Keywords: مهار آنزیم; Toxoplasma gondii; 1-Deoxy-d-xylulose-5-phosphate reductoisomerase; Protein expression; Enzyme inhibition; Structure-activity relationship;
مقالات ISI مهار آنزیم (ترجمه نشده)
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Keywords: مهار آنزیم; DDIJSDOLYBZWCO-UHFFFAOYSA-N; Diabetic complications; Aldose reductase; Enzyme inhibition; Imidazolidinediones; Hypoglycemic agents;
Keywords: مهار آنزیم; Nonsymmetrical aromatic disulfides; Acetohydroxyacid synthase; Branched-chain amino acids; Enzyme inhibition; Herbicidal activity;
Keywords: مهار آنزیم; Chorismate; Enzyme inhibition; Hydrolase;
Keywords: مهار آنزیم; BLC; bovine liver catalase; ECG; epicatechin gallate; EGC; epigallocatechin; EGCG; epigallocatechin gallate; Catalase; Enzyme inhibition; Flavonoids;
Keywords: مهار آنزیم; Chicken skin; Membrane ultrafiltration; Protein hydrolysates; Peptide profile; Angiotensin converting enzyme; Renin; Enzyme inhibition;
Keywords: مهار آنزیم; Block copolymer micelles; Lipase enzyme; Hydrolytic degradation; Enzyme interfacial activation; Enzyme inhibition;
Keywords: مهار آنزیم; MMP-2 and MMP-9; Ilomastat analogs; Benzamide groups; Enzyme inhibition; Non-zinc binding; HEY cell invasion
Keywords: مهار آنزیم; β-N-acetylhexosaminidase; Hex B; Enzyme inhibition; O-GlcNAcase; Pichia pastoris
Keywords: مهار آنزیم; Purinergic signaling; Mucociliary clearance; Bronchial epithelium; Mathematical model; Enzyme inhibition;
Antiradical, antimicrobial and enzyme inhibition evaluation of sulfonamide derived esters; synthesis, X-Ray analysis and DFT studies
Keywords: مهار آنزیم; Antioxidant; DFT; Enzyme inhibition; Ester; Sulfonamide;
Synthesis of novel 5-amino-1,3,4-thiadiazole-2-sulfonamide containing acridine sulfonamide/carboxamide compounds and investigation of their inhibition effects on human carbonic anhydrase I, II, IV and VII
Keywords: مهار آنزیم; Carbonic anhydrase; Acridine; Sulfonamide; Carboxamide; Enzyme inhibition; Isoforms CA I, II, IV and VII;
Assessment of the inhibitory activity of the pyrethroid pesticide deltamethrin against human placental glutathione transferase P1-1: A combined kinetic and docking study
Keywords: مهار آنزیم; Glutathione transferase P1-1; Detoxification; Deltamethrin; Pyrethroid insecticide; Enzyme inhibition; Molecular docking;
Investigations of anti-aging potential of Hypericum origanifolium Willd. for skincare formulations
Keywords: مهار آنزیم; Hypericum origanifolium; Anti-aging; Enzyme inhibition; Antioxidant; Antigenotoxicity;
Neuroprotective potential of Viburnum orientale Pallas through enzyme inhibition and antioxidant activity assays
Keywords: مهار آنزیم; Viburnum orientale; Enzyme inhibition; Antioxidant activity; Neuroprotective effect; Cholinesterase; Tyrosinase;
In vitro and in silico PTP-1B inhibition and in vivo antidiabetic activity of semisynthetic moronic acid derivatives
Keywords: مهار آنزیم; RGKMKULXFZOUPF-BQSMYOSZSA-N; SXYLITRDEAEYTJ-MGPMMZCJSA-N; Diabetes; Moronic acid derivatives; PTP-1B; Molecular docking; Enzyme inhibition;
Inhibition of UDP-glucuronosyltransferases (UGTs) by phthalate monoesters
Keywords: مهار آنزیم; Phthalate esters (PAEs); Phthalate monoesters; UDP-glucuronosyltransferases (UGTs); Enzyme inhibition;
Effects of dibutyl phthalate and di(2-ethylhexyl) phthalate with their metabolites on CYP2C9*1 and CYP2C19*1 activities in vitro
Keywords: مهار آنزیم; Cytochrome P450 enzyme; Enzyme inhibition; Dibutyl phthalate; Monoethylhexyl phthalate; Metabolites; Phthalates;
Concentrated hot water-infusion of phragmanthera incana improves muscle glucose uptake, inhibits carbohydrate digesting enzymes and abates Fe2+-induced oxidative stress in hepatic tissues
Keywords: مهار آنزیم; Antioxidants; Enzyme inhibition; Glucose uptake; Phragamenthra incana;
Mechanisms of acetylcholinesterase protection against sarin and soman by adenosine A1 receptor agonist N6-cyclopentyladenosine
Keywords: مهار آنزیم; Nerve agent; Antidote; Enzyme inhibition; Reactivation; Thermodynamic analysis; Density functional theory;
Lotus aegaeus (Gris.) Boiss and Iberis sempervirens L.: Chemical fingerprints, antioxidant potential, and inhibition activities and docking on key enzymes linked to global health problems
Keywords: مهار آنزیم; Polyphenols; Antioxidants; Enzyme inhibition; Medicinal plants; Pharmaceuticals; Molecular docking;
Crocus sativus L. stigmas and byproducts: Qualitative fingerprint, antioxidant potentials and enzyme inhibitory activities
