Keywords: آنتاگونیست; allosteric drug discovery; protocol; agonist; antagonist; driver atom; anchor atom; allostery
مقالات ISI آنتاگونیست (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: آنتاگونیست; Iminocoumarine; Coumarine; Galectin; Antagonist; Multicomponent reaction;
Keywords: آنتاگونیست; AR; androgen receptor; DMEM; Dulbecco's minimal essential medium; FCS; fetal calf serum; GR; glucocorticoid receptor; GRE; glucocorticoid response element; GST; glutathione S-transferase; HEK; human embryonic kidney; IPTG; isopropyl-β-d-thiogalactoside
Keywords: آنتاگونیست; Methamphetamine; α1-Adrenergic receptor; Antagonist; Memory consolidation; Conditioning; Sensitization;
Keywords: آنتاگونیست; Elderly; Skeletal muscle; Exercise; Voluntary activation; Co-activation; Antagonist; Strength training
Keywords: آنتاگونیست; alpha2-adrenergic agonist; antagonist; atipa-mezole; detomidine; equine; tolazoline; yohimbine;
Keywords: آنتاگونیست; Sphingosine-1-phosphate (S1P); Antagonist; Fluorination; [18F]-radiotracer; Molecular imaging; Positron emission tomography (PET);
Keywords: آنتاگونیست; Mineralocorticoid receptor; Antagonist; Aldosterone; Myocardium; Ischemia–reperfusion injury; Cardiac remodeling11βHSD1, 11-β-hydroxysteroid dehydrogenase type 1; 11βHSD2, 11-β-hydroxysteroid dehydrogenase type 2; ACS, acute coronary syndrome; IL, interle
Keywords: آنتاگونیست; Retinoid; Diphenylamine; Agonist; Antagonist; Synergist;
Keywords: آنتاگونیست; Nicotinic; Attention; Antagonist; α4β2; α7;
Keywords: آنتاگونیست; Antagonist; Cocontraction; Elderly; Electromyography; EMG; Incline; Decline;
Keywords: آنتاگونیست; Nicotinic receptors; Postsynaptic neurotoxins; Skeletal muscle; Snake venom; Antagonist;
Keywords: آنتاگونیست; GPR55; Neuropathic pain; GPCR; Antagonist; Cancer
Keywords: آنتاگونیست; Dopamine; Antagonist; DA D3 receptor; 7-TM; Morpholine
Repellence of nectar-thieving ants by a physical barrier: Adaptive role of petal hairs on Menyanthes trifoliata (Menyanthaceae)
Keywords: آنتاگونیست; Antagonist; Ants; Flower; Menyanthaceae; Plant-Insect Interactions;
Novel VDR antagonists based on the GW0742 scaffold
Keywords: آنتاگونیست; Nuclear receptor; Vitamin D receptor (VDR); Peroxisome proliferation-activated receptor δ (PPARδ); Antagonist; Steroid receptor coactivator 2;
2-Methylacrylamide as a bioisoster of thiourea group for 1,3-dibenzylthioureido TRPV1 receptor antagonists
Keywords: آنتاگونیست; 2-Methylacrylamide; Bioisoster; TRPV1; 1,3-Dibenzylthioureas; Antagonist; 45Ca2+-Influx assay;
Benzopyrone represents a privilege scaffold to identify novel adenosine A1/A2A receptor antagonists
Keywords: آنتاگونیست; Benzopyrone; Adenosine A2A receptor; Adenosine A1 receptor; Antagonist; GTP shift; Radioligand binding assay; Cancer; Parkinson's disease; AR; adenosine receptor; GTP; guanosine triphosphate; [3H]DPCPX; [3H]-dipropyl-8-cyclopentylxanthine; [3H]NECA; N-[3H
Gas-phase structural characterization of neuropeptides Y Y1 receptor antagonists using mass spectrometry: Orbitrap vs triple quadrupole
Keywords: آنتاگونیست; Obesity; Diabetes; Antagonist; Triple quadrupole; Orbitrap; Mass spectrometry;
Allosteric inhibition abrogates dysregulated LFA-1 activation: Structural insight into mechanisms of diminished immunologic disease
Keywords: آنتاگونیست; Affinity; Allosteric; Antagonist; Immunologic; Lifitegrast; LFA-1;
Assessment of androgen receptor agonistic/antagonistic effects on 25 chemicals in household applicants by OECD in vitro stably transfected transcriptional activation assays
Keywords: آنتاگونیست; Human androgen receptor; Transcriptional activation assay; OECD test guideline; Agonist; Antagonist;
Rac1 plays a role in CXCL12 but not CCL3-induced chemotaxis and Rac1 GEF inhibitor NSC23766 has off target effects on CXCR4
Keywords: آنتاگونیست; AUC; Area under Curve; EDTA; Ethylenediaminetetraacetic acid; FCS; Foetal calf serum; FSC; Forward scatter; GPCR; G protein-coupled receptor; PBS; Phosphate buffered saline; SEM; Standard Error of Means; SSC; Side scatter; Chemokine receptor; Chemotaxis;
