Keywords: کینازولین; Liver functions; Ulcers; Dexamesathone; Quinazoline; Acetamide; Ulcerative colitis;
مقالات ISI کینازولین (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: کینازولین; Leishmaniasis; Resistance; Oxindole; Benzimidazole; Quinazoline;
Keywords: کینازولین; Quinazoline; Structure-activity relationship; Drug design and development; Therapeutic agents; Pharmacological significance;
Quinazoline-directed selective ortho-iodination for the synthesis of 2-(2-iodoaryl)-4-arylquinazolines
Keywords: کینازولین; C-H activation; Selective iodination; Palladium catalysis; Quinazoline;
Keywords: کینازولین; DFT; ALIE; RDF; BDE; Quinazoline; Molecular docking;
Keywords: کینازولین; Quinazoline; Antihyperlipidemic; Hypoglycemic;
Keywords: کینازولین; Quinazoline; Supercritical water; Oxidation; Reaction mechanism;
Keywords: کینازولین; Ruthenium; Quinazoline; Transfer hydrogenation; Ketone; Secondary alcohols;
Keywords: کینازولین; Niementowski reaction; Quinazoline; Heterocycle; Cyclisation; Medium-ring;
Keywords: کینازولین; Cascade reaction; Tandem sequence; Beckmann rearrangement; Electrophilic aromatic substitution; Quinazoline;
Keywords: کینازولین; Trypanosoma cruzi; Leishmania mexicana; Plasmodium berghei; Quinazoline; Dihydrofolate reductase; Pteridin reductase;
Keywords: کینازولین; Carbonic anhydrase; Sulfonamide; Quinazoline; Tail approach;
Keywords: کینازولین; Leishmania mexicana; Quinazoline; Antiprotozoan activityPTR1, Pteridine reductase 1; DHFR, Dyhydrofolate reductase; IC50, Half inhibitory concentration; TAQ, Quinazoline-2,4,6-triamine; PDB, Protein Data Bank
Keywords: کینازولین; Solid-phase synthesis; Alkoxyamine Linker; Benzimidazole; Quinazoline; Quinazolinone;
Keywords: کینازولین; Quinazoline; Benzimidazole; Primary amines; Antitumor activity;
Keywords: کینازولین; Microwave irradiation; Ultrasonic; Ionic liquid; Quinazoline; Pyrimidine;
Keywords: کینازولین; Vasicinone; Quinazoline; Synthesis; Bronchodilator; Toxicity;
Keywords: کینازولین; Synthesis; Quinazoline; In-vitro antitumor evaluation; Selective activity; NCI
Keywords: کینازولین; Synthesis; Quinazoline; In-vitro antitumor evaluation; NCI; Molecular docking;
Keywords: کینازولین; TNNI3K; B-Raf; Quinazoline; Substituent effects; Kinase selectivity
Keywords: کینازولین; Quinazoline; N,N based ligand; Ruthenium; Asymmetric transfer hydrogenation
Keywords: کینازولین; Quinazoline; Sulfonamides; Sulfonylthioureas; Carbonic anhydrase; Antitumor
Discovery of selective 2,4-diaminoquinazoline toll-like receptor 7 (TLR 7) agonists
Keywords: کینازولین; HBV; TLR7; Quinazoline;
Discovery and lead identification of quinazoline-based BRD4 inhibitors
Keywords: کینازولین; BET inhibitor; BRD4; Bromodomain; Quinazoline; Cancer; Inflammation;
Novel quinazoline derivatives bearing various 6-benzamide moieties as highly selective and potent EGFR inhibitors
Keywords: کینازولین; EGFR; Kinase inhibitor; Quinazoline; High selectivity; Anti-cancer;
Synthesis, structural characterization, spectroscopic, and DFT studies of two penta-coordinated zinc(II) complexes containing quinazoline and 1, 10-phenanthroline as mixed ligands
Keywords: کینازولین; Spectroscopic studies; DFT calculations; Zinc(II) complexes; Quinazoline; 1,10-phenanthroline; Crystal structures;
Synthesis and biological evaluation of novel quinazoline-4-piperidinesulfamide derivatives as inhibitors of NPP1
Keywords: کینازولین; NPP1 inhibitor; Quinazoline; Sulfamide; Calcific aortic valve disease;
Quinazoline-1-deoxynojirimycin hybrids as high active dual inhibitors of EGFR and α-glucosidase
Keywords: کینازولین; Quinazoline; 1-Deoxynojirimycin; Hybrids; Epidermal growth factor receptor (EGFR); α-Glucosidase; Enzyme inhibitors;
Identification of quinazoline based inhibitors of IRAK4 for the treatment of inflammation
Keywords: کینازولین; IRAK4; Quinazoline; Serine-threonine kinase; Kinase inhibitor; Inflammatory disease; HVQXFGHHSFTACS-CXIWYSOXSA-N;
Iron-catalyzed Csp3Csp3 bond formation via dehydrative cross coupling reaction: Facile access to new hybrid dihydroquinazolines having quinoline, isoquinoline, quinoxaline and azoles
Keywords: کینازولین; Cross coupling; Dehydrative; Iron catalyst; Quinazoline;
An alternative synthesis of Vandetanib (Caprelsaâ¢) via a microwave accelerated Dimroth rearrangement
