasion; Metastasis; Lung adenocarcinomaDDP, cisplatin; CNTN-1, Contactin-1; EGFR, epidermal growth factor receptor; IHC, Immunohistochemistry; MDR, multidrug resistance; NCAM, neural cell adhesion molecule; NMJ, neurom
Keywords: مقاومت چنددارویی; ROS, reactive oxygen species; MDR, multidrug resistance; MTT, (3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide); FBS, fetal bovine serum; DMSO, dimethyl sulfoxide; ATCC, American Type Culture Collection; PI, propidium iodideAnthracycline deri
Keywords: مقاومت چنددارویی; PVC, polyvinyl chloride; TBT, tributyltin; DBT, dibutyltin; IC50, half inhibitory concentration; MDR, multidrug resistance; Pgp, P-glycoprotein; PEG, polyethylene glycol; GI50, growth inhibition 50%; ID50, the half-inhibition dose; NSAIDs, non-steroidal a
Keywords: مقاومت چنددارویی; Anthracyclines; Electron beam irradiation; Multidrug resistance; Apoptosis; Acute lymphoblastic leukemiaDAU, daunorubicin; DOX, doxorubicin; EPI, epirubicin; IR, irradiated; NIR, non-irradiated; MDR, multidrug resistance
Prediction and characterization of P-glycoprotein substrates potentially bound to different sites by emerging chemical pattern and hierarchical cluster analysis
Keywords: مقاومت چنددارویی; P-gp, P-glycoprotein; ABC, ATP-binding cassette; MDR, multidrug resistance; EP, emerging pattern; ECP, emerging chemical pattern; ECPG, emerging chemical pattern group; TM, transmembrane; TMD, transmembrane domain; NBD, nucleotide-binding domain; SBS, sub
Tangeretin, a citrus pentamethoxyflavone, antagonizes ABCB1-mediated multidrug resistance by inhibiting its transport function
Keywords: مقاومت چنددارویی; MDR, Multidrug resistance; P-gp, glycoprotein P; ABC, ATP-binding cassette; PTX, paclitaxel; DOX, doxorubicin; NSCLC, non-small cell lung cancer; CI, combination index; Rho 123, rhodamin123Tangeretin (PubChem CID: 69077); Paclitaxel (PubChem CID: 36314);
Inhibition of protein glycosylation reverses the MDR phenotype of cancer cell lines
Keywords: مقاومت چنددارویی; ABC, ATP binding cassette superfamily; BCRP/ABCG2, breast cancer resistance protein; BSA, bovine serum albumin; FBS, foetal bovine serum; GAPDH, glyceraldehydes-3-phosphate dehydrogenase; MDR, multidrug resistance; MEME, minimum essential medium eagle; PB
Decreased expression of nucleophosmin/B23 increases drug sensitivity of adriamycin-resistant Molt-4 leukemia cells through mdr-1 regulation and Akt/mTOR signaling
Keywords: مقاومت چنددارویی; NPM/B23, nucleophosmin/B23; ALL, acute lymphoblastic leukemia; MDR, multidrug resistance; P-gp, P-glycoprotein; ADM, adriamycin; DNR, daunorubicin; CTX, cyclophosphamide; VCR, vincristine; VP16, etoposide; IC50, half inhibitory concentration; RNAi, RNA in
Development of resistance to antiglioma agents in rat C6 cells caused collateral sensitivity to doxorubicin
Keywords: مقاومت چنددارویی; GBM, glioblastoma multiforme; MDR, multidrug resistance; BCNU, 1,3-Bis(2-chloroethyl)-1-nitrosourea; ROS, reactive oxygen species; NF-kB, nuclear factor kappa-light-chain-enhancer of activated B cells; Nrf2, nuclear factor (erythroid-derived 2)-like 2; HI
Exploiting a novel miR-519c–HuR–ABCG2 regulatory pathway to overcome chemoresistance in colorectal cancer
Keywords: مقاومت چنددارویی; ABCG2, ATP-binding cassette sub-family G member 2 transporter; CRC, colorectal cancer; FTC, fumitremorgin; HuR, ELAV-like protein 1 or human antigen R; MDR, multidrug resistance; PhA, pheophorbide A; 3′UTR, 3′untranslated region; 5-FU, 5-fluorouracilABCG2
Activity of the dietary flavonoid, apigenin, against multidrug-resistant tumor cells as determined by pharmacogenomics and molecular docking
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; MDR, multidrug resistance; BCRP, breast cancer resistance proteinChemotherapy; Flavonoids; Multidrug resistance; Natural products, Pharmacogenomics, Molecular docking and modelling.