In vitro and in vivo functional profile characterization of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6α-(isoquinoline-3-carboxamido)morphinan (NAQ) as a low efficacy mu opioid receptor modulator
Keywords: آنتاگونیست; NAQ; Mu opioid receptor; Opioid addiction; Antagonist; β-arrestin2 recruitment; Nalbuphine;
Pseudomonas graminis strain CPA-7 differentially modulates the oxidative response in fresh-cut 'Golden delicious' apple depending on the storage conditions
Keywords: آنتاگونیست; Antioxidant enzymes; Oxidative stress; Antagonist; Fruit defense response;
Impact of Pseudomonas graminis strain CPA-7 on respiration and ethylene production in fresh-cut 'Golden delicious' apple according to the maturity stage and the preservation strategy
Keywords: آنتاگونیست; Antagonist; Fresh-cut fruit physiology; Passive modified atmosphere packaging; MAP;
The preparation of novel histrionicotoxin analogues and their activity towards the α4β2 and α7 nicotinic acetylcholine receptors
Keywords: آنتاگونیست; Histrionicotoxin; Poison arrow frog toxin; Nicotinic acetylcholine receptor; Antagonist; 1,3-Dipolar cycloaddition;
Human GIP(3-30)NH2 inhibits G protein-dependent as well as G protein-independent signaling and is selective for the GIP receptor with high-affinity binding to primate but not rodent GIP receptors
Keywords: آنتاگونیست; Glucose-dependent insulinotropic polypeptide (GIP); GIP receptor; Antagonist; Human subcutaneous adipocytes; Signaling;
The tamoxifen derivative ridaifen-B is a high affinity selective CB2 receptor inverse agonist exhibiting anti-inflammatory and anti-osteoclastogenic effects
Keywords: آنتاگونیست; Cannabinoid receptors; G-protein coupled receptors; Inverse agonist; Antagonist; Drug action; AC; adenylyl cyclase; CB1R; cannabinoid receptor type 1; CB2R; cannabinoid receptor type 2; CHO; Chinese hamster ovary; CP-55,940; 5-(1,1-dimethylheptyl)-2-[5-hy
Synthesis and pharmacological characterization of functionalized 6-piperazin-1-yl-purines as cannabinoid receptor 1 (CB1) inverse agonists
Keywords: آنتاگونیست; BBB; Blood-Brain Barrier; CB1; Cannabinoid Receptor 1; CB2; Cannabinoid Receptor 2; CHO-K1; Chinese Hamster Ovary Cells; CNS; Central Nervous System; EtOH; ethanol; EtOAc; ethyl acetate; Ke; apparent affinity constant, MDCK-mdr1, Madin-Darby canine kidney
Synthetic studies of (23S,25R)-1α,25-dihydroxyvitamin D3 26,23-lactone (calcitriol lactone) and its derivatives
Keywords: آنتاگونیست; Calcitriol lactone; TEI-9647; Calcitriol lactam (DLAM); Antagonist; Side chain;
Yokukansan contains compounds that antagonize the 5-HT3 receptor
Keywords: آنتاگونیست; Yokukansan; Yi-Gan San; Serotonin receptor; Ion channel; Antagonist; 5-HT3; 5-HT; 5-hydroxytryptamine or serotonin;
Synthesis of 7β-hydroxy-8-ketone opioid derivatives with antagonist activity at mu- and delta-opioid receptors
Keywords: آنتاگونیست; Morphine; Oxidation; Supported permanganate; Hydroxy ketone; Antagonist; Opioid receptor; VZGNAZRFVZVYHM-DRDPLEBGSA-N; XOBHDVAWTNEDQE-UZUQFWOOSA-N;
CNS distribution, signalling properties and central effects of G-protein coupled receptor 4
Keywords: آنتاگونیست; GPR4; Antagonist; Lactate; Modulation; Respiration; Distribution;
Discovery and characterization of a potent Wnt and hedgehog signaling pathways dual inhibitor
Keywords: آنتاگونیست; Wnt signaling pathway; Hedgehog signaling pathway; Porcupine; Smoothened; Antagonist; Stem cell; Cancer therapy; AUC; area under the plasma time-concentration curve; BCC; basal cell carcinoma; BPO; benzoyl peroxide; CL; clearance; CSC; cancer stem cells;
Design, synthesis, and structure-activity-relationship of a novel series of CXCR4 antagonists
Keywords: آنتاگونیست; Chemokine; CXCR4; Antagonist; GPCR; Scaffold hybridization; Therapy; APC; allophycocyanin; BPO; benzoyl peroxide; CCD; charge coupled device; CYP; cytochrome P450; DC; dendritic cells; DCE; 1,2-dichloroethane; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbe
