Keywords: مهارکننده آنزیم; Silyl tacrine; Deprotonation of amine; Acetylcholinesterase; Butyrylcholinesterase; Carbonic anhydrase; Enzyme inhibitor;
مقالات ISI مهارکننده آنزیم (ترجمه نشده)
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Keywords: مهارکننده آنزیم; retinoic acid; aldehyde dehydrogenase 1A; enzyme inhibitor; pregnancy;
Keywords: مهارکننده آنزیم; Gypsophila; Natural products; Flavonoids; Antioxidant; Enzyme inhibitor;
Keywords: مهارکننده آنزیم; Folate pathway; Trypanosomatids; Structure-based drug design; Selective inhibition; Enzyme inhibitor; Anti-parasitic drug; PTR1; Pteridine reductase 1; DHFR; Dihydrofolate reductase; dUMP; Deoxyuridine monophosphate; dTMP; Deoxythymidine monophosphate; hD
Keywords: مهارکننده آنزیم; Biscoumarin; Enzyme inhibitor; Urease; Aromatase; α-Glucosidase; Steroid sulfatase; α-Amylase inhibitors; HIV-1 integrase inhibition; c-Met inhibitors; SAR;
Keywords: مهارکننده آنزیم; Carotenoids; Fungal lycopene; Enzyme inhibitor; Lycopene cyclase; Engineered microorganisms
Keywords: مهارکننده آنزیم; Glutaminyl cyclase; Flavonoids; Synthesis; Enzyme inhibitor; Alzheimer’s disease
Keywords: مهارکننده آنزیم; Sphingolipids; Enzyme inhibitor; Sphingosine lyase; Synthesis; Stereocontrolled;
Keywords: مهارکننده آنزیم; Proteins; Peptides; Insulin; Permeability; Enzyme inhibitor; Peroral
Keywords: مهارکننده آنزیم; Carbonic anhydrase; Glycine; Phenylalanine; Sulfonamide; Docking; Enzyme inhibitor
Keywords: مهارکننده آنزیم; Affinity selection mass spectrometry; Enzyme inhibitor; Rapid screening; Microextraction; Traditional Chinese medicine
Keywords: مهارکننده آنزیم; Capillary electrophoresis; Enzyme inhibitor; Pre-capillary enzyme assay; In-capillary enzyme assay; Review
Keywords: مهارکننده آنزیم; Carbonic anhydrase; Hydroxyl; Uracil; Enzyme inhibitor;
Keywords: مهارکننده آنزیم; Molecular docking; Scoring functions; Hydrophilic vs hydrophobic targets; Drug design; Enzyme inhibitor;
Keywords: مهارکننده آنزیم; Carbonic anhydrase; Enzyme inhibitor; Bisphosphonate; Bone resorption inhibitor; Matrix metalloproteinase inhibitor
Keywords: مهارکننده آنزیم; ATP; adenosine triphosphate; ADP; adenosine diphosphate; Cer; ceramide; ERK-1/2; extra-cellular signal-regulated kinase 1/2; HDAC; histone deacetylase; LDH; lactate dehydrogenase; S1P; sphingosine-1-phosphate; SAR; structure-activity relationship; Sph;
Keywords: مهارکننده آنزیم; Isostere; Purine; Triazine; Enzyme inhibitor; Anticancer; Antiviral
Keywords: مهارکننده آنزیم; Antibiotic resistance; Penicillinase; Enzyme inhibitor; Peptide inhibitor; Phage display; Surface plasmon resonance
Keywords: مهارکننده آنزیم; Tuberculosis; Enzyme inhibitor; Targeted therapy; Kinase inhibitor; Phenotypical screening
The extracellular bioactive substances of Arthrobotrys oligospora during the nematode-trapping process
Keywords: مهارکننده آنزیم; Nematode-trapping fungi; Arthrobotrys oligospora; Extracellular bioactive substances; Enzyme inhibitor; Protease
Design and synthesis of a series of bioavailable fatty acid synthase (FASN) KR domain inhibitors for cancer therapy
Keywords: مهارکننده آنزیم; FASN; Fatty acid synthase; LRS; lipid-reduced serum; NADPH; nicotinamide adenine dinucleotide phosphate; KR; ketoreductase domain; ER; enoylreductase domain; ÏME; pseudo-methyltransferase domain; ÏKR; pseudo-ketoreductase domain; Fatty acid synthase; En
Insight into the biological properties and phytochemical composition of Ballota macrodonta Boiss. et Balansa, - an endemic medicinal plant from Turkey
Keywords: مهارکننده آنزیم; Ballotama crodonta; Phenolics; Antimicrobial; Antioxidant; Enzyme inhibitor; Natural bioactive agents;
Synthesis, structure-activity relationships, and mechanistic studies of 5-arylazo-tropolone derivatives as novel xanthine oxidase (XO) inhibitors
Keywords: مهارکننده آنزیم; Xanthine oxidase; Enzyme inhibitor; Tropolone; Kinetic study; Docking-simulation study;