Evaluation of blood–brain barrier and blood–cerebrospinal fluid barrier permeability of 2-phenoxy-indan-1-one derivatives using in vitro cell models
Keywords: مقاومت چنددارویی; PIOs, 2-phenoxy-indan-1-one derivatives; AD, Alzheimer's disease; CNS, central nervous system; BBB, blood–brain barrier; BCSFB, blood–cerebrospinal fluid barrier; MDCK, Madin–Darby canine kidney; P-gp, P-glycoprotein; MDR, multidrug resistance; CP, choroi
New examples of membrane protein expression and purification using the yeast based Pdr1-3 expression strategy
Keywords: مقاومت چنددارویی; ATP binding cassette (ABC) transporters; Multidrug resistance; P-type ATPases; Floppases; Membrane protein overexpressionGPD, gylceraldehyde-3-phosphate dehydrogenase; LTE, lipid translocating enzyme; MDR, multidrug resistance; PDR, pleiotropic drug resis
L-1416, a novel MDR reversing agent with possible reduced calcium antagonism
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; VER, verapamil; VBL, vinblastine; DOX, doxorubicin; VCR, vincristineL-1416; P-gp inhibitor; Tumor therapy; Calcium antagonism
A comparative study of class 1 integrons in Acinetobacter baumannii
Keywords: مقاومت چنددارویی; DNA, deoxyribonucleic acid; MDR, multidrug resistance; IntI, integrase; HGT, horizontal gene transfer; IS, insertion sequence; AbaRs, antibiotic resistance islandsAcinetobacter baumannii; Integron; Integrase
Doxorubicin delivery enhanced by electroporation to gastrointestinal adenocarcinoma cells with P-gp overexpression
Keywords: مقاومت چنددارویی; EP, electroporation; ECT, electrochemotherapy; DOX, doxorubicin; MDR, multidrug resistance; MDR1, multidrug resistance protein 1; P-gp, permeability glycoprotein; TEM, transmission electron microscopy; CLSM, confocal laser microscopy; rER, rough endoplasm
Dioscin enhances methotrexate absorption by down-regulating MDR1 in vitro and in vivo
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; Caco-2 cells, human colon adenocarcinoma cells; MDR, multidrug resistance; MDR1, multidrug resistance 1; MTT, 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; MTX, methotrexate; ADR, adriamycin; Ver, verapamil; Rif,
Kinetic Analysis of Rhodamines Efflux Mediated by the Multidrug Resistance Protein (MRP1)
Keywords: مقاومت چنددارویی; MRP1, multidrug resistance associated protein; P-gp, P-glycoprotein; MDR, multidrug resistance; Rh 6G, Rhodamine 6G; TMR, tetramethylrosamine; Rh I, tetramethylrhodamine ethyl ester or rhodamine I; Rh II, tetramethylrhodamine methyl ester or rhodamine II;
Telatinib reverses chemotherapeutic multidrug resistance mediated by ABCG2 efflux transporter in vitro and in vivo
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; ABCB1, ABC transporter-subfamily B member 1; ABCG2, ABC transporter-subfamily G member 2; MDR, multidrug resistance; VEGFR, vascular endothelial growth factor receptor; TKI, tyrosine kinase inhibitorABC transporter; ABCG2; Multi
Human ATP-Binding Cassette transporters ABCB1 and ABCG2 confer resistance to CUDC-101, a multi-acting inhibitor of histone deacetylase, epidermal growth factor receptor and human epidermal growth factor receptor 2
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; ABC, ATP-binding cassette; HDAC, histone deacetylase; EGFR, epidermal growth factor receptor; HER2, human epidermal growth factor receptor 2Multidrug resistance; EGFR; HDAC; HER2; CUDC-101
Curcumin induces apoptosis of multidrug-resistant human leukemia HL60 cells by complex pathways leading to ceramide accumulation
