Keywords: مهارکننده کیناز ; Cancer chemoprevention; Liver cancer; Kinase inhibitor; Epidermal growth factor; Nanoparticle;
مقالات ISI مهارکننده کیناز (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهارکننده کیناز ; Fluorescence; Polydopamine nanospheres; Protein kinase activity; Kinase inhibitor;
Keywords: مهارکننده کیناز ; BAD phosphorylation; Apoptosis; kinase inhibitor; Bcl-2 family;
Keywords: مهارکننده کیناز ; Alloxazine; Antitumor; Kinase inhibitor; Docking; Apoptosis;
Keywords: مهارکننده کیناز ; Ruthenium-coordination complex; Ligand exchange rate; Kinase inhibitor; Ruthenium-glutathione-S-transferase inhibitors; DNA damage; Anticancer; 1-BI; 1-benzylimidazole; 2,3-dpp; 2,3-bis(2-pyridyl)pyrazine; 2-ap; 2-acetylpyridine; 3-pyha; 3-pyridinehydroxa
Keywords: مهارکننده کیناز ; Breast cancer; Raf; ERK; Bioinformatics; Kinase inhibitor;
Keywords: مهارکننده کیناز ; BTSC; Brain Tumor Stem Cell(s); DIPG; Diffuse Intrinsic Pontine Glioma; EGF; Epidermal Growth Factor; FBS; Fetal Bovine Serum; FGF; Fibroblast Growth Factor; PAGE; Parametric Analysis of Geneset Enrichment; PCA; Principle Component Analysis; PDGF; Platele
Keywords: مهارکننده کیناز ; Kinase inhibitor; Polo-like kinase 1; Ras-driven signaling pathways; Non-ATP competitive inhibition; Anti-cancer agents;
Keywords: مهارکننده کیناز ; LC-MS/MS; Chromatographic bioanalysis; Kinase inhibitor; Oncology;
Keywords: مهارکننده کیناز ; Canine; Cell lines; Kinase inhibitor; Osteosarcoma; Screening;
Keywords: مهارکننده کیناز ; Plasmodium; Schistosoma; Life cycle; Reproduction; Kinase; Kinase inhibitor
Keywords: مهارکننده کیناز ; Haemonchus contortus; Anthelmintic screening; Motility assay; Automated imaging analysis; Kinase inhibitor; Biphenyl amide; Pyrazolo[1,5-α]pyridine;
Keywords: مهارکننده کیناز ; Anti-influenza viral drug; Compound library screening; vRNP activity; Kinase inhibitor; Target database search; KINOMEscan;
Keywords: مهارکننده کیناز ; CLL; Fludarabine refractory; Microenvironment; Kinase inhibitor; Dasatinib; NOXA;
Keywords: مهارکننده کیناز ; Signal transduction; Rheumatoid arthritis; Inflammation; Kinase inhibitor; Tofacitinib; Kinase; Arthritis; Small molecule;
Keywords: مهارکننده کیناز ; c-Met; Kinase inhibitor; Anti-tumor; Quinoline; Semicarbazone;
Keywords: مهارکننده کیناز ; Solvatochromism; Photophysics; UV–Vis spectroscopy; SKF86002; Kinase inhibitor; Anti-inflammatory drug
Keywords: مهارکننده کیناز ; Tuberculosis; Enzyme inhibitor; Targeted therapy; Kinase inhibitor; Phenotypical screening
Preliminary in vitro and in vivo investigation of a potent platelet derived growth factor receptor (PDGFR) family kinase inhibitor
Keywords: مهارکننده کیناز ; Kinase inhibitor; PDGFR; KIT; Cancer; Systemic mastocytosis;
Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitors
Keywords: مهارکننده کیناز ; Bruton's tyrosine kinase; Kinase inhibitor; Kinase selectivity; Pyrimidine; Passive cutaneous anaphylaxis;
Discovery of a highly potent orally bioavailable imidazo-[1, 2-a]pyrazine Aurora inhibitor
Keywords: مهارکننده کیناز ; Aurora inhibitor; Kinase inhibitor; Imidazopyrazine;
Structural basis for the potent and selective binding of LDN-212854 to the BMP receptor kinase ALK2
Keywords: مهارکننده کیناز ; BMP; Heterotopic ossification; Kinase inhibitor; Crystal structure; Drug; Fibrodysplasia ossificans progressiva;
Novel Small-Molecule Inhibitors of Protein Kinase C Epsilon Reduce Ethanol Consumption in Mice