Evaluation of α-glucosidase inhibiting potentials with docking calculations of synthesized arylidene-pyrazolones
Keywords: مهارکننده آنزیم; Coumarins; Arylidenes; Antipyrine; Knoevenagel condensations; Enzyme Inhibitor;
7-Methylguanosine monophosphate analogues with 5â²-(1,2,3-triazoyl) moiety: Synthesis and evaluation as the inhibitors of cNIIIB nucleotidase
Keywords: مهارکننده آنزیم; ONHSLFXWBJKDSL-IDTAVKCVSA-N; OXYNPFVALCVOEE-JJNLEZRASA-O; RVESWCGOZRMDGX-QYVSTXNMSA-N; JDNSTJQSYYVVEA-QYVSTXNMSA-N; CRNXHGUBCVWODG-KQYNXXCUSA-O; ZHBLUYQJPJHFGX-PZKVIMCMSA-M; 5â² Nucleotidase cNIIIB; 7-Methylguanosine 5â²-monophosphate; Click chemistry;
A novel RPE65 inhibitor CU239 suppresses visual cycle and prevents retinal degeneration
Keywords: مهارکننده آنزیم; RPE; retinal pigment epithelium; IPM; inter-photoreceptor matrix; 11-cis-RAL; 11-cis-retinaldehyde; all-trans-RAL; all-trans-retinaldehyde; ABCA4; ATP-cassette transporter 4; atRDH; all-trans-retinol dehydrogenases; all-trans-ROL; all-trans-retinol; IRBP;
Class A β-lactamases and inhibitors: In silico analysis of the binding mode and the relationship with resistance
Keywords: مهارکننده آنزیم; β-lactamase; Enzyme inhibitor; Antimicrobial; Resistance; Molecular modeling;
CD73 inhibition by purine cytotoxic nucleoside analogue-based diphosphonates
Keywords: مهارکننده آنزیم; Enzyme inhibitor; CD73; Nucleotide; Cancer; Immunology; NXJDMDJDFQJJGS-GFCOJPQKSA-L; JUQZSESVGXFBBE-KBNQYOMWSA-L; OLCWZBFDIYXLAA-YNJARDAQSA-L; VPXFTBZVQMXNLH-FRSABSTQSA-L;
Region-specific bioconversion of dynorphin neuropeptide detected by in situ histochemistry and MALDI imaging mass spectrometry
Keywords: مهارکننده آنزیم; IMS; imaging mass spectrometry; DA; dopamine; PD; Parkinson's disease; LID; L-DOPA-induced dyskinesia; NEM; N-Ethylmaleimide; DynB; dynorphin B; Neuropeptide; Dynorphin; Bioconversion; Enzyme; Enzyme inhibitor; Histochemistry; MALDI imaging mass spectro
Structural basis for the inhibition of AKR1B10 by the C3 brominated TTNPB derivative UVI2008
Keywords: مهارکننده آنزیم; Cancer; Enzyme inhibitor; Psoriasis; RAR/RXR agonist; Retinoic acid; Skin disease; AR; Aldose Reductase; AKR; Aldo-Keto Reductase; AKR1B10; AKR family member 1B10; AKR1B15; AKR family member 1B15; AKR1A1; AKR family member 1A1 or aldehyde reductase; ARIs;
Characterisation of the fumarate hydratase repertoire in Trypanosoma cruzi
Keywords: مهارکننده آنزیم; Trypanosoma cruzi; Gene disruption; Tricarboxylic acid cycle; Drug design; Enzyme inhibitor; Iron-sulfur protein;
Treatment of estrogen-dependent diseases: Design, synthesis and profiling of a selective 17β-HSD1 inhibitor with sub-nanomolar IC50 for a proof-of-principle study
Keywords: مهارکننده آنزیم; 17β-Hydroxysteroid dehydrogenase type 1; Enzyme inhibitor; Steroidogenic enzymes; Estrogen-dependent disease; Intracrinology; (h)17β-HSD1; (human) 17β-hydroxysteroid dehydrogenase type 1; (h)17β-HSD2; (human) 17β-hydroxysteroid dehydrogenase type 2;
Dipeptidyl peptidase IV and quorum sensing signaling in biofilm-related virulence of Prevotella aurantiaca
Keywords: مهارکننده آنزیم; Autoinducer-2; Biofilm; Enzyme inhibitor; Estradiol; Pathogenicity; Prevotella;
Methanolic extract from red berry-like fruits of Hypericum androsaemum: Chemical characterization and inhibitory potential of central nervous system enzymes
Keywords: مهارکننده آنزیم; Hypericum androsaemum; Enzyme inhibitor; MAO-A; Tyrosinase; Polyphenols;
Correlative effect of dissolved oxygen and key enzyme inhibitors responsible for l-lactate production by immobilized Rhizopus oryzae NRRL395 cultivated in a static bed bioreactor
Keywords: مهارکننده آنزیم; Rhizopus oryzae; l-Lactic acid; Ethanol; Enzyme inhibitor; Dissolved oxygen; Alcohol dehydrogenase; Pyruvate decarboxylate; Static bed bioreactor;
Design, synthesis, and in vitro and biological evaluation of potent amino acid-derived thiol inhibitors of the metallo-β-lactamase IMP-1