Keywords: مقاومت چنددارویی; DGK, diacylglycerol kinase; FBS, fetal bovine serum; GCS, glucosylceramide synthase; MDR, multidrug resistance; MTT, 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide; nSMase, neutral sphingomyelinase; PDMP, D,L-threo-1-phenyl-2-decanoylamino-
Hydroxypropyl-Sulfobutyl-β-Cyclodextrin Improves the Oral Bioavailability of Edaravone by Modulating Drug Efflux Pump of Enterocytes
Keywords: مقاومت چنددارویی; cyclodextrins; edaravone; bioavailability; permeability; P-glycoprotein; lipid raft; Caco-2 cells; pharamcokinetics; solubility; CDs, cyclodextrins; HP-SBE-βCD, hydroxypropylsulfobutyl-β-cyclodextrin; HP-βCD, hydroxypropyl-β-cyclodextrin; SBE-βCD, su
The role of a Schiff base scaffold, N-(2-hydroxy acetophenone) glycinate-in overcoming multidrug resistance in cancer
Keywords: مقاومت چنددارویی; CuNG, Copper N-(2-hydroxyacetophenone)glycinate; EAC/Dox, Doxorubicin resistant Ehrlich ascites carcinoma cells; FeNG, Iron N-(2-hydroxy acetophenone)glycinate; FoxP3, Forkhead box P3; GSH, Glutathione; MDR, Multidrug resistance; MAPK, Mitogen-activated p
The novel pyrrolo-1,5-benzoxazepine, PBOX-6, synergistically enhances the apoptotic effects of carboplatin in drug sensitive and multidrug resistant neuroblastoma cells
Keywords: مقاومت چنددارویی; Bcl-2, B cell lymphoma-2; BCRP, breast cancer resistance protein; CML, chronic myeloid leukaemia; DTT, Dithiothreitol; FAC, fluorescence associated cell sorter; FBS, foetal bovine serum; Mcl-1, Myeloid cell leukaemia 1; MDR, multidrug resistance; MRP1, mu
Comparative evaluation of two dye probes in the rat everted gut sac model for unambiguous classification of P-gp substrate and inhibitor
Keywords: مقاومت چنددارویی; Ab, beta-amyloid; Ab-HiLyte, HiLyte Fluor™ TR-labeled; AD, Alzheimer's disease; BBB, blood–brain barrier; MDR, multidrug resistance; P-gp, P-glycoprotein; Rho, rhodamine 123Beta-amyloid; Rat everted gut sac assay; P-glycoprotein; MC18; MC266; HiLyte Fluor
MDR-selective microbial-based therapy: A novel approach to cancer treatment
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; MBT, MDR-selective bacterial therapy; BCG, Bacillus Calmete–Guerin; MRP, Multidrug resistance-associated protein; Pgp, P-glycoprotein; MIC, minimum inhibitory concentration; MHC, major histocompatibility complex; CADD, chlamydia
Influence of CYP3A4, CYP3A5 and MDR-1 polymorphisms on tacrolimus pharmacokinetics and early renal dysfunction in liver transplant recipients
Keywords: مقاومت چنددارویی; CYP450, cytochrome P450 enzymes; MDR, multidrug resistance; P-gp, P-glycoprotein; C/D ratio, tacrolimus concentration/dose ratio; ALT, alanine aminotransferase; ALP, alkaline phosphatase; CNI, calcineurin inhibitor; MA, microalbumin; IGU, urine immunoglob
In vivo effect of Schisandrin B on cytochrome P450 enzyme activity
Keywords: مقاومت چنددارویی; Sch A, Schisandrin A; Sch B, Schisandrin B; SchE, Schisandra sphenanthera extract; P-gp, P-glycoprotein; MDR, multidrug resistance; CYP, cytochrome P450; CYP3A, cytochrome P450 3A; CYP3A4, cytochrome P450 3A4; IC50, the half maximal (50%) inhibitory conce
Knockdown of nucleophosmin by RNA interference reverses multidrug resistance in resistant leukemic HL-60 cells
Keywords: مقاومت چنددارویی; ADR, adriamycin; AML, acute myeloid leukemia; DNR, daunorubicin; ECL, enhanced chemiluminescence; IC50, half inhibitory concentration; LV, lentivirus; MDR, multidrug resistance; NPM, nucleophosmin; NBT, nitroblue tetrazolium reduction; PI, propidium iodid
