Keywords: ریمونابانت، آکومپلیا; Magnesium carbonate; Mesoporous; Hydroxypropyl methylcellulose; Tolfenamic acid; Rimonabant; Supersaturation;
مقالات ISI ریمونابانت، آکومپلیا (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: ریمونابانت، آکومپلیا; Conditioned place preference; Ethanol; Rimonabant; Cannabinoid; Conditioning; Environment;
Keywords: ریمونابانت، آکومپلیا; Avoidance behavior; Response extinction; CB1 receptors; Dopamine D1 receptors; AM404; SDA; step-down inhibitory avoidance; C57BL/6N; C57BL/6NCrl; EBT; exposure based therapy; ECS; endocannabinoid system; D1-CB1â/â; conditional D1-CB1 knock-out mic
The effect of cannabinoid receptor 1 blockade on hepatic free fatty acid profile in mice with nonalcoholic fatty liver disease
Keywords: ریمونابانت، آکومپلیا; NAFLD; Endocannabinoid system; Rimonabant; CB1 receptor blockade; Free fatty acid profile; Mice;
Keywords: ریمونابانت، آکومپلیا; Drug repurposing; Tuberculosis; Rimonabant; BM212; Sila analogue; MmpL3 inhibitorMIC, Minimum Inhibitory Concentration; ADME, absorption, distribution, metabolism, excretion; CB1, Cannabinoid receptor Type 1; Mtb, Mycobacterium tuberculosis; CNS, Central
Keywords: ریمونابانت، آکومپلیا; AM251; 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(1-piperidyl)pyrazo-le-3-carboxamide; BSA; bovine serum albumin; DAMGO; [d-Ala2, N-MePhe4, Gly-ol]-enkephalin; DIEA; diisopropylethylamine; DMF; dimethylformamide; EGTA; ethylene glycol-bis(2-amino
Keywords: ریمونابانت، آکومپلیا; Sal; saline; Veh; vehicle; Rim; rimonabant; Eth; ethanol; Mor; morphine; Coc; cocaine; VTA; ventral tegmental area; NAc; nucleus accumbens; GABA; gamma-aminobutyric acid; Behavioral sensitization; Cocaine; Ethanol; Morphine; Rimonabant;
Keywords: ریمونابانت، آکومپلیا; Rimonabant; Naloxone; norBNI; Cannabinoid; Opioid; Mouse; Obesity; Diabetes;
Keywords: ریمونابانت، آکومپلیا; CB1R; Cannabis; Cannabinoid; Marijuana; PET; Rimonabant; Radioligand; Prefrontal cortex; Schizophrenia;
Keywords: ریمونابانت، آکومپلیا; 2-AG; 2-arachidonoylglycerol; AEA; N-arachidonylethanolamine anandamide; CB1R; cannabinoid type one receptor; CBG; corticosteroid-binding globulin; CRH; corticotrophin-releasing hormone; eCB; endocannabinoid; ECS; endocannabinoid signaling; epm; elevated
Keywords: ریمونابانت، آکومپلیا; Paced mating; Sexual motivation; THC; Anandamide; Locomotion; Rimonabant; AEA; SR141716A;
Keywords: ریمونابانت، آکومپلیا; Endocannabinoid; Cannabinoid 1 (CB1) receptor antagonists; Obesity; Rimonabant
Keywords: ریمونابانت، آکومپلیا; Anxiety; Depression; Palatability; Appetite; Cannabinoid; CB1; Tetrahydrocannabivarin; Cannabidiol; Cannabigerol; Rimonabant; Delta-9-tetrahydrocannabinol;
Keywords: ریمونابانت، آکومپلیا; Adjusting-delay procedure; Cannabinoids; Delay discounting; Impulsive choice; Obese Zucker rat; Rimonabant;
Keywords: ریمونابانت، آکومپلیا; Nucleus accumbens core; Cannabinoid system; Cannabinoid receptor 1; Conditioned place preference; Morphine withdrawal; Rimonabant;
Keywords: ریمونابانت، آکومپلیا; Δ9-Tetrahydrocannabinol; Dependence; Rimonabant; Sex differences
Melatonin attenuates Î9-tetrahydrocannabinol-induced reduction in rat sperm motility and kinematics in-vitro