Keywords: کینازولین; Vandetanib; Quinazoline; Dimroth rearrangement; Tyrosine kinase inhibitor;
Quinazolinone-benzimidazole conjugates: Synthesis, characterization, dihydrofolate reductase inhibition, DNA and protein binding properties
Keywords: کینازولین; Quinazoline; Benzimidazole; DHFR; Calf thymus DNA; Bovine serum albumin;
Supercritical water oxidation of quinazoline: Reaction kinetics and modeling
Keywords: کینازولین; Quinazoline; Supercritical water oxidation; Kinetics; Modeling; Reaction mechanism;
Structure-activity relationship studies of G9a-like protein (GLP) inhibitors
Keywords: کینازولین; GLP; G9a; Inhibitor; Quinazoline; Quinoline;
Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines
Keywords: کینازولین; Quinazoline; Quinone; α1-Adrenoreceptor antagonist; DNA fragmentation; Antiproliferative activity; α1-AR; α1-adrenoreceptor; BPH; benign prostatic hyperplasia; CHO; Chinese hamster ovary; Dox; doxazosin; GSH; glutathione; LUTS; lower urinary tract symp
Design and synthesis of quinazolinones as EGFR inhibitors to overcome EGFR resistance obstacle
Keywords: کینازولین; Quinazoline; Non Small Cell Lung Cancer; T790M EGFR;
Research paper2-Guanidino-quinazolines as a novel class of translation inhibitors
Keywords: کینازولین; Protein synthesis; Bacteria; Antibacterial; Translation; Reporter strain; Screening; Quinazoline;
Design, synthesis, and docking studies of quinazoline analogues bearing aryl semicarbazone scaffolds as potent EGFR inhibitors
Keywords: کینازولین; Quinazoline; Aryl semicarbazone scaffolds; Synthesis; Docking; Anti-tumor activity;
Ultrasonic treatment of CoFe2O4@B2O3-SiO2 as a new hybrid magnetic composite nanostructure and catalytic application in the synthesis of dihydroquinazolinones
Keywords: کینازولین; Ultrasonic irradiation; Hybrid magnetic nanocatalysts; Composite nanostructure; Glass-ceramic; Quinazoline;
A novel quinazoline-based analog induces G2/M cell cycle arrest and apoptosis in human A549 lung cancer cells via a ROS-dependent mechanism
Keywords: کینازولین; Reactive oxygen species; Cell cycle; G2/M arrest; Michael acceptor; Quinazoline;
Design and synthesis of quinazoline-3,4-(4H)-diamine endowed with thiazoline moiety as new class for DPP-4 and DPPH inhibitor
Keywords: کینازولین; Quinazoline; Thiazoline; DPP-4 inhibitors; DPPH; Molecular docking;
Quinazoline derivatives as selective CYP1B1 inhibitors
Keywords: کینازولین; Quinazoline; CYP1B1; Cancer chemoprevention; Sacchrosomes; Selective CYP1B1 inhibitor;
Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold
Keywords: کینازولین; Quinazoline; Quinoline; Quinoxaline; Thienopyrimidine; Trichloromethyl goup; Plasmodium falciparum; In vitro antiplasmodial activity; In vitro HepG2 cytotoxicity; Structure-activity relationships;
Spectroscopic and reactive properties of a newly synthesized quinazoline derivative: Combined experimental, DFT, molecular dynamics and docking study
Keywords: کینازولین; DFT; IR and Raman; BDE; RDF; Quinazoline; Molecular docking;
Stereoselective synthesis of benzosulfamidate-fused tetrahydroquinazoline scaffold via organocatalytic [4+2] cycloaddition of 2-amino-β-nitrostyrenses of cyclic N-sulfimines
Keywords: کینازولین; Benzosulfamidate; Quinazoline; Cycloaddition reaction; Michael reaction; Organocatalyst;
DABCO-catalyzed one-pot three component synthesis of dihydropyrano[3,2-c]chromene substituted quinazolines and their evaluation towards anticancer activity
Keywords: کینازولین; Multicomponent reaction; Knoevenagel–Michael reaction; Quinazoline; 4-Hydroxycoumarin; DABCO; Anti-cancer
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors
Keywords: کینازولین; EGFR inhibitors; NSCLC; Quinazoline; Molecular docking; Anti-cancer
Synthesis of aminomethyl quinazoline based ruthenium (II) complex and its application in asymmetric transfer hydrogenation under mild conditions
Keywords: کینازولین; Asymmetric transfer hydrogenation; NN ligand; Quinazoline; Ruthenium
Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma
Keywords: کینازولین; Carbonic anhydrase; Quinazoline; Sulfonamides; Mercaptan; Tumor-associated isoforms
Thermal [3Â + 2] cycloaddition of N-iminoquiazoline ylides with allenoates for synthesis of tetrahydropyrazoloquinazoline derivatives
Keywords: کینازولین; Cycloaddition; Allenoates; Azomethine imine; N-iminoquiazoline ylide; Quinazoline;