Naphthalenyl derivatives for hitting P-gp/MRP1/BCRP transporters
Keywords: مقاومت چنددارویی; MDR, MultiDrug Resistance; ABC, ATP Binding Cassette; P-gp, P-glycoprotein; BCRP, Breast Cancer Resistance Protein; MRP1, MultiDrug Resistance-associated Protein1; Papp, apparent permeability; Calcein-AM, Acetoxymethyl esters of calcein; MDCK, Madin-Darby
Oroxylin A reverses P-glycoprotein-mediated multidrug resistance of MCF7/ADR cells by G2/M arrest
Keywords: مقاومت چنددارویی; MCF7/ADR, Adriamycin resistant human breast cancer cell line; MDR, multidrug resistance; Chk2, checkpoint kinase 2; NF-κB, nuclear factor-kappa B; PMSF, phenylmethylsulfonyl fluorideOroxylin A; MCF7/ADR; G2/M; P-gp; Chk2
Overexpression of ATP-binding cassette transporter ABCG2 as a potential mechanism of acquired resistance to vemurafenib in BRAF(V600E) mutant cancer cells
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; ABC, ATP-binding cassette; EGFR, epidermal growth factor receptor; TKI, tyrosine kinase inhibitor; PBS, phosphate-buffered saline; FTC, Fumitremorgin C; IAAP, Iodoarylazidoprazosin; MTT, 3-(4,5-dimethylthiazol-yl)-2,5-diphenylla
Berberine analogue IMB-Y53 improves glucose-lowering efficacy by averting cellular efflux especially P-glycoprotein efflux
Keywords: مقاومت چنددارویی; P-gp, P-glycoprotein; MDR, multidrug resistance; MRP, multidrug resistance-associated protein; BBR, Berberine; LDLR, low-density-lipoprotein receptor; InsR, insulin receptor; AMPK, AMP-activated protein kinase; IMB-Y53, pseudo-berberine; Tet, tetrandrine;
Nilotinib potentiates anticancer drug sensitivity in murine ABCB1-, ABCG2-, and ABCC10-multidrug resistance xenograft models
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; ABC, ATP-binding cassette; ABCB1, also called P-gp (P-glycoprotein); ABCG2, also called BCRP (breast cancer resistance protein)/MXR (mitoxantrone resistance protein); ABCC1, also called MRP1 (multidrug resistance protein 1); EGF
A conserved interdomain communication pathway of pseudosymmetrically distributed residues affects substrate specificity of the fungal multidrug transporter Cdr1p
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; PDR, pleiotropic drug resistance; ABC, ATP-binding cassette; NBD, nucleotide binding domain; TMD, transmembrane domain; TM, transmembrane; SCA, statistical coupling analysis; 4-NQO, 4-nitroquinoline 1-oxide; DiOC6, 3,3′-dihexylo
Synthesis of N4-(substituted phenyl)-N4-alkyl/desalkyl-9H-pyrimido[4,5-b]indole-2,4-diamines and identification of new microtubule disrupting compounds that are effective against multidrug resistant cells
Keywords: مقاومت چنددارویی; CA-4, combretastatin A-4; MDR, multidrug resistance; Pgp, P-glycoprotein’; Rr, relative resistance; DAMA colchicine, N-deacetyl-N-(2-mercaptoacetyl)colchicinePyrimido[4,5-b]indole-2,4-diamines; Microtubules; Multidrug resistance
Alanine scanning of all cysteines and construction of a functional cysteine-less Cdr1p, a multidrug ABC transporter of Candida albicans
Keywords: مقاومت چنددارویی; ABC, ATP binding cassette; MFS, major facilitator superfamily; MDR, multidrug resistance; MIC, minimum inhibitory concentration; FLC, fluconazole; CYH, cycloheximide; ITR, itraconazole; KTC, ketoconazole; MIC, miconazole; ANI, anisomycin; DIC, differentia
Elucidation of the therapeutic enhancer mechanism of poly-S-nitrosated human serum albumin against multidrug-resistant tumor in animal models