Keywords: ریمونابانت، آکومپلیا; HAM; hyper-activated motility; SR141716; rimonabant; AM-630; iodopravadoline; THC; Î9-tetrahydrocannabinol; CB; cannabinoid receptor; CASA; computer-assisted sperm analyser; CSC; annabis sativa; ZP; zona pellucida; BWW; Biggers-Whitten-Whittingham; B
The quest for endothelial atypical cannabinoid receptor: BKCa channels act as cellular sensors for cannabinoids in in vitro and in situ endothelial cells
Keywords: ریمونابانت، آکومپلیا; N-arachidonoyl glycine; Abnormal cannabidiol; Rimonabant; Mouse aorta; Endothelial cells; BKCa channels;
Novel behavioral assays of spontaneous and precipitated THC withdrawal in mice
Keywords: ریمونابانت، آکومپلیا; 2-AG; 2-arachidonoylglycerol; CB1; Cannabinoid receptor subtype 1; CB2; Cannabinoid receptor subtype 2; FAAH; Fatty acid amide hydrolase; JZL184; 4-nitrophenyl-4-[bis(1,3-benzodioxol-5-yl)(hydroxy)methyl]piperidine-1-carboxylate; JWH-018; Naphthalen-1-yl-
Intra-accumbal blockade of endocannabinoid CB1 receptors impairs learning but not retention of conditioned relief
Keywords: ریمونابانت، آکومپلیا; Backward conditioning; Nucleus accumbens; Rats; Rimonabant; SR141716A; Startle response;
Rimonabant, a selective cannabinoid1 receptor antagonist, protects against light-induced retinal degeneration in vitro and in vivo
Keywords: ریمونابانت، آکومپلیا; Age-related macular degeneration; Cannabinoid; Oxidative stress; Photoreceptor; Rimonabant;
Research articlePost-sensitization treatment with rimonabant blocks the expression of cocaine-induced behavioral sensitization and c-Fos protein in mice
Keywords: ریمونابانت، آکومپلیا; Behavioral sensitization; Cannabinoid; C-Fos expression; Cocaine; Conditioning; Rimonabant;
Système endocannabinoïde : effets sur le métabolisme glucidique, mais aussi lipidique
Keywords: ریمونابانت، آکومپلیا; Système endocannabinoïde; récepteur cannabinoïde de type 1 (CB1-R); anandamide; rimonabant; lipides; tissu adipeux; stéatose hépatique; insulino-résistance; syndrome métabolique; diabète de type 2; Endocannabinoid system; cannabinoid type 1-recep
Pure Î9-tetrahydrocannabivarin and a Cannabis sativa extract with high content in Î9-tetrahydrocannabivarin inhibit nitrite production in murine peritoneal macrophages
Keywords: ریمونابانت، آکومپلیا; BSA; albumin bovine serum; CB1; cannabinoid receptor type 1; CB2; cannabinoid receptor type 2; CBC; cannabichromene; CBD; cannabidiol; CBG; cannabigerol; COX-2; cyclooxygenase-2; DAN; 2,3-diaminonaphthalene; DMSO; dimethyl sulfoxide (DMSO); DTT; 1,4-dithi
A PET study comparing receptor occupancy by five selective cannabinoid 1 receptor antagonists in non-human primates
Keywords: ریمونابانت، آکومپلیا; Cannabinoid 1 receptor (CB1R) antagonists; Obesity; Positron emission tomography (PET); Receptor occupancy; [11C]SD5024; Rimonabant; TaranabantAZ, AstraZeneca; AUC, area under the curve; BBB, blood–brain barrier; CB1R, cannabinoid 1 receptor; CD, candidat
Enhanced discriminative stimulus effects of Î9-THC in the presence of cannabidiol and 8-OH-DPAT in rhesus monkeys
Keywords: ریمونابانت، آکومپلیا; Cannabinoid; Rhesus monkey; Drug discrimination; Cannabidiol; 8-OH-DPAT; Serotonin; 5-HT1A; Rimonabant; Dependence;