Keywords: مهارکننده کیناز ; Addiction; Alcohol; Kinase inhibitor; Protein kinase C epsilon;
Developmental effects of the protein kinase inhibitor kenpaullone on the sea urchin embryo
Keywords: مهارکننده کیناز ; Embryonic development; Gene expression; Kenpaullone; Kinase inhibitor; Sea urchin;
Discovery and optimization of novel benzothiophene-3-carboxamides as highly potent inhibitors of Aurora kinases A and B
Keywords: مهارکننده کیناز ; Cancer; Targeted therapy; Aurora kinase; Kinase inhibitor; Benzothiophene-3-carboxamide;
In silico-in vitro discovery of untargeted kinase-inhibitor interactions from kinase-targeted therapies: A case study on the cancer MAPK signaling pathway
Keywords: مهارکننده کیناز ; Mitogen-activated protein kinase; Kinase inhibitor; Untargeted interaction; Biomolecular modeling; Cancer;
Design, synthesis, and biological evaluation of new B-RafV600E kinase inhibitors
Keywords: مهارکننده کیناز ; B-Raf; Molecular dynamics; Docking; Kinase inhibitor; Drug design;
3H-pyrazolo[4,3-f]quinoline haspin kinase inhibitors and anticancer properties
Keywords: مهارکننده کیناز ; Haspin; Kinase inhibitor; Doebner/Povarov reaction;
Discovery of novel 4-aryl-thieno[1,4]diazepin-2-one derivatives targeting multiple protein kinases as anticancer agents
Keywords: مهارکننده کیناز ; 4-Aryl-thieno[1,4]diazepin-2-one; Antiproliferative activity; Hematopoietic cell line; Kinase inhibitor; Multiple protein kinase inhibitor;
Novel quinazoline derivatives bearing various 6-benzamide moieties as highly selective and potent EGFR inhibitors
Keywords: مهارکننده کیناز ; EGFR; Kinase inhibitor; Quinazoline; High selectivity; Anti-cancer;
Mechanisms of mitochondrial toxicity of the kinase inhibitors ponatinib, regorafenib and sorafenib in human hepatic HepG2 cells
Keywords: مهارکننده کیناز ; MKI; multikinase inhibitor; ALT; alanine aminotransferase; AST; aspartate aminotransferase; DRP1; dynamin-related protein 1; FIS1; mitochondrial fission 1; ROS; reactive oxygen species; DMSO; dimethylsulfoxide; AK; adenylate kinase; PBS; phosphate buffere
Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases
Keywords: مهارکننده کیناز ; Palladium; Sphingosine kinase; Kinase inhibitor; Jaspine B; Structure-activity relationship;
Design and discovery of thioether and nicotinamide containing sorafenib analogues as multikinase inhibitors targeting B-Raf, B-RafV600E and VEGFR-2
Keywords: مهارکننده کیناز ; Nicotinamide; B-Raf; VEGFR-2; Kinase inhibitor; Antitumor;
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibitor for PDGFRα driving chronic eosinophilic leukemia
Keywords: مهارکننده کیناز ; PDGFR kinase; Type II inhibitor; Kinase inhibitor; CEL; PDGFR; platelet-derived growth factor receptor; RTK; Receptor Tyrosine Kinases; ABL kinase; Abelson kinase; KIT kinase; v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; RTK; receptor ty
Overcoming the stability, solubility and extraction challenges in reversed-phase UHPLC-MS/MS bioanalysis of a phosphate drug and its prodrug in blood lysate
Keywords: مهارکننده کیناز ; Sphingosine-1-phosphate (S1P); Phosphate compound; Blood lysate; Quantitative; Bioanalysis; LC-MS/MS; Phosphatase inhibitor; Kinase inhibitor;
Optogenetic control of focal adhesion kinase signaling
Keywords: مهارکننده کیناز ; CRY2; cryptochrome 2; FAK; focal adhesion kinase; FAT; focal adhesion targeting; FERM; band 4.1-ezrin-radixin-moesin; p130Cas; p130 Crk-associated substrate; SC; single clone; SFK; SRC family kinases; Optogenetics; Cryptochrome 2; Focal adhesion kinase; F
Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Keywords: مهارکننده کیناز ; Quinoxaline; Pim-1; Kinase inhibitor; Anticancer targeted therapy; IC50; 50% inhibitory concentration; SAR; structure-activity relationships; Pim; proviral integration site of Moloney murine leukemia virus; CML; chronic myeloid leukemia; DYRK1A; dual spec
Prognostic Testing Patterns and Outcomes of Chronic Lymphocytic Leukemia Patients Stratified by Fluorescence In Situ Hybridization/Cytogenetics: A Real-world Clinical Experience in the Connect CLL Registry
Keywords: مهارکننده کیناز ; Community setting; Cytogenetic testing; Kinase inhibitor; Prognosis; Unfavorable risk;
Design, synthesis, and biological evaluation of polo-like kinase 1/eukaryotic elongation factor 2 kinase (PLK1/EEF2K) dual inhibitors for regulating breast cancer cells apoptosis and autophagy
Keywords: مهارکننده کیناز ; Apoptosis; Autophagy; Breast cancer; EEF2K; Kinase inhibitor; PLK1;
The development of Bruton's tyrosine kinase (BTK) inhibitors from 2012 to 2017: A mini-review
Keywords: مهارکننده کیناز ; Bruton's tyrosine kinase (BTK); Kinase inhibitor; Irreversible inhibitor; Reversible covalent inhibitor;
Divergent synthesis of kinase inhibitor derivatives, leading to discovery of selective Gck inhibitors
Keywords: مهارکننده کیناز ; BAY 61-3606; Imidazo[1,2-c]pyrimidine; Gck; Indole; Kinase inhibitor;
Mutations in TP53, PIK3CA, PTEN and other genes in EGFR mutated lung cancers: Correlation with clinical outcomes
Keywords: مهارکننده کیناز ; Mutation; Lung cancer; Adenocarcinoma; EGFR; TP53; PIK3CA; PTEN; Kinase inhibitor; Erlotinib;
Identification of quinazoline based inhibitors of IRAK4 for the treatment of inflammation
Keywords: مهارکننده کیناز ; IRAK4; Quinazoline; Serine-threonine kinase; Kinase inhibitor; Inflammatory disease; HVQXFGHHSFTACS-CXIWYSOXSA-N;
A high throughput assay to identify substrate-selective inhibitors of the ERK protein kinases
Keywords: مهارکننده کیناز ; Protein kinase; Phosphorylation; Kinase inhibitor; High-throughput screening; Mitogen-activated protein kinase;
Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors
Keywords: مهارکننده کیناز ; AXL; 7-Azaindole; Receptor tyrosine kinase; Kinase inhibitor; Modeling study; Medicinal chemistry;
Synthesis and photophysical properties of a fluorescent cyanoquinoline probe for profiling ERBB2 kinase inhibitor response
Keywords: مهارکننده کیناز ; Receptor tyrosine kinase; Kinase inhibitor; Fluorescent probe; EGFR; ERBB;
Inhibition of protein kinases by anticancer DNA intercalator, 4-butylaminopyrimido[4â²,5â²:4,5]thieno(2,3-b)quinoline
Keywords: مهارکننده کیناز ; DNA intercalator; Molecular docking; Kinase inhibitor; Anticancer drugs; Apoptosis; Chemotherapy;
Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B
Keywords: مهارکننده کیناز ; Sphingosine kinase; Kinase inhibitor; Jaspine B; Structure-activity relationship;
Thiazolidine derivatives as potent and selective inhibitors of the PIM kinase family
Keywords: مهارکننده کیناز ; Thiazolidine; PIM kinase; Anti-cancer; High throughput screen; Kinase inhibitor;
Discovery and structure activity relationship of the first potent cryptosporidium FIKK kinase inhibitor
Keywords: مهارکننده کیناز ; Cryptosporidium; Kinase inhibitor; FIKK Kinase inhibitor;