Keywords: مقاومت چنددارویی; MDR, multidrug resistance; NO, Nitric oxide; HSA, human serum albumin; Poly-SNO-HSA, poly-S-nitrosated HSA; dx, doxorubicinHuman serum albumin; Nitric oxide; S-nitrosation; Anticancer; p-glycoprotein; HIF-1α
Reversal of P-glycoprotein-mediated multidrug resistance by a synthetic α-aminoxy peptidomimetic
Keywords: مقاومت چنددارویی; DMEM, Dulbecco's modified Eagle's medium; Dox, doxorubicin; ER, efflux ratio; FBS, fetal bovine serum; HBSS, Hanks’ balanced salt solution; IS, internal standard; Lys-P, lysine-peptidomimetic; MDR, multidrug resistance; MRP1, multidrug resistance-associat
Fabrication of magnetic nanoparticles with controllable drug loading and release through a simple assembly approach
Keywords: مقاومت چنددارویی; ABC, ATP-binding cassette; DA, dopamine; DOX, doxorubicin; MDR, multidrug resistance; MRI, magnetic resonance imaging; PEG, poly (ethylene glycol); NP-DOX, DOX-loaded nanoparticles; PBAE, poly (beta-amino ester); SPIONs, superparamagnetic iron oxide nanop
Up-regulation of FXR isoforms is not required for stimulation of the expression of genes involved in the lack of response of colon cancer to chemotherapy
Keywords: مقاومت چنددارویی; CDDP, cis-diamminedichloroplatinum(II); CRAC, colorectal adenocarcinoma; 5-FU, 5-fluorouracil; FXR, farnesoid X receptor; MDR, multidrug resistance; MOC, mechanism of chemoresistance; TKI, tyrosine kinase inhibitor; TLDA, Taqman Low-Density ArrayChemoresi
Minor structural modifications to alchemix influence mechanism of action and pharmacological activity
Keywords: مقاومت چنددارویی; CHO, Chinese hamster ovary; CT DNA, calf thymus DNA; DMSO, dimethyl sulphoxide; DSB, double strand break; H2AX, histone-2AX; MDR, multidrug resistance; MTT, (3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; TdT, terminal deoxynucleotidyl tran
Curcumin reverses cis-platin resistance and promotes human lung adenocarcinoma A549/DDP cell apoptosis through HIF-1α and caspase-3 mechanisms
Keywords: مقاومت چنددارویی; Cur, curcumin; DDP, cis-platin; HIF-1, hypoxia-inducible factor 1; MDR, multidrug resistance; MTT, 3-[4,5-dimethylthiazol-2-yl]2,5-diphenyltetrazolium bromide; DAPI, 4′,6-diamidino-2-phenylindole; DMSO, dimethyl sulfoxide; RT-PCR, reverse transcription po
Microparticles and their emerging role in cancer multidrug resistance
Keywords: مقاومت چنددارویی; DNR, daunorubicin; FCM, flow cytometry; MFI, mean fluorescence intensity; MPs, microparticles; MDR, multidrug resistance; MRP1, Multidrug Resistance-Associated Protein 1; P-gp, P-glycoproteinMicroparticles; Multidrug resistance; P-glycoprotein; Multidrug
Pharmacogenomic determination of genes associated with sensitivity or resistance of tumor cells to curcumin and curcumin derivatives
Keywords: مقاومت چنددارویی; ABC transporter, ATP-binding cassette (ABC) transporter; MDR, multidrug resistance; MDR1, multidrug resistance gene 1; MRP1, multidrug resistance-related protein 1; NCI, National Cancer Institute; TCM, traditional Chinese medicineCancer; Curcumin; ABC tra
Antitumor agents 292. Design, synthesis and pharmacological study of S- and O-substituted 7-mercapto- or hydroxy-coumarins and chromones as potent cytotoxic agents
Keywords: مقاومت چنددارویی; Coumarin; Synthesis; Cytotoxicity; Cell cycle arrestHIV, Human immunodeficiency virus; CYP, Cytochrome P450; MDR, Multidrug resistance; DMDCK, (±)-3′-O-4′-O-bis(3,4-dimethoxycinnamoyl)-cis-khellactone; DSP, 3′R,4′R-disubstituted-2′,2′-dimethyldihydropyran