Keywords: مهار آنزیم; Crocus sativus L.; Saffron byproducts; Enzyme inhibition; Oxidative stress; Antioxidant effect; Lipid peroxidation; CST; saffron stigmas; CTA; byproducts (tepals+anthers); IBD; inflammatory bowel disease; LPS; lipopolysaccharide; MDA; malondialdehyde; LDH
Inhibition of α-amylases by pentagalloyl glucose: Kinetics, molecular dynamics and consequences for starch absorption
Keywords: مهار آنزیم; Enzyme inhibition; Diabetes; Functional foods; Molecular docking; Molecular dynamics simulations;
Polyphenolic composition, enzyme inhibitory effects ex-vivo and in-vivo studies on two Brassicaceae of north-central Italy
Keywords: مهار آنزیم; Brassica oleracea L.; Broccolo Fiolaro di Creazzo; Cavolo Nero; Extractions; Enzyme inhibition; HPLC-PDA;
Activating effects on trypsin, α-chymotrypsin, and lipase and inhibitory effects on α-amylase and α-glucosidase as provided by low-molecular-weight compounds in the water extract of the earthworm Eisenia fetida
Keywords: مهار آنزیم; α-Amylase; Earthworm; Eisenia fetida; Enzyme activation; Enzyme inhibition; Trypsin;
Phytochemical characterization, antioxidant, antimicrobial and pharmacological activities of Feijoa sellowiana leaves growing in Tunisia
Keywords: مهار آنزیم; Feijoa sellowiana; HS-SPME/GC-MS; Antioxidant activity; Antimicrobial activity; Enzyme inhibition; Pharmacological activity;
Optimized allosteric inhibition of engineered protein tyrosine phosphatases with an expanded palette of biarsenical small molecules
Keywords: مهار آنزیم; AsCy3; FlAsH; Enzyme inhibition; Protein engineering; Protein tyrosine phosphatases;
Acyclic nucleoside phosphonates with unnatural nucleobases, favipiravir and allopurinol, designed as potential inhibitors of the human and Plasmodium falciparum 6-oxopurine phosphoribosyltransferases
Keywords: مهار آنزیم; Hypoxanthine-guanine-xanthine phosphoribosyltransferase; Regioselective Mitsunobu reaction; Acyclic nucleotide analogues; Enzyme inhibition;
Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX
Keywords: مهار آنزیم; 1,3,5-Triazine; Benzene sulfonamides; Amino acids; Carbonic anhydrase; Enzyme inhibition; Isoform selectivity;
Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action
Keywords: مهار آنزیم; 1,3,5-Triazine; Benzene sulfonamides; Carbonic anhydrase; Enzyme inhibition; Isoform selectivity; RBTRACBIJHXJOW-UHFFFAOYSA-N; YBEIEFLSBAECJS-UHFFFAOYSA-N; CEJPWNPQLGPPAS-UHFFFAOYSA-N; IKVVCANHSURSQN-UHFFFAOYSA-N; UJOHKJMLFDCSCH-UHFFFAOYSA-N; OOTLZKHMVNUK
Simultaneous detection of dual biomarkers from humans exposed to organophosphorus pesticides by combination of immunochromatographic test strip and ellman assay
Keywords: مهار آنزیم; Pesticides exposure; Biomarkers; BChE monoclonal antibody; Enzyme inhibition; Immunochromatographic test strip;
Synthesis and use of 6,6,6-trifluoro-L-fucose to block core-fucosylation in hybridoma cell lines
Keywords: مهار آنزیم; Fucose; Enzyme inhibition; Monoclonal antibody; Hybridoma;
DNA-binding, enzyme inhibition, and photochemical properties of chalcone-containing metallophthalocyanine compounds
Keywords: مهار آنزیم; Phthalocyanine; Chalcone; Enzyme inhibition; DNA-binding; Photochemical;
Antidiabetic and antiparasitic potentials: Inhibition effects of some natural antioxidant compounds on α-glycosidase, α-amylase and human glutathione S-transferase enzymes
Keywords: مهار آنزیم; Antidiabetic; Antiparasitic; Glutathione S-transferase; Enzyme inhibition;
Biological applications of Ru(II) polypyridyl complexes
Keywords: مهار آنزیم; FDA; United States Food and Drug Administration; PDT; photodynamic therapy; PS; photosensitizer; ROS; reactive oxygen species; PACT; photodynamic antimicrobial chemotherapy; NKP-1339; sodium salt of indazolium trans-[tetrachlorobis(1H-indazole)ruthenate(I
Kinetic, spectroscopic and computational docking study of the inhibitory effect of the pesticides 2,4,5-T, 2,4-D and glyphosate on the diphenolase activity of mushroom tyrosinase
Keywords: مهار آنزیم; Tyrosinase; Herbicides; Enzyme inhibition; Fluorescence spectroscopy; Computational Docking Analysis;
Biological effects and chemical characterization of Iris schachtii Markgr. extracts: A new source of bioactive constituents
Keywords: مهار آنزیم; Iris schachtii; Ornamental crops; Bioactive compounds; Enzyme inhibition; Herbal extracts;
Biological evaluation of p-toluene sulphonylhydrazone as carbonic anhydrase IX inhibitors: An approach to fight hypoxia-induced tumors
Keywords: مهار آنزیم; CAIX inhibitors; Tumor hypoxia; Enzyme inhibition;
Impact of different geographical locations on varying profile of bioactives and associated functionalities of caper (Capparis spinosa L.)