Phenotypic assessment of THC discriminative stimulus properties in fatty acid amide hydrolase knockout and wildtype mice
Keywords: ریمونابانت، آکومپلیا; Î9-Tetrahydrocannabinol; Anandamide; Fatty acid amide hydrolase; 2-arachidonoylglycerol; Drug discrimination; Rimonabant;
The intracerebroventricular injection of rimonabant inhibits systemic lipopolysaccharide-induced lung inflammation
Keywords: ریمونابانت، آکومپلیا; ICV; intracerebroventricular; CB1; cannabinoid receptor type 1; LPS; lipopolysaccharide; IV; intravenous; Ppc; pulmonary capillary pressure; TLR4; toll-like receptor 4; IRAK1; interleukin receptor-associated kinase-1; IκBα; inhibitor of nuclear factor o
Design, synthesis and in vitro evaluation of novel uni- and bivalent ligands for the cannabinoid receptor type 1 with variation of spacer length and structure
Keywords: ریمونابانت، آکومپلیا; Bivalent ligand; Cannabinoid receptor; CB1; Rimonabant;
Effects of the novel cannabinoid CB1 receptor antagonist PF 514273 on the acquisition and expression of ethanol conditioned place preference
Keywords: ریمونابانت، آکومپلیا; Ethanol; Reward; Place preference; Locomotor activity; CB1; PF 514273; Rimonabant; SR141716A; Inbred mice; DBA/2J;
Short communicationInfusion of cannabidiol into infralimbic cortex facilitates fear extinction via CB1 receptors
Keywords: ریمونابانت، آکومپلیا; Fear extinction; Cannabidiol; CB1 receptor; Infralimbic cortex; Rimonabant; Conditioned freezing;
Pain as a reward: Changing the meaning of pain from negative to positive co-activates opioid and cannabinoid systems
Keywords: ریمونابانت، آکومپلیا; Pain; Reward; Endogenous opioids; Endocannabinoids; Naltrexone; Rimonabant;
Novel antiobesity agents: Synthesis and pharmacological evaluation of analogues of Rimonabant and of LH21
Keywords: ریمونابانت، آکومپلیا; LH21; 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1H-1,2,4-triazole; Rimonabant; 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide; CB1; cannabinoid receptor 1; CB2; cannabinoid receptor 2; PPARα; perox
CB1 agonists, locally applied to the cortico-thalamic circuit of rats with genetic absence epilepsy, reduce epileptic manifestations
Keywords: ریمونابانت، آکومپلیا; Seizure; Anandamide; WIN55,212; CB receptors; Rimonabant; WAG/Rij rats;
Peripherally restricted CB1 receptor blockers
Keywords: ریمونابانت، آکومپلیا; Cannabinoid receptor blocker; Inverse agonist; Silent antagonist; Peripherally restricted; CB1-antagonist; Obesity; Diabetes; Metabolic disorders; Liver diseases; Rimonabant; AM6545; JD5037;
Additive effect of rimonabant and citalopram on extracellular serotonin levels monitored with in vivo microdialysis in rat brain
Keywords: ریمونابانت، آکومپلیا; Rimonabant; Citalopram; Microdialysis; Serotonin; Locus coeruleus; Prefrontal cortex
Tolerance to hypophagia induced by prolonged treatment with a CB1 antagonist is related to the reversion of anorexigenic neuropeptide gene expression in the hypothalamus
Keywords: ریمونابانت، آکومپلیا; Hypophagia; Rimonabant; CRF; CART
Expression of the cannabinoid receptor type 1 in the pituitary of rabbits and its role in the control of LH secretion
Keywords: ریمونابانت، آکومپلیا; CB1; Endocannabinoids; Rimonabant; LH; Rabbit