Evaluation of biocontrol capacity of Pseudomonas graminis CPA-7 against foodborne pathogens on fresh-cut pear and its effect on fruit volatile compounds
Keywords: آنتاگونیست; Listeria; Salmonella; Ethanol; Acetaldehyde; Antagonist;
Design and synthesis of aryloxypropanolamine as β3-adrenergic receptor antagonist in cancer and lipolysis
Keywords: آنتاگونیست; β-Adrenergic receptor; Antagonist; Cancer; Lipolysis and cachexia;
Dimethyl adenosine transferase (KsgA) contributes to cell-envelope fitness in Salmonella Enteritidis
Keywords: آنتاگونیست; KsgA; Dimethyl adenosine transferase; Salmonella; Cell-envelope; Fitness; Antagonist;
Synthesis and structure-activity relationships of quinolinone and quinoline-based P2X7 receptor antagonists and their anti-sphere formation activities in glioblastoma cells
Keywords: آنتاگونیست; P2X7 receptor; Antagonist; IL-1β; EtBr; Inflammation; Quinoline; Quinolinone; Anti-glioma;
Tools and drugs for uracil nucleotide-activated P2Y receptors
Keywords: آنتاگونیست; ADP; Adenosine 5â²-diphosphate; AP4A; P1,P4-Di(adenosine-5â²)-tetraphosphate; AR; Adenosine receptor; AR-C118925; 5-{[5-(2,8-Dimethyl-5H-dibenzo[a,d]cyclohepten-5-yl)-3,4-dihydro-2-oxo-4-thioxo-1(2H)-pyrimidinyl]methyl}-N-(1H-tetrazol-5-yl)-2-furancarbo
Design, synthesis and metabolic regulation effect of farnesoid X receptor (FXR) antagonistic benzoxepin-5-ones
Keywords: آنتاگونیست; Farnesoid X receptor; Antagonist; Benzoxepin-5-one; Triglyceride; Plasma ALT;
Antagonism of vasopressin V2 receptor improves albuminuria at the early stage of diabetic nephropathy in a mouse model of type 2 diabetes
Keywords: آنتاگونیست; Vasopressin; V2 receptor; Antagonist; Diabetic nephropathy; Type 2 diabetes;
Structure-activity relationships of 2-substituted phenyl-N-phenyl-2-oxoacetohydrazonoyl cyanides as novel antagonists of exchange proteins directly activated by cAMP (EPACs)
Keywords: آنتاگونیست; Exchange proteins directly activated by cAMP; EPAC; Antagonist; Molecular docking;
From UTP to AR-C118925, the discovery of a potent non nucleotide antagonist of the P2Y2 receptor
Keywords: آنتاگونیست; P2Y2; Purinergic; AR-C118925; P2; Antagonist;
Structure-activity relationships of benzothiazole GPR35 antagonists
Keywords: آنتاگونیست; GPR35; Antagonist; G protein-coupled receptor; Benzothiazole; SAR;
[11C]AZ10419096 - a full antagonist PET radioligand for imaging brain 5-HT1B receptors
Keywords: آنتاگونیست; 5-HT1B receptor; Antagonist; Radioligand; Carbon-11; PET;
Structure-activity relationship study of β-oxidation resistant indole-based 5-oxo-6,8,11,14-eicosatetraenoic acid (5-oxo-ETE) receptor antagonists
Keywords: آنتاگونیست; AA; arachidonic acid; 5-HETE; 5-hydroxy-6E,8Z,11Z,14Z-eicosatetraenoic acid; 5-oxo-ETE; 5-oxo-6E,8Z,11Z,14Z-eicosatetraenoic acid; 5-HEDH; 5-hydroxyeicosanoid dehydrogenase; 5-HpETE; 5-hydroperoxyeicosatetraenoic acid; LT; leukotriene; NADP+; nicotinamide
Identification of ligand-selective peptidic ActRIIB-antagonists using phage display technology
Keywords: آنتاگونیست; ActRIIB; activin receptor type-2B; MSTN; myostatin; GDF11; growth differentiation factor 11; BMP9; bone morphogenetic protein 9; PPI; protein-protein interaction; ALK; activin receptor type-1B; ActRIIB; Antagonist; Ligand-selectivity; Peptide; Phage displ
Virtual screening and experimental validation identify novel modulators of nuclear receptor RXRα from Drugbank database
Keywords: آنتاگونیست; RXRα; Old drug; Agonist; Antagonist; Virtual screening; QVVCZWKLXIGYPX-ZRYTXGOBSA-N; QMRFMKFSCAFNDM-BZCZYQESSA-N; KFJUEWQQCHWYIV-QPZJVCRCSA-N; HEILJUCIFZMCAH-QTDJRPCYSA-N;
Synthesis and evaluation of a 68Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography
Keywords: آنتاگونیست; Bradykinin B1 receptor; Agonist; Antagonist; Positron emission tomography; Gallium-68;