Keywords: مهار آنزیم; Capparis spinosa; Antioxidant; Enzyme inhibition; Fatty acids; Essential oils; Nutraceuticals;
Drug-drug interaction potential of antitumor acridine agent C-1748: The substrate of UDP-glucuronosyltransferases 2B7, 2B17 and the inhibitor of 1A9 and 2B7
Keywords: مهار آنزیم; Antitumor agent C-1748; Drug-drug interactions; II phase metabolism; Glucuronidation; Enzyme inhibition; UGT;
A connection between antimicrobial properties of venom peptides and microbial ATP synthase
Keywords: مهار آنزیم; E. coli F1Fo ATP synthase; Venom peptides; Enzyme inhibition;
Synthesis, characterization, antimicrobial activity, carbonic anhydrase enzyme inhibitor effects, and computational studies on new Schiff bases of Sulfa drugs and their Pd(II), Cu(II) complexes
Keywords: مهار آنزیم; Sulfamethoxazole; Sulfisoxazole; Enzyme inhibition; Antibacterial activity; DFT computation;
Cytochrome P4501-inhibiting chemicals amplify aryl hydrocarbon receptor activation and IL-22 production in T helper 17 cells
Keywords: مهار آنزیم; Aryl hydrocarbon receptor; Cytochrome P4501; T helper 17 cells; Interleukin 22; Enzyme inhibition; Synergistic receptor activation;
Design, synthesis and biological assessment of new thiazolylhydrazine derivatives as selective and reversible hMAO-A inhibitors
Keywords: مهار آنزیم; Thiazole; Hydrazine; hMAO enzymes; Enzyme inhibition; Docking;
Pancreatic lipase inhibitory activity of phenolic inhibitor from endophytic Diaporthe arengae
Keywords: مهار آنزیم; Kinetic data; Porcine pancreatic lipase; Enzyme inhibition; Phenol-rich fraction; Orlistat;
In vitro and in vivo cytochrome P450 3A enzyme inhibition by Aframomum melegueta and Denniettia tripetala extracts
Keywords: مهار آنزیم; Cytochrome P450 enzymes; CYP 3A; Enzyme inhibition; Herbal extracts;
A comprehensive study on chemical composition, antioxidant and enzyme inhibition activities of the essential oils of Chenopodium botrys collected from three different parts of Turkey
Keywords: مهار آنزیم; Chenopodium botrys; Essential oil; Chemical composition; Antioxidant activity; Enzyme inhibition;
Taxifolin inhibits rat and human 11β-hydroxysteroid dehydrogenase 2
Keywords: مهار آنزیم; Taxifolin; 11β-Hydroxysteroid dehydrogenase 2; Enzyme inhibition; Noncompetitive; Glucocorticoid;
A simple and novel colorimetric assay for tyrosinase and inhibitor screening using 3,3â²,5,5â²-tetramethylbenzidine as a chromogenic probe
Keywords: مهار آنزیم; Silver ion (Ag+); 3,3â²,5,5â²-tetramethylbenzidine (TMB); Tyrosinase; Enzyme inhibition; Colorimetric assay;
Phosphonodifluoropyruvate is a mechanism-based inhibitor of phosphonopyruvate decarboxylase from Bacteroides fragilis
Keywords: مهار آنزیم; Thiamin diphosphate; CD; UV-Vis; Phosphonate; Enzyme inhibition; PnDFP; phosphonodifluoropyruvate; Phtase; phosphonatase from P. putida; PDC; pyruvate decarboxylase; PnPDC; phosphonopyruvate decarboxylase; ThDP; thiamin diphosphate; YADH; yeast alcohol