Keywords: مهارکننده آنزیم; Metallo-β-lactamase; Enzyme inhibitor; Antibiotic resistance
Arylpiperidines as a new class of oxidosqualene cyclase inhibitors
Keywords: مهارکننده آنزیم; Oxidosqualene cyclase; Enzyme inhibitor; High energy intermediate; Arylpiperidine; Docking experiments
Impact of structural modifications at positions 13, 16 and 17 of 16β-(m-carbamoylbenzyl)-estradiol on 17β-hydroxysteroid dehydrogenase type 1 inhibition and estrogenic activity
Keywords: مهارکننده آنزیم; Steroid; Enzyme inhibitor; Estrogen; Chemical synthesis; Estradiol isomer
Synthesis, X-ray crystallography, spectroscopic (FT-IR, 1H &13C NMR and UV), computational (DFT/B3LYP) and enzymes inhibitory studies of 7-hydroximinocholest-5-en-3-ol acetate
Keywords: مهارکننده آنزیم; Steroidal oxime; Crystal structure; DFT; Enzyme inhibitor; Molecular docking
Synthesis, spectroscopic and computational studies of 2-(thiophen-2-yl)-2,3-dihydro-1H-perimidine: An enzymes inhibition study
Keywords: مهارکننده آنزیم; 2-(Thiophen-2-yl)-2,3-dihydro-1H-perimidine; B3LYP/6-311++G(d,p); Enzyme inhibitor; Molecular docking; Hirshfeld analysis
Le pamplemousse, un célèbre inhibiteur enzymatique
Keywords: مهارکننده آنزیم; effet indésirable; inhibiteur enzymatique; jus de pamplemousse; observance; pomelo; statineadverse effect; compliance; enzyme inhibitor; grapefruit juice; pomelo; statin
Label-free fluorometric detection of S1 nuclease activity by using polycytosine oligonucleotide-templated silver nanoclusters
Keywords: مهارکننده آنزیم; S1 nuclease; Silver nanoclusters; Fluorometry; Enzyme activity; Enzyme inhibitor;
Synthesis, molecular docking and Brugia malayi thymidylate kinase (BmTMK) enzyme inhibition study of novel derivatives of [6]-shogaol
Keywords: مهارکننده آنزیم; [6]-Shogaol; Zingiber officinale; Filariasis; Brugia malayi; Thymidylate kinase; Molecular modelling; Enzyme inhibitor
Identification of fused 16β,17β-oxazinone-estradiol derivatives as a new family of non-estrogenic 17β-hydroxysteroid dehydrogenase type 1 inhibitors
Keywords: مهارکننده آنزیم; Steroid; 17beta-hydroxysteroid dehydrogenase; Oxazinone; Enzyme inhibitor; Chemical synthesis; Molecular modeling
5-O-Acyl plumbagins inhibit DNA polymerase activity and suppress the inflammatory response
Keywords: مهارکننده آنزیم; 5-O-Acyl plumbagins; C22:6-acyl plumbagin; DNA polymerase λ; Enzyme inhibitor; Anti-inflammation
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors: Evaluation of potency and selectivity derived from distinct binding pockets
Keywords: مهارکننده آنزیم; Serine protease; Peptidomimetic; Benzamidine; Hepsin; Matriptase; HGFA; Small-molecule; Therapeutic; c-MET; RON; HGF; MSP; Receptor tyrosine kinase; Cancer; Cell-signaling; Growth factor; Structure-based drug design; Enzyme inhibitor;
Design, chemical synthesis and biological evaluation of 3-spiromorpholinone/3-spirocarbamate androsterone derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 3
Keywords: مهارکننده آنزیم; ADT; androsterone; AR; androgen receptor; Ar; aryl group; DBD; DNA binding domain; DCM; dichloromethane; DHT; dihydrotestosterone; DIPEA; N,N-diisopropylethylamine; DMF; dimethylformamide; DMSO; dimethylsulfoxide; Î4-dione; 4-androstene-3,17-dione; EtOAc
Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors
Keywords: مهارکننده آنزیم; Non-classical bioisostere; Pyrazole; Amide; Enzyme inhibitor; Prolylcarboxypeptidase (PrCP); Angiotensinase C;
Azide-alkyne cycloaddition affording enzymatically tunable bisubstrate based inhibitors of histone acetyltransferase PCAF
Keywords: مهارکننده آنزیم; Bisubstrate based inhibitor; Histone acetyltransferase; Enzyme inhibitor; Posttranslational modification; Protein acetylation;
Sulfonamide inhibition studies of the β carbonic anhydrase from Drosophila melanogaster
Keywords: مهارکننده آنزیم; Carbonic anhydrase; β-Class enzyme; Drosophila melanogaster; Sulfonamide; Enzyme inhibitor;