Rimonabant for neurocognition in schizophrenia: A 16-week double blind randomized placebo controlled trial
Keywords: ریمونابانت، آکومپلیا; Rimonabant; Cognition; Schizophrenia; CB1 receptor antagonist; Probabilistic learning;
Rimonabant attenuates amphetamine sensitisation in a CCK2 receptor-dependent manner
Keywords: ریمونابانت، آکومپلیا; CCK2 receptors; CB1 receptors; Rimonabant; Amphetamine; Motor sensitisation; Knockout mice
Interactions of CB1 and mGlu5 receptor antagonists in food intake, anxiety and memory models in rats
Keywords: ریمونابانت، آکومپلیا; MTEP; 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pridine; SIB-1757; 6-methyl-2-(phenylazo)-3-pyridinol); Rimonabant; (5-(4-Chlorophenyl)-1-(2,4-dichloro-phenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide)hydrochloride; USV; ultrasonic vocalization;
Rimonabant abolishes sensitivity to workload changes in a progressive ratio procedure
Keywords: ریمونابانت، آکومپلیا; THC; Rimonabant; Progressive ratio; Rat; Step size
The effects of chronic administration of tranylcypromine and rimonabant on behaviour and protein expression in brain regions of the rat
Keywords: ریمونابانت، آکومپلیا; Brain-derived neurotrophic factor (BDNF); Rimonabant; Depression; Endocannabinoids; Tranylcypromine (TCP);
Rimonabant reduces the essential value of food in the genetically obese Zucker rat: An exponential demand analysis
Keywords: ریمونابانت، آکومپلیا; Behavioral economics; Essential value; Fixed ratio schedule; Obese Zucker rat; Rimonabant; Sucrose reinforcement;
JD-5006 and JD-5037: Peripherally restricted (PR) cannabinoid-1 receptor blockers related to SLV-319 (Ibipinabant) as metabolic disorder therapeutics devoid of CNS liabilities
Keywords: ریمونابانت، آکومپلیا; CB1 receptor inverse agonist; Metabolic disorders; Diabetes; Liver diseases; Dyslipidemias; Obesity; JD-5006; JD-5037; SLV-319; Peripherally restricted cannabinoid-1 receptor blockers; Rimonabant; CB1 antagonist;
CB1 receptor antagonism/inverse agonism increases motor system excitability in humans
Keywords: ریمونابانت، آکومپلیا; Transcranial magnetic stimulation; Motor cortex; CB1; Rimonabant; Spinal cord
Structural analogs of pyrazole and sulfonamide cannabinoids: Effects on acute food intake in mice
Keywords: ریمونابانت، آکومپلیا; Antagonist; Cannabinoid; Feeding; Hemopressin; Pyrazole; Rimonabant; Sulfonamide; (Mouse)
Antidepressant-like effects of Î9-tetrahydrocannabinol and rimonabant in the olfactory bulbectomised rat model of depression
Keywords: ریمونابانت، آکومپلیا; Cannabinoids; Î9-tetrahydrocannabinol; Rimonabant; Olfactory bulbectomy;
Inhibition of forebrain μ-opioid receptor signaling by low concentrations of rimonabant does not require cannabinoid receptors and directly involves μ-opioid receptors
Keywords: ریمونابانت، آکومپلیا; Rimonabant; CB1 cannabinoid receptor; μ-Opioid receptor; [35S]GTPγS binding; Radioligand binding; Docking; CB1 receptor knockout mouse; CB1/CB2 receptor double knockout mouse; Forebrain;
Blocking the postpartum mouse dam's CB1 receptors impairs maternal behavior as well as offspring development and their adult social–emotional behavior
Keywords: ریمونابانت، آکومپلیا; CB1R; Rimonabant; SR141716; Maternal behavior; USVs; Mice; Anxiety