Synthesis of novel 15-membered 8a-azahomoerythromycin A acylides: Consequences of structural modification at the C-3 and C-6 position on antibacterial activity
Keywords: واکنش هک; Macrolide antibiotics; Macrolide resistance; Acylides; Structure-activity relationships; Antibacterial activity; Heck reaction; MLSB; macrolide-lincosamide-streptogramin B; Mef; macrolide efflux; SAR; structure-activity relationships; DABCO; 1,4-diazabicy